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—— 8-[(3-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(3-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(3-fluorophenyl)methyl]-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H36N4O3
8-(cyclohexylmethyl)-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2S)-1-(2-oxo-2-piperidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2S)-1-(2-oxo-2-piperidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-oxo-2-pyrazol-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-oxo-2-pyrazol-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-oxo-2-piperidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H33N5O2
8-benzyl-4-methyl-2-[(2R)-1-(2-oxo-2-piperidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H36N4O3
8-(cyclohexylmethyl)-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N6O2
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-propan-2-yloxyacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H36N4O3
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-propan-2-yloxyacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(oxan-4-yl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H26N6O2
8-benzyl-4-methyl-2-[(2R)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H30N4O3
8-benzyl-2-[(2S)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H37N5O2
8-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(2-oxo-2-pyrrolidin-1-ylethyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H30N4O2
8-benzyl-2-[(2S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-propan-2-yloxyacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-propan-2-yloxyacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2R)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H39N5O2
8-(cyclohexylmethyl)-2-[(2R)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propan-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N4O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propan-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H34N6O
8-(cyclohexylmethyl)-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(2-fluorophenyl)methyl]-2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O3
8-[(4-fluorophenyl)methyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(2R)-1-(2-pyrrolidin-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H31N5O2
8-benzyl-4-methyl-2-[(2R)-1-(2-pyrrolidin-1-ylacetyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H39N5O2
8-(cyclohexylmethyl)-2-[(2S)-1-[2-(diethylamino)acetyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H29FN4O
8-(cyclopropylmethyl)-2-[(2R)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[2-(3-oxopiperazin-1-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O3
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[2-(3-oxopiperazin-1-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(3R)-1-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(cyclopropylmethyl)-2-[(3R)-1-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-2-[(2R)-1-(2-methoxy-3-methylbenzoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C26H32N4O3
8-(cyclopropylmethyl)-2-[(2R)-1-(2-methoxy-3-methylbenzoyl)piperidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C27H30N4O2
8-benzyl-2-[(2R)-1-[(4-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(3S)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H32N4O3
8-benzyl-2-[(3S)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H29N5O2S
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(thiadiazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H24N6O2S
8-benzyl-4-methyl-2-[(3S)-1-(thiadiazole-4-carbonyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3R)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(3R)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H32N6O2
8-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H27FN4O2
8-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[2-(4-methylpiperidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H37N5O2
8-(cyclopropylmethyl)-4-methyl-2-[(2R)-1-[2-(4-methylpiperidin-1-yl)acetyl]piperidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-[2-(3-oxopiperazin-1-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H32N6O3
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-[2-(3-oxopiperazin-1-yl)acetyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-[(2-methylpyrazol-3-yl)methyl]pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-2-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H30N6O
8-benzyl-2-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-benzyl-4-methyl-2-[(3S)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H28N6O2
8-benzyl-4-methyl-2-[(3S)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclohexylmethyl)-2-[(2S)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C25H36N6O
8-(cyclohexylmethyl)-2-[(2S)-1-[(1-ethylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H27FN6O
8-[(2-fluorophenyl)methyl]-2-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propan-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N4O2
8-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propan-2-ylpyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C24H25FN6O2
8-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C23H30N6O3
8-(cyclopropylmethyl)-4-methyl-2-[(3R)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one
—— 8-(5-bromo-2-hydroxyphenyl)-7-ethenyl-2,3,8a-trimethyl-5,8-dihydro-4aH-naphthalene-1,4-dione —— C21H21BrO3
8-(5-bromo-2-hydroxyphenyl)-7-ethenyl-2,3,8a-trimethyl-5,8-dihydro-4aH-naphthalene-1,4-dione
—— 8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one —— C21H28N6O3S
8-(cyclopropylmethyl)-4-methyl-2-[(3S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]-5,6-dihydropyrido[2,3-d]pyrimidin-7-one