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中文名称 英文名称 CAS号 化学式 结构式图片
—— (8S)-3-(3-chlorophenyl)-8-(4-hydroxy-3-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C21H18ClN3O3S
(8S)-3-(3-chlorophenyl)-8-(4-hydroxy-3-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-8-(4-bromophenyl)-3-(2-fluorophenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C20H15BrFN3OS
(8R)-8-(4-bromophenyl)-3-(2-fluorophenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-3-(3-chlorophenyl)-8-(3,4-dimethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C22H20ClN3O3S
(8R)-3-(3-chlorophenyl)-8-(3,4-dimethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-8-(4-chlorophenyl)-3-(2-ethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C22H20ClN3O2S
(8R)-8-(4-chlorophenyl)-3-(2-ethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-8-(5-bromo-2-methoxyphenyl)-3-(2-ethylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C23H22BrN3O2S
(8S)-8-(5-bromo-2-methoxyphenyl)-3-(2-ethylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-8-(2,3-dimethoxyphenyl)-3-(2-ethylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C24H25N3O3S
(8S)-8-(2,3-dimethoxyphenyl)-3-(2-ethylphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-8-(2,5-dimethoxyphenyl)-3-(2-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C23H23N3O4S
(8S)-8-(2,5-dimethoxyphenyl)-3-(2-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-3-(3-chloro-2-methylphenyl)-6-oxo-8-(4-propan-2-ylphenyl)-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C24H24ClN3OS
(8S)-3-(3-chloro-2-methylphenyl)-6-oxo-8-(4-propan-2-ylphenyl)-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8R)-3-(4-fluorophenyl)-8-(2-methoxynaphthalen-1-yl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C25H20FN3O2S
(8R)-3-(4-fluorophenyl)-8-(2-methoxynaphthalen-1-yl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— (8S)-8-(3-ethoxy-4-hydroxyphenyl)-3-(2-fluorophenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile —— C22H20FN3O3S
(8S)-8-(3-ethoxy-4-hydroxyphenyl)-3-(2-fluorophenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrile
—— 8-[(3-hydroxypropyl)amino]-1,3-dimethyl-7-(propan-2-yl)-3,7-dihydro-1H-purine-2,6-dione —— C13H21N5O3
8-[(3-hydroxypropyl)amino]-1,3-dimethyl-7-(propan-2-yl)-3,7-dihydro-1H-purine-2,6-dione
—— 8-Chloro-3-(4-chlorophenyl)-6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine —— C13H6Cl2F3N3
8-Chloro-3-(4-chlorophenyl)-6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
—— 8-[(4-chlorobenzyl)sulfanyl]-1,3-dimethyl-7-pentyl-3,7-dihydro-1H-purine-2,6-dione —— C19H23ClN4O2S
8-[(4-chlorobenzyl)sulfanyl]-1,3-dimethyl-7-pentyl-3,7-dihydro-1H-purine-2,6-dione
—— 8,9-dimethoxy-5-[(2-methylbenzyl)sulfanyl]imidazo[1,2-c]quinazolin-2(3H)-one —— C20H19N3O3S
8,9-dimethoxy-5-[(2-methylbenzyl)sulfanyl]imidazo[1,2-c]quinazolin-2(3H)-one
—— 8-[2-[[4-(Dimethylamino)phenyl]methylidene]hydrazinyl]-7-(2-hydroxy-3-propan-2-yloxypropyl)-3-methylpurine-2,6-dione —— C21H29N7O4
8-[2-[[4-(Dimethylamino)phenyl]methylidene]hydrazinyl]-7-(2-hydroxy-3-propan-2-yloxypropyl)-3-methylpurine-2,6-dione
—— 8-[2-[(4-Bromophenyl)methylidene]hydrazinyl]-1,3-dimethyl-7-[(4-methylphenyl)methyl]purine-2,6-dione —— C22H21BrN6O2
8-[2-[(4-Bromophenyl)methylidene]hydrazinyl]-1,3-dimethyl-7-[(4-methylphenyl)methyl]purine-2,6-dione
—— 8-[2-(2,3-dihydro-1H-inden-2-yl)acetyl]-N-(1-naphthalen-1-ylethyl)-2,8-diazaspiro[4.5]decane-2-carboxamide —— C32H37N3O2
8-[2-(2,3-dihydro-1H-inden-2-yl)acetyl]-N-(1-naphthalen-1-ylethyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
—— 8-Benzoyl-7-(4-bromophenyl)-5-phenyl-3,4-dihydrochromen-2-one —— C28H19BrO3
8-Benzoyl-7-(4-bromophenyl)-5-phenyl-3,4-dihydrochromen-2-one
—— 8,8-Dimethyl-6-phenyl-8-azoniabicyclo[3.2.1]octan-2-one —— C15H20NO+
8,8-Dimethyl-6-phenyl-8-azoniabicyclo[3.2.1]octan-2-one
—— 8-methyl-1-[(naphthalen-1-ylmethyl)sulfanyl]-4-phenyl-6,7,8,9-tetrahydro[1]benzothieno[3,2-e][1,2,4]triazolo[4,3-a]pyrimidin-5(4H)-one —— C29H24N4OS2
8-methyl-1-[(naphthalen-1-ylmethyl)sulfanyl]-4-phenyl-6,7,8,9-tetrahydro[1]benzothieno[3,2-e][1,2,4]triazolo[4,3-a]pyrimidin-5(4H)-one
—— 8,15-Dibenzyl-26-methyl-22-propan-2-yl-13,20,27-trioxa-6,9,16,23,28,29,30-heptazapentacyclo[23.2.1.111,14.118,21.02,6]triaconta-1(28),14(30),21(29)-triene-7,10,17,24-tetrone —— C38H45N7O7
8,15-Dibenzyl-26-methyl-22-propan-2-yl-13,20,27-trioxa-6,9,16,23,28,29,30-heptazapentacyclo[23.2.1.111,14.118,21.02,6]triaconta-1(28),14(30),21(29)-triene-7,10,17,24-tetrone
—— 8-[2-(2-Bromo-3-phenylprop-2-enylidene)hydrazinyl]-3-methyl-7-[(4-methylphenyl)methyl]purine-2,6-dione —— C23H21BrN6O2
8-[2-(2-Bromo-3-phenylprop-2-enylidene)hydrazinyl]-3-methyl-7-[(4-methylphenyl)methyl]purine-2,6-dione
—— 8-(2-Fluorophenoxy)-7-isopentyl-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione —— C18H21FN4O3
8-(2-Fluorophenoxy)-7-isopentyl-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione
—— (8S,9S,10S,13R,14S,17R)-17-ethynyl-17-hydroxy-13-methyl-1,2,6,7,8,9,10,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthren-3-one —— C20H26O2
(8S,9S,10S,13R,14S,17R)-17-ethynyl-17-hydroxy-13-methyl-1,2,6,7,8,9,10,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthren-3-one
—— 8-Bromodibenzo[b,f]oxepin-3-amine —— C14H10BrNO
8-Bromodibenzo[b,f]oxepin-3-amine
—— (8R)-8-(4-ethoxy-3-methoxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one —— C25H24N2O3
(8R)-8-(4-ethoxy-3-methoxyphenyl)-8,10,11,12-tetrahydro-7H-benzo[a][4,7]phenanthrolin-9-one
—— 8-methyl-1-[2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-2-oxoethyl]chromeno[4,3-c]pyrazol-4-one —— C25H26N4O3
8-methyl-1-[2-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-2-oxoethyl]chromeno[4,3-c]pyrazol-4-one
—— 8-Bromo-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine —— C5H5BrN6
8-Bromo-[1,2,4]triazolo[1,5-c]pyrimidine-5,7-diamine
—— 8-methyl-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]thieno[3,2-c]chromen-4-one —— C25H24N2O3S
8-methyl-2-[(3S)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]thieno[3,2-c]chromen-4-one
—— 8-methyl-1-[2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-2-oxoethyl]chromeno[4,3-c]pyrazol-4-one —— C25H26N4O3
8-methyl-1-[2-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-2-oxoethyl]chromeno[4,3-c]pyrazol-4-one
—— 8-methyl-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]thieno[3,2-c]chromen-4-one —— C25H24N2O3S
8-methyl-2-[(3R)-3-methyl-4-(3-methylphenyl)piperazine-1-carbonyl]thieno[3,2-c]chromen-4-one
—— 8-[4-[(3S)-2,5-dioxo-1-phenylpyrrolidin-3-yl]piperazin-1-yl]-1,3-dimethyl-7H-purine-2,6-dione —— C21H23N7O4
8-[4-[(3S)-2,5-dioxo-1-phenylpyrrolidin-3-yl]piperazin-1-yl]-1,3-dimethyl-7H-purine-2,6-dione
—— 8-bromo-6-ethyl-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21BrN2OS
8-bromo-6-ethyl-N-[(1R)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H25BrN2OS
8-bromo-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-6-ethyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C24H21BrN2OS
8-bromo-6-ethyl-N-[(1S)-1-phenylethyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H25BrN2OS
8-bromo-N-[(1R,2R,3R)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-6-ethyl-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C21H21BrN2O2S
8-bromo-6-ethyl-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H35N3OS
8-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-6-methyl-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C20H19BrN2O2S
8-bromo-6-methyl-N-[[(2R)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-methyl-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C27H35N3OS
8-methyl-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-6-propylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H25BrN2OS
8-bromo-N-[(1S,2R,3R)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide —— C23H25BrN2OS
8-bromo-N-[(1R,2R,3S)-2,3-dimethylcyclohexyl]-6-methylbenzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-bromo-6-methyl-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide —— C20H19BrN2O2S
8-bromo-6-methyl-N-[[(2S)-oxolan-2-yl]methyl]benzo[b][1,4]benzothiazepine-3-carboxamide
—— 8-[(1R,3R)-3-hydroxycyclopentyl]-1,3-dimethyl-7H-purine-2,6-dione —— C12H16N4O3
8-[(1R,3R)-3-hydroxycyclopentyl]-1,3-dimethyl-7H-purine-2,6-dione
—— 8-[3-Chloro-5-(trifluoromethyl)-2-pyridinyl]-4-methyl-1-oxa-4,8-diazaspiro[4.5]decane —— C14H17ClF3N3O
8-[3-Chloro-5-(trifluoromethyl)-2-pyridinyl]-4-methyl-1-oxa-4,8-diazaspiro[4.5]decane
—— (8R,11S)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile —— C28H21N5O
(8R,11S)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile
—— (8S,11R)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile —— C28H21N5O
(8S,11R)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile
—— (8S,11S)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile —— C28H21N5O
(8S,11S)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile
—— (8R,11R)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile —— C28H21N5O
(8R,11R)-5-amino-9-oxo-11-phenyl-8-pyridin-3-yl-8,10,11,12-tetrahydroquinolino[1,2-a]quinazoline-7-carbonitrile
—— 8-(5-chloro-2-hydroxybenzoyl)-6-[[(2R)-oxolan-2-yl]methylamino]pyrido[2,1-b]quinazolin-11-one —— C24H20ClN3O4
8-(5-chloro-2-hydroxybenzoyl)-6-[[(2R)-oxolan-2-yl]methylamino]pyrido[2,1-b]quinazolin-11-one