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—— 8-[(4-Benzylpiperazin-1-yl)methyl]-7-[(4-chlorophenyl)methyl]-1,3-dimethylpurine-2,6-dione —— C26H29ClN6O2
8-[(4-Benzylpiperazin-1-yl)methyl]-7-[(4-chlorophenyl)methyl]-1,3-dimethylpurine-2,6-dione
—— 8-bromo-N-(4-chlorophenyl)-2-methyl-4-thioxo-3,4,5,6-tetrahydro-2H-2,6-methano-1,3,5-benzoxadiazocine-11-carboxamide —— C18H15BrClN3O2S
8-bromo-N-(4-chlorophenyl)-2-methyl-4-thioxo-3,4,5,6-tetrahydro-2H-2,6-methano-1,3,5-benzoxadiazocine-11-carboxamide
—— 8-cyclopropyl-4-(piperidin-1-yl)pyrido[2,3-d]pyrimidin-7(8H)-one —— C15H18N4O
8-cyclopropyl-4-(piperidin-1-yl)pyrido[2,3-d]pyrimidin-7(8H)-one
—— 8-cyclopropyl-4-methoxypyrido[2,3-d]pyrimidin-7(8H)-one —— C11H11N3O2
8-cyclopropyl-4-methoxypyrido[2,3-d]pyrimidin-7(8H)-one
—— 8-cyclopropyl-4-((2-hydroxyethyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one —— C12H14N4O2
8-cyclopropyl-4-((2-hydroxyethyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one
—— [8-(1,3-Benzodioxole-5-carbonyl)-1-thia-4,8-diazaspiro[4.5]decan-4-yl]-(4-bromophenyl)methanone —— C22H21BrN2O4S
[8-(1,3-Benzodioxole-5-carbonyl)-1-thia-4,8-diazaspiro[4.5]decan-4-yl]-(4-bromophenyl)methanone
—— 8-butyl-4-methoxypyrido[2,3-d]pyrimidin-7(8H)-one —— C12H15N3O2
8-butyl-4-methoxypyrido[2,3-d]pyrimidin-7(8H)-one
—— 8-cyclopropyl-4-morpholinopyrido[2,3-d]pyrimidin-7(8H)-one —— C14H16N4O2
8-cyclopropyl-4-morpholinopyrido[2,3-d]pyrimidin-7(8H)-one
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[3-methylbutyl(pentanoyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C27H38N2O7
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[3-methylbutyl(pentanoyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— 8-(Bromomethyl)-6a,9a-dichloro-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-(2-hydroxy-3-methylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C30H26BrCl2N5O9
8-(Bromomethyl)-6a,9a-dichloro-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-(2-hydroxy-3-methylphenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— [8-(2-Bromobenzoyl)-1-thia-4,8-diazaspiro[4.5]decan-4-yl]-(3-methylphenyl)methanone —— C22H23BrN2O2S
[8-(2-Bromobenzoyl)-1-thia-4,8-diazaspiro[4.5]decan-4-yl]-(3-methylphenyl)methanone
—— 8-(2,4-dichloroanilino)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-(4-methoxyphenyl)-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C46H37Cl2N3O7
8-(2,4-dichloroanilino)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-(4-methoxyphenyl)-2-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(4-hydroxy-3-iodo-5-methoxyphenyl)-6a-methyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C38H36ClIN4O6S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(4-hydroxy-3-iodo-5-methoxyphenyl)-6a-methyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-(2-hydroxy-3-prop-2-enylphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C38H33ClFN5O9
8-(3-chloro-4-fluorophenyl)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-(2-hydroxy-3-prop-2-enylphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chlorophenyl)-6-(4-hydroxynaphthalen-1-yl)-2-methyl-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H29ClN2O5
8-(3-chlorophenyl)-6-(4-hydroxynaphthalen-1-yl)-2-methyl-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-2-(4-ethylphenyl)-6-(4-hydroxynaphthalen-1-yl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C33H27BrCl2N2O5
8-(Bromomethyl)-6a,9a-dichloro-2-(4-ethylphenyl)-6-(4-hydroxynaphthalen-1-yl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(3-fluoro-2-hydroxyphenyl)-2-hydroxy-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C34H28ClFN4O6S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(3-fluoro-2-hydroxyphenyl)-2-hydroxy-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-2-(4-chlorophenyl)-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H27Cl2FN2O6
8-(3-chloro-4-fluorophenyl)-2-(4-chlorophenyl)-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-6-(3-fluoro-4-hydroxyphenyl)-2-hydroxy-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C27H21ClF2N2O6
8-(3-chloro-4-fluorophenyl)-6-(3-fluoro-4-hydroxyphenyl)-2-hydroxy-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-6-(2-hydroxy-3-methoxyphenyl)-2,6a-dimethyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H26ClFN2O6
8-(3-chloro-4-fluorophenyl)-6-(2-hydroxy-3-methoxyphenyl)-2,6a-dimethyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-2-ethyl-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C32H28ClFN2O6
8-(3-chloro-4-fluorophenyl)-2-ethyl-6-(6-hydroxy-4H-chromen-3-yl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-6-(4-hydroxy-3-iodo-5-methoxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide —— C29H24ClFIN3O7
8-(3-chloro-4-fluorophenyl)-6-(4-hydroxy-3-iodo-5-methoxyphenyl)-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide
—— 8-methyl-3-[[[2-methyl-1-[1-(oxolan-2-ylmethyl)tetrazol-5-yl]propyl]-(oxolan-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H36N6O3
8-methyl-3-[[[2-methyl-1-[1-(oxolan-2-ylmethyl)tetrazol-5-yl]propyl]-(oxolan-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[5-(hydroxymethyl)furan-2-yl]-6a-methyl-2-(4-morpholin-4-ylphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C43H40ClN5O7S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-[5-(hydroxymethyl)furan-2-yl]-6a-methyl-2-(4-morpholin-4-ylphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-6-(4-hydroxy-2,6-dimethoxyphenyl)-6a-methyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C34H30ClFN2O7S
8-(3-chloro-4-fluorophenyl)-6-(4-hydroxy-2,6-dimethoxyphenyl)-6a-methyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(bromomethyl)-6a,9a-dichloro-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(6-hydroxy-4H-chromen-3-yl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C31H23BrCl3F3N4O6
8-(bromomethyl)-6a,9a-dichloro-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-6-(6-hydroxy-4H-chromen-3-yl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(Bromomethyl)-6a,9a-dichloro-6-[4-(2-hydroxyethoxy)phenyl]-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H24BrCl2N3O8
8-(Bromomethyl)-6a,9a-dichloro-6-[4-(2-hydroxyethoxy)phenyl]-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-(4-ethenylphenyl)-6-(3-fluoro-4-hydroxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C42H34ClFN4O5S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-2-(4-ethenylphenyl)-6-(3-fluoro-4-hydroxyphenyl)-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(2,4-dichloroanilino)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-[2-(4-hydroxy-3-methoxyphenyl)ethenyl]-6a-(4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C44H38Cl2N6O11
8-(2,4-dichloroanilino)-2-[4-(dimethylamino)-3,5-dinitrophenyl]-6-[2-(4-hydroxy-3-methoxyphenyl)ethenyl]-6a-(4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chloro-4-fluorophenyl)-6-(4-hydroxy-3-methoxyphenyl)-2-[2-(4-hydroxyphenyl)ethyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H32ClFN2O7
8-(3-chloro-4-fluorophenyl)-6-(4-hydroxy-3-methoxyphenyl)-2-[2-(4-hydroxyphenyl)ethyl]-6a-methyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(3-chlorophenyl)-2-hydroxy-6-(6-hydroxy-4H-chromen-3-yl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C35H27ClN2O7
8-(3-chlorophenyl)-2-hydroxy-6-(6-hydroxy-4H-chromen-3-yl)-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— [8-(2-Chloro-6-methoxypyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-2-yl]-(2,3-dihydro-1,4-benzodioxin-3-yl)methanone —— C24H26ClN3O5
[8-(2-Chloro-6-methoxypyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-2-yl]-(2,3-dihydro-1,4-benzodioxin-3-yl)methanone
—— 8-(4-Chlorophenyl)sulfonyl-2-methyl-3-[3-(trifluoromethyl)phenyl]-1,4,8-triazaspiro[4.5]deca-1,3-diene —— C21H19ClF3N3O2S
8-(4-Chlorophenyl)sulfonyl-2-methyl-3-[3-(trifluoromethyl)phenyl]-1,4,8-triazaspiro[4.5]deca-1,3-diene
—— 8-(3-chloro-4-fluorophenyl)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-methyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H34ClFN2O6
8-(3-chloro-4-fluorophenyl)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-methyl-2-propyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(2-chloro-6-methoxypyridine-4-carbonyl)-N-[3-(diethylamino)propyl]-2,8-diazaspiro[4.5]decane-2-carbothioamide —— C23H36ClN5O2S
8-(2-chloro-6-methoxypyridine-4-carbonyl)-N-[3-(diethylamino)propyl]-2,8-diazaspiro[4.5]decane-2-carbothioamide
—— 8-Nitro-5-pyridin-2-yl-1,2,3,4,4a,6-hexahydrobenzo[c]quinolizine-5-carbonitrile —— C19H18N4O2
8-Nitro-5-pyridin-2-yl-1,2,3,4,4a,6-hexahydrobenzo[c]quinolizine-5-carbonitrile
—— 8-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-N-[2-fluoro-3-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decane-2-carboxamide —— C22H24F4N4O3
8-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-N-[2-fluoro-3-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decane-2-carboxamide
—— 8-ethoxy-N-[2-(2-ethoxyphenyl)ethyl]quinoline-5-sulfonamide —— C21H24N2O4S
8-ethoxy-N-[2-(2-ethoxyphenyl)ethyl]quinoline-5-sulfonamide
—— 8-(2,4-dichloroanilino)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-(4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H33Cl2N3O7
8-(2,4-dichloroanilino)-6-(2-hydroxy-4-phenylmethoxyphenyl)-6a-(4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-(2,5-dimethylphenyl)sulfonyl-N-(2-methyl-6-propan-2-ylphenyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide —— C27H37N3O2S2
8-(2,5-dimethylphenyl)sulfonyl-N-(2-methyl-6-propan-2-ylphenyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide
—— 8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(4-hydroxy-3-iodo-5-methoxyphenyl)-6a-methyl-2-(3-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H33ClIN5O8S
8-[5-(5-chloro-3-methyl-1-benzothiophen-2-yl)-2-methylpyrazol-3-yl]-6-(4-hydroxy-3-iodo-5-methoxyphenyl)-6a-methyl-2-(3-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 8-[3-(2-ethoxyphenyl)prop-2-enoyl]-N-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide —— C25H35N3O3S
8-[3-(2-ethoxyphenyl)prop-2-enoyl]-N-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decane-2-carbothioamide
—— (8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-[4-[1-[(2-methyl-1,3-thiazol-4-yl)methyl]imidazol-2-yl]piperidin-1-yl]methanone —— C25H30N4O2S
(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-[4-[1-[(2-methyl-1,3-thiazol-4-yl)methyl]imidazol-2-yl]piperidin-1-yl]methanone
—— 8-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2-[(2-methoxyphenyl)methylidene]-7,9-dihydrofuro[2,3-f][1,3]benzoxazin-3-one;1,4-dioxane —— C30H29NO8
8-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2-[(2-methoxyphenyl)methylidene]-7,9-dihydrofuro[2,3-f][1,3]benzoxazin-3-one;1,4-dioxane
—— 8-[(2-chlorophenyl)methyl]-2-(pyridin-3-ylmethylidene)-7,9-dihydrofuro[2,3-f][1,3]benzoxazin-3-one;1,4-dioxane —— C27H25ClN2O5
8-[(2-chlorophenyl)methyl]-2-(pyridin-3-ylmethylidene)-7,9-dihydrofuro[2,3-f][1,3]benzoxazin-3-one;1,4-dioxane
—— 8-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyridin-3-ylmethylidene)-7,9-dihydrofuro[2,3-f][1,3]benzoxazin-3-one;1,4-dioxane —— C28H26N2O7
8-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyridin-3-ylmethylidene)-7,9-dihydrofuro[2,3-f][1,3]benzoxazin-3-one;1,4-dioxane
—— 8-[2-[(2-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]-7-(2-hydroxypropyl)-3-methylpurine-2,6-dione —— C16H18N6O5
8-[2-[(2-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]-7-(2-hydroxypropyl)-3-methylpurine-2,6-dione
—— 8-[(3,5-Dimethylpiperidin-1-yl)sulfonyl]quinoline —— C16H20N2O2S
8-[(3,5-Dimethylpiperidin-1-yl)sulfonyl]quinoline
—— 8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[3-methylbutyl(oxolane-2-carbonyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide —— C27H36N2O8
8-formyl-4-hydroxy-N-(2-hydroxyethyl)-6-methoxy-3-[3-methylbutyl(oxolane-2-carbonyl)amino]-3,4,4a,9b-tetrahydrodibenzofuran-1-carboxamide
—— 8-Thiophen-2-ylsulfonyl-8-azabicyclo[3.2.1]octan-3-ol —— C11H15NO3S2
8-Thiophen-2-ylsulfonyl-8-azabicyclo[3.2.1]octan-3-ol