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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R,9R)-6-(5-bromo-2-methoxyphenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H22BrClN2O2
(6R,9R)-6-(5-bromo-2-methoxyphenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[(4S)-6-methoxy-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one —— C18H20N4O4
6-[(4S)-6-methoxy-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one
—— (6R)-2-cyclopropyl-8-(4-prop-2-enylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N2O2
(6R)-2-cyclopropyl-8-(4-prop-2-enylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-methyl-1,3-oxazole-4-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N3O3
(6R)-8-(5-methyl-1,3-oxazole-4-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O2
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H26N4O2
6-methyl-N-[1-[[(2R)-oxolan-2-yl]methyl]piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— (6S)-1-methyl-4-[4-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H28N6O
(6S)-1-methyl-4-[4-(methylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R,9S)-9-(4-methoxyphenyl)-6-(2-phenylmethoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C33H30N2O3
(6R,9S)-9-(4-methoxyphenyl)-6-(2-phenylmethoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[(3S)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]-N-methylpyridine-2-carboxamide —— C19H23N3O2
6-[(3S)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]-N-methylpyridine-2-carboxamide
—— (6R)-N-(2-chlorophenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C18H25ClN4O2
(6R)-N-(2-chlorophenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-[3-(tetrazol-1-yl)propyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H31N7O
(6S)-10-(cyclopropylmethyl)-1-methyl-4-[3-(tetrazol-1-yl)propyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(4R)-6-methoxy-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one —— C18H20N4O4
6-[(4R)-6-methoxy-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one
—— 6-methyl-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H26N4O2
6-methyl-N-[1-[[(2S)-oxolan-2-yl]methyl]piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-1,3-dihydroimidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N6O3
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-1,3-dihydroimidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-1,10-dimethyl-4-(2-thiophen-2-ylacetyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N3O2S
(6R)-1,10-dimethyl-4-(2-thiophen-2-ylacetyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-2-cyclopropyl-8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N2O3
(6R)-2-cyclopropyl-8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[(2E)-3,7-dimethylocta-2,6-dienyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H35N3O
(6S)-4-[(2E)-3,7-dimethylocta-2,6-dienyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-methyl-2-[[[(1S)-2-methyl-1-pyridin-2-ylpropyl]amino]methyl]-1H-quinolin-4-one —— C20H23N3O
6-methyl-2-[[[(1S)-2-methyl-1-pyridin-2-ylpropyl]amino]methyl]-1H-quinolin-4-one
—— 6-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine —— C18H21N7
6-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine
—— (6S)-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N6O
(6S)-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-N-(2-chlorophenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C18H25ClN4O2
(6S)-N-(2-chlorophenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— 6-[4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C21H28N4O3
6-[4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-1,10-dimethyl-4-(2-thiophen-2-ylacetyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N3O2S
(6S)-1,10-dimethyl-4-(2-thiophen-2-ylacetyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N6O
(6R)-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-(cyclopropylmethyl)-4-ethylsulfonyl-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H29N3O3S
(6S)-10-(cyclopropylmethyl)-4-ethylsulfonyl-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethylamino)-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C19H19N5O
6-[4-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethylamino)-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-methyl-2-[[[(1R)-2-methyl-1-pyridin-2-ylpropyl]amino]methyl]-1H-quinolin-4-one —— C20H23N3O
6-methyl-2-[[[(1R)-2-methyl-1-pyridin-2-ylpropyl]amino]methyl]-1H-quinolin-4-one
—— (6R,9R)-9-(4-methoxyphenyl)-6-naphthalen-1-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C30H26N2O2
(6R,9R)-9-(4-methoxyphenyl)-6-naphthalen-1-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine —— C18H21N7
6-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine
—— (6R,9S)-6-[4-(diethylamino)phenyl]-9-phenyl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C29H31N3O
(6R,9S)-6-[4-(diethylamino)phenyl]-9-phenyl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-10-ethyl-1-methyl-4-(3-pyridin-4-ylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H30N4O2
(6R)-10-ethyl-1-methyl-4-(3-pyridin-4-ylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-10-ethyl-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H26N4O2
(6R)-10-ethyl-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-[(4-ethoxyphenyl)methyl]-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C22H33N3O2
(6S)-4-[(4-ethoxyphenyl)methyl]-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-1-methyl-4-(3-phenylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H27N3O2
(6S)-1-methyl-4-(3-phenylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-1-methyl-4-(3-phenylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H27N3O2
(6R)-1-methyl-4-(3-phenylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S,9S)-6-[4-(diethylamino)phenyl]-9-phenyl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C29H31N3O
(6S,9S)-6-[4-(diethylamino)phenyl]-9-phenyl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-4-[2-(2,3-dimethylphenoxy)ethyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H33N3O2
(6S)-4-[2-(2,3-dimethylphenoxy)ethyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-10-ethyl-1-methyl-4-[[3-(trifluoromethyl)phenyl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H28F3N3O
(6R)-10-ethyl-1-methyl-4-[[3-(trifluoromethyl)phenyl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R,9R)-6-(3-bromophenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H20BrClN2O
(6R,9R)-6-(3-bromophenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-1-methyl-4-(5-methyl-2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C14H22N6O2
(6S)-1-methyl-4-(5-methyl-2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-1-methyl-4-(5-methyl-2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C14H22N6O2
(6R)-1-methyl-4-(5-methyl-2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-2-cyclopropyl-8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N2O3
(6S)-2-cyclopropyl-8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-3-acetyl-2-[4-(dimethylamino)phenyl]-4-hydroxy-5-oxo-2H-pyrrol-1-yl]hexanoic acid —— C20H26N2O5
6-[(2R)-3-acetyl-2-[4-(dimethylamino)phenyl]-4-hydroxy-5-oxo-2H-pyrrol-1-yl]hexanoic acid
—— 6-[6-methyl-4-(2-pyrrolidin-1-ylethylamino)-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H22N4O
6-[6-methyl-4-(2-pyrrolidin-1-ylethylamino)-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H31N3O2
(6S)-4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-(4-cyclopentylpyrimidin-2-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H29N5O
(6S)-4-(4-cyclopentylpyrimidin-2-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-2-cyclopropyl-8-[2-[(4-fluorophenyl)methyl-methylamino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H30FN3O2
(6R)-2-cyclopropyl-8-[2-[(4-fluorophenyl)methyl-methylamino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-ethyl-1-methyl-4-(3-pyridin-4-ylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H30N4O2
(6S)-10-ethyl-1-methyl-4-(3-pyridin-4-ylpropanoyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-ethyl-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H26N4O2
(6S)-10-ethyl-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]hexanoic acid —— C15H19NO4
6-[(1R,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]hexanoic acid