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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-(Bromomethyl)-6a,9a-dichloro-6-(2-chloro-4-hydroxyphenyl)-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide —— C22H17BrCl3N3O6
8-(Bromomethyl)-6a,9a-dichloro-6-(2-chloro-4-hydroxyphenyl)-1,3,7,9-tetraoxo-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-2-carboxamide
—— 8-benzyl-2-[(2S)-1-(2-cyclopentylacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H34N4O2
8-benzyl-2-[(2S)-1-(2-cyclopentylacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[1-(1H-pyrazole-5-carbonyl)piperidin-4-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(2-cyclopentylacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H34N4O2
8-benzyl-2-[(2R)-1-(2-cyclopentylacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-[1-[2-(Dimethylamino)acetyl]indol-3-yl]ethyl]-4-methyl-2-(methylaminomethyl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N6O2
8-[2-[1-[2-(Dimethylamino)acetyl]indol-3-yl]ethyl]-4-methyl-2-(methylaminomethyl)-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N4O3
8-benzyl-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-phenyl-N-(pyridin-4-ylmethyl)-1,6-naphthyridine-2-carboxamide —— C21H16N4O
8-phenyl-N-(pyridin-4-ylmethyl)-1,6-naphthyridine-2-carboxamide
—— 8-(6-Phenyl-2-pyridin-3-ylpyrimidin-4-yl)-1,4-dioxa-8-azaspiro[4.5]decane —— C22H22N4O2
8-(6-Phenyl-2-pyridin-3-ylpyrimidin-4-yl)-1,4-dioxa-8-azaspiro[4.5]decane
—— 8-(Allylthio)-1,3-dimethyl-7-(2-phenylethyl)-3,7-dihydro-1H-purine-2,6-dione —— C18H20N4O2S
8-(Allylthio)-1,3-dimethyl-7-(2-phenylethyl)-3,7-dihydro-1H-purine-2,6-dione
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(3-hydroxy-4-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H31ClN4O6S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(3-hydroxy-4-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-((4-(furan-2-carbonyl)piperazin-1-yl)methyl)-7-heptyl-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione —— C24H34N6O4
8-((4-(furan-2-carbonyl)piperazin-1-yl)methyl)-7-heptyl-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione
—— 8-[(4-Benzhydrylpiperazin-1-yl)methyl]-7-heptyl-1,3-dimethylpurine-2,6-dione —— C32H42N6O2
8-[(4-Benzhydrylpiperazin-1-yl)methyl]-7-heptyl-1,3-dimethylpurine-2,6-dione
—— 8-[(4-Benzylpiperazin-1-yl)methyl]-7-heptyl-1,3-dimethylpurine-2,6-dione —— C26H38N6O2
8-[(4-Benzylpiperazin-1-yl)methyl]-7-heptyl-1,3-dimethylpurine-2,6-dione
—— 8-Benzoyl-3-(1-cyclopentylpiperidin-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione —— C24H32N4O3
8-Benzoyl-3-(1-cyclopentylpiperidin-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
—— 8-[(3-Methoxyphenyl)methyl]-4-methyl-2-[[methyl(2-phenylethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H30N4O2
8-[(3-Methoxyphenyl)methyl]-4-methyl-2-[[methyl(2-phenylethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-Methoxyphenyl)methyl]-4-methyl-2-[[methyl-[(1-methylpyrazol-4-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H28N6O2
8-[(3-Methoxyphenyl)methyl]-4-methyl-2-[[methyl-[(1-methylpyrazol-4-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(2,4-dichloroanilino)-6-(2-hydroxy-3-methylphenyl)-6a-(4-methoxyphenyl)-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide —— C35H30Cl2N4O7
8-(2,4-dichloroanilino)-6-(2-hydroxy-3-methylphenyl)-6a-(4-methoxyphenyl)-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide
—— 8-Benzyl-4-methyl-2-[[methyl-[(2-propan-2-yloxyphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H32N4O2
8-Benzyl-4-methyl-2-[[methyl-[(2-propan-2-yloxyphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[[methyl-[(2-propoxyphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H32N4O2
8-Benzyl-4-methyl-2-[[methyl-[(2-propoxyphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-Fluorophenyl)methyl]-2-[[(2-methoxy-4-methylphenyl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H29FN4O2
8-[(4-Fluorophenyl)methyl]-2-[[(2-methoxy-4-methylphenyl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[[methyl-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6OS
8-Benzyl-4-methyl-2-[[methyl-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-2-[[[2-(dimethylamino)pyridin-3-yl]methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-Benzyl-2-[[[2-(dimethylamino)pyridin-3-yl]methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[[methyl-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H28N6O
8-Benzyl-4-methyl-2-[[methyl-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[[methyl-[(3R)-3-phenylbutyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H31FN4O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[[methyl-[(3R)-3-phenylbutyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[[methyl-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H30N4O2
8-benzyl-4-methyl-2-[[methyl-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-(3-chloro-4-methylphenyl)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H33Cl2F3N4O6S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-(3-chloro-4-methylphenyl)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[(4-Fluorophenyl)methyl]-4-methyl-2-[[methyl-[(2-methyl-1,3-thiazol-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C22H24FN5OS
8-[(4-Fluorophenyl)methyl]-4-methyl-2-[[methyl-[(2-methyl-1,3-thiazol-5-yl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-Fluorophenyl)methyl]-2-[[(2-methoxy-3-methylphenyl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H29FN4O2
8-[(4-Fluorophenyl)methyl]-2-[[(2-methoxy-3-methylphenyl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Benzyl-4-methyl-2-[[methyl(2-phenylethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N4O
8-Benzyl-4-methyl-2-[[methyl(2-phenylethyl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-Fluorophenyl)methyl]-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H27FN4O
8-[(4-Fluorophenyl)methyl]-4-methyl-2-[[methyl-[(2-methylphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-morpholin-4-ylsulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H31N5O4S
8-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-morpholin-4-ylsulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-morpholin-4-ylsulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H31N5O4S
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-morpholin-4-ylsulfonylpiperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-cyclopropyl-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C19H26N4O3
8-cyclopropyl-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[2-(1H-indol-3-yl)ethyl]-4-methyl-2-[[methyl(oxan-4-yl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31N5O2
8-[2-(1H-indol-3-yl)ethyl]-4-methyl-2-[[methyl(oxan-4-yl)amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(3-methoxypropyl)-4-methyl-2-[[methyl-[(E)-2-methyl-3-phenylprop-2-enyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N4O2
8-(3-methoxypropyl)-4-methyl-2-[[methyl-[(E)-2-methyl-3-phenylprop-2-enyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-4-methyl-2-[[methyl-[(4-pyrrolidin-1-ylphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H33N5O
8-(Cyclopropylmethyl)-4-methyl-2-[[methyl-[(4-pyrrolidin-1-ylphenyl)methyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(Cyclopropylmethyl)-2-[[[3-(3-fluorophenyl)phenyl]methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H29FN4O
8-(Cyclopropylmethyl)-2-[[[3-(3-fluorophenyl)phenyl]methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-Methoxy-2,3,5,6-tetrahydro-pyrido(3,2,1-IJ)quinoline-1,7-dione —— C13H13NO3
8-Methoxy-2,3,5,6-tetrahydro-pyrido(3,2,1-IJ)quinoline-1,7-dione
—— 8-(3-chlorophenyl)-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C46H35Cl2F3N4O6
8-(3-chlorophenyl)-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Cyclopropylmethyl)-2-[[(7-methoxy-1-benzofuran-2-yl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H28N4O3
8-(Cyclopropylmethyl)-2-[[(7-methoxy-1-benzofuran-2-yl)methyl-methylamino]methyl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(2,4-dichloroanilino)-6-(1-hydroxynaphthalen-2-yl)-6a-(4-methoxyphenyl)-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H35Cl2N3O6
8-(2,4-dichloroanilino)-6-(1-hydroxynaphthalen-2-yl)-6a-(4-methoxyphenyl)-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Cyclopropylmethyl)-4-methyl-2-[[methyl-[2-[3-(trifluoromethyl)phenoxy]ethyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27F3N4O2
8-(Cyclopropylmethyl)-4-methyl-2-[[methyl-[2-[3-(trifluoromethyl)phenoxy]ethyl]amino]methyl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(3-chlorophenyl)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(4-hydroxy-3,5-dimethylphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C48H42ClN5O5
8-(3-chlorophenyl)-2-[4-[[4-(dimethylamino)phenyl]diazenyl]phenyl]-6-(4-hydroxy-3,5-dimethylphenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-2-(4-ethenylphenyl)-6-(2-hydroxy-4-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H30ClFN2O6
8-(3-chloro-4-fluorophenyl)-2-(4-ethenylphenyl)-6-(2-hydroxy-4-methoxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(1-benzofuran-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]-1,6-naphthyridine-2-carboxamide —— C23H17N5O2
8-(1-benzofuran-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]-1,6-naphthyridine-2-carboxamide
—— 8,8-Dimethyl-2-(methylsulfanyl)-5-phenyl-3H,4H,5H,6H,7H,8H,9H,10H-pyrimido[4,5-B]quinoline-4,6-dione —— C20H21N3O2S
8,8-Dimethyl-2-(methylsulfanyl)-5-phenyl-3H,4H,5H,6H,7H,8H,9H,10H-pyrimido[4,5-B]quinoline-4,6-dione
—— 8-(3-chloro-4-fluorophenyl)-6-(2-hydroxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide —— C28H23ClFN3O6
8-(3-chloro-4-fluorophenyl)-6-(2-hydroxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide
—— 8-(3-chloro-4-fluorophenyl)-2-ethyl-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C30H25ClF4N2O6
8-(3-chloro-4-fluorophenyl)-2-ethyl-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(2,4-dichloroanilino)-6-(4-hydroxy-3,5-dimethoxyphenyl)-6a-(4-methoxyphenyl)-2-(4-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H34Cl2N4O10
8-(2,4-dichloroanilino)-6-(4-hydroxy-3,5-dimethoxyphenyl)-6a-(4-methoxyphenyl)-2-(4-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chlorophenyl)-6-(2-hydroxynaphthalen-1-yl)-2-(4-iodophenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H30ClIN2O5
8-(3-chlorophenyl)-6-(2-hydroxynaphthalen-1-yl)-2-(4-iodophenyl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone