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—— (8S)-8-(4-chlorophenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C19H16ClN3O2S
(8S)-8-(4-chlorophenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-3-(3,4-dimethylphenyl)-6-oxo-8-(3,4,5-trimethoxyphenyl)-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C25H27N3O4S
(8R)-3-(3,4-dimethylphenyl)-6-oxo-8-(3,4,5-trimethoxyphenyl)-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-[1-[3-Fluoro-8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H30F7NO3
8-[1-[3-Fluoro-8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-(4-Benzylpiperazin-4-ium-1-yl)-3-methyl-7-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl]purine-2,6-dione —— C22H27N8O2S2+
8-(4-Benzylpiperazin-4-ium-1-yl)-3-methyl-7-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl]purine-2,6-dione
—— (8S)-3-(3-chlorophenyl)-8-(2,4-dimethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C22H20ClN3O3S
(8S)-3-(3-chlorophenyl)-8-(2,4-dimethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-methyl-N-(pyridin-3-ylmethyl)-6,7,8,9-tetrahydropyrido[4',3':4,5]thieno[3,2-e]tetrazolo[1,5-a]pyrimidin-5-amine —— C16H16N8S
8-methyl-N-(pyridin-3-ylmethyl)-6,7,8,9-tetrahydropyrido[4',3':4,5]thieno[3,2-e]tetrazolo[1,5-a]pyrimidin-5-amine
—— 8-[2-[3-Fluoro-8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H30F7NO3
8-[2-[3-Fluoro-8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— (8R)-8-(4-chlorophenyl)-3-(furan-2-ylmethyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile —— C19H17ClN3O2S+
(8R)-8-(4-chlorophenyl)-3-(furan-2-ylmethyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile
—— 8-[1-[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]propyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H36ClNO3
8-[1-[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]propyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— (8S,9S,10R,13S,14S,17S)-17-acetyl-1-hydroxy-10,13-dimethyl-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-3-one;(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-1-[(2S)-2-[(carbamoylamino)carbamoyl]pyrrolidin-1-yl]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-[(2-methylpropan-2-yl)oxy]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide —— C80H114N18O17
(8S,9S,10R,13S,14S,17S)-17-acetyl-1-hydroxy-10,13-dimethyl-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-3-one;(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-1-[(2S)-2-[(carbamoylamino)carbamoyl]pyrrolidin-1-yl]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-[(2-methylpropan-2-yl)oxy]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide
—— (8R)-8-(5-methylfuran-2-yl)-3-(3-methylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C20H19N3O2S
(8R)-8-(5-methylfuran-2-yl)-3-(3-methylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-3-benzyl-8-(2-chloro-6-fluorophenyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile —— C21H18ClFN3OS+
(8S)-3-benzyl-8-(2-chloro-6-fluorophenyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile
—— (8R)-8-(4-chlorophenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C19H16ClN3O2S
(8R)-8-(4-chlorophenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-[3-[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]propyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H36ClNO3
8-[3-[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]propyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[[4-(2-Fluorophenyl)piperazin-1-ium-1-yl]methyl]-1,3-dimethyl-7-propylpurine-2,6-dione —— C21H28FN6O2+
8-[[4-(2-Fluorophenyl)piperazin-1-ium-1-yl]methyl]-1,3-dimethyl-7-propylpurine-2,6-dione
—— (8S)-8-(5-methylfuran-2-yl)-3-(3-methylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C20H19N3O2S
(8S)-8-(5-methylfuran-2-yl)-3-(3-methylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-Trifluoromethyl-7-(4-trifluoromethyl-cyclohexyloxy)-naphthalene-2-carbaldehyde —— C19H16F6O2
8-Trifluoromethyl-7-(4-trifluoromethyl-cyclohexyloxy)-naphthalene-2-carbaldehyde
—— 8-Methoxy-3-prop-2-enyl-2-propylchromeno[2,3-d]pyrimidine-4,5-dione —— C18H18N2O4
8-Methoxy-3-prop-2-enyl-2-propylchromeno[2,3-d]pyrimidine-4,5-dione
—— 8-{(S)-1-[7-(cis-4-methyl-cyclohexyloxy)-8-trifluoromethyl-naphthalen-2-yl]-ethyl}-8-aza-bicyclo[3.2.1]octane-3-carboxylic acid —— C28H34F3NO3
8-{(S)-1-[7-(cis-4-methyl-cyclohexyloxy)-8-trifluoromethyl-naphthalen-2-yl]-ethyl}-8-aza-bicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[3-[7-(4-Methylcyclohexyl)oxy-8-(trifluoromethyl)naphthalen-2-yl]propyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C29H36F3NO3
8-[3-[7-(4-Methylcyclohexyl)oxy-8-(trifluoromethyl)naphthalen-2-yl]propyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[2-[7-(4-Ethylcyclohexyl)oxy-8-(trifluoromethyl)naphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C29H36F3NO3
8-[2-[7-(4-Ethylcyclohexyl)oxy-8-(trifluoromethyl)naphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[[3-Fluoro-8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C27H28F7NO3
8-[[3-Fluoro-8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[1-[8-(Difluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H32F5NO3
8-[1-[8-(Difluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[2-[8-(Difluoromethyl)-7-(4-ethylcyclohexyl)oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C29H37F2NO3
8-[2-[8-(Difluoromethyl)-7-(4-ethylcyclohexyl)oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— (8aR,9S)-6,6-dimethyl-2-methylsulfanyl-9-thiophen-2-yl-1,7,8a,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C16H18N4OS2
(8aR,9S)-6,6-dimethyl-2-methylsulfanyl-9-thiophen-2-yl-1,7,8a,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 8,9-Dimethoxy-3-(4-methoxyphenyl)-5-methyl-[1,2,4]triazolo[4,3-c]quinazoline —— C19H18N4O3
8,9-Dimethoxy-3-(4-methoxyphenyl)-5-methyl-[1,2,4]triazolo[4,3-c]quinazoline
—— 8-[1-[8-(Difluoromethyl)-7-(4-ethylcyclohexyl)oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C29H37F2NO3
8-[1-[8-(Difluoromethyl)-7-(4-ethylcyclohexyl)oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-(2-methoxy-4-nitrophenyl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazine —— C14H19N3O4
8-(2-methoxy-4-nitrophenyl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazine
—— 8-[2-[8-(Difluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H32F5NO3
8-[2-[8-(Difluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-(Difluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalene-2-carbaldehyde —— C19H17F5O2
8-(Difluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalene-2-carbaldehyde
—— 8-Propanoyloxyoctadec-9-enoic acid —— C21H38O4
8-Propanoyloxyoctadec-9-enoic acid
—— (8aS,9R)-6,6-dimethyl-2-methylsulfanyl-9-thiophen-2-yl-1,7,8a,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C16H18N4OS2
(8aS,9R)-6,6-dimethyl-2-methylsulfanyl-9-thiophen-2-yl-1,7,8a,9-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 8-[[7-(4-Ethylcyclohexyl)oxy-8-(trifluoromethyl)naphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H34F3NO3
8-[[7-(4-Ethylcyclohexyl)oxy-8-(trifluoromethyl)naphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[(1S)-2,2,2-trideuterio-1-[8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H31F6NO3
8-[(1S)-2,2,2-trideuterio-1-[8-(trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[2-[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C27H34ClNO3
8-[2-[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[[8-Cyano-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C27H29F3N2O3
8-[[8-Cyano-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C26H32ClNO3
8-[[8-Chloro-7-(4-methylcyclohexyl)oxynaphthalen-2-yl]methyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— (8R)-8-(3-ethoxy-4-hydroxyphenyl)-3-(4-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C23H23N3O4S
(8R)-8-(3-ethoxy-4-hydroxyphenyl)-3-(4-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-(4-nitrophenyl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazine —— C13H17N3O3
8-(4-nitrophenyl)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazine
—— (8S)-8-(3-ethoxy-4-hydroxyphenyl)-3-(4-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C23H23N3O4S
(8S)-8-(3-ethoxy-4-hydroxyphenyl)-3-(4-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-[(4-ethylpiperazin-4-ium-1-yl)methyl]-7-[(4-fluorophenyl)methyl]-1,3-dimethylpurine-2,6-dione —— C21H28FN6O2+
8-[(4-ethylpiperazin-4-ium-1-yl)methyl]-7-[(4-fluorophenyl)methyl]-1,3-dimethylpurine-2,6-dione
—— (8S)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile —— C21H22N3O4S+
(8S)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile
—— 8-[[4-(2-fluorophenyl)piperazin-1-ium-1-yl]methyl]-1,3-dimethyl-7-[(4-methylphenyl)methyl]purine-2,6-dione —— C26H30FN6O2+
8-[[4-(2-fluorophenyl)piperazin-1-ium-1-yl]methyl]-1,3-dimethyl-7-[(4-methylphenyl)methyl]purine-2,6-dione
—— 8-[7-(4-Methylcyclohexyl)oxy-8-(trifluoromethyl)naphthalene-2-carbonyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C27H30F3NO4
8-[7-(4-Methylcyclohexyl)oxy-8-(trifluoromethyl)naphthalene-2-carbonyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— (8R)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C21H21N3O4S
(8R)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile —— C21H22N3O4S+
(8R)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-3,4,7,8-tetrahydro-2H-pyrido[2,1-b][1,3,5]thiadiazin-3-ium-9-carbonitrile
—— 8-[2-[8-Cyano-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H31F3N2O3
8-[2-[8-Cyano-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— (8S)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C21H21N3O4S
(8S)-8-(2,3-dimethoxyphenyl)-3-(furan-2-ylmethyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-[1-[8-Cyano-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H31F3N2O3
8-[1-[8-Cyano-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8-[2-[8-(Trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C28H31F6NO3
8-[2-[8-(Trifluoromethyl)-7-[4-(trifluoromethyl)cyclohexyl]oxynaphthalen-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid