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—— (E)-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-3-(5-phenylthiophen-2-yl)prop-2-enamide —— C23H28N2O3S
(E)-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]-3-(5-phenylthiophen-2-yl)prop-2-enamide
—— (E)-3-(3-chlorophenyl)-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]prop-2-enamide —— C19H25ClN2O3
(E)-3-(3-chlorophenyl)-N-[(2R)-2-morpholin-4-yl-2-[(3S)-oxolan-3-yl]ethyl]prop-2-enamide
—— (E)-3-(4-bromophenyl)-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]prop-2-enamide —— C19H25BrN2O3
(E)-3-(4-bromophenyl)-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]prop-2-enamide
—— ethyl 4-[3-[(3R)-3-[(4-ethylphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H37N3O4
ethyl 4-[3-[(3R)-3-[(4-ethylphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-(3-chlorophenyl)-N-[(2R)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]prop-2-enamide —— C19H25ClN2O3
(E)-3-(3-chlorophenyl)-N-[(2R)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]prop-2-enamide
—— (E)-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-3-(5-phenylthiophen-2-yl)prop-2-enamide —— C23H28N2O3S
(E)-N-[(2S)-2-morpholin-4-yl-2-[(3R)-oxolan-3-yl]ethyl]-3-(5-phenylthiophen-2-yl)prop-2-enamide
—— ethyl 4-[3-[(3S)-3-[2-(4-ethoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H39N3O5
ethyl 4-[3-[(3S)-3-[2-(4-ethoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-[(3S)-3-[(5-methylfuran-2-yl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate —— C24H33N3O5
ethyl 3,5-dimethyl-4-[3-[(3S)-3-[(5-methylfuran-2-yl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3S)-3-[(4-chlorophenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H32ClN3O4
ethyl 4-[3-[(3S)-3-[(4-chlorophenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-[3-ethoxy-4-[(1S)-1-phenylethoxy]phenyl]-2-(4-nitrophenyl)prop-2-enenitrile —— C25H22N2O4
(E)-3-[3-ethoxy-4-[(1S)-1-phenylethoxy]phenyl]-2-(4-nitrophenyl)prop-2-enenitrile
—— ethyl 4-[3-[(3R)-3-(1,3-benzodioxol-5-ylmethylcarbamoyl)piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H33N3O6
ethyl 4-[3-[(3R)-3-(1,3-benzodioxol-5-ylmethylcarbamoyl)piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-[(3S)-3-[(3-methylphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate —— C26H35N3O4
ethyl 3,5-dimethyl-4-[3-[(3S)-3-[(3-methylphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[(3-fluorophenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H32FN3O4
ethyl 4-[3-[(3R)-3-[(3-fluorophenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[(2,5-dimethoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H37N3O6
ethyl 4-[3-[(3R)-3-[(2,5-dimethoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[(4-ethoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H37N3O5
ethyl 4-[3-[(3R)-3-[(4-ethoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[(3R)-3-(2-phenylethylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C26H35N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[(3R)-3-(2-phenylethylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[(3S)-3-(2-phenylethylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C26H35N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[(3S)-3-(2-phenylethylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3S)-3-[(2-methoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H35N3O5
ethyl 4-[3-[(3S)-3-[(2-methoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[2-(4-ethoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C28H39N3O5
ethyl 4-[3-[(3R)-3-[2-(4-ethoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-[(3S)-3-[(2-methylphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate —— C26H35N3O4
ethyl 3,5-dimethyl-4-[3-[(3S)-3-[(2-methylphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[4-[[(1R)-1-phenylethyl]carbamoyl]piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C26H35N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[4-[[(1R)-1-phenylethyl]carbamoyl]piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[2-(2-methoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H37N3O5
ethyl 4-[3-[(3R)-3-[2-(2-methoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[(4-fluorophenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H32FN3O4
ethyl 4-[3-[(3R)-3-[(4-fluorophenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[4-[[(2S)-2-phenylpropyl]carbamoyl]piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C27H37N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[4-[[(2S)-2-phenylpropyl]carbamoyl]piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[4-[[(2R)-4-phenylbutan-2-yl]carbamoyl]piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C28H39N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[4-[[(2R)-4-phenylbutan-2-yl]carbamoyl]piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— (E)-3-[2-(2-methylfuran-3-carbonyl)hydrazinyl]-N,N-di(propan-2-yl)but-2-enamide —— C16H25N3O3
(E)-3-[2-(2-methylfuran-3-carbonyl)hydrazinyl]-N,N-di(propan-2-yl)but-2-enamide
—— ethyl 4-[3-[(3S)-3-[2-(2-methoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H37N3O5
ethyl 4-[3-[(3S)-3-[2-(2-methoxyphenyl)ethylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-3-(4-chlorophenyl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)phenyl]prop-2-enamide —— C23H17ClN2O2
(E)-3-(4-chlorophenyl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)phenyl]prop-2-enamide
—— ethyl 4-[3-[(3R)-3-(cycloheptylcarbamoyl)piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H39N3O4
ethyl 4-[3-[(3R)-3-(cycloheptylcarbamoyl)piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3S)-3-[3-(diethylamino)propylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H42N4O4
ethyl 4-[3-[(3S)-3-[3-(diethylamino)propylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C22H28N2O5
ethyl 4-[3-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino]-3-oxopropyl]-1,3,5-trimethylpyrrole-2-carboxylate —— C23H30N2O5
ethyl 4-[3-[[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]amino]-3-oxopropyl]-1,3,5-trimethylpyrrole-2-carboxylate
—— ethyl 4-[3-[(3S)-3-(azepane-1-carbonyl)piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H37N3O4
ethyl 4-[3-[(3S)-3-(azepane-1-carbonyl)piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[[(1R)-1-(1-adamantyl)ethyl]amino]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H36N2O3
ethyl 4-[3-[[(1R)-1-(1-adamantyl)ethyl]amino]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[(3R)-3-(3-phenylpropylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C27H37N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[(3R)-3-(3-phenylpropylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[[(1S)-1-(1-adamantyl)ethyl]amino]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H36N2O3
ethyl 4-[3-[[(1S)-1-(1-adamantyl)ethyl]amino]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3S)-3-[(2,5-dimethoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C27H37N3O6
ethyl 4-[3-[(3S)-3-[(2,5-dimethoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— Ethyl 2-(3-methoxybenzamido)-5-phenylthiophene-3-carboxylate —— C21H19NO4S
Ethyl 2-(3-methoxybenzamido)-5-phenylthiophene-3-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[(3S)-3-(2-thiophen-2-ylethylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C24H33N3O4S
ethyl 3,5-dimethyl-4-[3-oxo-3-[(3S)-3-(2-thiophen-2-ylethylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl (5E)-2-(4-ethylanilino)-4-oxo-5-[(4-phenylmethoxyphenyl)methylidene]thiophene-3-carboxylate —— C29H27NO4S
ethyl (5E)-2-(4-ethylanilino)-4-oxo-5-[(4-phenylmethoxyphenyl)methylidene]thiophene-3-carboxylate
—— ethyl 3,5-dimethyl-4-[3-oxo-3-[(3S)-3-(3-phenylpropylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate —— C27H37N3O4
ethyl 3,5-dimethyl-4-[3-oxo-3-[(3S)-3-(3-phenylpropylcarbamoyl)piperidin-1-yl]propyl]-1H-pyrrole-2-carboxylate
—— ethyl N-[(3R)-1-[(4-cyanophenyl)methylcarbamoyl]piperidin-3-yl]carbamate —— C17H22N4O3
ethyl N-[(3R)-1-[(4-cyanophenyl)methylcarbamoyl]piperidin-3-yl]carbamate
—— ethyl 4-[3-[4-[[(2R)-1-(furan-2-yl)propan-2-yl]carbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H35N3O5
ethyl 4-[3-[4-[[(2R)-1-(furan-2-yl)propan-2-yl]carbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 3,5-dimethyl-4-[3-[(3R)-3-[(5-methylfuran-2-yl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate —— C24H33N3O5
ethyl 3,5-dimethyl-4-[3-[(3R)-3-[(5-methylfuran-2-yl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[[(2S)-butan-2-yl]amino]-3-oxopropyl]-1,3,5-trimethylpyrrole-2-carboxylate —— C17H28N2O3
ethyl 4-[3-[[(2S)-butan-2-yl]amino]-3-oxopropyl]-1,3,5-trimethylpyrrole-2-carboxylate
—— ethyl 4-[3-[(3S)-3-[furan-2-ylmethyl(methyl)carbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C24H33N3O5
ethyl 4-[3-[(3S)-3-[furan-2-ylmethyl(methyl)carbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— (E)-2-cyano-N-[(1R,2R)-2-methylcyclohexyl]-3-(4-prop-2-enoxyphenyl)prop-2-enamide —— C20H24N2O2
(E)-2-cyano-N-[(1R,2R)-2-methylcyclohexyl]-3-(4-prop-2-enoxyphenyl)prop-2-enamide
—— ethyl 4-[3-[4-[[(2S)-butan-2-yl]carbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C22H35N3O4
ethyl 4-[3-[4-[[(2S)-butan-2-yl]carbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[(3-methoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H35N3O5
ethyl 4-[3-[(3R)-3-[(3-methoxyphenyl)methylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— ethyl 4-[3-[(3R)-3-[3-(diethylamino)propylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C25H42N4O4
ethyl 4-[3-[(3R)-3-[3-(diethylamino)propylcarbamoyl]piperidin-1-yl]-3-oxopropyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate