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—— Ethyl 4-[[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]-(3-morpholin-4-ylpropyl)amino]-4-oxobutanoate —— C19H30N4O5S
Ethyl 4-[[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]-(3-morpholin-4-ylpropyl)amino]-4-oxobutanoate
—— Ethyl 4-[3-[5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]-2,5-dioxopyrrolidin-1-yl]benzoate —— C23H17FN2O6S
Ethyl 4-[3-[5-[(4-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]-2,5-dioxopyrrolidin-1-yl]benzoate
—— Ethyl 4-(2,6-dipyridin-2-ylpyrimidin-4-yl)piperazine-1-carboxylate —— C21H22N6O2
Ethyl 4-(2,6-dipyridin-2-ylpyrimidin-4-yl)piperazine-1-carboxylate
—— (E)-3-(4-acetamidophenyl)-N-[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]prop-2-enamide —— C21H18FN3O3S
(E)-3-(4-acetamidophenyl)-N-[4-(3-fluoro-4-methoxyphenyl)-1,3-thiazol-2-yl]prop-2-enamide
—— ethyl 2-[[1-[(3,4-dichlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-8,8a-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H33Cl2N3O3S
ethyl 2-[[1-[(3,4-dichlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-8,8a-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl N-[1-(3-aminophenyl)ethylideneamino]carbamate —— C11H15N3O2
ethyl N-[1-(3-aminophenyl)ethylideneamino]carbamate
—— (E)-N-[3-(2-methylbenzimidazol-1-yl)propyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C24H26N4O2
(E)-N-[3-(2-methylbenzimidazol-1-yl)propyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— (E)-2-cyano-3-[2,5-dimethyl-1-(3-methylbutyl)pyrrol-3-yl]-N-[2-oxo-2-(propylamino)ethyl]prop-2-enamide —— C20H30N4O2
(E)-2-cyano-3-[2,5-dimethyl-1-(3-methylbutyl)pyrrol-3-yl]-N-[2-oxo-2-(propylamino)ethyl]prop-2-enamide
—— Ethyl 6-tert-butyl-2-{[(3-methyl-4-nitrophenyl)carbonyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H28N2O5S
Ethyl 6-tert-butyl-2-{[(3-methyl-4-nitrophenyl)carbonyl]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-(5-methylpyridin-2-yl)-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C20H19N3O2S
(E)-N-(5-methylpyridin-2-yl)-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— Ethyl 1-[2-[4-[methyl-(4-methylphenyl)sulfonylamino]phenoxy]acetyl]piperidine-3-carboxylate —— C24H30N2O6S
Ethyl 1-[2-[4-[methyl-(4-methylphenyl)sulfonylamino]phenoxy]acetyl]piperidine-3-carboxylate
—— (E)-2-cyano-3-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]prop-2-enamide —— C23H36N4O2
(E)-2-cyano-3-[1-[(2R)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]prop-2-enamide
—— (E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-(5-methylpyridin-2-yl)prop-2-enamide —— C20H18N4O2S
(E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-(5-methylpyridin-2-yl)prop-2-enamide
—— (E)-N-[2-(dimethylamino)-2-oxoethyl]-3-[3-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C18H21N3O3S
(E)-N-[2-(dimethylamino)-2-oxoethyl]-3-[3-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— Ethyl 2-[2-({8-oxo-5H,6H,7H,8H-[1,3,4]thiadiazolo[3,2-A][1,3]diazepin-2-YL}sulfanyl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C19H22N4O4S3
Ethyl 2-[2-({8-oxo-5H,6H,7H,8H-[1,3,4]thiadiazolo[3,2-A][1,3]diazepin-2-YL}sulfanyl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-2-cyano-3-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]prop-2-enamide —— C23H36N4O2
(E)-2-cyano-3-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]prop-2-enamide
—— Ethyl 4-[(1-methylsulfonylpiperidine-4-carbonyl)amino]piperidine-1-carboxylate —— C15H27N3O5S
Ethyl 4-[(1-methylsulfonylpiperidine-4-carbonyl)amino]piperidine-1-carboxylate
—— Ethyl 6-acetyl-2-(4-butoxybenzamido)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxylate —— C23H28N2O5S
Ethyl 6-acetyl-2-(4-butoxybenzamido)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxylate
—— (E)-3-(4-acetamidophenyl)-N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]prop-2-enamide —— C21H22N2O4
(E)-3-(4-acetamidophenyl)-N-[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]prop-2-enamide
—— (E)-N-(4-chloro-3-methylbenzo[d]thiazol-2(3H)-ylidene)-4-(2,5-dioxopyrrolidin-1-yl)benzamide —— C19H14ClN3O3S
(E)-N-(4-chloro-3-methylbenzo[d]thiazol-2(3H)-ylidene)-4-(2,5-dioxopyrrolidin-1-yl)benzamide
—— Ethyl 3-[(4-methoxyphenyl)hydrazinylidene]-2-methyl-4,5-dioxo-1-phenylpyrrolidine-2-carboxylate —— C21H21N3O5
Ethyl 3-[(4-methoxyphenyl)hydrazinylidene]-2-methyl-4,5-dioxo-1-phenylpyrrolidine-2-carboxylate
—— Ethyl 4-[furan-2-carbonyl-[(2-oxopyrrolidin-1-yl)methyl]amino]benzoate —— C19H20N2O5
Ethyl 4-[furan-2-carbonyl-[(2-oxopyrrolidin-1-yl)methyl]amino]benzoate
—— (E)-2-cyano-3-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-N-(4-methylpyridin-2-yl)prop-2-enamide —— C20H24N4O2
(E)-2-cyano-3-[1-[(2S)-1-methoxypropan-2-yl]-2,5-dimethylpyrrol-3-yl]-N-(4-methylpyridin-2-yl)prop-2-enamide
—— Ethyl 2-[[2-[[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C22H22ClN3O4S2
Ethyl 2-[[2-[[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-[2-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]sulfonylacetyl]imino-3-prop-2-ynyl-1,3-benzothiazole-6-carboxylate —— C25H23N3O6S2
Ethyl 2-[2-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]sulfonylacetyl]imino-3-prop-2-ynyl-1,3-benzothiazole-6-carboxylate
—— (E)-3-(3-cyanophenyl)-N-[(1S)-1-(2,5-difluorophenyl)ethyl]-N-methylprop-2-enamide —— C19H16F2N2O
(E)-3-(3-cyanophenyl)-N-[(1S)-1-(2,5-difluorophenyl)ethyl]-N-methylprop-2-enamide
—— (E)-N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-3-(furan-2-yl)prop-2-enamide —— C18H22N2O3
(E)-N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl N-[2-[[4-[butyl(ethyl)sulfamoyl]benzoyl]amino]-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonyl]carbamate —— C27H38N4O6S2
ethyl N-[2-[[4-[butyl(ethyl)sulfamoyl]benzoyl]amino]-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonyl]carbamate
—— ethyl 2-[[3-[4-[4-[4-(hydroxymethyl)phenyl]-6-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate —— C42H47N5O7
ethyl 2-[[3-[4-[4-[4-(hydroxymethyl)phenyl]-6-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylcarbamoylamino]acetate
—— ethyl 6-methyl-2-oxo-4-pyridin-4-yl-3,4-dihydro-1H-pyridine-5-carboxylate —— C14H16N2O3
ethyl 6-methyl-2-oxo-4-pyridin-4-yl-3,4-dihydro-1H-pyridine-5-carboxylate
—— Ethyl 2-[2-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]sulfonylacetyl]imino-3-prop-2-ynyl-1,3-benzothiazole-6-carboxylate —— C20H18N4O6S3
Ethyl 2-[2-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]sulfonylacetyl]imino-3-prop-2-ynyl-1,3-benzothiazole-6-carboxylate
—— Ethyl 5-carbamoyl-4-methyl-2-[(2,2,2-trifluoroacetyl)amino]thiophene-3-carboxylate —— C11H11F3N2O4S
Ethyl 5-carbamoyl-4-methyl-2-[(2,2,2-trifluoroacetyl)amino]thiophene-3-carboxylate
—— (E)-N-[3-[4-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]-3-oxopropyl]-3-(furan-2-yl)prop-2-enamide —— C20H30N4O4
(E)-N-[3-[4-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]-3-oxopropyl]-3-(furan-2-yl)prop-2-enamide
—— Ethyl 2-[[2-[2-oxo-2-[(3-prop-2-enyl-1,3-benzothiazol-2-ylidene)amino]ethyl]sulfonylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H27N3O6S3
Ethyl 2-[[2-[2-oxo-2-[(3-prop-2-enyl-1,3-benzothiazol-2-ylidene)amino]ethyl]sulfonylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[4-[benzyl(propan-2-yl)sulfamoyl]benzoyl]amino]-3-(methylcarbamoylcarbamoyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate —— C30H35N5O7S2
ethyl 2-[[4-[benzyl(propan-2-yl)sulfamoyl]benzoyl]amino]-3-(methylcarbamoylcarbamoyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate
—— Ethyl 2-[6-bromo-2-(naphthalene-1-carbonylimino)-1,3-benzothiazol-3-yl]acetate —— C22H17BrN2O3S
Ethyl 2-[6-bromo-2-(naphthalene-1-carbonylimino)-1,3-benzothiazol-3-yl]acetate
—— ethyl 2-[[2-[2-[(3-ethyl-6-methoxy-1,3-benzothiazol-2-ylidene)amino]-2-oxoethyl]sulfanylacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C24H27N3O5S3
ethyl 2-[[2-[2-[(3-ethyl-6-methoxy-1,3-benzothiazol-2-ylidene)amino]-2-oxoethyl]sulfanylacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— Ethyl 2-cyano-4-[1-[(2,4-dichlorophenyl)methyl]pyridin-4-ylidene]but-2-enoate —— C19H16Cl2N2O2
Ethyl 2-cyano-4-[1-[(2,4-dichlorophenyl)methyl]pyridin-4-ylidene]but-2-enoate
—— ethyl 2-[[2-[[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C26H31N3O4S2
ethyl 2-[[2-[[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— (E)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C15H16N2O7S
(E)-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— (E)-N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-3-(furan-2-yl)prop-2-enamide —— C18H22N2O3
(E)-N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl 2-[(3,5-diiodo-4-prop-2-ynoxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H18I2N2O4S2
ethyl 2-[(3,5-diiodo-4-prop-2-ynoxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(4-acetamidophenyl)-N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]prop-2-enamide —— C22H27N3O3
(E)-3-(4-acetamidophenyl)-N-[(2S)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]prop-2-enamide
—— (E)-2-Cyano-3-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]-N-(2,2,2-trifluoroethyl)prop-2-enamide —— C15H18F3N3O2
(E)-2-Cyano-3-[1-(2-methoxyethyl)-2,5-dimethylpyrrol-3-yl]-N-(2,2,2-trifluoroethyl)prop-2-enamide
—— (E)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C15H16N2O7S
(E)-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[4-(difluoromethylsulfonyl)phenyl]prop-2-enamide —— C18H16F2N2O4S
(E)-3-(4-acetamidophenyl)-N-[4-(difluoromethylsulfonyl)phenyl]prop-2-enamide
—— Ethyl 5-[2-(3-chlorophenoxy)propanoylamino]-1-phenylpyrazole-4-carboxylate —— C21H20ClN3O4
Ethyl 5-[2-(3-chlorophenoxy)propanoylamino]-1-phenylpyrazole-4-carboxylate
—— (E)-N-[(2R)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C20H25N3O2S
(E)-N-[(2R)-2-(2-methoxyphenyl)-2-pyrrolidin-1-ylethyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— Ethyl 3-(1-oxo-4-phenyl-1H-isochromene-3-amido)benzoate —— C25H19NO5
Ethyl 3-(1-oxo-4-phenyl-1H-isochromene-3-amido)benzoate
—— (E)-3-(4-acetamidophenyl)-N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]prop-2-enamide —— C22H27N3O3
(E)-3-(4-acetamidophenyl)-N-[(2R)-2-(dimethylamino)-2-(3-methoxyphenyl)ethyl]prop-2-enamide