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—— ethyl (4S)-6-(diethylaminomethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H25N3O3
ethyl (4S)-6-(diethylaminomethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[3-chloro-4-(3-oxopiperazin-1-yl)phenyl]-3-(3-cyanophenyl)prop-2-enamide —— C20H17ClN4O2
(E)-N-[3-chloro-4-(3-oxopiperazin-1-yl)phenyl]-3-(3-cyanophenyl)prop-2-enamide
—— ethyl 4-[(2R)-2-hydroxy-3-(4-methylpiperidin-1-yl)propoxy]benzoate —— C18H27NO4
ethyl 4-[(2R)-2-hydroxy-3-(4-methylpiperidin-1-yl)propoxy]benzoate
—— (E)-N-[(1R)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-thiophen-3-ylprop-2-enamide —— C16H18N2O3S2
(E)-N-[(1R)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-thiophen-3-ylprop-2-enamide
—— (E)-N-[(1S)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-thiophen-3-ylprop-2-enamide —— C16H18N2O3S2
(E)-N-[(1S)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-thiophen-3-ylprop-2-enamide
—— (E)-N-[(1R)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-phenylprop-2-enamide —— C18H20N2O3S
(E)-N-[(1R)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-phenylprop-2-enamide
—— Ethyl 4-[[2-(4-bromo-2-fluorophenoxy)acetyl]amino]benzoate —— C17H15BrFNO4
Ethyl 4-[[2-(4-bromo-2-fluorophenoxy)acetyl]amino]benzoate
—— ethyl (4R)-6-(diethylaminomethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H25N3O3
ethyl (4R)-6-(diethylaminomethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-2-cyano-3-[4-(dimethylamino)phenyl]-N-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C21H23N3O4
(E)-2-cyano-3-[4-(dimethylamino)phenyl]-N-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— ethyl 1-[3-[[(2R)-2-benzamidopropanoyl]amino]phenyl]pyrazole-3-carboxylate —— C22H22N4O4
ethyl 1-[3-[[(2R)-2-benzamidopropanoyl]amino]phenyl]pyrazole-3-carboxylate
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[(1R)-1-[3-(methanesulfonamido)phenyl]ethyl]prop-2-enamide —— C19H19N3O4S
(E)-3-(1,3-benzoxazol-2-yl)-N-[(1R)-1-[3-(methanesulfonamido)phenyl]ethyl]prop-2-enamide
—— ethyl 1-[3-[[(2S)-2-benzamidopropanoyl]amino]phenyl]pyrazole-3-carboxylate —— C22H22N4O4
ethyl 1-[3-[[(2S)-2-benzamidopropanoyl]amino]phenyl]pyrazole-3-carboxylate
—— (E)-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-[(4-pyrazol-1-ylphenyl)methyl]prop-2-enamide —— C20H16ClN5O
(E)-3-(2-chloroimidazo[1,2-a]pyridin-3-yl)-N-[(4-pyrazol-1-ylphenyl)methyl]prop-2-enamide
—— (E)-N-[(1S)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-phenylprop-2-enamide —— C18H20N2O3S
(E)-N-[(1S)-1-[3-(methanesulfonamido)phenyl]ethyl]-3-phenylprop-2-enamide
—— ethyl 4-[(2S)-2-hydroxy-3-(4-methylpiperidin-1-yl)propoxy]benzoate —— C18H27NO4
ethyl 4-[(2S)-2-hydroxy-3-(4-methylpiperidin-1-yl)propoxy]benzoate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[3-chloro-4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide —— C20H18ClN3O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[3-chloro-4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide
—— (E)-3-(3-cyanophenyl)-N-[3-cyano-4-(2,2,2-trifluoroethoxy)phenyl]prop-2-enamide —— C19H12F3N3O2
(E)-3-(3-cyanophenyl)-N-[3-cyano-4-(2,2,2-trifluoroethoxy)phenyl]prop-2-enamide
—— (E)-3-(2,6-difluorophenyl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide —— C19H17F2N3O2
(E)-3-(2,6-difluorophenyl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide
—— ethyl 2-[[2-[(5S,6R)-6-methyl-2,4-dioxo-1,3-diazaspiro[4.5]decan-3-yl]acetyl]amino]-4-(5-methylfuran-2-yl)thiophene-3-carboxylate —— C23H27N3O6S
ethyl 2-[[2-[(5S,6R)-6-methyl-2,4-dioxo-1,3-diazaspiro[4.5]decan-3-yl]acetyl]amino]-4-(5-methylfuran-2-yl)thiophene-3-carboxylate
—— (E)-3-(4-cyanophenyl)-N-[3-cyano-4-(2,2,2-trifluoroethoxy)phenyl]prop-2-enamide —— C19H12F3N3O2
(E)-3-(4-cyanophenyl)-N-[3-cyano-4-(2,2,2-trifluoroethoxy)phenyl]prop-2-enamide
—— Ethyl 4-(2-hydroxy-3-methoxybenzoyl)piperazine-1-carboxylate —— C15H20N2O5
Ethyl 4-(2-hydroxy-3-methoxybenzoyl)piperazine-1-carboxylate
—— (E)-3-(5-bromothiophen-2-yl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide —— C17H16BrN3O2S
(E)-3-(5-bromothiophen-2-yl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide
—— ethyl 5-[2-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H26N4O4S
ethyl 5-[2-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 2-[(2-benzoyloxyacetyl)amino]-4-methyl-5-(methylcarbamoyl)thiophene-3-carboxylate —— C19H20N2O6S
Ethyl 2-[(2-benzoyloxyacetyl)amino]-4-methyl-5-(methylcarbamoyl)thiophene-3-carboxylate
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[[3-(2,2,2-trifluoroethoxy)phenyl]methyl]prop-2-enamide —— C20H17F3N2O3
(E)-3-[4-(cyanomethoxy)phenyl]-N-[[3-(2,2,2-trifluoroethoxy)phenyl]methyl]prop-2-enamide
—— (E)-N-[4-(3-oxopiperazin-1-yl)phenyl]-3-(2,4,5-trimethylphenyl)prop-2-enamide —— C22H25N3O2
(E)-N-[4-(3-oxopiperazin-1-yl)phenyl]-3-(2,4,5-trimethylphenyl)prop-2-enamide
—— (E)-3-(1-benzyltriazol-4-yl)-N-[[3-(2,2,2-trifluoroethoxy)phenyl]methyl]prop-2-enamide —— C21H19F3N4O2
(E)-3-(1-benzyltriazol-4-yl)-N-[[3-(2,2,2-trifluoroethoxy)phenyl]methyl]prop-2-enamide
—— ethyl 2-[(2-benzoyloxyacetyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C19H19NO5S
ethyl 2-[(2-benzoyloxyacetyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— (E)-3-(4-bromophenyl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide —— C19H18BrN3O2
(E)-3-(4-bromophenyl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide
—— ethyl N-[(2R)-1-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylethylamino]-3-methyl-1-oxobutan-2-yl]carbamate —— C16H31N3O6S
ethyl N-[(2R)-1-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylethylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl N-[(2R)-1-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylethylamino]-3-methyl-1-oxobutan-2-yl]carbamate —— C16H31N3O6S
ethyl N-[(2R)-1-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylethylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl (6R)-6-methyl-2-[[(2R)-2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C18H24N4O3S2
ethyl (6R)-6-methyl-2-[[(2R)-2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-(4-cyanophenyl)-N-[[3-(pyridin-2-ylmethoxy)phenyl]methyl]prop-2-enamide —— C23H19N3O2
(E)-3-(4-cyanophenyl)-N-[[3-(pyridin-2-ylmethoxy)phenyl]methyl]prop-2-enamide
—— (E)-4-[(3R)-3-methylpiperidin-1-yl]-4-oxobut-2-enoic acid —— C10H15NO3
(E)-4-[(3R)-3-methylpiperidin-1-yl]-4-oxobut-2-enoic acid
—— (E)-N-[4-(dimethylamino)-2-methylphenyl]-3-[4-(methanesulfonamido)phenyl]prop-2-enamide —— C19H23N3O3S
(E)-N-[4-(dimethylamino)-2-methylphenyl]-3-[4-(methanesulfonamido)phenyl]prop-2-enamide
—— (E)-1-[4-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperazin-1-yl]-3-thiophen-2-ylprop-2-en-1-one —— C18H22N2O2S
(E)-1-[4-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperazin-1-yl]-3-thiophen-2-ylprop-2-en-1-one
—— (E)-3-(2-cyanophenyl)-N-[(1R)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide —— C21H22N2O4
(E)-3-(2-cyanophenyl)-N-[(1R)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide —— C24H28N2O4
(E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide
—— (E)-N-[2-methyl-5-(propanoylamino)phenyl]-3-(4-nitrophenyl)prop-2-enamide —— C19H19N3O4
(E)-N-[2-methyl-5-(propanoylamino)phenyl]-3-(4-nitrophenyl)prop-2-enamide
—— ethyl N-[(2R)-3-methyl-1-[[(2S)-2-(4-methylpiperidin-1-yl)-2-thiophen-2-ylethyl]amino]-1-oxobutan-2-yl]carbamate —— C20H33N3O3S
ethyl N-[(2R)-3-methyl-1-[[(2S)-2-(4-methylpiperidin-1-yl)-2-thiophen-2-ylethyl]amino]-1-oxobutan-2-yl]carbamate
—— (E)-3-(1-benzyltriazol-4-yl)-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide —— C22H23N5O2
(E)-3-(1-benzyltriazol-4-yl)-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide
—— (E)-4-[(3R)-3-methylpiperidin-1-yl]-4-oxobut-2-enoate —— C10H14NO3-
(E)-4-[(3R)-3-methylpiperidin-1-yl]-4-oxobut-2-enoate
—— (E)-3-(4-chloro-3-nitrophenyl)-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide —— C19H18ClN3O4
(E)-3-(4-chloro-3-nitrophenyl)-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide
—— ethyl 2-[[2-(2,6-dimethoxybenzoyl)oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C21H23NO7S
ethyl 2-[[2-(2,6-dimethoxybenzoyl)oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— Ethyl 2-[[2-(cyclopropanecarbonyloxy)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C17H21NO5S
Ethyl 2-[[2-(cyclopropanecarbonyloxy)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[4-(dimethylamino)-2-methylphenyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C21H24N2O4
(E)-N-[4-(dimethylamino)-2-methylphenyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— (E)-3-(2-cyanophenyl)-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide —— C21H22N2O4
(E)-3-(2-cyanophenyl)-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide
—— ethyl N-[(2S)-1-[4-[(4-methoxyphenyl)methyl]-1,4-diazepan-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C21H33N3O4
ethyl N-[(2S)-1-[4-[(4-methoxyphenyl)methyl]-1,4-diazepan-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl N-[(2S)-3-methyl-1-[[(2R)-2-(4-methylpiperidin-1-yl)-2-thiophen-2-ylethyl]amino]-1-oxobutan-2-yl]carbamate —— C20H33N3O3S
ethyl N-[(2S)-3-methyl-1-[[(2R)-2-(4-methylpiperidin-1-yl)-2-thiophen-2-ylethyl]amino]-1-oxobutan-2-yl]carbamate
—— (E)-3-(2,4-dimethylphenyl)-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide —— C22H27NO4
(E)-3-(2,4-dimethylphenyl)-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide