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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H31N5O3
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H24N6O2S
8-benzyl-4-methyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(cyclohexylmethyl)-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-2-[(2S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[3-(5-methyl-3,4-dihydropyrazol-2-yl)propanoyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[3-(5-methyl-3,4-dihydropyrazol-2-yl)propanoyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H23FN6O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H31N5O2
8-(cyclopropylmethyl)-2-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H23FN6O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(cyclopentanecarbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O2
8-benzyl-2-[(2R)-1-(cyclopentanecarbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-2-[(2R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O2
8-benzyl-2-[(2R)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(cyclohexylmethyl)-2-[(2S)-1-[(1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O
8-(cyclopropylmethyl)-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H34N4O3
8-(cyclohexylmethyl)-2-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H27N5O2
8-benzyl-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(1,3-dimethylpyrazole-4-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-2-[(2S)-1-(1,3-dimethylpyrazole-4-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclopropylmethyl)-2-[(2R)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N6O2
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H22FN5O3
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-pyridin-2-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-pyridin-2-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclohexylmethyl)-4-methyl-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N6O2
8-(Cyclohexylmethyl)-4-methyl-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-pyrrolidin-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H37N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-pyrrolidin-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H28N4O3
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25N5O2S
8-benzyl-4-methyl-2-[(2S)-1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H26N6O2
8-benzyl-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H23FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N6O2
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H24FN5O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H23FN6O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(cyclohexylmethyl)-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-(3-methoxybenzoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N4O3
8-(cyclopropylmethyl)-2-[(2R)-1-(3-methoxybenzoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-2-[(2S)-1-[(1,5-dimethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2S)-1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(3-methylbutanoyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H32N4O2
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(3-methylbutanoyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(1,3-dimethylpyrazole-4-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-2-[(2R)-1-(1,3-dimethylpyrazole-4-carbonyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H26N6O2
8-benzyl-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H38N4O3
8-(cyclohexylmethyl)-4-methyl-2-[(3R)-1-(2-propan-2-yloxyacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H24N6O2S
8-benzyl-4-methyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H23FN6O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one