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—— 8-[(2-Fluorophenyl)methyl]-4-methyl-2-[1-(3-methylbutanoyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[(2-Fluorophenyl)methyl]-4-methyl-2-[1-(3-methylbutanoyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-4-methyl-2-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O
8-(Cyclopropylmethyl)-4-methyl-2-[1-(2-phenylethyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclohexylmethyl)-4-methyl-2-[1-(2-propan-2-yloxyacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H38N4O3
8-(Cyclohexylmethyl)-4-methyl-2-[1-(2-propan-2-yloxyacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-3-[2-(1H-indol-2-yl)ethyl-(oxolane-2-carbonyl)amino]-6-methoxy-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C32H35N3O8
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-3-[2-(1H-indol-2-yl)ethyl-(oxolane-2-carbonyl)amino]-6-methoxy-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— 8-Cyclopentyl-2-[1-[(1-ethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-Cyclopentyl-2-[1-[(1-ethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-(cyclohexylmethyl)-2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclohexylmethyl)-4-methyl-2-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(Cyclohexylmethyl)-4-methyl-2-[1-[(2-methylpyrazol-3-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O2
8-(Cyclopropylmethyl)-2-[1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-4-methyl-2-[1-(4-pyridin-2-ylbutanoyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-(Cyclopropylmethyl)-4-methyl-2-[1-(4-pyridin-2-ylbutanoyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[1-(4-ethylthiadiazole-5-carbonyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H28N6O2S
8-(Cyclopropylmethyl)-2-[1-(4-ethylthiadiazole-5-carbonyl)piperidin-4-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-Benzyl-4-methyl-2-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[1-(2-pyrazol-1-ylacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-Benzyl-4-methyl-2-[1-(2-pyrazol-1-ylacetyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Cyclopentyl-4-methyl-2-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H36N6O
8-Cyclopentyl-4-methyl-2-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-{[3-Methyl-2-(pyrrolidine-1-carbonyl)-1-benzofuran-5-YL]sulfonyl}-1,4-dioxa-8-azaspiro[4.5]decane —— C21H26N2O6S
8-{[3-Methyl-2-(pyrrolidine-1-carbonyl)-1-benzofuran-5-YL]sulfonyl}-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-(3-chloro-4-fluorophenyl)-6-(2-hydroxy-3-methoxyphenyl)-6a-methyl-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C34H28ClFN2O6
8-(3-chloro-4-fluorophenyl)-6-(2-hydroxy-3-methoxyphenyl)-6a-methyl-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-2-carboxamide —— C20H23N5O2
8-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-[2-[1-(4-Methoxyphenyl)ethylidene]hydrazinyl]-3-methyl-7-(2-methylpropyl)purine-2,6-dione —— C19H24N6O3
8-[2-[1-(4-Methoxyphenyl)ethylidene]hydrazinyl]-3-methyl-7-(2-methylpropyl)purine-2,6-dione
—— 8-[(2S)-2-(4-ethoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-quinolin-4-one —— C23H24N2O3
8-[(2S)-2-(4-ethoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-quinolin-4-one
—— 8-(2,4-dichloroanilino)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(2-hydroxy-6-methoxyphenyl)-6a-(4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C48H42Cl2N6O7
8-(2,4-dichloroanilino)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(2-hydroxy-6-methoxyphenyl)-6a-(4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-bromo-N-(4-chlorophenyl)-3-ethyl-2-methyl-4-thioxo-3,4,5,6-tetrahydro-2H-2,6-methano-1,3,5-benzoxadiazocine-11-carboxamide —— C20H19BrClN3O2S
8-bromo-N-(4-chlorophenyl)-3-ethyl-2-methyl-4-thioxo-3,4,5,6-tetrahydro-2H-2,6-methano-1,3,5-benzoxadiazocine-11-carboxamide
—— 8-[(2R)-2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-quinolin-4-one —— C22H22N2O3
8-[(2R)-2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-quinolin-4-one
—— 8-[(2R)-2-(4-ethoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-quinolin-4-one —— C23H24N2O3
8-[(2R)-2-(4-ethoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-quinolin-4-one
—— 8-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-2-carboxamide —— C20H23N5O2
8-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-methyl-N-[5-[(1R)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H17N5O2S
8-methyl-N-[5-[(1R)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-chloro-N-(4-chlorophenyl)-3-(4-ethylphenyl)-2-methyl-4-thioxo-3,4,5,6-tetrahydro-2H-2,6-methano-1,3,5-benzoxadiazocine-11-carboxamide —— C26H23Cl2N3O2S
8-chloro-N-(4-chlorophenyl)-3-(4-ethylphenyl)-2-methyl-4-thioxo-3,4,5,6-tetrahydro-2H-2,6-methano-1,3,5-benzoxadiazocine-11-carboxamide
—— 8-methyl-N-[5-[(1S)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H17N5O2S
8-methyl-N-[5-[(1S)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— 8-methyl-N-[(1R)-3-morpholin-4-yl-1-phenylpropyl]imidazo[1,2-a]pyridine-2-carboxamide —— C22H26N4O2
8-methyl-N-[(1R)-3-morpholin-4-yl-1-phenylpropyl]imidazo[1,2-a]pyridine-2-carboxamide
—— (8-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone —— C24H27N5O
(8-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone
—— 8-(Bromomethyl)-6a,9a-dichloro-2-(3-chloro-4-methylphenyl)-6-(3-ethoxy-4-hydroxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C30H26BrCl3N2O6
8-(Bromomethyl)-6a,9a-dichloro-2-(3-chloro-4-methylphenyl)-6-(3-ethoxy-4-hydroxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(2-chloro-4-hydroxyphenyl)-2-(4-ethylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H24BrCl3N2O5
8-(Bromomethyl)-6a,9a-dichloro-6-(2-chloro-4-hydroxyphenyl)-2-(4-ethylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-[4-(2-hydroxyethoxy)phenyl]-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C23H21BrCl2N2O6
8-(Bromomethyl)-6a,9a-dichloro-6-[4-(2-hydroxyethoxy)phenyl]-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8a-(4-bromophenyl)-4,5-diphenylhexahydropyrimido[4,5-d]pyrimidine-2,7(1H,3H)-dione —— C24H21BrN4O2
8a-(4-bromophenyl)-4,5-diphenylhexahydropyrimido[4,5-d]pyrimidine-2,7(1H,3H)-dione
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(1-hydroxynaphthalen-2-yl)-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide —— C26H20BrCl2N3O6
8-(Bromomethyl)-6a,9a-dichloro-6-(1-hydroxynaphthalen-2-yl)-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide
—— 8-(3-chlorophenyl)-6-(2-hydroxy-3-methylphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C33H27ClN2O5
8-(3-chlorophenyl)-6-(2-hydroxy-3-methylphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(4-hydroxyphenyl)-2-(thiophen-2-ylmethyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C26H21BrCl2N2O5S
8-(Bromomethyl)-6a,9a-dichloro-6-(4-hydroxyphenyl)-2-(thiophen-2-ylmethyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(4-hydroxy-3,5-dimethoxyphenyl)-2-(4-iodophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H24BrCl2IN2O7
8-(Bromomethyl)-6a,9a-dichloro-6-(4-hydroxy-3,5-dimethoxyphenyl)-2-(4-iodophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-[5-(hydroxymethyl)furan-2-yl]-2-(4-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C26H20BrCl2N3O8
8-(Bromomethyl)-6a,9a-dichloro-6-[5-(hydroxymethyl)furan-2-yl]-2-(4-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-(4-hydroxy-3-methoxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C38H33BrCl2N2O8
8-(Bromomethyl)-6a,9a-dichloro-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-(4-hydroxy-3-methoxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(4-Chlorophenyl)-9-(trifluoromethyl)-2,3-dihydropyrano[3,2-h][1,4]benzodioxin-7-one —— C18H10ClF3O4
8-(4-Chlorophenyl)-9-(trifluoromethyl)-2,3-dihydropyrano[3,2-h][1,4]benzodioxin-7-one
—— 8-Ethyl-2-[4-[[4-[(3-methoxypyrazin-2-yl)sulfamoyl]phenyl]carbamothioyl]piperazin-1-ium-1-yl]-5-oxopyrido[2,3-d]pyrimidine-6-carboxylate —— C26H27N9O6S2
8-Ethyl-2-[4-[[4-[(3-methoxypyrazin-2-yl)sulfamoyl]phenyl]carbamothioyl]piperazin-1-ium-1-yl]-5-oxopyrido[2,3-d]pyrimidine-6-carboxylate
—— 8-methyl-2-pyridin-2-yl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]quinoline-4-carboxamide —— C25H27N5O
8-methyl-2-pyridin-2-yl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]quinoline-4-carboxamide
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(2-hydroxy-4-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H31ClN4O6S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(2-hydroxy-4-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-methyl-2-pyridin-3-yl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]quinoline-4-carboxamide —— C25H27N5O
8-methyl-2-pyridin-3-yl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]quinoline-4-carboxamide
—— 8-methyl-2-pyridin-3-yl-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]quinoline-4-carboxamide —— C25H27N5O
8-methyl-2-pyridin-3-yl-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]quinoline-4-carboxamide
—— 8-(Bromomethyl)-2-tert-butyl-6a,9a-dichloro-6-(4-hydroxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C25H25BrCl2N2O5
8-(Bromomethyl)-2-tert-butyl-6a,9a-dichloro-6-(4-hydroxyphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-methyl-2-pyridin-3-yl-N-[(2R)-1-pyrrolidin-1-ylpropan-2-yl]quinoline-4-carboxamide —— C23H26N4O
8-methyl-2-pyridin-3-yl-N-[(2R)-1-pyrrolidin-1-ylpropan-2-yl]quinoline-4-carboxamide
—— 8-(3-chlorophenyl)-6-(2-hydroxy-3-methylphenyl)-1,3,7,9-tetraoxo-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide —— C34H28ClN3O6
8-(3-chlorophenyl)-6-(2-hydroxy-3-methylphenyl)-1,3,7,9-tetraoxo-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide
—— 8-methyl-2-pyridin-3-yl-N-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]quinoline-4-carboxamide —— C23H26N4O
8-methyl-2-pyridin-3-yl-N-[(2S)-1-pyrrolidin-1-ylpropan-2-yl]quinoline-4-carboxamide
—— 8-(3-chloro-4-fluorophenyl)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(4-hydroxynaphthalen-1-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C45H37ClFN5O5
8-(3-chloro-4-fluorophenyl)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(4-hydroxynaphthalen-1-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chlorophenyl)-6-(3-fluoro-4-hydroxyphenyl)-2-(4-morpholin-4-ylphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H35ClFN3O6
8-(3-chlorophenyl)-6-(3-fluoro-4-hydroxyphenyl)-2-(4-morpholin-4-ylphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone