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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-benzyl-4-methyl-2-[(2S)-1-pyrimidin-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O
8-benzyl-4-methyl-2-[(2S)-1-pyrimidin-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5OS
8-benzyl-4-methyl-2-[(2S)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-methylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H32N4O
8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-methylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2S)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclopropylmethyl)-2-[(2S)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O2
8-benzyl-2-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(3-morpholin-4-ylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H35N5O3
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(3-morpholin-4-ylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O3
8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O3
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C20H30N4O
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H27N5O3
8-benzyl-2-[(2R)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2S)-1-[2-(4-methoxy-3-methylphenyl)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-cyclopropyl-2-[(2S)-1-[2-(4-methoxy-3-methylphenyl)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(2-pyridin-2-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29N5O2
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(2-pyridin-2-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(2-pyrrolidin-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(3R)-1-(2-pyrrolidin-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O
8-(cyclopropylmethyl)-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclopropylmethyl)-2-[(3S)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O3
8-benzyl-4-methyl-2-[(3S)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H28N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(3R)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H34N6O
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(2-pyrrolidin-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(3S)-1-(2-pyrrolidin-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-pyrazol-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2R)-1-(2-pyrazol-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(3S)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N6O
8-benzyl-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-(cyclopropylmethyl)-2-[(3S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[3-(5-methyl-3,4-dihydropyrazol-2-yl)propanoyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[3-(5-methyl-3,4-dihydropyrazol-2-yl)propanoyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(thiadiazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H24N6O2S
8-benzyl-4-methyl-2-[(3R)-1-(thiadiazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O
8-(cyclopropylmethyl)-2-[(3S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2R)-1-[2-(2-fluorophenoxy)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN4O3
8-cyclopropyl-2-[(2R)-1-[2-(2-fluorophenoxy)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Bromomethyl)-2-(4-bromophenyl)-6a,9a-dichloro-6-(5-chloro-2-hydroxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C27H19Br2Cl3N2O5
8-(Bromomethyl)-2-(4-bromophenyl)-6a,9a-dichloro-6-(5-chloro-2-hydroxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-cyclopropyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrimidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H26N6O3
8-cyclopropyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrimidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H29N5OS
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H28N6O3S
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H34N6O
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-4-methyl-2-[(2S)-1-[2-(2-oxopyrimidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H26N6O3
8-cyclopropyl-4-methyl-2-[(2S)-1-[2-(2-oxopyrimidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O
8-(cyclopropylmethyl)-2-[(3R)-1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(2-pyridin-2-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29N5O2
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(2-pyridin-2-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— (8-Methyl-2-oxo-4-phenylchromen-7-yl) 3-(4-fluorophenyl)prop-2-enoate —— C25H17FO4
(8-Methyl-2-oxo-4-phenylchromen-7-yl) 3-(4-fluorophenyl)prop-2-enoate
—— 8-cyclopropyl-2-[(2S)-1-[2-(2-fluorophenoxy)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN4O3
8-cyclopropyl-2-[(2S)-1-[2-(2-fluorophenoxy)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-pyrrolidin-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2R)-1-(2-pyrrolidin-1-ylacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O3
8-benzyl-4-methyl-2-[(3R)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-propylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N4O2
8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-propylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(2-propan-2-yloxyacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-4-methyl-2-[(2S)-1-(2-propan-2-yloxyacetyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2R)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H26N6O2
8-cyclopropyl-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one