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—— (E)-3-(3-chloro-5-methoxy-4-propoxyphenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide —— C21H29ClN2O4
(E)-3-(3-chloro-5-methoxy-4-propoxyphenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide
—— ethyl 5-[[(2S)-1-(furan-2-carbonyl)pyrrolidine-2-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C21H20N2O5S
ethyl 5-[[(2S)-1-(furan-2-carbonyl)pyrrolidine-2-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— (E)-3-[2-chloro-5-(trifluoromethyl)phenyl]-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide —— C18H20ClF3N2O2
(E)-3-[2-chloro-5-(trifluoromethyl)phenyl]-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide
—— (E)-3-(2,5-dichlorophenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide —— C17H20Cl2N2O2
(E)-3-(2,5-dichlorophenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide
—— (E)-N-(3-oxo-3-piperidin-1-ylpropyl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C20H28N2O5
(E)-N-(3-oxo-3-piperidin-1-ylpropyl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide —— C22H26N4O2
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide
—— (E)-3-(4-bromophenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide —— C17H21BrN2O2
(E)-3-(4-bromophenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide
—— (E)-N-(3-oxo-3-piperidin-1-ylpropyl)-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C20H28N2O5
(E)-N-(3-oxo-3-piperidin-1-ylpropyl)-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-cyclopropyl-N-[(2R)-3-methylbutan-2-yl]prop-2-enamide —— C22H27N3O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-cyclopropyl-N-[(2R)-3-methylbutan-2-yl]prop-2-enamide
—— (E)-N-(2-cyclopentylsulfanylethyl)-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C18H25NO3S
(E)-N-(2-cyclopentylsulfanylethyl)-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— ethyl 5-[[(3S)-1-(2-methylpropanoyl)piperidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C21H26N2O4S
ethyl 5-[[(3S)-1-(2-methylpropanoyl)piperidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— ethyl 5-[[2-(4-oxo-3H-phthalazin-1-yl)acetyl]amino]-1-benzothiophene-2-carboxylate —— C21H17N3O4S
ethyl 5-[[2-(4-oxo-3H-phthalazin-1-yl)acetyl]amino]-1-benzothiophene-2-carboxylate
—— (E)-N-(2-cyclopentylsulfanylethyl)-3-(4-methoxyphenyl)prop-2-enamide —— C17H23NO2S
(E)-N-(2-cyclopentylsulfanylethyl)-3-(4-methoxyphenyl)prop-2-enamide
—— ethyl 5-[[(3R)-1-(2-methylpropanoyl)piperidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C21H26N2O4S
ethyl 5-[[(3R)-1-(2-methylpropanoyl)piperidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— ethyl 5-[[(2R)-1-acetylpyrrolidine-2-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C18H20N2O4S
ethyl 5-[[(2R)-1-acetylpyrrolidine-2-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— ethyl 4-[(2S)-3-[benzyl(methyl)amino]-2-hydroxypropoxy]benzoate —— C20H25NO4
ethyl 4-[(2S)-3-[benzyl(methyl)amino]-2-hydroxypropoxy]benzoate
—— (E,2R)-5-(2-methoxyphenyl)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-3-oxopent-4-enenitrile —— C22H18N2O2S
(E,2R)-5-(2-methoxyphenyl)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-3-oxopent-4-enenitrile
—— ethyl 2-[(2-chloroacetyl)amino]-5-methyl-4-[(2R)-2-methylbutyl]thiophene-3-carboxylate —— C15H22ClNO3S
ethyl 2-[(2-chloroacetyl)amino]-5-methyl-4-[(2R)-2-methylbutyl]thiophene-3-carboxylate
—— (E,2S)-5-(2-methoxyphenyl)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-3-oxopent-4-enenitrile —— C22H18N2O2S
(E,2S)-5-(2-methoxyphenyl)-2-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-3-oxopent-4-enenitrile
—— ethyl 4-[(2S)-3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]benzoate —— C18H28N2O4
ethyl 4-[(2S)-3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]benzoate
—— (E)-3-(4-bromophenyl)-N-[4-methoxy-3-(2-methoxyethoxy)phenyl]prop-2-enamide —— C19H20BrNO4
(E)-3-(4-bromophenyl)-N-[4-methoxy-3-(2-methoxyethoxy)phenyl]prop-2-enamide
—— (E)-N-(2-cyclopentylsulfanylethyl)-3-(2-methoxyphenyl)prop-2-enamide —— C17H23NO2S
(E)-N-(2-cyclopentylsulfanylethyl)-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-[1-(4-fluorophenyl)-2,5-dimethylpyrrol-3-yl]prop-2-enoate —— C16H12FN2O2-
(E)-2-cyano-3-[1-(4-fluorophenyl)-2,5-dimethylpyrrol-3-yl]prop-2-enoate
—— ethyl 5-[[(3R)-1-pyrimidin-2-ylpiperidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C21H22N4O3S
ethyl 5-[[(3R)-1-pyrimidin-2-ylpiperidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— (E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide —— C20H26F2N2O4
(E)-3-[4-(difluoromethoxy)-3-ethoxyphenyl]-N-(3-oxo-3-piperidin-1-ylpropyl)prop-2-enamide
—— (E)-3-(2,3-dimethoxyphenyl)-N-(4-ethoxyphenyl)prop-2-enamide —— C19H21NO4
(E)-3-(2,3-dimethoxyphenyl)-N-(4-ethoxyphenyl)prop-2-enamide
—— ethyl 4-[(2R)-3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]benzoate —— C18H28N2O4
ethyl 4-[(2R)-3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]benzoate
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[4-methoxy-3-(2-methoxyethoxy)phenyl]prop-2-enamide —— C20H20N2O5
(E)-3-(1,3-benzoxazol-2-yl)-N-[4-methoxy-3-(2-methoxyethoxy)phenyl]prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-cyclopropyl-N-[(2S)-3-methylbutan-2-yl]prop-2-enamide —— C22H27N3O
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-cyclopropyl-N-[(2S)-3-methylbutan-2-yl]prop-2-enamide
—— (E)-3-[4-(4-tert-butylphenoxy)-3-nitrophenyl]-2-cyano-N-(3,4-dimethoxyphenyl)prop-2-enamide —— C28H27N3O6
(E)-3-[4-(4-tert-butylphenoxy)-3-nitrophenyl]-2-cyano-N-(3,4-dimethoxyphenyl)prop-2-enamide
—— ethyl (2Z)-2-[(5Z)-5-[(4-methylphenyl)methylidene]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C23H28N2O4S
ethyl (2Z)-2-[(5Z)-5-[(4-methylphenyl)methylidene]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 4-[(2R)-3-[benzyl(methyl)amino]-2-hydroxypropoxy]benzoate —— C20H25NO4
ethyl 4-[(2R)-3-[benzyl(methyl)amino]-2-hydroxypropoxy]benzoate
—— Ethyl 4-methyl-2-[[2-(4-methylsulfonyl-3-nitrobenzoyl)oxyacetyl]amino]-5-phenylthiophene-3-carboxylate —— C24H22N2O9S2
Ethyl 4-methyl-2-[[2-(4-methylsulfonyl-3-nitrobenzoyl)oxyacetyl]amino]-5-phenylthiophene-3-carboxylate
—— ethyl 5-[[(3S)-1-(cyclopropylmethyl)-5-oxopyrrolidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C20H22N2O4S
ethyl 5-[[(3S)-1-(cyclopropylmethyl)-5-oxopyrrolidine-3-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— (E)-N-(3-pyrazol-1-ylpropyl)-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide —— C21H22N4O2
(E)-N-(3-pyrazol-1-ylpropyl)-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-(2-cyclopentylsulfanylethyl)prop-2-enamide —— C17H21NO3S
(E)-3-(1,3-benzodioxol-5-yl)-N-(2-cyclopentylsulfanylethyl)prop-2-enamide
—— ethyl 5-[[(2S)-1-acetylpyrrolidine-2-carbonyl]amino]-1-benzothiophene-2-carboxylate —— C18H20N2O4S
ethyl 5-[[(2S)-1-acetylpyrrolidine-2-carbonyl]amino]-1-benzothiophene-2-carboxylate
—— (E)-N-[(3,4-dimethoxyphenyl)methyl]-3-(2-methoxyphenyl)prop-2-enamide —— C19H21NO4
(E)-N-[(3,4-dimethoxyphenyl)methyl]-3-(2-methoxyphenyl)prop-2-enamide
—— ethyl (2S)-2-[(5-ethylfuran-2-carbonyl)amino]-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]acetate —— C22H24FN3O4
ethyl (2S)-2-[(5-ethylfuran-2-carbonyl)amino]-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]acetate
—— ethyl 4-[(4Z)-4-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C26H20BrNO6
ethyl 4-[(4Z)-4-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— (E)-N-(6-bromo-1,3-benzothiazol-2-yl)-3-(3-fluorophenyl)prop-2-enamide —— C16H10BrFN2OS
(E)-N-(6-bromo-1,3-benzothiazol-2-yl)-3-(3-fluorophenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-1-(4-naphthalen-2-ylsulfonylpiperazin-1-yl)prop-2-en-1-one —— C24H22N2O5S
(E)-3-(1,3-benzodioxol-5-yl)-1-(4-naphthalen-2-ylsulfonylpiperazin-1-yl)prop-2-en-1-one
—— (E)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide —— C20H19N3O2S
(E)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide
—— (E,2S)-2-(1H-benzimidazol-2-yl)-5-(4-chlorophenyl)-3-oxopent-4-enenitrile —— C18H12ClN3O
(E,2S)-2-(1H-benzimidazol-2-yl)-5-(4-chlorophenyl)-3-oxopent-4-enenitrile
—— ethyl (2R)-2-[(5-ethylfuran-2-carbonyl)amino]-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]acetate —— C22H24FN3O4
ethyl (2R)-2-[(5-ethylfuran-2-carbonyl)amino]-2-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]acetate
—— (E)-N-(5-propyl-1,3,4-thiadiazol-2-yl)-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide —— C20H20N4O2S
(E)-N-(5-propyl-1,3,4-thiadiazol-2-yl)-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide
—— Ethyl 5-amino-3-[3-(1,3-benzothiazol-2-yl)propanoyloxymethyl]-4-cyanothiophene-2-carboxylate —— C19H17N3O4S2
Ethyl 5-amino-3-[3-(1,3-benzothiazol-2-yl)propanoyloxymethyl]-4-cyanothiophene-2-carboxylate
—— ethyl N-[(3R)-1-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propylcarbamoyl]piperidin-3-yl]carbamate —— C21H32N4O3
ethyl N-[(3R)-1-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propylcarbamoyl]piperidin-3-yl]carbamate
—— ethyl 2-[[2-(diethylamino)acetyl]amino]-5-(dimethylcarbamoyl)-4-methylthiophene-3-carboxylate —— C17H27N3O4S
ethyl 2-[[2-(diethylamino)acetyl]amino]-5-(dimethylcarbamoyl)-4-methylthiophene-3-carboxylate
—— (E,2R)-2-(1H-benzimidazol-2-yl)-5-(4-chlorophenyl)-3-oxopent-4-enenitrile —— C18H12ClN3O
(E,2R)-2-(1H-benzimidazol-2-yl)-5-(4-chlorophenyl)-3-oxopent-4-enenitrile