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—— (E)-3-(5-bromofuran-2-yl)-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]prop-2-enamide —— C16H13BrF3NO3
(E)-3-(5-bromofuran-2-yl)-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(1S)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide —— C22H22N2O3
(E)-3-(4-acetamidophenyl)-N-[(1S)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide
—— (E)-3-(1-benzyltriazol-4-yl)-N-[(1S)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide —— C23H22N4O2
(E)-3-(1-benzyltriazol-4-yl)-N-[(1S)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(1R)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide —— C22H22N2O3
(E)-3-(4-acetamidophenyl)-N-[(1R)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide
—— (E)-3-(5-bromofuran-2-yl)-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]prop-2-enamide —— C16H13BrF3NO3
(E)-3-(5-bromofuran-2-yl)-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]ethyl]prop-2-enamide
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[(1S)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide —— C22H20N2O3
(E)-3-[4-(cyanomethoxy)phenyl]-N-[(1S)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide
—— (E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]prop-2-enamide —— C23H21F2N3O2
(E)-3-[1-(2-cyanoethyl)indol-3-yl]-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]prop-2-enamide
—— ethyl 4-[[(3R)-1-(2,4-difluorophenyl)-5-oxopyrrolidine-3-carbonyl]amino]benzoate —— C20H18F2N2O4
ethyl 4-[[(3R)-1-(2,4-difluorophenyl)-5-oxopyrrolidine-3-carbonyl]amino]benzoate
—— (E)-N-[2-[[2-(3,5-dimethylphenoxy)pyridin-4-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C23H23N3O4
(E)-N-[2-[[2-(3,5-dimethylphenoxy)pyridin-4-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]prop-2-enamide —— C28H26N2O2
(E)-3-(4-acetamidophenyl)-N-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]prop-2-enamide
—— Ethyl 2-[[2-(2-chlorophenyl)sulfanylacetyl]amino]-5-(diethylcarbamoyl)-4-methylthiophene-3-carboxylate —— C21H25ClN2O4S2
Ethyl 2-[[2-(2-chlorophenyl)sulfanylacetyl]amino]-5-(diethylcarbamoyl)-4-methylthiophene-3-carboxylate
—— ethyl (6S)-6-methyl-2-[[(2R)-2-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H27N5O3S2
ethyl (6S)-6-methyl-2-[[(2R)-2-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C21H21F2NO5
(E)-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— (E)-N-methyl-N-(3-phenylpropyl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C22H27NO4
(E)-N-methyl-N-(3-phenylpropyl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-[(1R)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide —— C22H20N2O3
(E)-3-[4-(cyanomethoxy)phenyl]-N-[(1R)-1-(3-methyl-1-benzofuran-2-yl)ethyl]prop-2-enamide
—— (E)-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide —— C20H19F2NO4
(E)-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide
—— ethyl (6S)-6-methyl-2-[[(2S)-2-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H27N5O3S2
ethyl (6S)-6-methyl-2-[[(2S)-2-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methoxyphenyl)prop-2-enamide —— C23H27NO5
(E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methoxyphenyl)prop-2-enamide
—— (E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methylphenyl)prop-2-enamide —— C23H27NO4
(E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methylphenyl)prop-2-enamide
—— ethyl 1-[2-(1H-benzimidazol-2-ylsulfanyl)acetyl]piperidine-4-carboxylate —— C17H21N3O3S
ethyl 1-[2-(1H-benzimidazol-2-ylsulfanyl)acetyl]piperidine-4-carboxylate
—— (E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methylphenyl)prop-2-enamide —— C23H27NO4
(E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methylphenyl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[(2-phenylmethoxypyridin-4-yl)methylamino]ethyl]prop-2-enamide —— C22H21N3O4
(E)-3-(furan-2-yl)-N-[2-oxo-2-[(2-phenylmethoxypyridin-4-yl)methylamino]ethyl]prop-2-enamide
—— Ethyl 2-[(2-quinazolin-4-yloxyacetyl)amino]benzoate —— C19H17N3O4
Ethyl 2-[(2-quinazolin-4-yloxyacetyl)amino]benzoate
—— ethyl 4-[2-(quinoline-2-carbonyl)hydrazinyl]-3,6-dihydro-2H-pyridine-1-carboxylate —— C18H20N4O3
ethyl 4-[2-(quinoline-2-carbonyl)hydrazinyl]-3,6-dihydro-2H-pyridine-1-carboxylate
—— ethyl (3S)-1-[4-chloro-3-(dimethylsulfamoyl)benzoyl]piperidine-3-carboxylate —— C17H23ClN2O5S
ethyl (3S)-1-[4-chloro-3-(dimethylsulfamoyl)benzoyl]piperidine-3-carboxylate
—— (E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylthiophen-2-yl)prop-2-enamide —— C21H25NO4S
(E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylthiophen-2-yl)prop-2-enamide
—— (E)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide —— C22H22N4O4
(E)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide
—— (E)-3-(4-cyanophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide —— C23H19N3O2
(E)-3-(4-cyanophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide
—— (E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methoxyphenyl)prop-2-enamide —— C23H27NO5
(E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(3-methoxyphenyl)prop-2-enamide
—— (E)-3-(3-nitrophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide —— C22H19N3O4
(E)-3-(3-nitrophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide
—— ethyl 4-[2-[[7-(dimethylsulfamoyl)-[1,2,4]triazolo[3,4-b][1,3]benzoxazol-1-yl]sulfanyl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C21H23N5O6S2
ethyl 4-[2-[[7-(dimethylsulfamoyl)-[1,2,4]triazolo[3,4-b][1,3]benzoxazol-1-yl]sulfanyl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C21H25NO5
(E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]prop-2-enamide —— C22H24FNO4
(E)-3-(4-fluorophenyl)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]prop-2-enamide
—— (E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(4-methoxyphenyl)prop-2-enamide —— C23H27NO5
(E)-N-[[3-methoxy-4-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(4-methoxyphenyl)prop-2-enamide
—— ethyl (3R)-1-[4-chloro-3-(dimethylsulfamoyl)benzoyl]piperidine-3-carboxylate —— C17H23ClN2O5S
ethyl (3R)-1-[4-chloro-3-(dimethylsulfamoyl)benzoyl]piperidine-3-carboxylate
—— Ethyl 3-[[2-(2,5-dimethylphenyl)sulfanylacetyl]amino]-5-phenylthiophene-2-carboxylate —— C23H23NO3S2
Ethyl 3-[[2-(2,5-dimethylphenyl)sulfanylacetyl]amino]-5-phenylthiophene-2-carboxylate
—— (E)-3-(3-cyanophenyl)-N-[[4-(pyridin-3-ylmethoxy)phenyl]methyl]prop-2-enamide —— C23H19N3O2
(E)-3-(3-cyanophenyl)-N-[[4-(pyridin-3-ylmethoxy)phenyl]methyl]prop-2-enamide
—— Ethyl 3-[(5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanylmethyl]-1-benzofuran-2-carboxylate —— C24H22N4O4S
Ethyl 3-[(5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanylmethyl]-1-benzofuran-2-carboxylate
—— Ethyl 2-[(5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]acetate —— C16H18N4O3S
Ethyl 2-[(5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]acetate
—— ethyl 4-[2-[(4-amino-6-methyl-5-oxo-1,2,4-triazin-3-yl)sulfanyl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C15H19N5O4S
ethyl 4-[2-[(4-amino-6-methyl-5-oxo-1,2,4-triazin-3-yl)sulfanyl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl N-[2-[(5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]acetyl]carbamate —— C17H19N5O4S
ethyl N-[2-[(5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazolin-1-yl)sulfanyl]acetyl]carbamate
—— (E)-N-[3-[(2R)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-3-oxopropyl]-3-(furan-2-yl)prop-2-enamide —— C21H23FN2O3
(E)-N-[3-[(2R)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-3-oxopropyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl 2,4-dimethyl-5-[2-[2-[(4-oxo-2,3-dihydro-1H-cyclopenta[c]chromen-7-yl)oxy]acetyl]oxyacetyl]-1H-pyrrole-3-carboxylate —— C25H25NO8
ethyl 2,4-dimethyl-5-[2-[2-[(4-oxo-2,3-dihydro-1H-cyclopenta[c]chromen-7-yl)oxy]acetyl]oxyacetyl]-1H-pyrrole-3-carboxylate
—— [(E)-3-cyano-4-(4-fluorophenyl)-2-oxo-4-piperidin-1-ylbut-3-enyl] 1H-indazole-3-carboxylate —— C24H21FN4O3
[(E)-3-cyano-4-(4-fluorophenyl)-2-oxo-4-piperidin-1-ylbut-3-enyl] 1H-indazole-3-carboxylate
—— Ethyl 5-acetyl-4-methyl-2-[[2-(3-methyl-4-oxoquinazolin-2-yl)sulfanylacetyl]amino]thiophene-3-carboxylate —— C21H21N3O5S2
Ethyl 5-acetyl-4-methyl-2-[[2-(3-methyl-4-oxoquinazolin-2-yl)sulfanylacetyl]amino]thiophene-3-carboxylate
—— ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C22H26ClN3O7S2
ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-3-(5-bromofuran-2-yl)-N-(thiophen-2-ylmethyl)prop-2-enamide —— C12H10BrNO2S
(E)-3-(5-bromofuran-2-yl)-N-(thiophen-2-ylmethyl)prop-2-enamide
—— (E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(5-ethylthiophen-2-yl)methyl]prop-2-enamide —— C21H21N3O2S2
(E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(5-ethylthiophen-2-yl)methyl]prop-2-enamide
—— (E)-3-[4-(2-oxopyrrolidin-1-yl)phenyl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C23H26N4O2
(E)-3-[4-(2-oxopyrrolidin-1-yl)phenyl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-N-[(5-ethylthiophen-2-yl)methyl]-3-[4-(methylsulfamoyl)phenyl]prop-2-enamide —— C17H20N2O3S2
(E)-N-[(5-ethylthiophen-2-yl)methyl]-3-[4-(methylsulfamoyl)phenyl]prop-2-enamide