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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-benzyl-4-methyl-2-[(2R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29N5OS
8-benzyl-4-methyl-2-[(2R)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2S)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N6O
8-(cyclopropylmethyl)-2-[(2S)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H27N5O3
8-benzyl-2-[(2R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(3S)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N6O3
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-2-[(2R)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-ethylsulfonylpyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H32N4O3S
8-(cyclohexylmethyl)-2-[(2S)-1-ethylsulfonylpyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclopropylmethyl)-2-[(3R)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H28N6O
8-benzyl-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H28N6O
8-benzyl-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H30N4O2
8-benzyl-2-[(2S)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H33N5O2
8-benzyl-2-[(2R)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C20H30N4O
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H28N6O3S
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(4-fluorophenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O3
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(3S)-1-(2-hydroxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O3
8-(cyclohexylmethyl)-2-[(3S)-1-(2-hydroxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H34N6O
8-(cyclopropylmethyl)-2-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H33N5O2
8-benzyl-2-[(2S)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-2-[(2S)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(4-fluorophenyl)ethyl]-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29FN6O
8-[2-(4-fluorophenyl)ethyl]-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-2-[(2S)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-ethylsulfonylpyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H32N4O3S
8-(cyclohexylmethyl)-2-[(2R)-1-ethylsulfonylpyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H27N5O3
8-benzyl-2-[(2S)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H29N5O2S
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N6O2
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O2
8-benzyl-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O2
8-(cyclopropylmethyl)-2-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-(cyclohexylmethyl)-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-methylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H32N4O
8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-methylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(1H-imidazol-2-ylmethyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H28N6O
8-benzyl-2-[(2S)-1-(1H-imidazol-2-ylmethyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H31N5O2
8-(cyclopropylmethyl)-2-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O
8-(cyclopropylmethyl)-2-[(3R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N6O
8-benzyl-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O2
8-benzyl-2-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-(cyclopropylmethyl)-2-[(3R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(4-fluorophenyl)ethyl]-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29FN6O
8-[2-(4-fluorophenyl)ethyl]-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H26N6O2
8-cyclopropyl-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-[(2-methylpyrazol-3-yl)methyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-4-methyl-2-[(3R)-1-[(2-methylpyrazol-3-yl)methyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one