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—— [(8aR)-1,3,4,5,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-5-ium-2-yl]-[7-(difluoromethyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]methanone —— C22H24F2N5O+
[(8aR)-1,3,4,5,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-5-ium-2-yl]-[7-(difluoromethyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]methanone
—— (8,8-Dibromo-2-methoxyoctyl) prop-2-enoate —— C12H20Br2O3
(8,8-Dibromo-2-methoxyoctyl) prop-2-enoate
—— 8-phenoxy-9-(trifluoromethyl)-2,3-dihydro-7H-[1,4]dioxino[2,3-h]chromen-7-one —— C18H11F3O5
8-phenoxy-9-(trifluoromethyl)-2,3-dihydro-7H-[1,4]dioxino[2,3-h]chromen-7-one
—— (8R)-6-amino-8-(2-nitrophenyl)-2,4-dioxo-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile —— C14H9N5O5
(8R)-6-amino-8-(2-nitrophenyl)-2,4-dioxo-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile
—— (8S)-6-amino-8-(2-nitrophenyl)-2,4-dioxo-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile —— C14H9N5O5
(8S)-6-amino-8-(2-nitrophenyl)-2,4-dioxo-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile
—— (8R)-6-amino-8-(4-nitrophenyl)-2,4-dioxo-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile —— C14H9N5O5
(8R)-6-amino-8-(4-nitrophenyl)-2,4-dioxo-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile
—— (8S)-8-(5-chloro-2-methoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C17H14ClNO4
(8S)-8-(5-chloro-2-methoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (8S)-8-(4-propan-2-ylphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H19NO3
(8S)-8-(4-propan-2-ylphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (8R)-8-(5-chloro-2-methoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C17H14ClNO4
(8R)-8-(5-chloro-2-methoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 8-bromo-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C18H17BrClN3O
8-bromo-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— (8R)-8-(4-propan-2-ylphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H19NO3
(8R)-8-(4-propan-2-ylphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 8-chloro-N-(4-chlorophenyl)-7-methoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C19H19Cl2N3O2
8-chloro-N-(4-chlorophenyl)-7-methoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-(((3R,3aR,6R,6aS)-6-((tert-butyldimethylsilyl)oxy)hexahydrofuro[3,2-b]furan-3-yl)oxy)-2-chloro-7-((2-(trimethylsilyl)ethoxy)methyl)-7H-purine —— C23H39ClN4O5Si2
8-(((3R,3aR,6R,6aS)-6-((tert-butyldimethylsilyl)oxy)hexahydrofuro[3,2-b]furan-3-yl)oxy)-2-chloro-7-((2-(trimethylsilyl)ethoxy)methyl)-7H-purine
—— (±)-8-chloro-N,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)phenyl]-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide —— C24H27ClF3N5O2
(±)-8-chloro-N,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)phenyl]-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide
—— (±)-8-chloro-N,4-dimethyl-1-[4-(piperazin-1-yl)phenyl]-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide —— C23H25ClF3N5O2
(±)-8-chloro-N,4-dimethyl-1-[4-(piperazin-1-yl)phenyl]-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide
—— (±)-8-chloro-1-[4-(4-hydroxypiperidin-1-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide —— C24H26ClF3N4O3
(±)-8-chloro-1-[4-(4-hydroxypiperidin-1-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide
—— (±)-8-methoxy-N,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)phenyl]-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide —— C25H30F3N5O3
(±)-8-methoxy-N,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)phenyl]-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide
—— 8-acetamido-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C20H21ClN4O2
8-acetamido-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-(1,1-dihydroxy-1,4-thiazinan-4-yl)-1-[4-(1,1-dihydroxy-1,4-thiazinan-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C27H36F3N5O6S2
8-(1,1-dihydroxy-1,4-thiazinan-4-yl)-1-[4-(1,1-dihydroxy-1,4-thiazinan-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-chloro-1-[4-(1,1-dihydroxy-1,4-thiazinan-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C23H26ClF3N4O4S
8-chloro-1-[4-(1,1-dihydroxy-1,4-thiazinan-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-(1,1-dioxo-1,4-thiazinan-4-yl)-1-[4-(1,1-dioxo-1,4-thiazinan-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C27H32F3N5O6S2
8-(1,1-dioxo-1,4-thiazinan-4-yl)-1-[4-(1,1-dioxo-1,4-thiazinan-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-chloro-N-(4-chlorophenyl)-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C19H16Cl2F3N3O2
8-chloro-N-(4-chlorophenyl)-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— (±)-8-chloro-1-[4-(1,1-dioxidothiomorpholin-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide —— C23H24ClF3N4O4S
(±)-8-chloro-1-[4-(1,1-dioxidothiomorpholin-4-yl)phenyl]-N,4-dimethyl-7-(trifluoromethoxy)-4,5-dihydro-3H-2,3-benzodiazepine-3-carboxamide
—— 8-[1-(3-chloro-4-fluorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C24H23ClFNO4S
8-[1-(3-chloro-4-fluorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— (8R)-6-amino-2,4-dioxo-8-(3,4,5-trimethoxyphenyl)-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile —— C17H16N4O6
(8R)-6-amino-2,4-dioxo-8-(3,4,5-trimethoxyphenyl)-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile
—— (8S)-6-amino-2,4-dioxo-8-(3,4,5-trimethoxyphenyl)-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile —— C17H16N4O6
(8S)-6-amino-2,4-dioxo-8-(3,4,5-trimethoxyphenyl)-1,8-dihydropyrano[3,2-d]pyrimidine-7-carbonitrile
—— 8-tert-butyl-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C22H26ClN3O
8-tert-butyl-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-Fluoro-6-methoxy-3-methyl-7-(2-methylpyridin-3-yl)pyrazolo[3,4-c]cinnoline —— C17H14FN5O
8-Fluoro-6-methoxy-3-methyl-7-(2-methylpyridin-3-yl)pyrazolo[3,4-c]cinnoline
—— 8-hydroxy-N,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)phenyl]-7-oxo-4,5-dihydro-2H-2,3-benzodiazepine-3-carboxamide —— C23H29N5O3
8-hydroxy-N,4-dimethyl-1-[4-(4-methylpiperazin-1-yl)phenyl]-7-oxo-4,5-dihydro-2H-2,3-benzodiazepine-3-carboxamide
—— 8-[1-(3,5-difluorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C24H23F2NO4S
8-[1-(3,5-difluorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— 8-(2-chloro-4-fluoro-6-methoxy-3-methylphenyl)-3H-pyrazolo[3,4-c]cinnoline —— C17H12ClFN4O
8-(2-chloro-4-fluoro-6-methoxy-3-methylphenyl)-3H-pyrazolo[3,4-c]cinnoline
—— [(8R,9S,10R,13S,14S,17R)-17-acetyl-10,13-dimethyl-3-oxo-2,6,7,8,9,11,12,14,15,16-decahydro-1H-cyclopenta[a]phenanthren-17-yl] hexanoate;(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[(2S)-2-(ethylcarbamoyl)pyrrolidin-1-yl]-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide —— C86H124N16O16
[(8R,9S,10R,13S,14S,17R)-17-acetyl-10,13-dimethyl-3-oxo-2,6,7,8,9,11,12,14,15,16-decahydro-1H-cyclopenta[a]phenanthren-17-yl] hexanoate;(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[(2S)-2-(ethylcarbamoyl)pyrrolidin-1-yl]-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide
—— 8-(1-((4-chlorophenyl)sulfonyl)cyclobutyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-23-4 C23H26ClNO4S
8-(1-((4-chlorophenyl)sulfonyl)cyclobutyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 8-Fluoro-6-methoxy-3-methyl-9-(2-methylpyridin-3-yl)pyrazolo[3,4-c]cinnoline —— C17H14FN5O
8-Fluoro-6-methoxy-3-methyl-9-(2-methylpyridin-3-yl)pyrazolo[3,4-c]cinnoline
—— (8S)-8-(4-ethoxyphenyl)-11,11-dimethyl-7,8,10,12-tetrahydrobenzo[a][4,7]phenanthrolin-9-one —— C26H26N2O2
(8S)-8-(4-ethoxyphenyl)-11,11-dimethyl-7,8,10,12-tetrahydrobenzo[a][4,7]phenanthrolin-9-one
—— 8-[1-(Benzenesulfinyl)cyclopentyl]-3,3-dimethyl-2,5-dihydro-1,5-benzoxazepin-4-one —— C22H25NO3S
8-[1-(Benzenesulfinyl)cyclopentyl]-3,3-dimethyl-2,5-dihydro-1,5-benzoxazepin-4-one
—— 8-amino-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide —— C18H19ClN4O
8-amino-N-(4-chlorophenyl)-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide
—— 8-(1-((3,4-dichlorophenyl)sulfonyl)cyclopentyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-00-7 C24H27Cl2NO4S
8-(1-((3,4-dichlorophenyl)sulfonyl)cyclopentyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 8-[1-(3-chloro-5-fluorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C24H23ClFNO4S
8-[1-(3-chloro-5-fluorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— 8-(1-((3-chloro-5-fluorophenyl)sulfonyl)cyclopentyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563205-95-7 C24H27ClFNO4S
8-(1-((3-chloro-5-fluorophenyl)sulfonyl)cyclopentyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 8-[1-(3,4-dichlorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one —— C24H23Cl2NO4S
8-[1-(3,4-dichlorophenyl)sulfonylcyclopenta-2,4-dien-1-yl]-5-ethyl-3,3-dimethyl-2H-1,5-benzoxazepin-4-one
—— [(8S,9R,10S,11S,13S,14S,16S,17R)-17-(2-chloroacetyl)-9-fluoro-10,13,16-trimethyl-3-oxo-17-propanoyloxy-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-11-yl] 2-hydroxypropanoate —— C28H36ClFO7
[(8S,9R,10S,11S,13S,14S,16S,17R)-17-(2-chloroacetyl)-9-fluoro-10,13,16-trimethyl-3-oxo-17-propanoyloxy-6,7,8,11,12,14,15,16-octahydrocyclopenta[a]phenanthren-11-yl] 2-hydroxypropanoate
—— 8-(1-((4-chlorophenyl)sulfonyl)cyclohexyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-16-5 C25H30ClNO4S
8-(1-((4-chlorophenyl)sulfonyl)cyclohexyl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— (8S)-8-(4-propoxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one —— C25H24N2O2
(8S)-8-(4-propoxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one
—— (8S)-8-(3-ethoxy-4-hydroxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one —— C24H22N2O3
(8S)-8-(3-ethoxy-4-hydroxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one
—— (8R)-8-(3-ethoxy-4-hydroxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one —— C24H22N2O3
(8R)-8-(3-ethoxy-4-hydroxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one
—— 8-(4-((4-chlorophenyl)sulfonyl)tetrahydro-2H-pyran-4-yl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one 1563206-24-5 C24H26F3NO4S
8-(4-((4-chlorophenyl)sulfonyl)tetrahydro-2H-pyran-4-yl)-5-ethyl-3,3-dimethyl-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— 8-Phenyl-6-azaspiro[2.5]octane —— C13H17N
8-Phenyl-6-azaspiro[2.5]octane
—— 8-[3-Fluoro-4-(trifluoromethoxy)phenyl]-6,7-dihydropyrano[2,3-b]pyrazin-8-amine;hydrochloride —— C14H12ClF4N3O2
8-[3-Fluoro-4-(trifluoromethoxy)phenyl]-6,7-dihydropyrano[2,3-b]pyrazin-8-amine;hydrochloride
—— 8-(3-(1-benzyl-1H-benzo[d]imidazol-2-yl)propoxy)quinoline 1568975-52-9 C26H23N3O
8-(3-(1-benzyl-1H-benzo[d]imidazol-2-yl)propoxy)quinoline