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—— ethyl 2-[[2-(2-amino-2-oxoethoxy)-5-bromophenyl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28BrN3O5S
ethyl 2-[[2-(2-amino-2-oxoethoxy)-5-bromophenyl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 2-[[[2-[[1-[(4-bromophenyl)methyl]pyrrol-2-yl]methyl-butylamino]-2-oxoethyl]-propan-2-ylcarbamoyl]amino]acetate —— C26H37BrN4O4
Ethyl 2-[[[2-[[1-[(4-bromophenyl)methyl]pyrrol-2-yl]methyl-butylamino]-2-oxoethyl]-propan-2-ylcarbamoyl]amino]acetate
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[(2S)-2-[methyl(2-methylpropyl)amino]propyl]prop-2-enamide —— C18H25N3O2
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[(2S)-2-[methyl(2-methylpropyl)amino]propyl]prop-2-enamide
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-(3,5-dimethylphenyl)prop-2-enamide —— C18H16N2O3
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-(3,5-dimethylphenyl)prop-2-enamide
—— ethyl 4-[[(2R)-2-bromopropanoyl]amino]piperidine-1-carboxylate —— C11H19BrN2O3
ethyl 4-[[(2R)-2-bromopropanoyl]amino]piperidine-1-carboxylate
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(2R)-1-methoxypropan-2-yl]prop-2-enamide —— C14H16N2O4
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(2R)-1-methoxypropan-2-yl]prop-2-enamide
—— Ethyl 1-[[4-(furan-2-ylmethylcarbamoyl)phenyl]methyl]-6-methyl-4-(3-methylphenyl)-2-oxo-3,4-dihydropyridine-5-carboxylate —— C29H30N2O5
Ethyl 1-[[4-(furan-2-ylmethylcarbamoyl)phenyl]methyl]-6-methyl-4-(3-methylphenyl)-2-oxo-3,4-dihydropyridine-5-carboxylate
—— (E)-N-[2-(azepan-1-yl)ethyl]-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide —— C18H23N3O2
(E)-N-[2-(azepan-1-yl)ethyl]-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide
—— Ethyl 4-{4-(2-{[4-(ethoxycarbonyl)phenyl]amino}-2-oxoethyl)-5-oxo-2-thioxo-3-[4-(trifluoromethoxy)benzyl]imidazolidin-1-yl}benzoate —— C31H28F3N3O7S
Ethyl 4-{4-(2-{[4-(ethoxycarbonyl)phenyl]amino}-2-oxoethyl)-5-oxo-2-thioxo-3-[4-(trifluoromethoxy)benzyl]imidazolidin-1-yl}benzoate
—— (E)-2-cyano-N-[(2S)-1-(furan-2-yl)propan-2-yl]-3-(3-hydroxyphenyl)prop-2-enamide —— C17H16N2O3
(E)-2-cyano-N-[(2S)-1-(furan-2-yl)propan-2-yl]-3-(3-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-(2-phenoxyethyl)prop-2-enamide —— C18H16N2O3
(E)-2-cyano-3-(3-hydroxyphenyl)-N-(2-phenoxyethyl)prop-2-enamide
—— (E)-2-cyano-N-(2-ethylphenyl)-3-(3-hydroxyphenyl)prop-2-enamide —— C18H16N2O2
(E)-2-cyano-N-(2-ethylphenyl)-3-(3-hydroxyphenyl)prop-2-enamide
—— Ethyl 4-(4-hexanoyl-3-methylpiperazine-1-carbonyl)-2-methyl-6-propylpyrimidine-5-carboxylate —— C23H36N4O4
Ethyl 4-(4-hexanoyl-3-methylpiperazine-1-carbonyl)-2-methyl-6-propylpyrimidine-5-carboxylate
—— Ethyl 5-(dimethylcarbamoyl)-4-methyl-2-[[2-(2-naphthalen-1-yloxyacetyl)oxyacetyl]amino]thiophene-3-carboxylate —— C25H26N2O7S
Ethyl 5-(dimethylcarbamoyl)-4-methyl-2-[[2-(2-naphthalen-1-yloxyacetyl)oxyacetyl]amino]thiophene-3-carboxylate
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[2-(4-methylpiperazin-1-yl)ethyl]prop-2-enamide —— C17H22N4O2
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[2-(4-methylpiperazin-1-yl)ethyl]prop-2-enamide
—— (E)-2-cyano-N-[(1S)-1-cyclopropylethyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C15H16N2O3
(E)-2-cyano-N-[(1S)-1-cyclopropylethyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-[3-(diethylamino)propyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C17H23N3O3
(E)-2-cyano-N-[3-(diethylamino)propyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— (E)-3-(4-butan-2-ylphenyl)-N-(3-chloro-2-methylphenyl)-3-hydroxy-2-pyridin-1-ium-1-ylprop-2-enethioamide —— C25H26ClN2OS+
(E)-3-(4-butan-2-ylphenyl)-N-(3-chloro-2-methylphenyl)-3-hydroxy-2-pyridin-1-ium-1-ylprop-2-enethioamide
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]prop-2-enamide —— C15H13N3O2S
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]prop-2-enamide
—— ethyl 4-[[(2S)-2-bromopropanoyl]amino]piperidine-1-carboxylate —— C11H19BrN2O3
ethyl 4-[[(2S)-2-bromopropanoyl]amino]piperidine-1-carboxylate
—— (E)-2-cyano-N-(2-cyclohexylethyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C18H22N2O3
(E)-2-cyano-N-(2-cyclohexylethyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-(4-hydroxyphenyl)-N-[(2-hydroxyphenyl)methyl]prop-2-enamide —— C17H14N2O3
(E)-2-cyano-3-(4-hydroxyphenyl)-N-[(2-hydroxyphenyl)methyl]prop-2-enamide
—— (E)-3-(naphthalen-1-ylamino)-1-phenyl-2-pyridin-1-ium-1-yl-3-sulfanylideneprop-1-en-1-olate —— C24H18N2OS
(E)-3-(naphthalen-1-ylamino)-1-phenyl-2-pyridin-1-ium-1-yl-3-sulfanylideneprop-1-en-1-olate
—— (E)-N-[(2-chlorophenyl)methyl]-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide —— C17H13ClN2O2
(E)-N-[(2-chlorophenyl)methyl]-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-3-(4-hydroxyphenyl)prop-2-enamide —— C16H20N4O3
(E)-2-cyano-N-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-3-(4-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-3-(4-hydroxyphenyl)prop-2-enamide —— C17H18N4O2
(E)-2-cyano-N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-3-(4-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1R)-1-(1,3-thiazol-5-yl)ethyl]prop-2-enamide —— C15H13N3O2S
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1R)-1-(1,3-thiazol-5-yl)ethyl]prop-2-enamide
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-(2-oxo-2-piperidin-1-ylethyl)prop-2-enamide —— C17H19N3O3
(E)-2-cyano-3-(3-hydroxyphenyl)-N-(2-oxo-2-piperidin-1-ylethyl)prop-2-enamide
—— Ethyl 2-{[(2-methoxyphenyl)methyl]amino}-7-oxo-4H,7H-[1,2,4]triazolo[1,5-A]pyrimidine-6-carboxylate —— C16H17N5O4
Ethyl 2-{[(2-methoxyphenyl)methyl]amino}-7-oxo-4H,7H-[1,2,4]triazolo[1,5-A]pyrimidine-6-carboxylate
—— (E)-2-cyano-N-[2-(dipropylamino)ethyl]-3-(3-hydroxyphenyl)prop-2-enamide —— C18H25N3O2
(E)-2-cyano-N-[2-(dipropylamino)ethyl]-3-(3-hydroxyphenyl)prop-2-enamide
—— (E)-3-(4-hydroxyphenyl)-2-[(3R)-3-methylpiperidine-1-carbonyl]prop-2-enenitrile —— C16H18N2O2
(E)-3-(4-hydroxyphenyl)-2-[(3R)-3-methylpiperidine-1-carbonyl]prop-2-enenitrile
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[(5-methyl-1,3-thiazol-2-yl)methyl]prop-2-enamide —— C15H13N3O2S
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[(5-methyl-1,3-thiazol-2-yl)methyl]prop-2-enamide
—— Ethyl 2-[[2-[[5-(3-bromophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H20BrN3O4S2
Ethyl 2-[[2-[[5-(3-bromophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 1-[2-[4-chloro-6-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylacetyl]piperidine-4-carboxylate —— C23H34ClN5O4S
Ethyl 1-[2-[4-chloro-6-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]pyrimidin-2-yl]sulfanylacetyl]piperidine-4-carboxylate
—— (E)-2-cyano-N-[(2R)-1-(dimethylamino)butan-2-yl]-3-(4-hydroxyphenyl)prop-2-enamide —— C16H21N3O2
(E)-2-cyano-N-[(2R)-1-(dimethylamino)butan-2-yl]-3-(4-hydroxyphenyl)prop-2-enamide
—— (E)-3-(3,4-dihydroxyphenyl)-2-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]prop-2-enenitrile —— C17H20N2O3
(E)-3-(3,4-dihydroxyphenyl)-2-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]prop-2-enenitrile
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-(2-thiophen-2-ylpropan-2-yl)prop-2-enamide —— C17H16N2O2S
(E)-2-cyano-3-(3-hydroxyphenyl)-N-(2-thiophen-2-ylpropan-2-yl)prop-2-enamide
—— (E)-2-cyano-N-[(2R)-1-(furan-2-yl)propan-2-yl]-3-(3-hydroxyphenyl)prop-2-enamide —— C17H16N2O3
(E)-2-cyano-N-[(2R)-1-(furan-2-yl)propan-2-yl]-3-(3-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-N-[(1R)-1-cyclopropylethyl]-3-(3-hydroxyphenyl)prop-2-enamide —— C15H16N2O2
(E)-2-cyano-N-[(1R)-1-cyclopropylethyl]-3-(3-hydroxyphenyl)prop-2-enamide
—— ethyl (2R)-2-(3-chloropropanoylamino)-3-phenylpropanoate —— C14H18ClNO3
ethyl (2R)-2-(3-chloropropanoylamino)-3-phenylpropanoate
—— Ethyl 2-[[2-cyano-3-[5-(2,5-dichloro-4-nitrophenyl)furan-2-yl]prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H19Cl2N3O6S
Ethyl 2-[[2-cyano-3-[5-(2,5-dichloro-4-nitrophenyl)furan-2-yl]prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[2-(bromomethoxy)benzoyl]amino]acetate —— C12H14BrNO4
ethyl 2-[[2-(bromomethoxy)benzoyl]amino]acetate
—— (E)-2-cyano-N-[(1S)-1-cyclopropylethyl]-3-(3-hydroxyphenyl)prop-2-enamide —— C15H16N2O2
(E)-2-cyano-N-[(1S)-1-cyclopropylethyl]-3-(3-hydroxyphenyl)prop-2-enamide
—— ethyl (2R)-2-[(2-bromo-2-methylpropanoyl)amino]-3-methylbutanoate —— C11H20BrNO3
ethyl (2R)-2-[(2-bromo-2-methylpropanoyl)amino]-3-methylbutanoate
—— ethyl (2R)-2-[[(2S)-2-chloro-2-phenylacetyl]amino]propanoate —— C13H16ClNO3
ethyl (2R)-2-[[(2S)-2-chloro-2-phenylacetyl]amino]propanoate
—— (E)-3-(3,4-dihydroxyphenyl)-2-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]prop-2-enenitrile —— C17H20N2O3
(E)-3-(3,4-dihydroxyphenyl)-2-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]prop-2-enenitrile
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]prop-2-enamide —— C15H13N3O3S
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]prop-2-enamide
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]prop-2-enamide —— C20H18N2O2
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]prop-2-enamide
—— ethyl (2S)-2-[(2-bromo-2-methylpropanoyl)amino]-4-methylpentanoate —— C12H22BrNO3
ethyl (2S)-2-[(2-bromo-2-methylpropanoyl)amino]-4-methylpentanoate
—— Ethyl 5-(diethylcarbamoyl)-4-methyl-2-[[2-(4-thiophen-2-ylsulfonylpiperazin-1-yl)acetyl]amino]thiophene-3-carboxylate —— C23H32N4O6S3
Ethyl 5-(diethylcarbamoyl)-4-methyl-2-[[2-(4-thiophen-2-ylsulfonylpiperazin-1-yl)acetyl]amino]thiophene-3-carboxylate