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—— ethyl (2Z,5R)-2-[(2,3-dimethoxyphenyl)methylidene]-5-(2-methoxyphenyl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H30N2O6S
ethyl (2Z,5R)-2-[(2,3-dimethoxyphenyl)methylidene]-5-(2-methoxyphenyl)-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-5-(2-ethoxy-3-methoxyphenyl)-7-methyl-3-oxo-2-[(4-phenylmethoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O6S
ethyl (2E,5R)-5-(2-ethoxy-3-methoxyphenyl)-7-methyl-3-oxo-2-[(4-phenylmethoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-5-(2-methoxyphenyl)-2-[(3-methylthiophen-2-yl)methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H26N2O4S2
ethyl (2E,5S)-5-(2-methoxyphenyl)-2-[(3-methylthiophen-2-yl)methylidene]-3-oxo-7-propyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 1-[(1S)-1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-4-carboxylate —— C15H25N3O3
ethyl 1-[(1S)-1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-4-carboxylate
—— (E)-N-cyclopropyl-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide —— C20H26N4O4S
(E)-N-cyclopropyl-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-[(1-methylimidazol-2-yl)methyl]prop-2-enamide
—— ethyl N-[(2E)-2-[(2-methoxy-5-nitroanilino)methylidene]-3-oxobutanoyl]carbamate —— C15H17N3O7
ethyl N-[(2E)-2-[(2-methoxy-5-nitroanilino)methylidene]-3-oxobutanoyl]carbamate
—— (E)-N-[(1S)-2-anilino-2-oxo-1-phenylethyl]-3-(3-cyanophenyl)prop-2-enamide —— C24H19N3O2
(E)-N-[(1S)-2-anilino-2-oxo-1-phenylethyl]-3-(3-cyanophenyl)prop-2-enamide
—— ethyl (2Z,5S)-2-[(3-ethoxyphenyl)methylidene]-5-(4-methylsulfanylphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28N2O4S2
ethyl (2Z,5S)-2-[(3-ethoxyphenyl)methylidene]-5-(4-methylsulfanylphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[(3S)-1-pyrimidin-2-ylpiperidine-3-carbonyl]piperazine-1-carboxylate —— C17H25N5O3
ethyl 4-[(3S)-1-pyrimidin-2-ylpiperidine-3-carbonyl]piperazine-1-carboxylate
—— ethyl 4-[(3R)-1-pyrimidin-2-ylpiperidine-3-carbonyl]piperazine-1-carboxylate —— C17H25N5O3
ethyl 4-[(3R)-1-pyrimidin-2-ylpiperidine-3-carbonyl]piperazine-1-carboxylate
—— ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-7-methyl-2-[(5-morpholin-4-ylfuran-2-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H25N3O7S
ethyl (2E,5R)-5-(1,3-benzodioxol-5-yl)-7-methyl-2-[(5-morpholin-4-ylfuran-2-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-5-(4-fluorophenyl)-2-[(5-methylfuran-2-yl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H21FN2O4S
ethyl (2Z,5R)-5-(4-fluorophenyl)-2-[(5-methylfuran-2-yl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (4Z)-4-[(3-ethoxy-4-propoxyphenyl)methylidene]-2-methyl-1-(4-methylphenyl)-5-oxopyrrole-3-carboxylate —— C27H31NO5
ethyl (4Z)-4-[(3-ethoxy-4-propoxyphenyl)methylidene]-2-methyl-1-(4-methylphenyl)-5-oxopyrrole-3-carboxylate
—— ethyl (2Z,5S)-2-[[1-(cyanomethyl)indol-3-yl]methylidene]-5-(3-methoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H26N4O4S
ethyl (2Z,5S)-2-[[1-(cyanomethyl)indol-3-yl]methylidene]-5-(3-methoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5E)-5-[[2,5-dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-2-(4-methylanilino)-4-oxothiophene-3-carboxylate —— C28H28N2O3S
ethyl (5E)-5-[[2,5-dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-2-(4-methylanilino)-4-oxothiophene-3-carboxylate
—— ethyl (2E,5R)-5-(2,4-dimethoxyphenyl)-7-methyl-2-[(5-morpholin-4-ylfuran-2-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O7S
ethyl (2E,5R)-5-(2,4-dimethoxyphenyl)-7-methyl-2-[(5-morpholin-4-ylfuran-2-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(5E)-5-[(4-hydroxy-3-nitrophenyl)methylidene]-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate —— C20H17N3O6S
ethyl 4-[[(5E)-5-[(4-hydroxy-3-nitrophenyl)methylidene]-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate
—— ethyl (2E,5R)-5-(3-methoxy-2-propoxyphenyl)-7-methyl-2-(naphthalen-1-ylmethylidene)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H30N2O5S
ethyl (2E,5R)-5-(3-methoxy-2-propoxyphenyl)-7-methyl-2-(naphthalen-1-ylmethylidene)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-2-[(5-bromo-3-chloro-2-hydroxyphenyl)methylidene]-5-(2-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H17BrCl2N2O4S
ethyl (2Z,5S)-2-[(5-bromo-3-chloro-2-hydroxyphenyl)methylidene]-5-(2-chlorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(5E)-5-[(3-chloro-5-methoxy-4-prop-2-ynoxyphenyl)methylidene]-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate —— C24H21ClN2O5S
ethyl 4-[[(5E)-5-[(3-chloro-5-methoxy-4-prop-2-ynoxyphenyl)methylidene]-3-methyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate
—— ethyl (2E,5R)-2-[(3-chloro-5-methoxy-4-prop-2-enoxyphenyl)methylidene]-5-(4-ethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H29ClN2O6S
ethyl (2E,5R)-2-[(3-chloro-5-methoxy-4-prop-2-enoxyphenyl)methylidene]-5-(4-ethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 3-[5-[(E)-[5-oxo-1-(4-sulfamoylphenyl)-3-(trifluoromethyl)pyrazol-4-ylidene]methyl]furan-2-yl]benzoate —— C24H18F3N3O6S
ethyl 3-[5-[(E)-[5-oxo-1-(4-sulfamoylphenyl)-3-(trifluoromethyl)pyrazol-4-ylidene]methyl]furan-2-yl]benzoate
—— ethyl (2E,5R)-5-(4-ethoxyphenyl)-2-[[1-(3-methoxycarbonylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H33N3O6S
ethyl (2E,5R)-5-(4-ethoxyphenyl)-2-[[1-(3-methoxycarbonylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(2-hydroxyphenyl)methylidene]-5-(3-methoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H24N2O5S
ethyl (2E,5R)-2-[(2-hydroxyphenyl)methylidene]-5-(3-methoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(5E)-5-benzylidene-3-ethyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate —— C21H20N2O3S
ethyl 4-[[(5E)-5-benzylidene-3-ethyl-4-oxo-1,3-thiazolidin-2-ylidene]amino]benzoate
—— ethyl (2Z,5S)-2-[[4-(dimethylamino)phenyl]methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O3S
ethyl (2Z,5S)-2-[[4-(dimethylamino)phenyl]methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 4-[4-[(E)-1-(3,4-dimethoxyphenyl)methylidene]-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-1-YL]benzoate —— C22H19F3N2O5
Ethyl 4-[4-[(E)-1-(3,4-dimethoxyphenyl)methylidene]-5-oxo-3-(trifluoromethyl)-4,5-dihydro-1H-pyrazol-1-YL]benzoate
—— ethyl 4-{[(2E,5Z)-5-(2,5-dimethoxybenzylidene)-3-ethyl-4-oxo-1,3-thiazolidin-2-ylidene]amino}benzoate —— C23H24N2O5S
ethyl 4-{[(2E,5Z)-5-(2,5-dimethoxybenzylidene)-3-ethyl-4-oxo-1,3-thiazolidin-2-ylidene]amino}benzoate
—— ethyl (2Z,5R)-2-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H25FN4O5S
ethyl (2Z,5R)-2-[[2,5-dimethyl-1-(4-nitrophenyl)pyrrol-3-yl]methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(3,4-dichlorophenyl)-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide —— C16H22Cl2N2O3S
(E)-3-(3,4-dichlorophenyl)-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide
—— ethyl (2Z,5R)-5-(4-methoxyphenyl)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H24N2O6S
ethyl (2Z,5R)-5-(4-methoxyphenyl)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(3-nitrophenyl)-1-[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]prop-2-en-1-one —— C22H19N3O3
(E)-3-(3-nitrophenyl)-1-[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]prop-2-en-1-one
—— ethyl (2Z,5R)-5-(1,3-benzodioxol-5-yl)-2-[(2-methyl-1H-indol-3-yl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H25N3O5S
ethyl (2Z,5R)-5-(1,3-benzodioxol-5-yl)-2-[(2-methyl-1H-indol-3-yl)methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide —— C18H25N3O4S
(E)-3-[4-(cyanomethoxy)phenyl]-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide
—— (E)-3-(2,6-dichlorophenyl)-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]prop-2-enamide —— C17H11Cl2N3O2
(E)-3-(2,6-dichlorophenyl)-N-[4-(1,3,4-oxadiazol-2-yl)phenyl]prop-2-enamide
—— ethyl 3-[[(2R)-1-ethylpyrrolidin-2-yl]methylcarbamoyl]-5-nitrobenzoate —— C17H23N3O5
ethyl 3-[[(2R)-1-ethylpyrrolidin-2-yl]methylcarbamoyl]-5-nitrobenzoate
—— ethyl 3-[[(3S)-1-methylsulfonylpiperidine-3-carbonyl]amino]propanoate —— C12H22N2O5S
ethyl 3-[[(3S)-1-methylsulfonylpiperidine-3-carbonyl]amino]propanoate
—— ethyl (2Z,5R)-5-(2-chlorophenyl)-2-[(2,3-dichlorophenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H17Cl3N2O3S
ethyl (2Z,5R)-5-(2-chlorophenyl)-2-[(2,3-dichlorophenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 3-[[(2S)-1-ethylpyrrolidin-2-yl]methylcarbamoyl]-5-nitrobenzoate —— C17H23N3O5
ethyl 3-[[(2S)-1-ethylpyrrolidin-2-yl]methylcarbamoyl]-5-nitrobenzoate
—— ethyl (2Z,5S)-2-[(3-bromo-4-hydroxy-5-nitrophenyl)methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H17BrFN3O6S
ethyl (2Z,5S)-2-[(3-bromo-4-hydroxy-5-nitrophenyl)methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylidene]-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H24N2O5S2
ethyl (2Z,5R)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylidene]-5-(4-methylsulfanylphenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H20N2O5S2
ethyl (2Z,5S)-7-methyl-2-[(6-methyl-1,3-benzodioxol-5-yl)methylidene]-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (4S)-2-amino-6-chloro-4-(4-fluorophenyl)-4H-benzo[h]chromene-3-carboxylate —— C22H17ClFNO3
ethyl (4S)-2-amino-6-chloro-4-(4-fluorophenyl)-4H-benzo[h]chromene-3-carboxylate
—— ethyl (2E,5R)-5-(4-fluorophenyl)-2-[(4-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H19FN2O4S
ethyl (2E,5R)-5-(4-fluorophenyl)-2-[(4-hydroxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 4-[4-oxo-7-(2-oxo-2-propan-2-yloxyethoxy)chromen-3-yl]oxybenzoate —— C23H22O8
Ethyl 4-[4-oxo-7-(2-oxo-2-propan-2-yloxyethoxy)chromen-3-yl]oxybenzoate
—— ethyl (2Z,5R)-2-[(5-bromo-2-prop-2-ynoxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H19BrN2O4S2
ethyl (2Z,5R)-2-[(5-bromo-2-prop-2-ynoxyphenyl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2S,4R)-1,4-dimethylpiperidine-2-carboxylate —— C10H19NO2
ethyl (2S,4R)-1,4-dimethylpiperidine-2-carboxylate
—— ethyl {[(2Z)-3-oxo-2-(2,3,4-trimethoxybenzylidene)-2,3-dihydro-1-benzofuran-6-yl]oxy}acetate —— C22H22O8
ethyl {[(2Z)-3-oxo-2-(2,3,4-trimethoxybenzylidene)-2,3-dihydro-1-benzofuran-6-yl]oxy}acetate
—— ethyl (4aR,9bR)-1,3,4,4a,5,9b-hexahydropyrido[4,3-b]indole-2-carboxylate —— C14H18N2O2
ethyl (4aR,9bR)-1,3,4,4a,5,9b-hexahydropyrido[4,3-b]indole-2-carboxylate
—— ethyl (4aS,9bS)-1,3,4,4a,5,9b-hexahydropyrido[4,3-b]indole-2-carboxylate —— C14H18N2O2
ethyl (4aS,9bS)-1,3,4,4a,5,9b-hexahydropyrido[4,3-b]indole-2-carboxylate