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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8aR)-2-(3-amino-5-fluoropyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one —— C12H15FN4O
(8aR)-2-(3-amino-5-fluoropyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one
—— (8aS)-2-(3-amino-5-fluoropyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one —— C12H15FN4O
(8aS)-2-(3-amino-5-fluoropyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one
—— 8-[4-(Diethylamino)-2-[8-(3-pentyloctanoyloxy)octoxy]butoxy]octyl 3-pentyloctanoate —— C50H99NO6
8-[4-(Diethylamino)-2-[8-(3-pentyloctanoyloxy)octoxy]butoxy]octyl 3-pentyloctanoate
—— 8-(4-ethoxyphenyl)-6-oxo-3,4-dihydro-2H,6H-pyrimido[2,1-b][1,3]thiazine-7-carbonitrile —— C16H15N3O2S
8-(4-ethoxyphenyl)-6-oxo-3,4-dihydro-2H,6H-pyrimido[2,1-b][1,3]thiazine-7-carbonitrile
—— 8-Ethyl-6-[2-fluoro-4-(2-fluoropyridin-3-yl)phenyl]-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C32H30F2N6O
8-Ethyl-6-[2-fluoro-4-(2-fluoropyridin-3-yl)phenyl]-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 8-Ethyl-6-[2-methyl-6-(1-propan-2-ylpyrrolidin-3-yl)pyridin-3-yl]-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C33H39N7O
8-Ethyl-6-[2-methyl-6-(1-propan-2-ylpyrrolidin-3-yl)pyridin-3-yl]-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(Dimethylamino)ethyl]-6-[4-methyl-2-(1-methylpiperidin-2-yl)phenyl]-2-(4-piperidin-4-ylanilino)pyrido[2,3-d]pyrimidin-7-one —— C35H45N7O
8-[2-(Dimethylamino)ethyl]-6-[4-methyl-2-(1-methylpiperidin-2-yl)phenyl]-2-(4-piperidin-4-ylanilino)pyrido[2,3-d]pyrimidin-7-one
—— 8-Ethyl-6-(2-fluoro-4-pyrazin-2-ylphenyl)-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C31H30FN7O
8-Ethyl-6-(2-fluoro-4-pyrazin-2-ylphenyl)-2-[4-(1-methylpiperidin-4-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-6-[3-methyl-5-(1,3-oxazol-4-yl)pyridin-2-yl]-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one —— C31H32N8O2
8-(Cyclopropylmethyl)-6-[3-methyl-5-(1,3-oxazol-4-yl)pyridin-2-yl]-2-[4-(4-methylpiperazin-1-yl)anilino]pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-[Methyl(methylsulfanyl)amino]ethyl]-2-[4-(1-methylpiperidin-3-yl)oxyanilino]-6-[4-pyridin-4-yl-2-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-7-one —— C35H36F3N7O2S
8-[2-[Methyl(methylsulfanyl)amino]ethyl]-2-[4-(1-methylpiperidin-3-yl)oxyanilino]-6-[4-pyridin-4-yl-2-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(Dimethylamino)ethyl]-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-6-(5-methyl-2-pyrrolidin-2-ylpyrimidin-4-yl)pyrido[2,3-d]pyrimidin-7-one —— C31H39N9O2
8-[2-(Dimethylamino)ethyl]-2-[4-(1-methylpyrrolidin-3-yl)oxyanilino]-6-(5-methyl-2-pyrrolidin-2-ylpyrimidin-4-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-Phenyl-2-(4-piperidin-3-yloxyanilino)-6-[4-(1-prop-1-en-2-ylpyrrolidin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one —— C37H38N6O2
8-Phenyl-2-(4-piperidin-3-yloxyanilino)-6-[4-(1-prop-1-en-2-ylpyrrolidin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(Dimethylamino)ethyl]-6-[1-methyl-4-(1,3,4-oxadiazol-2-yl)imidazol-2-yl]-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one —— C27H31N11O2
8-[2-(Dimethylamino)ethyl]-6-[1-methyl-4-(1,3,4-oxadiazol-2-yl)imidazol-2-yl]-2-(4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one
—— 8-Methyl-2-[4-(1-methylpiperidin-4-yl)anilino]-6-(2-methyl-5-pyridin-3-ylphenyl)pyrido[2,3-d]pyrimidin-7-one 1428760-01-3 C32H32N6O
8-Methyl-2-[4-(1-methylpiperidin-4-yl)anilino]-6-(2-methyl-5-pyridin-3-ylphenyl)pyrido[2,3-d]pyrimidin-7-one
—— 8-(1-methylsulfinylpiperidin-4-yl)-2-(4-piperidin-3-yloxyanilino)-6-(5-pyridin-4-yl-1H-imidazol-2-yl)pyrido[2,3-d]pyrimidin-7-one —— C32H35N9O3S
8-(1-methylsulfinylpiperidin-4-yl)-2-(4-piperidin-3-yloxyanilino)-6-(5-pyridin-4-yl-1H-imidazol-2-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[4-(4-methylmorpholin-2-yl)anilino]-6-[4-(1-methylpyrrol-2-yl)-2-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-7-one —— C35H35F3N6O2
8-Cyclopentyl-2-[4-(4-methylmorpholin-2-yl)anilino]-6-[4-(1-methylpyrrol-2-yl)-2-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-7-one
—— 8-Ethyl-2-[3-fluoro-4-(3-methylpiperazin-1-yl)anilino]-6-[2-(2-methylpyrazol-3-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one —— C30H31FN8O
8-Ethyl-2-[3-fluoro-4-(3-methylpiperazin-1-yl)anilino]-6-[2-(2-methylpyrazol-3-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one
—— 8-Propan-2-yl-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)-3-(trifluoromethyl)anilino]-6-[4-(1,3-thiazol-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one —— C31H27F3N6OS
8-Propan-2-yl-2-[4-(1,2,3,6-tetrahydropyridin-4-yl)-3-(trifluoromethyl)anilino]-6-[4-(1,3-thiazol-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-6-[2,6-dichloro-4-(1-methylpiperidin-2-yl)phenyl]-2-(3-methyl-4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one —— C34H39Cl2N7O
8-(Cyclopropylmethyl)-6-[2,6-dichloro-4-(1-methylpiperidin-2-yl)phenyl]-2-(3-methyl-4-piperazin-1-ylanilino)pyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[4-(1-methylpiperidin-4-yl)anilino]-6-(5-methyl-2-thiophen-3-ylpyrimidin-4-yl)pyrido[2,3-d]pyrimidin-7-one —— C32H33N7OS
8-(Cyclopropylmethyl)-2-[4-(1-methylpiperidin-4-yl)anilino]-6-(5-methyl-2-thiophen-3-ylpyrimidin-4-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-[Methyl(methylsulfanyl)amino]ethyl]-2-[4-(1-methylpiperidin-3-yl)anilino]-6-(5-piperidin-4-ylpyridin-2-yl)pyrido[2,3-d]pyrimidin-7-one —— C33H42N8OS
