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—— ethyl 2-[(4-ethoxyphenyl)methylidene]-7-methyl-3-oxo-5-(2-propan-2-yloxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H30N2O5S
ethyl 2-[(4-ethoxyphenyl)methylidene]-7-methyl-3-oxo-5-(2-propan-2-yloxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 2-(2-iodobenzamido)benzo[d]thiazole-6-carboxylate —— C17H13IN2O3S
Ethyl 2-(2-iodobenzamido)benzo[d]thiazole-6-carboxylate
—— Ethyl 5-[(2,3-dimethoxyphenyl)methylidene]-2-methylidene-4-oxopyrrolidine-3-carboxylate —— C17H19NO5
Ethyl 5-[(2,3-dimethoxyphenyl)methylidene]-2-methylidene-4-oxopyrrolidine-3-carboxylate
—— Ethyl 6-(3-{[(3,4-dichlorophenyl)carbamoyl]amino}phenyl)-8-methyl-2H,3H,4H,6H-pyrimido[2,1-B][1,3]thiazine-7-carboxylate —— C24H24Cl2N4O3S
Ethyl 6-(3-{[(3,4-dichlorophenyl)carbamoyl]amino}phenyl)-8-methyl-2H,3H,4H,6H-pyrimido[2,1-B][1,3]thiazine-7-carboxylate
—— ethyl (2R)-2-[[4-(chloromethyl)-5-methylfuran-2-carbonyl]amino]-4-methylpentanoate —— C15H22ClNO4
ethyl (2R)-2-[[4-(chloromethyl)-5-methylfuran-2-carbonyl]amino]-4-methylpentanoate
—— ethyl 2-benzylsulfanyl-5-[4-(dimethylamino)phenyl]-7-methyl-4-oxo-5,8-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carboxylate —— C26H28N4O3S
ethyl 2-benzylsulfanyl-5-[4-(dimethylamino)phenyl]-7-methyl-4-oxo-5,8-dihydro-3H-pyrido[2,3-d]pyrimidine-6-carboxylate
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(3R)-octan-3-yl]prop-2-enamide —— C18H24N2O3
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(3R)-octan-3-yl]prop-2-enamide
—— (E)-N-[2-(butylamino)-2-oxoethyl]-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C16H19N3O4
(E)-N-[2-(butylamino)-2-oxoethyl]-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— Ethyl 4-{[3-(2,4-dimethylphenyl)-6-(4-fluorophenyl)-7-oxo-2-sulfanylidene-2H,3H,6H,7H-[1,3]thiazolo[4,5-D]pyrimidin-5-YL]sulfanyl}-3-oxobutanoate —— C25H22FN3O4S3
Ethyl 4-{[3-(2,4-dimethylphenyl)-6-(4-fluorophenyl)-7-oxo-2-sulfanylidene-2H,3H,6H,7H-[1,3]thiazolo[4,5-D]pyrimidin-5-YL]sulfanyl}-3-oxobutanoate
—— (E)-2-cyano-3-(4-hydroxyphenyl)-N-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)prop-2-enamide —— C15H14N4O3
(E)-2-cyano-3-(4-hydroxyphenyl)-N-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)prop-2-enamide
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-thiophen-2-ylethyl]prop-2-enamide —— C16H14N2O3S
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-thiophen-2-ylethyl]prop-2-enamide
—— Ethyl 2-{2-[(5-{[2-(4-chlorophenoxy)acetamido]methyl}-4-(2,3-dimethylphenyl)-4H-1,2,4-triazol-3-YL)sulfanyl]acetamido}-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate —— C31H32ClN5O5S2
Ethyl 2-{2-[(5-{[2-(4-chlorophenoxy)acetamido]methyl}-4-(2,3-dimethylphenyl)-4H-1,2,4-triazol-3-YL)sulfanyl]acetamido}-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate
—— (E)-N-(3-ethyl-4-methoxybenzo[d]thiazol-2(3H)-ylidene)-2,6-dimethoxybenzamide —— C19H20N2O4S
(E)-N-(3-ethyl-4-methoxybenzo[d]thiazol-2(3H)-ylidene)-2,6-dimethoxybenzamide
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[3-(dimethylamino)propyl]prop-2-enamide —— C15H19N3O3
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[3-(dimethylamino)propyl]prop-2-enamide
—— ethyl 2-({[3-bromo-5-(4-methoxyphenyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]carbonyl}amino)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C25H20BrF3N4O4S
