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—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(4-hydroxy-2-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H35Cl2F3N6O6S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(4-hydroxy-2-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-chloro-N-[2-[(8-chloro-2,2,3,3,4,4,5,5,6,6,7,7,8,8-tetradecafluorooctanoyl)amino]propyl]-2,2,3,3,4,4,5,5,6,6,7,7,8,8-tetradecafluorooctanamide —— C19H8Cl2F28N2O2
8-chloro-N-[2-[(8-chloro-2,2,3,3,4,4,5,5,6,6,7,7,8,8-tetradecafluorooctanoyl)amino]propyl]-2,2,3,3,4,4,5,5,6,6,7,7,8,8-tetradecafluorooctanamide
—— 8-[(3-bromo-4-methoxyphenyl)carbonyl]-10-(3,5-dichlorophenyl)-11a,11b-dihydro-8H-pyrrolo[3',4':3,4]pyrrolo[2,1-a]isoquinoline-9,11(8aH,10H)-dione —— C28H19BrCl2N2O4
8-[(3-bromo-4-methoxyphenyl)carbonyl]-10-(3,5-dichlorophenyl)-11a,11b-dihydro-8H-pyrrolo[3',4':3,4]pyrrolo[2,1-a]isoquinoline-9,11(8aH,10H)-dione
—— 8-(Bromomethyl)-6a,9a-dichloro-6-[2-(4-hydroxy-3,5-dimethoxyphenyl)ethenyl]-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C31H26BrCl2N3O9
8-(Bromomethyl)-6a,9a-dichloro-6-[2-(4-hydroxy-3,5-dimethoxyphenyl)ethenyl]-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-6-(4-hydroxyphenyl)-6a-methyl-2-(3-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C33H25ClFN3O7
8-(3-chloro-4-fluorophenyl)-6-(4-hydroxyphenyl)-6a-methyl-2-(3-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-Methylpiperidin-1-yl)sulfonylquinoline —— C15H18N2O2S
8-(3-Methylpiperidin-1-yl)sulfonylquinoline
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(2-hydroxy-3-methylphenyl)-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide —— C23H20BrCl2N3O6
8-(Bromomethyl)-6a,9a-dichloro-6-(2-hydroxy-3-methylphenyl)-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide
—— 8-(Bromomethyl)-2-(4-bromophenyl)-6a,9a-dichloro-6-(4-hydroxy-2,6-dimethoxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H24Br2Cl2N2O7
8-(Bromomethyl)-2-(4-bromophenyl)-6a,9a-dichloro-6-(4-hydroxy-2,6-dimethoxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-(2-hydroxy-3-methoxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C38H33BrCl2N2O8
8-(Bromomethyl)-6a,9a-dichloro-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-(2-hydroxy-3-methoxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(2-hydroxy-6-methoxyphenyl)-2-(4-morpholin-4-ylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C32H30BrCl2N3O7
8-(Bromomethyl)-6a,9a-dichloro-6-(2-hydroxy-6-methoxyphenyl)-2-(4-morpholin-4-ylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-benzyl-2-(2-methylpropoxy)-3,3a,4,5,6,7-hexahydro-2H-[1,2]oxazolo[2,3-a]pyridin-8-ium —— C18H28NO2+
8-benzyl-2-(2-methylpropoxy)-3,3a,4,5,6,7-hexahydro-2H-[1,2]oxazolo[2,3-a]pyridin-8-ium
—— 8-N-(1,3-benzothiazol-2-yl)-6-(4-hydroxyphenyl)-5'-[2-(4-methoxyphenyl)ethynyl]-1,2'-dioxo-3,4-diphenyl-1-N'-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1',8-dicarboxamide —— C58H45N5O7S
8-N-(1,3-benzothiazol-2-yl)-6-(4-hydroxyphenyl)-5'-[2-(4-methoxyphenyl)ethynyl]-1,2'-dioxo-3,4-diphenyl-1-N'-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1',8-dicarboxamide
—— 8-(2-Cyclopentylidenehydrazinyl)-7-[2-(4-methoxyphenyl)ethyl]-3-methylpurine-2,6-dione —— C20H24N6O3
8-(2-Cyclopentylidenehydrazinyl)-7-[2-(4-methoxyphenyl)ethyl]-3-methylpurine-2,6-dione
—— 8-[5-(2-Bromo-4-nitrophenyl)furan-2-yl]-3-butyl-7-(3-methylbutyl)purine-2,6-dione —— C24H26BrN5O5
8-[5-(2-Bromo-4-nitrophenyl)furan-2-yl]-3-butyl-7-(3-methylbutyl)purine-2,6-dione
—— 8-(2-Benzylidenehydrazinyl)-7-[(3-bromophenyl)methyl]-1,3-dimethylpurine-2,6-dione —— C21H19BrN6O2
8-(2-Benzylidenehydrazinyl)-7-[(3-bromophenyl)methyl]-1,3-dimethylpurine-2,6-dione
—— 8-Methyl-2-(5-methylthiophen-2-yl)indolizine-3-carbaldehyde —— C15H13NOS
8-Methyl-2-(5-methylthiophen-2-yl)indolizine-3-carbaldehyde
—— 8-(2,5-dimethoxybenzoyl)-N-(3,5-dimethoxyphenyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide —— C26H33N3O5S
8-(2,5-dimethoxybenzoyl)-N-(3,5-dimethoxyphenyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide
—— 8-(4-ethoxybenzoyl)-N-(1-phenylethyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide —— C26H33N3O2S
8-(4-ethoxybenzoyl)-N-(1-phenylethyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide
—— 8-(2-Ethylpiperidin-1-yl)sulfonylquinoline —— C16H20N2O2S
8-(2-Ethylpiperidin-1-yl)sulfonylquinoline
—— 8-(2,3-Dimethoxybenzoyl)-2-(4-fluorophenyl)-1,2,4,8-tetraazaspiro[4.5]decan-3-one —— C21H23FN4O4
8-(2,3-Dimethoxybenzoyl)-2-(4-fluorophenyl)-1,2,4,8-tetraazaspiro[4.5]decan-3-one
—— 8-[(1-Acetyl-4-piperidyl)carbonyl]-2-(4-fluorophenyl)-1,2,4,8-tetraazaspiro[4.5]decan-3-one —— C20H26FN5O3
8-[(1-Acetyl-4-piperidyl)carbonyl]-2-(4-fluorophenyl)-1,2,4,8-tetraazaspiro[4.5]decan-3-one
—— 8-[2-(4-Fluorophenoxy)acetyl]-2-(4-fluorophenyl)-1,2,4,8-tetrazaspiro[4.5]decan-3-one —— C20H20F2N4O3
8-[2-(4-Fluorophenoxy)acetyl]-2-(4-fluorophenyl)-1,2,4,8-tetrazaspiro[4.5]decan-3-one
—— 8-[(6-Methoxy-3-pyridyl)carbonyl]-2-phenyl-1,2,4,8-tetraazaspiro[4.5]decan-3-one —— C19H21N5O3
8-[(6-Methoxy-3-pyridyl)carbonyl]-2-phenyl-1,2,4,8-tetraazaspiro[4.5]decan-3-one
—— 8-[(1-ethyl-1H-pyrazol-5-yl)carbonyl]-2-(4-fluorophenyl)-1,2,4,8-tetraazaspiro[4.5]decan-3-one —— C18H21FN6O2
8-[(1-ethyl-1H-pyrazol-5-yl)carbonyl]-2-(4-fluorophenyl)-1,2,4,8-tetraazaspiro[4.5]decan-3-one
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[propanoyl(3-propan-2-yloxypropyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C26H36N2O8
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[propanoyl(3-propan-2-yloxypropyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— 8-(2-Aminoethylamino)-1,7-bis[(4-chlorophenyl)methyl]-3-methylpurine-2,6-dione —— C22H22Cl2N6O2
8-(2-Aminoethylamino)-1,7-bis[(4-chlorophenyl)methyl]-3-methylpurine-2,6-dione
—— 8-[3-(Dimethylamino)benzoyl]-2-(3-fluorophenyl)-1,2,4,8-tetrazaspiro[4.5]decan-3-one —— C21H24FN5O2
8-[3-(Dimethylamino)benzoyl]-2-(3-fluorophenyl)-1,2,4,8-tetrazaspiro[4.5]decan-3-one
—— 8-[3-(3-Methoxyphenyl)propanoyl]-2-phenyl-1,2,4,8-tetraazaspiro[4.5]decan-3-one —— C22H26N4O3
8-[3-(3-Methoxyphenyl)propanoyl]-2-phenyl-1,2,4,8-tetraazaspiro[4.5]decan-3-one
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[2-(2-methoxyphenyl)ethyl-(3-methoxypropanoyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C30H36N2O9
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[2-(2-methoxyphenyl)ethyl-(3-methoxypropanoyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— [8-bromo-6-(2-chlorophenyl)-3-oxo-2,4-dihydro-1H-1,5-benzodiazocin-4-yl] 3-aminopropanoate —— C19H17BrClN3O3
[8-bromo-6-(2-chlorophenyl)-3-oxo-2,4-dihydro-1H-1,5-benzodiazocin-4-yl] 3-aminopropanoate
—— 8-(4-Benzylpiperazin-1-yl)-3-methyl-7-octylpurine-2,6-dione —— C25H36N6O2
8-(4-Benzylpiperazin-1-yl)-3-methyl-7-octylpurine-2,6-dione
—— 8-(Bromomethyl)-2-(4-bromophenyl)-6a,9a-dichloro-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C28H19Br2Cl2F3N2O6
8-(Bromomethyl)-2-(4-bromophenyl)-6a,9a-dichloro-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-Chlorobenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene —— C20H20ClN3O2
8-(3-Chlorobenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene
—— 8-(3,4-Difluorobenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene —— C20H19F2N3O2
8-(3,4-Difluorobenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene
—— 8-(3-Fluoro-4-methoxybenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene —— C21H22FN3O3
8-(3-Fluoro-4-methoxybenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene
—— 8-(3-Methylbenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene —— C21H23N3O2
8-(3-Methylbenzoyl)-3-(4-methylphenyl)-1-oxa-2,4,8-triazaspiro[4.5]dec-2-ene
—— 8-methyl-6-[4-(nonanoylamino)phenyl]-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C30H38N4O2S
8-methyl-6-[4-(nonanoylamino)phenyl]-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 8-(4-Butylbenzoyl)-3-(2-morpholin-4-yl-2-oxoethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one —— C30H38N4O4
8-(4-Butylbenzoyl)-3-(2-morpholin-4-yl-2-oxoethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
—— [8-[2-[[2-(4-tert-butylphenoxy)acetyl]amino]-6-oxo-4,5-dihydro-1H-purin-9-yl]-2,2,4,4-tetra(propan-2-yl)-6a,8,9,9a-tetrahydro-6H-furo[3,2-f][1,3,5,2,4]trioxadisilocin-9-yl] 2-(4-tert-butylphenoxy)acetate —— C46H69N5O10Si2
[8-[2-[[2-(4-tert-butylphenoxy)acetyl]amino]-6-oxo-4,5-dihydro-1H-purin-9-yl]-2,2,4,4-tetra(propan-2-yl)-6a,8,9,9a-tetrahydro-6H-furo[3,2-f][1,3,5,2,4]trioxadisilocin-9-yl] 2-(4-tert-butylphenoxy)acetate
—— 8-(2-Benzylidenehydrazinyl)-3-methyl-7-(naphthalen-1-ylmethyl)purine-2,6-dione —— C24H20N6O2
8-(2-Benzylidenehydrazinyl)-3-methyl-7-(naphthalen-1-ylmethyl)purine-2,6-dione
—— 8-(4-(2-hydroxyethyl)piperazin-1-yl)-3-methyl-7-(2-((1-phenyl-1H-tetrazol-5-yl)thio)ethyl)-1H-purine-2,6(3H,7H)-dione —— C21H26N10O3S
8-(4-(2-hydroxyethyl)piperazin-1-yl)-3-methyl-7-(2-((1-phenyl-1H-tetrazol-5-yl)thio)ethyl)-1H-purine-2,6(3H,7H)-dione
—— 8-bromo-4-[3-(trifluoromethyl)phenyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-6-carboxylic acid —— C20H15BrF3NO2
8-bromo-4-[3-(trifluoromethyl)phenyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-6-carboxylic acid
—— 8-(3-chlorophenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H31ClF3N5O10
8-(3-chlorophenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-bromo-4-[3-(trifluoromethyl)phenyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-6-carboxylate —— C20H14BrF3NO2-
8-bromo-4-[3-(trifluoromethyl)phenyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-6-carboxylate
—— 8-(Bromomethyl)-6a,9a-dichloro-6-[4-(2-hydroxyethoxy)phenyl]-2-(4-morpholin-4-ylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C33H32BrCl2N3O7
8-(Bromomethyl)-6a,9a-dichloro-6-[4-(2-hydroxyethoxy)phenyl]-2-(4-morpholin-4-ylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[(6-aminohexyl)amino]-7-(2-chlorobenzyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione —— C20H27ClN6O2
8-[(6-aminohexyl)amino]-7-(2-chlorobenzyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione
—— 8-(Bromomethyl)-6a,9a-dichloro-6-[2-(4-hydroxy-3-methoxyphenyl)ethenyl]-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide —— C25H22BrCl2N3O7
8-(Bromomethyl)-6a,9a-dichloro-6-[2-(4-hydroxy-3-methoxyphenyl)ethenyl]-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide
—— 8-benzyl-1,3-dimethyl-7-(naphthalen-2-yl)-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione —— C26H21N5O2
8-benzyl-1,3-dimethyl-7-(naphthalen-2-yl)-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione
—— 8-N-(1,3-benzothiazol-2-yl)-5'-[3-[benzyl(methyl)amino]prop-1-ynyl]-6-(4-hydroxyphenyl)-1,2'-dioxo-3,4-diphenyl-1-N'-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1',8-dicarboxamide —— C60H50N6O6S
8-N-(1,3-benzothiazol-2-yl)-5'-[3-[benzyl(methyl)amino]prop-1-ynyl]-6-(4-hydroxyphenyl)-1,2'-dioxo-3,4-diphenyl-1-N'-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1',8-dicarboxamide
—— 8-[[4-[4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid —— C29H36N4O6S
8-[[4-[4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid