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—— 8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N4O3
8-(cyclohexylmethyl)-4-methyl-2-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(pyridine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H27N5O2
8-benzyl-4-methyl-2-[(3S)-1-(pyridine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H30N4O3
8-(cyclopropylmethyl)-4-methyl-2-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O3
8-Cyclopentyl-2-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H28N4O4S
8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H28N4O4S
8-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H32N4O3S
8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N4O3
8-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-Cyclopentyl-2-[1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-Benzyl-4-methyl-2-[1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(3-fluorophenyl)methyl]-2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N6O2
8-(cyclohexylmethyl)-4-methyl-2-[(3S)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H25FN4O3S
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-Cyclopentyl-2-[1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-Fluorophenyl)methyl]-2-[1-(2-hydroxy-2-methylpropanoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(3-Fluorophenyl)methyl]-2-[1-(2-hydroxy-2-methylpropanoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-benzyl-4-methyl-2-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[1-[(1S)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H32N4O2
8-benzyl-2-[1-[(1S)-cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-3-[2-(1H-indol-2-yl)ethyl-pent-4-enoylamino]-6-methoxy-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C32H35N3O7
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-3-[2-(1H-indol-2-yl)ethyl-pent-4-enoylamino]-6-methoxy-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— 8-Benzyl-4-methyl-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H27N5O2
8-Benzyl-4-methyl-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O3
8-[(4-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-Fluorophenyl)methyl]-2-[1-(3-methoxypropanoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(3-Fluorophenyl)methyl]-2-[1-(3-methoxypropanoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O3
8-Cyclopentyl-2-[1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O3
8-Benzyl-4-methyl-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-Fluorophenyl)methyl]-4-methyl-2-(1-methylsulfonylpiperidin-4-yl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H25FN4O3S
8-[(2-Fluorophenyl)methyl]-4-methyl-2-(1-methylsulfonylpiperidin-4-yl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(3-methylbutanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(3-methylbutanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H34N6O
8-(Cyclopropylmethyl)-2-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H36N6O
8-Cyclopentyl-2-[1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-Fluorophenyl)methyl]-2-[1-(2-methoxyacetyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O3
8-[(3-Fluorophenyl)methyl]-2-[1-(2-methoxyacetyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-ethylsulfonylpiperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C19H28N4O3S
8-(cyclopropylmethyl)-2-[(3R)-1-ethylsulfonylpiperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-4-methyl-2-[1-(2-pyrrolidin-1-ylacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H35N5O2
8-Cyclopentyl-4-methyl-2-[1-(2-pyrrolidin-1-ylacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H25FN4O3S
8-[(2-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H34N4O2
8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-2-[1-(2-methoxy-2-methylpropanoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H34N4O3
8-Cyclopentyl-2-[1-(2-methoxy-2-methylpropanoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(3R)-1-ethylsulfonylpiperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H34N4O3S
8-(cyclohexylmethyl)-2-[(3R)-1-ethylsulfonylpiperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H27FN4O3S
8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3S)-1-methylsulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[1-(2-methoxy-3-methylbenzoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-(Cyclopropylmethyl)-2-[1-(2-methoxy-3-methylbenzoyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O2
8-benzyl-2-[1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-4-methyl-2-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H34N6O
8-(Cyclopropylmethyl)-4-methyl-2-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3S)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(3S)-1-propanoylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-Fluorophenyl)methyl]-4-methyl-2-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H29FN6O
8-[(3-Fluorophenyl)methyl]-4-methyl-2-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one