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—— 8-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C24H32N6O4
8-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[cyclohexyl-[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C25H34N6O3
8-[[cyclohexyl-[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C25H27N7O4
8-[[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-cyclopentyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C26H27FN6O3
8-[[(1-cyclopentyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[1,3-benzodioxol-5-ylmethyl-[(1-cyclohexyltetrazol-5-yl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C28H30N6O5
8-[[1,3-benzodioxol-5-ylmethyl-[(1-cyclohexyltetrazol-5-yl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-methoxy-N-[2-[2-[2-(4-methoxyphenyl)-2-oxoethyl]tetrazol-5-yl]phenyl]-2-oxochromene-3-carboxamide —— C27H21N5O6
8-methoxy-N-[2-[2-[2-(4-methoxyphenyl)-2-oxoethyl]tetrazol-5-yl]phenyl]-2-oxochromene-3-carboxamide
—— 8-Methyl-thieno[2,3-b]quinoline-2-carboxylic acid cyclopentylcarbamoylmethyl-(2,3-dimethyl-phenyl)-amide —— C28H29N3O2S
8-Methyl-thieno[2,3-b]quinoline-2-carboxylic acid cyclopentylcarbamoylmethyl-(2,3-dimethyl-phenyl)-amide
—— 8-Methyl-thieno[2,3-b]quinoline-2-carboxylic acid cyclopentylcarbamoylmethyl-(2,5-dimethyl-phenyl)-amide —— C28H29N3O2S
8-Methyl-thieno[2,3-b]quinoline-2-carboxylic acid cyclopentylcarbamoylmethyl-(2,5-dimethyl-phenyl)-amide
—— 8-methoxy-4-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]tetrazolo[1,5-a]quinoline —— C27H32N10O
8-methoxy-4-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]tetrazolo[1,5-a]quinoline
—— 8-[4-[(1-Benzyltetrazol-5-yl)methyl]piperazin-1-yl]-1,3,7-trimethylpurine-2,6-dione —— C21H26N10O2
8-[4-[(1-Benzyltetrazol-5-yl)methyl]piperazin-1-yl]-1,3,7-trimethylpurine-2,6-dione
—— 8-[4-[(1-Cyclopentyltetrazol-5-yl)methyl]piperazin-1-yl]-1,3,7-trimethylpurine-2,6-dione —— C19H28N10O2
8-[4-[(1-Cyclopentyltetrazol-5-yl)methyl]piperazin-1-yl]-1,3,7-trimethylpurine-2,6-dione
—— 8-Methyl-2-phenyl-4-piperidin-1-ylquinazoline —— C20H21N3
8-Methyl-2-phenyl-4-piperidin-1-ylquinazoline
—— 8-[(S)-(4-methylpiperazin-1-yl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C26H29N7O3
8-[(S)-(4-methylpiperazin-1-yl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[(S)-morpholin-4-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C25H26N6O4
8-[(S)-morpholin-4-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— (8aR)-2-[(S)-(4-methylphenyl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine —— C24H30N6
(8aR)-2-[(S)-(4-methylphenyl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine
—— (8aR)-2-[(R)-(4-chlorophenyl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine —— C23H27ClN6
(8aR)-2-[(R)-(4-chlorophenyl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine
—— 8-[(R)-morpholin-4-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C25H26N6O4
8-[(R)-morpholin-4-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[(R)-(4-methylpiperazin-1-yl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C26H29N7O3
8-[(R)-(4-methylpiperazin-1-yl)-[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— (8aS)-2-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine —— C17H24N6
(8aS)-2-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine
—— 8-Methyl-7-(2-(piperidin-1-yl)ethylthio)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline —— C19H24N2O2S
8-Methyl-7-(2-(piperidin-1-yl)ethylthio)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline
—— 8-methoxy-2-oxo-N-(4-piperazin-1-ylphenyl)chromene-3-carboxamide —— C21H21N3O4
8-methoxy-2-oxo-N-(4-piperazin-1-ylphenyl)chromene-3-carboxamide
—— 8-(3-Benzyl-5-methyltriazolo[4,5-d]pyrimidin-7-yl)-1,4-dioxa-8-azaspiro[4.5]decane —— C19H22N6O2
8-(3-Benzyl-5-methyltriazolo[4,5-d]pyrimidin-7-yl)-1,4-dioxa-8-azaspiro[4.5]decane
—— (8-Methyl-2-morpholin-4-ylquinolin-3-yl)methanamine —— C15H19N3O
(8-Methyl-2-morpholin-4-ylquinolin-3-yl)methanamine
—— 8-methyl-3-[(R)-[2-phenylethyl(thiophen-2-ylmethyl)amino]-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C28H30N6OS
8-methyl-3-[(R)-[2-phenylethyl(thiophen-2-ylmethyl)amino]-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— 8-methyl-3-[(R)-(4-methylpiperidin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C21H28N6O
8-methyl-3-[(R)-(4-methylpiperidin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— 8-methyl-3-[(S)-(4-methylpiperidin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C21H28N6O
8-methyl-3-[(S)-(4-methylpiperidin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— 8-methyl-3-[(S)-[2-phenylethyl(thiophen-2-ylmethyl)amino]-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C28H30N6OS
8-methyl-3-[(S)-[2-phenylethyl(thiophen-2-ylmethyl)amino]-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— 8-methyl-3-[(R)-(4-methylpiperazin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C20H27N7O
8-methyl-3-[(R)-(4-methylpiperazin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— 8-methoxy-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)chromene-3-carboxamide —— C21H21NO5S
8-methoxy-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)chromene-3-carboxamide
—— 8-methyl-3-[(S)-(4-methylpiperazin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C20H27N7O
8-methyl-3-[(S)-(4-methylpiperazin-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— 8-methoxy-2-oxo-N,N-bis(thiophen-2-ylmethyl)chromene-3-carboxamide —— C21H17NO4S2
8-methoxy-2-oxo-N,N-bis(thiophen-2-ylmethyl)chromene-3-carboxamide
—— 8-methoxy-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)chromene-3-carboxamide —— C21H21NO5S
8-methoxy-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-2-ylmethyl)chromene-3-carboxamide
—— 8-methoxy-N-[3-methoxy-4-(tetrazol-1-yl)phenyl]-2-oxochromene-3-carboxamide —— C19H15N5O5
8-methoxy-N-[3-methoxy-4-(tetrazol-1-yl)phenyl]-2-oxochromene-3-carboxamide
—— 8-[2-(3,5-Dimethoxyphenyl)-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-9-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C25H30N4O4
8-[2-(3,5-Dimethoxyphenyl)-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-9-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-methoxy-N-[3-methyl-4-(tetrazol-1-yl)phenyl]-2-oxochromene-3-carboxamide —— C19H15N5O4
8-methoxy-N-[3-methyl-4-(tetrazol-1-yl)phenyl]-2-oxochromene-3-carboxamide
—— 8-methoxy-N-[(4-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-2-oxochromene-3-carboxamide —— C27H25NO5
8-methoxy-N-[(4-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-2-oxochromene-3-carboxamide
—— 8-[2-(3-Fluoro-phenyl)-5-phenyl-pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-aza-spiro[4.5]decane —— C25H23FN4O2
8-[2-(3-Fluoro-phenyl)-5-phenyl-pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-aza-spiro[4.5]decane
—— 8-[2-(3,4-Dimethoxyphenyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C27H28N4O4
8-[2-(3,4-Dimethoxyphenyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[11-(3,5-Dimethoxyphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C24H28N4O4
8-[11-(3,5-Dimethoxyphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-(5-Phenyl-2-p-tolyl-pyrazolo[1,5-a]pyrimidin-7-yl)-1,4-dioxa-8-aza-spiro[4.5]decane —— C26H26N4O2
8-(5-Phenyl-2-p-tolyl-pyrazolo[1,5-a]pyrimidin-7-yl)-1,4-dioxa-8-aza-spiro[4.5]decane
—— 8-[11-(3-Methoxyphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C23H26N4O3
8-[11-(3-Methoxyphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[2-(3,4-Dimethoxyphenyl)-6-ethyl-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C24H30N4O4
8-[2-(3,4-Dimethoxyphenyl)-6-ethyl-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[11-(3-Methylphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C23H26N4O2
8-[11-(3-Methylphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[11-(4-Methoxyphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C23H26N4O3
8-[11-(4-Methoxyphenyl)-1,8,12-triazatricyclo[7.3.0.03,7]dodeca-2,7,9,11-tetraen-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[5-Methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C21H24N4O2
8-[5-Methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[2-(4-Methoxyphenyl)-5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane —— C22H26N4O3
8-[2-(4-Methoxyphenyl)-5,6-dimethylpyrazolo[1,5-a]pyrimidin-7-yl]-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione —— C18H27N5O3S
8-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione
—— 8-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione —— C18H27N5O3S
8-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione
—— 8-[2-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione —— C18H27N5O3S
8-[2-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione
—— 8-[2-(3,4-Dimethylphenyl)-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione —— C19H22N4O3S
8-[2-(3,4-Dimethylphenyl)-2-oxoethyl]sulfanyl-1-ethyl-3,7-dimethylpurine-2,6-dione