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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-Methyl-2-[3-(trifluoromethyl)phenyl]imidazo[1,2-a]pyridine —— C15H11F3N2
8-Methyl-2-[3-(trifluoromethyl)phenyl]imidazo[1,2-a]pyridine
—— (8-chloro-6-methylbenzo[b][1,4]benzothiazepin-3-yl)-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methanone —— C27H26ClN3OS
(8-chloro-6-methylbenzo[b][1,4]benzothiazepin-3-yl)-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methanone
—— (8-chloro-6-methylbenzo[b][1,4]benzothiazepin-3-yl)-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methanone —— C27H26ClN3OS
(8-chloro-6-methylbenzo[b][1,4]benzothiazepin-3-yl)-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methanone
—— (8S)-6-methyl-11-(2-morpholin-4-ylethyl)-4,8-diphenyl-2-oxa-4,5,11,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3(7),5,12-tetraen-10-imine —— C27H28N6O2
(8S)-6-methyl-11-(2-morpholin-4-ylethyl)-4,8-diphenyl-2-oxa-4,5,11,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3(7),5,12-tetraen-10-imine
—— (8R)-6-methyl-11-(2-morpholin-4-ylethyl)-4,8-diphenyl-2-oxa-4,5,11,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3(7),5,12-tetraen-10-imine —— C27H28N6O2
(8R)-6-methyl-11-(2-morpholin-4-ylethyl)-4,8-diphenyl-2-oxa-4,5,11,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),3(7),5,12-tetraen-10-imine
—— 8-[[[(1S)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C29H28FN7O3
8-[[[(1S)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[2-hydroxyethyl-[[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C21H26N6O5
8-[[2-hydroxyethyl-[[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-cyclohexyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C27H29FN6O3
8-[[(1-cyclohexyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-benzyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C29H28N6O4
8-[[(1-benzyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[2-hydroxyethyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C24H26N6O4
8-[[2-hydroxyethyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C28H27FN6O3S
8-[[[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[benzyl-[(1-benzyltetrazol-5-yl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C28H26N6O3
8-[[benzyl-[(1-benzyltetrazol-5-yl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[[(1R)-1-(1-benzyltetrazol-5-yl)propyl]-[(4-methylphenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C31H32N6O3
8-[[[(1R)-1-(1-benzyltetrazol-5-yl)propyl]-[(4-methylphenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(4-methylphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C30H30N6O3
8-[[(4-methylphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[furan-2-ylmethyl-[[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C24H26N6O5
8-[[furan-2-ylmethyl-[[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[cyclopentyl-[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C28H31FN6O3
8-[[cyclopentyl-[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-cyclopentyltetrazol-5-yl)methyl-(pyridin-3-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C25H27N7O3
8-[[(1-cyclopentyltetrazol-5-yl)methyl-(pyridin-3-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-cyclopentyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C27H30N6O4
8-[[(1-cyclopentyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-benzyltetrazol-5-yl)methyl-(thiophen-2-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C26H24N6O3S
8-[[(1-benzyltetrazol-5-yl)methyl-(thiophen-2-ylmethyl)amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[(1-cyclohexyltetrazol-5-yl)methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C25H32N6O4
8-[[(1-cyclohexyltetrazol-5-yl)methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[[2-(3,4-dimethoxyphenyl)ethyl-[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C29H36N6O5
8-[[2-(3,4-dimethoxyphenyl)ethyl-[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-methoxy-4-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]tetrazolo[1,5-a]quinoline —— C27H32N10O
8-methoxy-4-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]tetrazolo[1,5-a]quinoline
—— 8-(5-Phenyl-2-m-tolyl-pyrazolo[1,5-a]pyrimidin-7-yl)-1,4-dioxa-8-aza-spiro[4.5]decane —— C26H26N4O2
8-(5-Phenyl-2-m-tolyl-pyrazolo[1,5-a]pyrimidin-7-yl)-1,4-dioxa-8-aza-spiro[4.5]decane
—— 8-[[benzyl-[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]butyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C29H36N6O3
8-[[benzyl-[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]butyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— (8aR)-2-[(S)-(1-cyclopentyltetrazol-5-yl)-(2-methoxyphenyl)methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine —— C21H30N6O
(8aR)-2-[(S)-(1-cyclopentyltetrazol-5-yl)-(2-methoxyphenyl)methyl]-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazine
—— 8-[[[(1S)-1-(1-tert-butyltetrazol-5-yl)butyl]-[(4-fluorophenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one —— C28H33FN6O3
8-[[[(1S)-1-(1-tert-butyltetrazol-5-yl)butyl]-[(4-fluorophenyl)methyl]amino]methyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-one
—— 8-[4-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]sulfonyl-1,4-dioxa-8-azaspiro[4.5]decane —— C19H28N2O6S2
8-[4-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]sulfonyl-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-methyl-3-[3-(2-methylbutan-2-ylamino)imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C22H24N4O
8-methyl-3-[3-(2-methylbutan-2-ylamino)imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 896683-84-4 (Racemate) —— C27H32N4O4S
896683-84-4 (Racemate)
—— 8-[2-[(4-Fluorophenyl)methylidene]hydrazinyl]-1,3-dimethyl-7-propan-2-ylpurine-2,6-dione —— C17H19FN6O2
8-[2-[(4-Fluorophenyl)methylidene]hydrazinyl]-1,3-dimethyl-7-propan-2-ylpurine-2,6-dione
—— (8R,8aS)-6-amino-2-benzyl-8-(4-chloro-2-nitrophenyl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C25H19ClN6O2
(8R,8aS)-6-amino-2-benzyl-8-(4-chloro-2-nitrophenyl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8S,8aR)-6-amino-8-(3,4-diethoxyphenyl)-2,3,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile —— C22H23N5O2
(8S,8aR)-6-amino-8-(3,4-diethoxyphenyl)-2,3,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile
—— 8-Bromo-7-[(2-chlorophenyl)methyl]-3-methyl-1-[(3-methylphenyl)methyl]purine-2,6-dione —— C21H18BrClN4O2
8-Bromo-7-[(2-chlorophenyl)methyl]-3-methyl-1-[(3-methylphenyl)methyl]purine-2,6-dione
—— 8,9-Dimethoxy-3-(4-methoxy-phenyl)-5,5-dimethyl-5,6-dihydro-[1,2,4]triazolo[3,4-a]isoquinoline —— C21H23N3O3
8,9-Dimethoxy-3-(4-methoxy-phenyl)-5,5-dimethyl-5,6-dihydro-[1,2,4]triazolo[3,4-a]isoquinoline
—— 8-{[4-(2-Methoxyphenyl)piperazin-1-yl]sulfonyl}quinoline —— C20H21N3O3S
8-{[4-(2-Methoxyphenyl)piperazin-1-yl]sulfonyl}quinoline
—— 8-(4-benzhydrylpiperazin-1-yl)-3-methyl-7-(3-methylbenzyl)-1H-purine-2,6(3H,7H)-dione —— C31H32N6O2
8-(4-benzhydrylpiperazin-1-yl)-3-methyl-7-(3-methylbenzyl)-1H-purine-2,6(3H,7H)-dione
—— 8-[(2R)-butan-2-yl]-12-[4-(3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyl]-5-thia-1,8,10,11-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,9,11-tetraen-7-one —— C24H27N5O2S
8-[(2R)-butan-2-yl]-12-[4-(3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyl]-5-thia-1,8,10,11-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,9,11-tetraen-7-one
—— 8-[(2S)-butan-2-yl]-12-[4-(3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyl]-5-thia-1,8,10,11-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,9,11-tetraen-7-one —— C24H27N5O2S
8-[(2S)-butan-2-yl]-12-[4-(3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyl]-5-thia-1,8,10,11-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),3,9,11-tetraen-7-one
—— 8-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-3-methyl-7-[2-(1-phenyltetrazol-5-yl)sulfanylethyl]purine-2,6-dione —— C22H27N9O2S
8-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-3-methyl-7-[2-(1-phenyltetrazol-5-yl)sulfanylethyl]purine-2,6-dione
—— 8-[2-[1-(4-Methoxyphenyl)ethylidene]hydrazinyl]-1,3-dimethyl-7-(naphthalen-1-ylmethyl)purine-2,6-dione —— C27H26N6O3
8-[2-[1-(4-Methoxyphenyl)ethylidene]hydrazinyl]-1,3-dimethyl-7-(naphthalen-1-ylmethyl)purine-2,6-dione
—— (8aR)-4-phenacylsulfanyl-6,7,8,8a-tetrahydropyrrolo[1,2-a]pyrimidine-3-carbonitrile —— C16H15N3OS
(8aR)-4-phenacylsulfanyl-6,7,8,8a-tetrahydropyrrolo[1,2-a]pyrimidine-3-carbonitrile
—— 8-[2-[(4-methoxyphenyl)methylidene]hydrazinyl]-1,3-dimethyl-7-(naphthalen-1-ylmethyl)purine-2,6-dione —— C26H24N6O3
8-[2-[(4-methoxyphenyl)methylidene]hydrazinyl]-1,3-dimethyl-7-(naphthalen-1-ylmethyl)purine-2,6-dione
—— 8-Morpholin-4-yl-4,11-dioxa-1,3,5,7,10-pentazatricyclo[7.3.0.02,6]dodeca-2,5,7,9-tetraen-12-one —— C9H8N6O4
8-Morpholin-4-yl-4,11-dioxa-1,3,5,7,10-pentazatricyclo[7.3.0.02,6]dodeca-2,5,7,9-tetraen-12-one
—— (8R,8aR)-6-amino-8-(2-fluoro-5-methoxyphenyl)-2-propan-2-yl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C22H22FN5O
(8R,8aR)-6-amino-8-(2-fluoro-5-methoxyphenyl)-2-propan-2-yl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8S,8aS)-6-amino-8-(2,5-dichlorophenyl)-2-ethyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C20H17Cl2N5
(8S,8aS)-6-amino-8-(2,5-dichlorophenyl)-2-ethyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— 8-Methyl-13-phenyl-8,10,12,15,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,13-heptaene —— C18H13N5
8-Methyl-13-phenyl-8,10,12,15,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,13-heptaene
—— 8-(Azepan-1-ylmethyl)-3-(4-methoxyphenoxy)-4-oxochromen-7-olate —— C23H24NO5-
8-(Azepan-1-ylmethyl)-3-(4-methoxyphenoxy)-4-oxochromen-7-olate
—— 8,8-dimethyl-2-thioxo-2,3,7,8-tetrahydro-1H-pyrano[3'',4'':5',6']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(10H)-one —— C14H13N3O2S2
8,8-dimethyl-2-thioxo-2,3,7,8-tetrahydro-1H-pyrano[3'',4'':5',6']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(10H)-one
—— 8-(4-benzylpiperidin-1-yl)-7-(2,4-dichlorobenzyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione —— C26H27Cl2N5O2
8-(4-benzylpiperidin-1-yl)-7-(2,4-dichlorobenzyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione
—— 8-methyl-2-[(4-methylphenyl)methyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-4,5-dihydrofuro[2,3-g]indazole-7-carboxamide —— C27H34N4O2
8-methyl-2-[(4-methylphenyl)methyl]-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-4,5-dihydrofuro[2,3-g]indazole-7-carboxamide