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—— [8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-[1-(phenoxymethyl)pyrazol-3-yl]methanone —— C18H17F3N6O2
[8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-[1-(phenoxymethyl)pyrazol-3-yl]methanone
—— [8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(4-propan-2-yloxy-1-benzofuran-6-yl)methanone —— C19H19F3N4O3
[8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(4-propan-2-yloxy-1-benzofuran-6-yl)methanone
—— [8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(1,2,3-trimethylindol-5-yl)methanone —— C19H20F3N5O
[8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(1,2,3-trimethylindol-5-yl)methanone
—— 8-methyl-7-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C17H19F3N4O2S
8-methyl-7-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[3-methoxypropanoyl(3-methylbutyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C26H36N2O8
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[3-methoxypropanoyl(3-methylbutyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— [8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-pyrazin-2-ylmethanone —— C12H11F3N6O
[8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-pyrazin-2-ylmethanone
—— [8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(5-thiophen-2-yl-1H-pyrazol-3-yl)methanone —— C15H13F3N6OS
[8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-(5-thiophen-2-yl-1H-pyrazol-3-yl)methanone
—— [8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-[4-(pyrazol-1-ylmethyl)phenyl]methanone —— C18H17F3N6O
[8-methyl-3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-[4-(pyrazol-1-ylmethyl)phenyl]methanone
—— 8-(3-chlorophenyl)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C39H31ClN2O6
8-(3-chlorophenyl)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(2,4-dichloroanilino)-6-(2-hydroxy-3-methoxyphenyl)-6a-(4-methoxyphenyl)-2-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H31Cl2N3O7
8-(2,4-dichloroanilino)-6-(2-hydroxy-3-methoxyphenyl)-6a-(4-methoxyphenyl)-2-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[Benzyl(methyl)amino]-7-[(3-bromophenyl)methyl]-1,3-dimethylpurine-2,6-dione —— C22H22BrN5O2
8-[Benzyl(methyl)amino]-7-[(3-bromophenyl)methyl]-1,3-dimethylpurine-2,6-dione
—— 8-(3-chlorophenyl)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-[2-(4-hydroxy-3,5-dimethoxyphenyl)ethenyl]-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C50H44ClN5O7
8-(3-chlorophenyl)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-[2-(4-hydroxy-3,5-dimethoxyphenyl)ethenyl]-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8a-Hydroxy-1-(propan-2-ylideneamino)spiro[3,4a,5,6,7,8-hexahydroquinazoline-4,1'-cyclohexane]-2-thione —— C16H27N3OS
8a-Hydroxy-1-(propan-2-ylideneamino)spiro[3,4a,5,6,7,8-hexahydroquinazoline-4,1'-cyclohexane]-2-thione
—— 8-[4-(2-hydroxyethyl)piperazin-1-yl]-13-(4-methylphenyl)-15-thia-9,17-diaza-10-azoniatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),2,4,6,8,12(16),13-heptaen-11-one —— C26H26N5O2S+
8-[4-(2-hydroxyethyl)piperazin-1-yl]-13-(4-methylphenyl)-15-thia-9,17-diaza-10-azoniatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),2,4,6,8,12(16),13-heptaen-11-one
—— 8-[4-(2-hydroxyethyl)piperazin-1-yl]-13,14-dimethyl-15-thia-9,17-diaza-10-azoniatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),2,4,6,8,12(16),13-heptaen-11-one —— C21H24N5O2S+
8-[4-(2-hydroxyethyl)piperazin-1-yl]-13,14-dimethyl-15-thia-9,17-diaza-10-azoniatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),2,4,6,8,12(16),13-heptaen-11-one
—— 8-(Piperidine-1-carbonyl)pyrido[2,1-b]quinazolin-11-one —— C18H17N3O2
8-(Piperidine-1-carbonyl)pyrido[2,1-b]quinazolin-11-one
—— 8-[(4-Benzylpiperidin-1-YL)methyl]-7-[(2-chlorophenyl)methyl]-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C27H30ClN5O2
8-[(4-Benzylpiperidin-1-YL)methyl]-7-[(2-chlorophenyl)methyl]-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 8-(2-Chlorobenzylidene)-6,10-dioxaspiro(4.5)decane-7,9-dione —— C15H13ClO4
8-(2-Chlorobenzylidene)-6,10-dioxaspiro(4.5)decane-7,9-dione
—— 8-(biphenyl-4-yloxy)-7-(4-methoxybenzyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione —— C27H24N4O4
8-(biphenyl-4-yloxy)-7-(4-methoxybenzyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione
—— 8-Benzoyl-4-(4-chlorobenzoyl)-2-phenyl-3a,4,9a,9b-tetrahydropyrrolo[3,4-a]indolizine-1,3-dione —— C30H21ClN2O4
8-Benzoyl-4-(4-chlorobenzoyl)-2-phenyl-3a,4,9a,9b-tetrahydropyrrolo[3,4-a]indolizine-1,3-dione
—— 8-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-5'-[3-[benzyl(methyl)amino]prop-1-ynyl]-6-(4-hydroxyphenyl)-1,2'-dioxo-3,4-diphenyl-N-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1'-carboxamide —— C65H60N6O8
8-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-5'-[3-[benzyl(methyl)amino]prop-1-ynyl]-6-(4-hydroxyphenyl)-1,2'-dioxo-3,4-diphenyl-N-(1-phenylethyl)spiro[4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine-7,3'-indole]-1'-carboxamide
—— 8-[3,5-bis(trifluoromethyl)benzoyl]-N-(2-phenylethyl)-1-thia-4,8-diazaspiro[4.5]decane-3-carboxamide —— C25H25F6N3O2S
8-[3,5-bis(trifluoromethyl)benzoyl]-N-(2-phenylethyl)-1-thia-4,8-diazaspiro[4.5]decane-3-carboxamide
—— 8-(Hexylamino)-7-[2-hydroxy-3-(4-methylphenoxy)propyl]-1,3-dimethylpurine-2,6-dione —— C23H33N5O4
8-(Hexylamino)-7-[2-hydroxy-3-(4-methylphenoxy)propyl]-1,3-dimethylpurine-2,6-dione
—— 8-Chloro-4-(1,3-thiazol-2-ylmethylamino)quinoline-3-carbonitrile —— C14H9ClN4S
8-Chloro-4-(1,3-thiazol-2-ylmethylamino)quinoline-3-carbonitrile
—— 8-Chloro-4-(3-indol-1-ylpropylamino)quinoline-3-carbonitrile —— C21H17ClN4
8-Chloro-4-(3-indol-1-ylpropylamino)quinoline-3-carbonitrile
—— 8-Chloro-4-(2-methyl-2,3-dihydroindol-1-yl)quinoline-3-carbonitrile —— C19H14ClN3
8-Chloro-4-(2-methyl-2,3-dihydroindol-1-yl)quinoline-3-carbonitrile
—— 8-Methoxy-4-[3-(4-methylindazol-1-yl)propylamino]quinoline-3-carbonitrile —— C22H21N5O
8-Methoxy-4-[3-(4-methylindazol-1-yl)propylamino]quinoline-3-carbonitrile
—— 8-methoxy-4-(6-methyl-3,4-dihydro-2H-quinolin-1-yl)quinoline-3-carbonitrile —— C21H19N3O
8-methoxy-4-(6-methyl-3,4-dihydro-2H-quinolin-1-yl)quinoline-3-carbonitrile
—— 8-Methoxy-4-(2-methyl-2,3-dihydroindol-1-yl)quinoline-3-carbonitrile —— C20H17N3O
8-Methoxy-4-(2-methyl-2,3-dihydroindol-1-yl)quinoline-3-carbonitrile
—— 8-methoxy-5-oxo-N-[1-(2,2,2-trifluoroacetyl)piperidin-4-yl]-2,4-dihydro-1H-chromeno[3,4-c]pyridine-3-carboxamide —— C21H22F3N3O5
8-methoxy-5-oxo-N-[1-(2,2,2-trifluoroacetyl)piperidin-4-yl]-2,4-dihydro-1H-chromeno[3,4-c]pyridine-3-carboxamide
—— 8-(benzyloxy)-N-tert-butyl-2-(3-methylphenyl)imidazo[1,2-a]pyridin-3-amine —— C25H27N3O
8-(benzyloxy)-N-tert-butyl-2-(3-methylphenyl)imidazo[1,2-a]pyridin-3-amine
—— 8-Methoxy-4-[(4-methyl-1,3-thiazol-2-yl)methylamino]quinoline-3-carbonitrile —— C16H14N4OS
8-Methoxy-4-[(4-methyl-1,3-thiazol-2-yl)methylamino]quinoline-3-carbonitrile
—— 8-(3-Methylpiperidin-1-yl)-1,6-naphthyridine —— C14H17N3
8-(3-Methylpiperidin-1-yl)-1,6-naphthyridine
—— 8-Piperidin-1-yl-1,6-naphthyridine —— C13H15N3
8-Piperidin-1-yl-1,6-naphthyridine
—— 8-[4-(2-Methoxyethylsulfonyl)piperazin-1-yl]-1,6-naphthyridine —— C15H20N4O3S
8-[4-(2-Methoxyethylsulfonyl)piperazin-1-yl]-1,6-naphthyridine
—— 8-Methoxy-4-[3-(6-methylindazol-1-yl)propylamino]quinoline-3-carbonitrile —— C22H21N5O
8-Methoxy-4-[3-(6-methylindazol-1-yl)propylamino]quinoline-3-carbonitrile
—— 8-(2,3-Dihydroindol-1-yl)-1,6-naphthyridine —— C16H13N3
8-(2,3-Dihydroindol-1-yl)-1,6-naphthyridine
—— 8-chloro-4-(3,4-dihydro-1H-isoquinolin-2-yl)quinoline-3-carbonitrile —— C19H14ClN3
8-chloro-4-(3,4-dihydro-1H-isoquinolin-2-yl)quinoline-3-carbonitrile
—— 8-(6-methyl-3,4-dihydro-2H-quinolin-1-yl)-1,6-naphthyridine —— C18H17N3
8-(6-methyl-3,4-dihydro-2H-quinolin-1-yl)-1,6-naphthyridine
—— 8-(3,5-Dimethylpiperidin-1-yl)-1,6-naphthyridine —— C15H19N3
8-(3,5-Dimethylpiperidin-1-yl)-1,6-naphthyridine
—— 8-(2-Methylpiperidin-1-yl)-1,6-naphthyridine —— C14H17N3
8-(2-Methylpiperidin-1-yl)-1,6-naphthyridine
—— 8-[4-[(4-Methylphenyl)methyl]piperazin-1-yl]-1,6-naphthyridine —— C20H22N4
8-[4-[(4-Methylphenyl)methyl]piperazin-1-yl]-1,6-naphthyridine
—— 8-Methoxy-4-(oxolan-2-ylmethylamino)quinoline-3-carbonitrile —— C16H17N3O2
8-Methoxy-4-(oxolan-2-ylmethylamino)quinoline-3-carbonitrile
—— 8-Methoxy-4-[3-(2-methylimidazol-1-yl)propylamino]quinoline-3-carbonitrile —— C18H19N5O
8-Methoxy-4-[3-(2-methylimidazol-1-yl)propylamino]quinoline-3-carbonitrile
—— 8-(4-Ethylsulfonylpiperazin-1-yl)-1,6-naphthyridine —— C14H18N4O2S
8-(4-Ethylsulfonylpiperazin-1-yl)-1,6-naphthyridine
—— 8-Methoxy-4-(1,3-thiazol-2-ylmethylamino)quinoline-3-carbonitrile —— C15H12N4OS
8-Methoxy-4-(1,3-thiazol-2-ylmethylamino)quinoline-3-carbonitrile
—— 8-Pyrrolidin-1-yl-1,6-naphthyridine —— C12H13N3
8-Pyrrolidin-1-yl-1,6-naphthyridine
—— 8-(4-Phenylpiperazin-1-yl)-1,6-naphthyridine —— C18H18N4
8-(4-Phenylpiperazin-1-yl)-1,6-naphthyridine
—— 8-methoxy-4-[2-(2,5,7-trimethyl-1H-indol-3-yl)ethylamino]quinoline-3-carbonitrile —— C24H24N4O
8-methoxy-4-[2-(2,5,7-trimethyl-1H-indol-3-yl)ethylamino]quinoline-3-carbonitrile
—— 8-(4-Methylpiperazin-1-yl)-1,6-naphthyridine —— C13H16N4
8-(4-Methylpiperazin-1-yl)-1,6-naphthyridine