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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8S,9aS)-8-(4-nitrobenzoyl)oxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylate —— C16H16N3O7-
(8S,9aS)-8-(4-nitrobenzoyl)oxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylate
—— (8R,9aS)-5-oxo-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid —— C15H16F3N3O4
(8R,9aS)-5-oxo-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid
—— [(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-(trifluoromethyl)phenyl]methanone —— C23H25F3N4O2
[(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-(trifluoromethyl)phenyl]methanone
—— (8R,9aR)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,5,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-7-one —— C21H19F6N3O4S
(8R,9aR)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,5,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-7-one
—— (8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[2-fluoro-3-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C23H22F4N4O3
(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[2-fluoro-3-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[4-(trifluoromethyl)phenyl]methanone —— C23H25F3N4O2
[(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[4-(trifluoromethyl)phenyl]methanone
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C22H23F3N4O2
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8R,9aR)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C21H19F6N3O4S
(8R,9aR)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[5-(trifluoromethyl)pyridin-2-yl]-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine —— C21H24F3N5O
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[5-(trifluoromethyl)pyridin-2-yl]-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine
—— (8S,9aS)-8-(4-nitrobenzoyl)oxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid —— C16H17N3O7
(8S,9aS)-8-(4-nitrobenzoyl)oxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid
—— [(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[5-(trifluoromethyl)pyridin-2-yl]methanone —— C22H24F3N5O2
[(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[5-(trifluoromethyl)pyridin-2-yl]methanone
—— (8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C23H24F4N4O2
(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C22H23F3N4O4S
(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C23H24F4N4O2
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8S,9aR)-8-hydroxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid —— C9H14N2O4
(8S,9aR)-8-hydroxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C23H25F3N4O2
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine —— C22H25F3N4O3S
(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine —— C22H25F3N4O3S
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine
—— [(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-(4-fluorophenyl)methanone —— C22H25FN4O2
[(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-(4-fluorophenyl)methanone
—— (8R,9aR)-2-[3-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C21H19F6N3O4S
(8R,9aR)-2-[3-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8R,9aR)-8-hydroxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid —— C9H14N2O4
(8R,9aR)-8-hydroxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid
—— (8R,9aS)-8-[(5-cyclopropylpyrazin-2-yl)oxy]-2-{[4-(trifluoromethyl)phenyl]sulfonyl}octahydro-1H-pyrrolo[1,2-a][1,4]diazepane 1613627-88-5 C22H25F3N4O3S
(8R,9aS)-8-[(5-cyclopropylpyrazin-2-yl)oxy]-2-{[4-(trifluoromethyl)phenyl]sulfonyl}octahydro-1H-pyrrolo[1,2-a][1,4]diazepane
—— (8R,10S)-5-(3-fluorophenyl)-1,3,8-trimethyl-10-(5-methylfuran-2-yl)-7,8,9,10-tetrahydropyrimido[4,5-a]indolizine-2,4-dione —— C24H24FN3O3
(8R,10S)-5-(3-fluorophenyl)-1,3,8-trimethyl-10-(5-methylfuran-2-yl)-7,8,9,10-tetrahydropyrimido[4,5-a]indolizine-2,4-dione
—— (8S,9aS)-2-[3-(trifluoromethyl)phenyl]sulfonyl-8-[6-(trifluoromethyl)pyridin-3-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C21H19F6N3O4S
(8S,9aS)-2-[3-(trifluoromethyl)phenyl]sulfonyl-8-[6-(trifluoromethyl)pyridin-3-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-(trifluoromethyl)phenyl]methanone —— C23H25F3N4O2
[(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-(trifluoromethyl)phenyl]methanone
—— [(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[4-(trifluoromethyl)phenyl]methanone —— C23H25F3N4O2
[(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[4-(trifluoromethyl)phenyl]methanone
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C23H24F4N4O2
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[4-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C23H25F3N4O2
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[4-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8S,9aS)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C21H19F6N3O4S
(8S,9aS)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[5-(trifluoromethyl)pyridin-2-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-fluoro-4-(trifluoromethyl)phenyl]methanone —— C23H24F4N4O2
[(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-fluoro-4-(trifluoromethyl)phenyl]methanone
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C23H25F3N4O2
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[[3-(trifluoromethyl)phenyl]methyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— [(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-(4-fluorophenyl)methanone —— C22H25FN4O2
[(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-(4-fluorophenyl)methanone
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[4-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C23H23F3N4O3
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[4-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[4-(trifluoromethyl)phenyl]methanone —— C23H25F3N4O2
[(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[4-(trifluoromethyl)phenyl]methanone
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C22H23F3N4O4S
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[5-(trifluoromethyl)pyridin-2-yl]methanone —— C22H24F3N5O2
[(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[5-(trifluoromethyl)pyridin-2-yl]methanone
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-fluoro-4-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C23H22F4N4O3
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-fluoro-4-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[6-(trifluoromethyl)pyridin-2-yl]-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine —— C21H24F3N5O
(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[6-(trifluoromethyl)pyridin-2-yl]-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one —— C22H23F3N4O2
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]-4,5,7,8,9,9a-hexahydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[2-(methylamino)-2-[3-(trifluoromethyl)phenyl]acetyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C25H28F3N5O3
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[2-(methylamino)-2-[3-(trifluoromethyl)phenyl]acetyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8R,9aR)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[6-(trifluoromethyl)pyridin-3-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C21H19F6N3O4S
(8R,9aR)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[6-(trifluoromethyl)pyridin-3-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine —— C22H25F3N4O3S
(8S,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-(trifluoromethyl)phenyl]sulfonyl-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine
—— (8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[2-hydroxy-2-[3-(trifluoromethyl)phenyl]acetyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C24H25F3N4O4
(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[2-hydroxy-2-[3-(trifluoromethyl)phenyl]acetyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— (8R,9aS)-8-hydroxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid —— C9H16N2O3
(8R,9aS)-8-hydroxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid
—— (8S,9aR)-8-(4-nitrobenzoyl)oxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid —— C16H17N3O7
(8S,9aR)-8-(4-nitrobenzoyl)oxy-5-oxo-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxylic acid
—— [(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[6-(trifluoromethyl)pyridin-2-yl]methanone —— C22H24F3N5O2
[(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[6-(trifluoromethyl)pyridin-2-yl]methanone
—— (8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-fluoro-4-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C23H22F4N4O3
(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-2-[3-fluoro-4-(trifluoromethyl)benzoyl]-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-(trifluoromethoxy)phenyl]methanone —— C23H25F3N4O3
[(8S,9aS)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[3-(trifluoromethoxy)phenyl]methanone
—— (8S,9aS)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[6-(trifluoromethyl)pyridin-3-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one —— C21H19F6N3O4S
(8S,9aS)-2-[4-(trifluoromethyl)phenyl]sulfonyl-8-[6-(trifluoromethyl)pyridin-3-yl]oxy-3,4,7,8,9,9a-hexahydro-1H-pyrrolo[1,2-a][1,4]diazepin-5-one
—— [(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[2-fluoro-4-(trifluoromethyl)phenyl]methanone —— C23H24F4N4O2
[(8R,9aR)-8-(5-cyclopropylpyrazin-2-yl)oxy-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-[2-fluoro-4-(trifluoromethyl)phenyl]methanone