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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-[2-(azetidin-3-yl-oxy)ethyl]-6-[2-chloro-4-(6-methyl-2-pyridyl)phenyl]-2-(ethylamino)pyrido[2,3-d]pyrimidin-7-one —— C26H27ClN6O2
8-[2-(azetidin-3-yl-oxy)ethyl]-6-[2-chloro-4-(6-methyl-2-pyridyl)phenyl]-2-(ethylamino)pyrido[2,3-d]pyrimidin-7-one
—— 8-[3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-1H-quinolin-2-one —— C22H20N6O2
8-[3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-1H-quinolin-2-one
—— 8-(6-(3,4-dimethoxyphenyl)isothiazolo[4,3-b]pyridin-3-yl)-1,4-dioxa-8-azaspiro[4.5]decane —— C21H23N3O4S
8-(6-(3,4-dimethoxyphenyl)isothiazolo[4,3-b]pyridin-3-yl)-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[(4-Aminocyclohexyl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(propan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one —— C29H33ClN6O
8-[(4-Aminocyclohexyl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(propan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one
—— 8-Chloro-7-methoxy-1-(3-methylpentyl)pyrimido[5,4-c]quinoline-2,4-dione —— C18H20ClN3O3
8-Chloro-7-methoxy-1-(3-methylpentyl)pyrimido[5,4-c]quinoline-2,4-dione
—— 8-methoxy-4-[[(3R)-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-3-yl]amino]quinoline-3-carboxylic acid —— C20H25N3O5
8-methoxy-4-[[(3R)-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-3-yl]amino]quinoline-3-carboxylic acid
—— 8-Bromo-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-2-carbaldehyde;8-bromo-2-ethynyl-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole —— C25H16Br2N2O3S2
8-Bromo-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole-2-carbaldehyde;8-bromo-2-ethynyl-4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazole
—— 8-bromo-2-[2-(1-methylpiperidin-4-yl)-1,2,4-triazol-3-yl]-4,5-dihydro-1H-[1]benzoxepino[5,4-d][1,2]thiazole —— C19H22BrN5OS
8-bromo-2-[2-(1-methylpiperidin-4-yl)-1,2,4-triazol-3-yl]-4,5-dihydro-1H-[1]benzoxepino[5,4-d][1,2]thiazole
—— 8-[2-(4-Acetyl-2-methylphenyl)ethylsulfonyl]-2-[3-hydroxy-5-(trifluoromethyl)phenyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C25H26F3N3O5S
8-[2-(4-Acetyl-2-methylphenyl)ethylsulfonyl]-2-[3-hydroxy-5-(trifluoromethyl)phenyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-[2-[Bis(8-hydroxyoctyl)amino]ethyl-(8-hydroxyoctyl)amino]octan-1-ol —— C34H72N2O4
8-[2-[Bis(8-hydroxyoctyl)amino]ethyl-(8-hydroxyoctyl)amino]octan-1-ol
—— 8-[(E)-2-(4-tert-butyl-2,6-dimethylphenyl)ethenoxy]-2-nonyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C30H47N3O2
8-[(E)-2-(4-tert-butyl-2,6-dimethylphenyl)ethenoxy]-2-nonyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-Butylsulfinyl-2-(2,4-dichlorophenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C17H21Cl2N3O2S
8-Butylsulfinyl-2-(2,4-dichlorophenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-[(S)-(3-chlorophenyl)sulfinyl]-2-piperidin-3-yl-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C18H23ClN4O2S
8-[(S)-(3-chlorophenyl)sulfinyl]-2-piperidin-3-yl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-[2-(1-Butylindol-4-yl)ethylsulfonyl]-2-cyclohexyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C27H38N4O3S
8-[2-(1-Butylindol-4-yl)ethylsulfonyl]-2-cyclohexyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-[(E)-2-[4-(hydroxymethylamino)-2-methylphenyl]ethenyl]sulfonyl-2-(4-methylcyclohexyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C24H34N4O4S
8-[(E)-2-[4-(hydroxymethylamino)-2-methylphenyl]ethenyl]sulfonyl-2-(4-methylcyclohexyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-[(E)-2-[4-[[2-[tert-butyl(dimethyl)silyl]oxyethylamino]methyl]-2-methylphenyl]ethenyl]sulfonyl-2-cyclohexyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C31H50N4O4SSi
8-[(E)-2-[4-[[2-[tert-butyl(dimethyl)silyl]oxyethylamino]methyl]-2-methylphenyl]ethenyl]sulfonyl-2-cyclohexyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-[2-[4-(3-Hydroxypropoxy)-2,6-dimethylphenyl]ethylsulfonyl]-2-(3-methylphenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one —— C27H35N3O5S
8-[2-[4-(3-Hydroxypropoxy)-2,6-dimethylphenyl]ethylsulfonyl]-2-(3-methylphenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
—— 8-Chloro-1-[4-(2,3-dihydropyridin-2-yl)cyclohexyl]-5-methyl-4,6-dihydro-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine —— C22H26ClN5
8-Chloro-1-[4-(2,3-dihydropyridin-2-yl)cyclohexyl]-5-methyl-4,6-dihydro-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine
—— [(8S,9S,10R,13R,14S,17R)-10,13-dimethyl-17-[(2R)-6-methylheptan-2-yl]-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3-yl] 2-[(2R)-2-carbamoylbutyl]sulfanylacetate —— C34H57NO3S
[(8S,9S,10R,13R,14S,17R)-10,13-dimethyl-17-[(2R)-6-methylheptan-2-yl]-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3-yl] 2-[(2R)-2-carbamoylbutyl]sulfanylacetate
—— 8-[5-chloro-3-ethyl-1-[1-[(5-methoxypyrazin-2-yl)amino]prop-1-enyl]-2H-indol-3-yl]octan-2-one —— C26H35ClN4O2
8-[5-chloro-3-ethyl-1-[1-[(5-methoxypyrazin-2-yl)amino]prop-1-enyl]-2H-indol-3-yl]octan-2-one
—— 8-[1-[(Z)-1-[(3-chloro-6-methyl-2-thiabicyclo[3.1.1]hept-3-en-1-yl)amino]prop-1-enyl]-3-ethyl-5-propyl-2H-indol-3-yl]octan-2-one —— C31H45ClN2OS
8-[1-[(Z)-1-[(3-chloro-6-methyl-2-thiabicyclo[3.1.1]hept-3-en-1-yl)amino]prop-1-enyl]-3-ethyl-5-propyl-2H-indol-3-yl]octan-2-one
—— 8-ethyl-2-methyl-10-oxo-3H-chromeno[3,2-c]pyridine-3-carboxylic acid —— C16H15NO4
8-ethyl-2-methyl-10-oxo-3H-chromeno[3,2-c]pyridine-3-carboxylic acid
—— 8,8,10-Triethyl-7,9,11-trimethyl-10-propyl-1,5-dioxa-9-phosphaspiro[5.5]undecane —— C20H39O2P
8,8,10-Triethyl-7,9,11-trimethyl-10-propyl-1,5-dioxa-9-phosphaspiro[5.5]undecane
—— [(8S)-5-(5-chloropyridin-2-yl)-3,4,6,12-tetrazatricyclo[6.3.1.02,6]dodeca-1,4-dien-3-yl]-[2-chloro-3-(trifluoromethyl)phenyl]methanone —— C21H16Cl2F3N5O
[(8S)-5-(5-chloropyridin-2-yl)-3,4,6,12-tetrazatricyclo[6.3.1.02,6]dodeca-1,4-dien-3-yl]-[2-chloro-3-(trifluoromethyl)phenyl]methanone
—— 8-[1-(2-Phenylquinolin-4-yl)ethyl]-1,4-dioxa-8-azaspiro[4.5]decane —— C24H26N2O2
8-[1-(2-Phenylquinolin-4-yl)ethyl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[1-hydroxy-2-methyl-1-[5-(tetrazol-1-yl)pyridin-2-yl]propan-2-yl]-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C23H29N7O4
8-[1-hydroxy-2-methyl-1-[5-(tetrazol-1-yl)pyridin-2-yl]propan-2-yl]-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-{2-[4-(hydroxymethyl)-6-(1H-tetrazol-1-yl)pyridin-3-yl]ethyl}-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-1-oxo-2-aza-8-azoniaspiro[4.5]decane —— C22H27N7O4
8-{2-[4-(hydroxymethyl)-6-(1H-tetrazol-1-yl)pyridin-3-yl]ethyl}-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-1-oxo-2-aza-8-azoniaspiro[4.5]decane
—— 8-(1-methyl-1H-imidazol-4-yl)-2-(2,2,2-trifluoroethoxy)pyrido[3,4-d]pyrimidin-4-ol —— C13H10F3N5O2
8-(1-methyl-1H-imidazol-4-yl)-2-(2,2,2-trifluoroethoxy)pyrido[3,4-d]pyrimidin-4-ol
—— [8-[2-Fluoro-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-2-yl]purin-9-yl]carbamic acid —— C20H8F10N6O2
[8-[2-Fluoro-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-2-yl]purin-9-yl]carbamic acid
—— 8-{(2R)-2-[2-fluoro-4-(1H-tetrazol-1-yl)phenyl]-2-hydroxyethyl}-1-oxo-2-(5-oxo-2,5-dihydrofuran-3-yl)-2-aza-8-azoniaspiro[4.5]decane —— C21H23FN6O4
8-{(2R)-2-[2-fluoro-4-(1H-tetrazol-1-yl)phenyl]-2-hydroxyethyl}-1-oxo-2-(5-oxo-2,5-dihydrofuran-3-yl)-2-aza-8-azoniaspiro[4.5]decane
—— 8-[2-hydroxy-2-[5-(tetrazol-1-yl)pyrazin-2-yl]ethyl]-2-[4-(methoxymethyl)-5-oxo-2H-furan-3-yl]-2,8-diazaspiro[4.5]decan-1-one —— C21H26N8O5
8-[2-hydroxy-2-[5-(tetrazol-1-yl)pyrazin-2-yl]ethyl]-2-[4-(methoxymethyl)-5-oxo-2H-furan-3-yl]-2,8-diazaspiro[4.5]decan-1-one
—— 8-ethoxy-2-oxo-N-(2,2,6,6-tetramethylpiperidin-4-yl)chromene-3-carboxamide —— C21H28N2O4
8-ethoxy-2-oxo-N-(2,2,6,6-tetramethylpiperidin-4-yl)chromene-3-carboxamide
—— 8-(1-methyl-1H-imidazol-4-yl)-2-{[2-(trifluoromethyl)phenyl]methoxy}pyrido[3,4-d]pyrimidin-4-ol —— C19H14F3N5O2
8-(1-methyl-1H-imidazol-4-yl)-2-{[2-(trifluoromethyl)phenyl]methoxy}pyrido[3,4-d]pyrimidin-4-ol
—— 8-[2-hydroxy-2-[5-(tetrazol-1-yl)pyrazin-2-yl]ethyl]-6-methoxy-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C21H26N8O5
8-[2-hydroxy-2-[5-(tetrazol-1-yl)pyrazin-2-yl]ethyl]-6-methoxy-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-[2-hydroxy-2-[5-(tetrazol-1-yl)pyrazin-2-yl]ethyl]-4'-methoxy-1'-(4-methyl-5-oxo-2H-furan-3-yl)spiro[8-azabicyclo[3.2.1]octane-3,3'-pyrrolidine]-2'-one —— C23H28N8O5
8-[2-hydroxy-2-[5-(tetrazol-1-yl)pyrazin-2-yl]ethyl]-4'-methoxy-1'-(4-methyl-5-oxo-2H-furan-3-yl)spiro[8-azabicyclo[3.2.1]octane-3,3'-pyrrolidine]-2'-one
—— 8-(1-(6-(1H-tetrazol-1-yl)pyridin-3-yl)-3-hydroxypropan-2-yl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C22H27N7O4
8-(1-(6-(1H-tetrazol-1-yl)pyridin-3-yl)-3-hydroxypropan-2-yl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-ethoxy-2-oxo-N-(2,2,6,6-tetramethylpiperidin-1-ium-4-yl)chromene-3-carboxamide —— C21H29N2O4+
8-ethoxy-2-oxo-N-(2,2,6,6-tetramethylpiperidin-1-ium-4-yl)chromene-3-carboxamide
—— 8-[2-hydroxy-2-[6-(tetrazol-1-yl)pyridin-3-yl]ethyl]-3-methyl-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C22H27N7O4
8-[2-hydroxy-2-[6-(tetrazol-1-yl)pyridin-3-yl]ethyl]-3-methyl-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-(1-methyl-1H-imidazol-4-yl)-2-(oxan-4-ylmethoxy)pyrido[3,4-d]pyrimidin-4-ol —— C17H19N5O3
8-(1-methyl-1H-imidazol-4-yl)-2-(oxan-4-ylmethoxy)pyrido[3,4-d]pyrimidin-4-ol
—— 8-(1-(5-(1H-tetrazol-1-yl)pyrazin-2-yl)-1-hydroxy-2-methylpropan-2-yl)-3-methyl-2-(5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C22H28N8O4
8-(1-(5-(1H-tetrazol-1-yl)pyrazin-2-yl)-1-hydroxy-2-methylpropan-2-yl)-3-methyl-2-(5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-[2-hydroxy-2-[2-methoxy-6-(tetrazol-1-yl)pyridin-3-yl]ethyl]-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C22H27N7O5
8-[2-hydroxy-2-[2-methoxy-6-(tetrazol-1-yl)pyridin-3-yl]ethyl]-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-((R)-1-cyclohexylethyl)-8-azabicyclo[3.2.1]octan-3-one —— C15H25NO
8-((R)-1-cyclohexylethyl)-8-azabicyclo[3.2.1]octan-3-one
—— 8-(2-(6-(1H-tetrazol-1-yl)pyridazin-3-yl)propyl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C21H26N8O3
8-(2-(6-(1H-tetrazol-1-yl)pyridazin-3-yl)propyl)-2-(4-methyl-5-oxo-2,5-dihydrofuran-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— [(8R,9S,10R,13S,14S)-17-(benzimidazol-1-yl)-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15-decahydro-1H-cyclopenta[a]phenanthren-3-yl] methanesulfonate —— C27H34N2O3S
[(8R,9S,10R,13S,14S)-17-(benzimidazol-1-yl)-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15-decahydro-1H-cyclopenta[a]phenanthren-3-yl] methanesulfonate
—— 8-[2-hydroxy-2-[6-(tetrazol-1-yl)pyridin-3-yl]ethyl]-6-methoxy-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one —— C22H27N7O5
8-[2-hydroxy-2-[6-(tetrazol-1-yl)pyridin-3-yl]ethyl]-6-methoxy-2-(4-methyl-5-oxo-2H-furan-3-yl)-2,8-diazaspiro[4.5]decan-1-one
—— 8-[2-hydroxy-2-[6-(tetrazol-1-yl)pyridazin-3-yl]ethyl]-2-[4-(methoxymethyl)-5-oxo-2H-furan-3-yl]-2,8-diazaspiro[4.5]decan-1-one —— C21H26N8O5
8-[2-hydroxy-2-[6-(tetrazol-1-yl)pyridazin-3-yl]ethyl]-2-[4-(methoxymethyl)-5-oxo-2H-furan-3-yl]-2,8-diazaspiro[4.5]decan-1-one
—— 8-(1-methyl-1H-imidazol-4-yl)-2-{[4-(trifluoromethyl)phenyl]methoxy}pyrido[3,4-d]pyrimidin-4-ol —— C19H14F3N5O2
8-(1-methyl-1H-imidazol-4-yl)-2-{[4-(trifluoromethyl)phenyl]methoxy}pyrido[3,4-d]pyrimidin-4-ol
—— 8-Bromo-7-phenylmethoxy-[1,2,4]triazolo[4,3-a]pyridine —— C13H10BrN3O
8-Bromo-7-phenylmethoxy-[1,2,4]triazolo[4,3-a]pyridine
—— 8-[1-[5-[(3,5-Dichlorophenyl)methoxycarbonyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid —— C25H30Cl2N4O4
8-[1-[5-[(3,5-Dichlorophenyl)methoxycarbonyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-2-yl]ethyl]-8-azabicyclo[3.2.1]octane-3-carboxylic acid
—— 8,9,10,10a-tetrahydro-7H-pyrido[1,2-b][1,2]benzothiazole —— C11H13NS
8,9,10,10a-tetrahydro-7H-pyrido[1,2-b][1,2]benzothiazole