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—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoate —— C24H27N3O5S
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoate
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C20H17N3O4S
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 2-[(2S)-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— (8-methylimidazo[1,2-a]pyridin-2-yl)methyl 4-methoxy-3-[(2S)-2-methylpiperidin-1-yl]sulfonylbenzoate —— C23H27N3O5S
(8-methylimidazo[1,2-a]pyridin-2-yl)methyl 4-methoxy-3-[(2S)-2-methylpiperidin-1-yl]sulfonylbenzoate
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoate —— C24H27N3O5S
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylbenzoate
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-chloro-3-[methyl(phenyl)sulfamoyl]benzoate —— C24H20ClN3O5S
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-chloro-3-[methyl(phenyl)sulfamoyl]benzoate
—— 8-[[2-[4-[4-[4-(hydroxymethyl)phenyl]-6-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-8-oxooctanoic acid —— C45H52N4O7
8-[[2-[4-[4-[4-(hydroxymethyl)phenyl]-6-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-8-oxooctanoic acid
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 2-(4-benzoylphenoxy)acetate —— C25H20N2O5
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 2-(4-benzoylphenoxy)acetate
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl (2S)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate —— C25H23N3O3
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl (2S)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-[ethyl(phenyl)sulfamoyl]benzoate —— C25H23N3O5S
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl 4-[ethyl(phenyl)sulfamoyl]benzoate
—— (8-methyl-4-oxo-1H-quinazolin-2-yl)methyl (2R)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate —— C25H23N3O3
(8-methyl-4-oxo-1H-quinazolin-2-yl)methyl (2R)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate
—— (8-methylimidazo[1,2-a]pyridin-2-yl)methyl 3-methoxy-4-[2-(4-methoxyanilino)-2-oxoethoxy]benzoate —— C26H25N3O6
(8-methylimidazo[1,2-a]pyridin-2-yl)methyl 3-methoxy-4-[2-(4-methoxyanilino)-2-oxoethoxy]benzoate
—— (8-methylimidazo[1,2-a]pyridin-2-yl)methyl 4-[ethyl(phenyl)sulfamoyl]benzoate —— C24H23N3O4S
(8-methylimidazo[1,2-a]pyridin-2-yl)methyl 4-[ethyl(phenyl)sulfamoyl]benzoate
—— 8-Hexanoyl-3-(2-morpholin-4-yl-2-oxoethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one —— C25H36N4O4
8-Hexanoyl-3-(2-morpholin-4-yl-2-oxoethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
—— 8-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-8-oxooctanoic acid —— C41H49N5O6
8-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-pyrimidin-2-ylpiperazin-1-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-8-oxooctanoic acid
—— 8-methoxy-3-{5-[(3-methylphenyl)amino]-1,3,4-thiadiazol-2-yl}-2H-chromen-2-one —— C19H15N3O3S
8-methoxy-3-{5-[(3-methylphenyl)amino]-1,3,4-thiadiazol-2-yl}-2H-chromen-2-one
—— 8-Bromo-3-methyl-7-(1-oxo-1-phenylbutan-2-yl)purine-2,6-dione —— C16H15BrN4O3
8-Bromo-3-methyl-7-(1-oxo-1-phenylbutan-2-yl)purine-2,6-dione
—— 8-[(2R)-1-(azepan-1-yl)-1-oxopropan-2-yl]sulfanyl-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-3-one —— C25H31N5O2S
8-[(2R)-1-(azepan-1-yl)-1-oxopropan-2-yl]sulfanyl-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-3-one
—— 8-[(2S)-1-(azepan-1-yl)-1-oxopropan-2-yl]sulfanyl-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-3-one —— C25H31N5O2S
8-[(2S)-1-(azepan-1-yl)-1-oxopropan-2-yl]sulfanyl-4-phenyl-4,5,7,9-tetrazatricyclo[7.5.0.02,6]tetradeca-1,5,7-trien-3-one
—— 8-(2,4-Dichlorobenzoyl)-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one —— C26H28Cl2N4O3
8-(2,4-Dichlorobenzoyl)-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
—— 8'-(azocane-1-carbonyl)-6'-[4-(2-hydroxyethoxy)phenyl]-5-[2-(4-methoxyphenyl)ethynyl]-3',4'-diphenylspiro[1H-indole-3,7'-4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine]-1',2-dione —— C51H49N3O7
8'-(azocane-1-carbonyl)-6'-[4-(2-hydroxyethoxy)phenyl]-5-[2-(4-methoxyphenyl)ethynyl]-3',4'-diphenylspiro[1H-indole-3,7'-4,6,8,8a-tetrahydro-3H-pyrrolo[2,1-c][1,4]oxazine]-1',2-dione
—— (8-methoxy-4-methyl-6-oxobenzo[c]chromen-3-yl) (2S,3S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate —— C26H31NO7
(8-methoxy-4-methyl-6-oxobenzo[c]chromen-3-yl) (2S,3S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate
—— (8-methoxy-6-oxobenzo[c]chromen-3-yl) (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylpropanoate —— C28H27NO7
(8-methoxy-6-oxobenzo[c]chromen-3-yl) (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylpropanoate
—— (8R)-2,2,6-trimethyl-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione —— C17H19N3O2
(8R)-2,2,6-trimethyl-3,6,17-triazatetracyclo[8.7.0.03,8.011,16]heptadeca-1(10),11,13,15-tetraene-4,7-dione
—— (8-methoxy-4-methyl-6-oxobenzo[c]chromen-3-yl) (2R,3R)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate —— C26H31NO7
(8-methoxy-4-methyl-6-oxobenzo[c]chromen-3-yl) (2R,3R)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate
—— (8-methoxy-6-oxobenzo[c]chromen-3-yl) (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]propanoate —— C22H23NO7
(8-methoxy-6-oxobenzo[c]chromen-3-yl) (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]propanoate
—— [(8R,9R,13R,14R,17S)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate —— C30H37FO3
[(8R,9R,13R,14R,17S)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate
—— (8-methyl-2-oxo-4-phenylchromen-7-yl) (2S,3S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate —— C27H31NO6
(8-methyl-2-oxo-4-phenylchromen-7-yl) (2S,3S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate
—— (8-methyl-2-oxo-4-phenylchromen-7-yl) (2R,3R)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate —— C27H31NO6
(8-methyl-2-oxo-4-phenylchromen-7-yl) (2R,3R)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate
—— [(8R,9R,13R,14S,17R)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate —— C30H37FO3
[(8R,9R,13R,14S,17R)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate
—— [(8R,9R,13R,14S,17S)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate —— C30H37FO3
[(8R,9R,13R,14S,17S)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate
—— (8-methyl-2-oxo-4-phenylchromen-7-yl) (2R,3S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate —— C27H31NO6
(8-methyl-2-oxo-4-phenylchromen-7-yl) (2R,3S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]pentanoate
—— (8S,8aS)-6-amino-8-(4-chloro-2-nitrophenyl)-2-ethyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C20H17ClN6O2
(8S,8aS)-6-amino-8-(4-chloro-2-nitrophenyl)-2-ethyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8S,8aS)-6-amino-8-(3-ethoxy-4-propoxyphenyl)-2-propyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C26H31N5O2
(8S,8aS)-6-amino-8-(3-ethoxy-4-propoxyphenyl)-2-propyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8R,8aS)-6-amino-2-(2-phenylethyl)-8-thiophen-2-yl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C24H21N5S
(8R,8aS)-6-amino-2-(2-phenylethyl)-8-thiophen-2-yl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— [(8R,9R,13R,14R,17R)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate —— C30H37FO3
[(8R,9R,13R,14R,17R)-3-[(2-fluorophenyl)methoxy]-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] pentanoate
—— (8S,8aS)-6-amino-8-(4-chloro-2-nitrophenyl)-2-methyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C19H15ClN6O2
(8S,8aS)-6-amino-8-(4-chloro-2-nitrophenyl)-2-methyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8R,8aS)-6-amino-8-(2,3-difluorophenyl)-2-propyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C21H19F2N5
(8R,8aS)-6-amino-8-(2,3-difluorophenyl)-2-propyl-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— (8R,8aS)-6-amino-2-ethyl-8-(2-methoxyphenyl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile —— C21H21N5O
(8R,8aS)-6-amino-2-ethyl-8-(2-methoxyphenyl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrile
—— 8-bromo-3-methyl-7-[(2S)-2-methyl-3-(4-methylpyrimidin-2-yl)sulfanylpropyl]purine-2,6-dione —— C15H17BrN6O2S
8-bromo-3-methyl-7-[(2S)-2-methyl-3-(4-methylpyrimidin-2-yl)sulfanylpropyl]purine-2,6-dione
—— 8-bromo-3-methyl-7-[(2R)-2-methyl-3-(4-methylpyrimidin-2-yl)sulfanylpropyl]purine-2,6-dione —— C15H17BrN6O2S
8-bromo-3-methyl-7-[(2R)-2-methyl-3-(4-methylpyrimidin-2-yl)sulfanylpropyl]purine-2,6-dione
—— 8-(Benzyloxy)-2-(pyridin-2-YL)-N-(2,4,4-trimethylpentan-2-YL)imidazo[1,2-A]pyridin-3-amine —— C27H32N4O
8-(Benzyloxy)-2-(pyridin-2-YL)-N-(2,4,4-trimethylpentan-2-YL)imidazo[1,2-A]pyridin-3-amine
—— 8-[[2-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-8-oxooctanoic acid —— C46H54N4O7
8-[[2-[4-[4-[4-(Hydroxymethyl)phenyl]-6-[(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-8-oxooctanoic acid
—— (8aS,10R,11R)-11-acetyl-10-(2-ethoxyphenyl)spiro[10,11-dihydro-8aH-pyrrolo[1,2-a][1,10]phenanthroline-9,2'-indene]-1',3'-dione —— C33H26N2O4
(8aS,10R,11R)-11-acetyl-10-(2-ethoxyphenyl)spiro[10,11-dihydro-8aH-pyrrolo[1,2-a][1,10]phenanthroline-9,2'-indene]-1',3'-dione
—— 8-[[4-[4-[4-(Hydroxymethyl)phenyl]-6-[[2-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid —— C36H50N2O8
8-[[4-[4-[4-(Hydroxymethyl)phenyl]-6-[[2-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-8-oxooctanoic acid
—— 8-(3-nitrobenzoyl)-N-(2-phenylethyl)-1-thia-4,8-diazaspiro[4.5]decane-3-carboxamide —— C23H26N4O4S
8-(3-nitrobenzoyl)-N-(2-phenylethyl)-1-thia-4,8-diazaspiro[4.5]decane-3-carboxamide
—— (8R,9R,13S,14R,17Z)-17-[(E)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8R,9R,13S,14R,17Z)-17-[(E)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol
—— 8-[4-[4-(1,4-Dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid —— C33H44N2O8
8-[4-[4-(1,4-Dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-8-oxooctanoic acid
—— 8-methoxy-3-[(E)-[(1R,2S,6S)-2,4,6-trimethylcyclohex-3-en-1-yl]methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione —— C21H24N4O3
8-methoxy-3-[(E)-[(1R,2S,6S)-2,4,6-trimethylcyclohex-3-en-1-yl]methylideneamino]-1,5-dihydropyrimido[5,4-b]indole-2,4-dione
—— 8-benzyl-1,3-dimethyl-7H-purine-2,6-dithione —— C14H14N4S2
8-benzyl-1,3-dimethyl-7H-purine-2,6-dithione
—— (8R,9R,13S,14R,17E)-17-[(Z)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol —— C25H32N4O
(8R,9R,13S,14R,17E)-17-[(Z)-(1-ethyl-3-methylpyrazol-4-yl)methylidenehydrazinylidene]-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-3-ol