8-[2-[Methyl(methylsulfanyl)amino]ethyl]-2-[4-(1-methylpiperidin-3-yl)anilino]-6-(5-piperidin-4-ylpyridin-2-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[4-(1-methylpiperidin-3-yl)anilino]-6-(4-methyl-2-thiophen-3-ylpyrimidin-5-yl)pyrido[2,3-d]pyrimidin-7-one —— C33H35N7OS
8-Cyclopentyl-2-[4-(1-methylpiperidin-3-yl)anilino]-6-(4-methyl-2-thiophen-3-ylpyrimidin-5-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(Dimethylamino)ethyl]-2-[4-(4-methylmorpholin-2-yl)anilino]-6-[2-(1,2-oxazol-4-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one —— C31H33N7O3
8-[2-(Dimethylamino)ethyl]-2-[4-(4-methylmorpholin-2-yl)anilino]-6-[2-(1,2-oxazol-4-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(Dimethylamino)ethyl]-2-[4-(1-methylpiperidin-4-yl)anilino]-6-(2-pyridin-2-ylpyrimidin-5-yl)pyrido[2,3-d]pyrimidin-7-one —— C32H35N9O
8-[2-(Dimethylamino)ethyl]-2-[4-(1-methylpiperidin-4-yl)anilino]-6-(2-pyridin-2-ylpyrimidin-5-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-6-[4-methyl-6-(1,3,4-oxadiazol-2-yl)pyridin-3-yl]-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C31H32N8O3
8-Cyclopentyl-6-[4-methyl-6-(1,3,4-oxadiazol-2-yl)pyridin-3-yl]-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[4-(4-methylmorpholin-2-yl)anilino]-6-(3-methyl-5-pyrazin-2-ylpyridin-2-yl)pyrido[2,3-d]pyrimidin-7-one —— C32H32N8O2
8-(Cyclopropylmethyl)-2-[4-(4-methylmorpholin-2-yl)anilino]-6-(3-methyl-5-pyrazin-2-ylpyridin-2-yl)pyrido[2,3-d]pyrimidin-7-one
—— 8-(2-morpholin-4-ylethyl)-2-(4-pyrrolidin-3-yloxyanilino)-6-[2-(3H-pyrrol-5-yl)-4,5-dihydropyrimidin-5-yl]-8H-quinazolin-7-one —— C32H36N8O3
8-(2-morpholin-4-ylethyl)-2-(4-pyrrolidin-3-yloxyanilino)-6-[2-(3H-pyrrol-5-yl)-4,5-dihydropyrimidin-5-yl]-8H-quinazolin-7-one
—— 8-(Cyclopropylmethyl)-6-(2-methyl-4-piperidin-4-ylphenyl)-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C34H40N6O2
8-(Cyclopropylmethyl)-6-(2-methyl-4-piperidin-4-ylphenyl)-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(Dimethylamino)ethyl]-6-[2-fluoro-4-(oxan-4-yl)phenyl]-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one —— C33H39FN6O3
8-[2-(Dimethylamino)ethyl]-6-[2-fluoro-4-(oxan-4-yl)phenyl]-2-(4-piperidin-3-yloxyanilino)pyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[4-(1-methylpiperidin-3-yl)anilino]-6-[1-(2-methylpyrazol-3-yl)imidazol-2-yl]pyrido[2,3-d]pyrimidin-7-one —— C30H33N9O
8-(Cyclopropylmethyl)-2-[4-(1-methylpiperidin-3-yl)anilino]-6-[1-(2-methylpyrazol-3-yl)imidazol-2-yl]pyrido[2,3-d]pyrimidin-7-one
—— 8-methoxy-3-[4-(3-methoxyphenyl)-1,3-thiazol-2-yl]-2H-chromen-2-one —— C20H15NO4S
8-methoxy-3-[4-(3-methoxyphenyl)-1,3-thiazol-2-yl]-2H-chromen-2-one
—— 8-Methoxy-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]chromen-2-one —— C19H12N2O5S
8-Methoxy-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]chromen-2-one
—— 8-methoxy-3-[4-(2-oxo-2H-chromen-3-yl)-1,3-thiazol-2-yl]-2H-chromen-2-one —— C22H13NO5S
8-methoxy-3-[4-(2-oxo-2H-chromen-3-yl)-1,3-thiazol-2-yl]-2H-chromen-2-one
—— (8aR)-2-(3-amino-5-methylpyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one —— C13H18N4O
(8aR)-2-(3-amino-5-methylpyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one
—— (8aS)-2-(3-amino-5-methylpyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one —— C13H18N4O
(8aS)-2-(3-amino-5-methylpyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one
—— 8-(3-Amino-5-methylpyridin-4-yl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one —— C14H20N4O2
8-(3-Amino-5-methylpyridin-4-yl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
—— 8-(3-Aminopyridin-4-yl)-1-methyl-1,8-diazaspiro[4.5]decan-2-one —— C14H20N4O
8-(3-Aminopyridin-4-yl)-1-methyl-1,8-diazaspiro[4.5]decan-2-one
—— (8aR)-2-(3-aminopyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one —— C12H16N4O
(8aR)-2-(3-aminopyridin-4-yl)-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-6-one
—— (8aR)-7-(3-amino-5-methylpyridin-4-yl)-5,6,8,8a-tetrahydro-1H-[1,3]oxazolo[3,4-a]pyrazin-3-one —— C12H16N4O2
(8aR)-7-(3-amino-5-methylpyridin-4-yl)-5,6,8,8a-tetrahydro-1H-[1,3]oxazolo[3,4-a]pyrazin-3-one
—— 8-Tert-butyl-4,4-dimethyltetrazolo[5,1-c][1,4]benzoxazine —— C14H18N4O
8-Tert-butyl-4,4-dimethyltetrazolo[5,1-c][1,4]benzoxazine
—— [(8E)-8-[2,2-dimethyl-3-[(E)-(2-methyl-6,7-dihydro-5H-quinolin-8-ylidene)amino]oxypropoxy]imino-2-methyl-6,7-dihydro-5H-quinolin-4-yl]methanol —— C26H34N4O3
[(8E)-8-[2,2-dimethyl-3-[(E)-(2-methyl-6,7-dihydro-5H-quinolin-8-ylidene)amino]oxypropoxy]imino-2-methyl-6,7-dihydro-5H-quinolin-4-yl]methanol
—— 8-Chloro-2-oxa-8-azaspiro[3.5]nonane —— C7H12ClNO
8-Chloro-2-oxa-8-azaspiro[3.5]nonane
—— 8-Methyl-3-oxabicyclo[3.2.1]octane —— C8H14O
8-Methyl-3-oxabicyclo[3.2.1]octane
—— 8-Chloro-2-cyclobutyl-3-methylimidazo[1,2-a]pyridine —— C12H13ClN2
8-Chloro-2-cyclobutyl-3-methylimidazo[1,2-a]pyridine
—— 8-Chloro-3-methyl-2-(trideuteriomethoxymethyl)imidazo[1,2-a]pyridine —— C10H11ClN2O
8-Chloro-3-methyl-2-(trideuteriomethoxymethyl)imidazo[1,2-a]pyridine
—— 8-Tert-butyl-2-oxa-8-azaspiro[3.5]nonane —— C11H21NO
8-Tert-butyl-2-oxa-8-azaspiro[3.5]nonane
—— [8-(2,2-Dimethylpropanoyl)naphthalen-2-yl]-methylborinic acid —— C16H19BO2
[8-(2,2-Dimethylpropanoyl)naphthalen-2-yl]-methylborinic acid
—— 8-(2,2-Dimethylpropyl)-3-methyl-3-azabicyclo[3.2.1]octane —— C13H25N
8-(2,2-Dimethylpropyl)-3-methyl-3-azabicyclo[3.2.1]octane
—— [8-[4-[3-(Aminomethyl)phenyl]piperidine-1-carbonyl]-4-fluoronaphthalen-2-yl]boronic acid —— C23H24BFN2O3
[8-[4-[3-(Aminomethyl)phenyl]piperidine-1-carbonyl]-4-fluoronaphthalen-2-yl]boronic acid
—— [8-[4-[3-(Aminomethyl)phenyl]piperidine-1-carbonyl]quinolin-2-yl]boronic acid —— C22H24BN3O3
[8-[4-[3-(Aminomethyl)phenyl]piperidine-1-carbonyl]quinolin-2-yl]boronic acid