ethyl 2-({[3-bromo-5-(4-methoxyphenyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]carbonyl}amino)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]prop-2-enamide —— C18H23N3O2
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]prop-2-enamide
—— ethyl 2-[[4-[(4-bromophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H29BrN2O6S
ethyl 2-[[4-[(4-bromophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-{[({5-[(4-chloro-1H-pyrazol-1-yl)methyl]furan-2-yl}carbonyl)carbamothioyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H21ClN4O4S2
ethyl 2-{[({5-[(4-chloro-1H-pyrazol-1-yl)methyl]furan-2-yl}carbonyl)carbamothioyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 8-methyl-4-oxo-6-phenyl-2-(pyridin-4-yl)-4H,6H-pyrimido[2,1-b][1,3]thiazine-7-carboxylate —— C22H19N3O3S
ethyl 8-methyl-4-oxo-6-phenyl-2-(pyridin-4-yl)-4H,6H-pyrimido[2,1-b][1,3]thiazine-7-carboxylate
—— ethyl 3-(benzo[d]thiazol-2-yl)-2-(4-(tert-butyl)benzamido)-4,5-dihydrothieno[2,3-c]pyridine-6(7H)-carboxylate —— C28H29N3O3S2
ethyl 3-(benzo[d]thiazol-2-yl)-2-(4-(tert-butyl)benzamido)-4,5-dihydrothieno[2,3-c]pyridine-6(7H)-carboxylate
—— Ethyl 6-acetyl-3-(4-methoxybenzoyl)-1-indolizinecarboxylate —— C21H19NO5
Ethyl 6-acetyl-3-(4-methoxybenzoyl)-1-indolizinecarboxylate
—— ethyl 2-[[6-[(3-ethoxycarbonyl-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)carbamoyl]pyridine-2-carbonyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C31H35N3O6S2
ethyl 2-[[6-[(3-ethoxycarbonyl-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)carbamoyl]pyridine-2-carbonyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— Ethyl 7-chloro-2-methyl-5-(naphthalene-2-sulfonamido)benzofuran-3-carboxylate —— C22H18ClNO5S
Ethyl 7-chloro-2-methyl-5-(naphthalene-2-sulfonamido)benzofuran-3-carboxylate
—— Ethyl 4-{[3-(4-bromophenyl)-[1,2,4]triazolo[3,4-B][1,3]thiazol-6-YL]methyl}piperazine-1-carboxylate —— C18H20BrN5O2S
Ethyl 4-{[3-(4-bromophenyl)-[1,2,4]triazolo[3,4-B][1,3]thiazol-6-YL]methyl}piperazine-1-carboxylate
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[2-[(3R)-3-methylpiperidin-1-yl]ethyl]prop-2-enamide —— C18H23N3O2
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[2-[(3R)-3-methylpiperidin-1-yl]ethyl]prop-2-enamide
—— Ethyl 2-[3-oxo-1-(2-oxo-6-thia-1,8-diazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carbonyl)piperazin-2-yl]acetate —— C19H18N4O5S
Ethyl 2-[3-oxo-1-(2-oxo-6-thia-1,8-diazatricyclo[7.4.0.03,7]trideca-3(7),4,8,10,12-pentaene-5-carbonyl)piperazin-2-yl]acetate
—— Ethyl 5-methyl-4-(4-methylphenyl)-2-[[2-(2-nitropyridin-3-yl)oxyacetyl]amino]thiophene-3-carboxylate —— C22H21N3O6S
Ethyl 5-methyl-4-(4-methylphenyl)-2-[[2-(2-nitropyridin-3-yl)oxyacetyl]amino]thiophene-3-carboxylate
—— ethyl (2R)-2-(3-bromopropanoylamino)-3-methylbutanoate —— C10H18BrNO3
ethyl (2R)-2-(3-bromopropanoylamino)-3-methylbutanoate
—— ethyl (2S)-2-[[5-[(1R)-1-chloroethyl]furan-2-carbonyl]amino]-3-methylbutanoate —— C14H20ClNO4
ethyl (2S)-2-[[5-[(1R)-1-chloroethyl]furan-2-carbonyl]amino]-3-methylbutanoate
—— (E)-2-cyano-N-(3-fluorophenyl)-3-(4-hydroxyphenyl)prop-2-enamide —— C16H11FN2O2
(E)-2-cyano-N-(3-fluorophenyl)-3-(4-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-(4-hydroxyphenyl)-N-[(1R)-1-(2-methyl-1,3-thiazol-5-yl)ethyl]prop-2-enamide —— C16H15N3O2S
(E)-2-cyano-3-(4-hydroxyphenyl)-N-[(1R)-1-(2-methyl-1,3-thiazol-5-yl)ethyl]prop-2-enamide
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-pyridin-2-ylprop-2-enamide —— C15H11N3O3
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-pyridin-2-ylprop-2-enamide
—— (E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(3S)-octan-3-yl]prop-2-enamide —— C18H24N2O3
(E)-2-cyano-3-(3,4-dihydroxyphenyl)-N-[(3S)-octan-3-yl]prop-2-enamide
—— (E)-2-cyano-3-(4-hydroxyphenyl)-N-[4-oxo-4-(propylamino)butyl]prop-2-enamide —— C17H21N3O3
(E)-2-cyano-3-(4-hydroxyphenyl)-N-[4-oxo-4-(propylamino)butyl]prop-2-enamide
—— ethyl 2-[[(2S)-2-chloro-2-(4-methoxyphenyl)acetyl]amino]acetate —— C13H16ClNO4
ethyl 2-[[(2S)-2-chloro-2-(4-methoxyphenyl)acetyl]amino]acetate
—— ethyl (2R,3R)-2-(3-chloropropanoylamino)-3-methylpentanoate —— C11H20ClNO3
ethyl (2R,3R)-2-(3-chloropropanoylamino)-3-methylpentanoate
—— ethyl (2R)-2-[[5-[(1S)-1-chloroethyl]furan-2-carbonyl]amino]-3-methylbutanoate —— C14H20ClNO4
ethyl (2R)-2-[[5-[(1S)-1-chloroethyl]furan-2-carbonyl]amino]-3-methylbutanoate
—— (E)-2-cyano-3-(4-hydroxyphenyl)-N-(2-phenoxyethyl)prop-2-enamide —— C18H16N2O3
(E)-2-cyano-3-(4-hydroxyphenyl)-N-(2-phenoxyethyl)prop-2-enamide
—— (E)-2-cyano-3-(4-hydroxyphenyl)-N-[(1S)-1-(2-methyl-1,3-thiazol-5-yl)ethyl]prop-2-enamide —— C16H15N3O2S
(E)-2-cyano-3-(4-hydroxyphenyl)-N-[(1S)-1-(2-methyl-1,3-thiazol-5-yl)ethyl]prop-2-enamide
—— ethyl (2S)-2-[[4-(chloromethyl)-5-methylfuran-2-carbonyl]amino]-4-methylpentanoate —— C15H22ClNO4
ethyl (2S)-2-[[4-(chloromethyl)-5-methylfuran-2-carbonyl]amino]-4-methylpentanoate
—— ethyl (2S)-2-(3-bromopropanoylamino)-3-methylbutanoate —— C10H18BrNO3
ethyl (2S)-2-(3-bromopropanoylamino)-3-methylbutanoate
—— (E)-2-cyano-N-(cyclopentylmethyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C16H18N2O3
(E)-2-cyano-N-(cyclopentylmethyl)-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— ethyl (2R)-2-[[5-[(1R)-1-chloroethyl]furan-2-carbonyl]amino]-3-methylbutanoate —— C14H20ClNO4
ethyl (2R)-2-[[5-[(1R)-1-chloroethyl]furan-2-carbonyl]amino]-3-methylbutanoate
—— (E)-2-cyano-N-(2-hydroxy-5-methylphenyl)-3-(3-hydroxyphenyl)prop-2-enamide —— C17H14N2O3
(E)-2-cyano-N-(2-hydroxy-5-methylphenyl)-3-(3-hydroxyphenyl)prop-2-enamide
—— ethyl 2-[[(2R)-2-chloro-2-(4-methoxyphenyl)acetyl]amino]acetate —— C13H16ClNO4
ethyl 2-[[(2R)-2-chloro-2-(4-methoxyphenyl)acetyl]amino]acetate
—— ethyl 3-cyano-2-[[2-[(4-methylphenyl)sulfonylamino]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate —— C25H24N4O5S2
ethyl 3-cyano-2-[[2-[(4-methylphenyl)sulfonylamino]benzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate
—— ethyl (2S)-2-[[(2R)-2-bromopropanoyl]amino]-4-methylsulfanylbutanoate —— C10H18BrNO3S
ethyl (2S)-2-[[(2R)-2-bromopropanoyl]amino]-4-methylsulfanylbutanoate
—— ethyl (2R,3S)-2-(3-chloropropanoylamino)-3-methylpentanoate —— C11H20ClNO3
ethyl (2R,3S)-2-(3-chloropropanoylamino)-3-methylpentanoate
—— ethyl 1-[5-[(1S)-1-chloroethyl]furan-2-carbonyl]piperidine-4-carboxylate —— C15H20ClNO4
ethyl 1-[5-[(1S)-1-chloroethyl]furan-2-carbonyl]piperidine-4-carboxylate
—— Ethyl 2-[[2-[2-[(3,6-dimethyl-1,3-benzothiazol-2-ylidene)amino]-2-oxoethyl]sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H27N3O4S3
Ethyl 2-[[2-[2-[(3,6-dimethyl-1,3-benzothiazol-2-ylidene)amino]-2-oxoethyl]sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate