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—— 6-(4-ethylpiperazin-1-yl)-4-methyl-2-oxo-5-[(Z)-[4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1-propylpyridine-3-carbonitrile —— C28H33N5O2S2
6-(4-ethylpiperazin-1-yl)-4-methyl-2-oxo-5-[(Z)-[4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1-propylpyridine-3-carbonitrile
—— 6-[(5Z)-5-[[5-cyano-2-(3-ethoxycarbonylpiperidin-1-yl)-1,4-dimethyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C26H32N4O6S2
6-[(5Z)-5-[[5-cyano-2-(3-ethoxycarbonylpiperidin-1-yl)-1,4-dimethyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-[(5Z)-5-[[5-cyano-2-(4-ethylpiperazin-1-yl)-1,4-dimethyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C24H31N5O4S2
6-[(5Z)-5-[[5-cyano-2-(4-ethylpiperazin-1-yl)-1,4-dimethyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— (6,8-dichloro-3,4-dihydro-1H-isoquinolin-2-yl)-[(2R)-4-methylmorpholin-2-yl]methanone —— C15H18Cl2N2O2
(6,8-dichloro-3,4-dihydro-1H-isoquinolin-2-yl)-[(2R)-4-methylmorpholin-2-yl]methanone
—— 6-chloro-8-[[(S)-[3-(trifluoromethyl)phenyl]methylsulfinyl]methyl]-3,4-dihydro-2H-1,5-benzodioxepine —— C18H16ClF3O3S
6-chloro-8-[[(S)-[3-(trifluoromethyl)phenyl]methylsulfinyl]methyl]-3,4-dihydro-2H-1,5-benzodioxepine
—— 6-(3,5-dimethylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-(4-oxo-3-propyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile —— C22H28N4O2S2
6-(3,5-dimethylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-(4-oxo-3-propyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile
—— 6-(3,5-dimethylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-[4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile —— C27H30N4O2S2
6-(3,5-dimethylpiperidin-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-[4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile
—— 6-(4-benzylpiperazin-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-[4-oxo-3-(1-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile —— C31H31N5O2S2
6-(4-benzylpiperazin-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-[4-oxo-3-(1-phenylethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile
—— 6-(3,5-dimethylpiperidin-1-yl)-1-ethyl-4-methyl-2-oxo-5-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile —— C25H34N4O2S2
6-(3,5-dimethylpiperidin-1-yl)-1-ethyl-4-methyl-2-oxo-5-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile
—— 6-(4-ethylpiperazin-1-yl)-4-methyl-5-[(Z)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-oxo-1-propylpyridine-3-carbonitrile —— C28H33N5O2S2
6-(4-ethylpiperazin-1-yl)-4-methyl-5-[(Z)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-oxo-1-propylpyridine-3-carbonitrile
—— 6-(3,5-dimethylpiperidin-1-yl)-4-methyl-5-[(Z)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-oxo-1-propylpyridine-3-carbonitrile —— C29H34N4O2S2
6-(3,5-dimethylpiperidin-1-yl)-4-methyl-5-[(Z)-[3-[(4-methylphenyl)methyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-oxo-1-propylpyridine-3-carbonitrile
—— 6-methyl-4-oxo-N-[(5R)-2,3,4,5-tetrahydrobenzo[i][1]benzoxepin-5-yl]-1H-pyridine-3-carboxamide —— C21H20N2O3
6-methyl-4-oxo-N-[(5R)-2,3,4,5-tetrahydrobenzo[i][1]benzoxepin-5-yl]-1H-pyridine-3-carboxamide
—— 6-methyl-4-oxo-N-[(5S)-2,3,4,5-tetrahydrobenzo[i][1]benzoxepin-5-yl]-1H-pyridine-3-carboxamide —— C21H20N2O3
6-methyl-4-oxo-N-[(5S)-2,3,4,5-tetrahydrobenzo[i][1]benzoxepin-5-yl]-1H-pyridine-3-carboxamide
—— 6-(4-benzylpiperazin-1-yl)-4-methyl-2-oxo-5-[(Z)-(4-oxo-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-propylpyridine-3-carbonitrile —— C28H33N5O2S2
6-(4-benzylpiperazin-1-yl)-4-methyl-2-oxo-5-[(Z)-(4-oxo-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-propylpyridine-3-carbonitrile
—— 6-[4-(2-fluorophenyl)piperazin-1-yl]-1,4-dimethyl-5-[(Z)-(3-octyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-2-oxopyridine-3-carbonitrile —— C30H36FN5O2S2
6-[4-(2-fluorophenyl)piperazin-1-yl]-1,4-dimethyl-5-[(Z)-(3-octyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-2-oxopyridine-3-carbonitrile
—— 6-[(5Z)-5-[[5-cyano-2-(3,5-dimethylpiperidin-1-yl)-1,4-dimethyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C25H32N4O4S2
6-[(5Z)-5-[[5-cyano-2-(3,5-dimethylpiperidin-1-yl)-1,4-dimethyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-(azepan-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-[4-oxo-3-(oxolan-2-ylmethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile —— C23H28N4O3S2
6-(azepan-1-yl)-1,4-dimethyl-2-oxo-5-[(Z)-[4-oxo-3-(oxolan-2-ylmethyl)-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]pyridine-3-carbonitrile
—— 6-(4-benzylpiperazin-1-yl)-1-ethyl-4-methyl-2-oxo-5-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile —— C29H35N5O2S2
6-(4-benzylpiperazin-1-yl)-1-ethyl-4-methyl-2-oxo-5-[(Z)-(4-oxo-3-pentyl-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]pyridine-3-carbonitrile
—— 6-(4-benzylpiperazin-1-yl)-5-[(Z)-[3-(2-ethylhexyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-methyl-2-oxo-1-propylpyridine-3-carbonitrile —— C33H43N5O2S2
6-(4-benzylpiperazin-1-yl)-5-[(Z)-[3-(2-ethylhexyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-4-methyl-2-oxo-1-propylpyridine-3-carbonitrile
—— 6-(4-benzylpiperazin-1-yl)-1-ethyl-5-[(Z)-(3-ethyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-4-methyl-2-oxopyridine-3-carbonitrile —— C26H29N5O2S2
6-(4-benzylpiperazin-1-yl)-1-ethyl-5-[(Z)-(3-ethyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-4-methyl-2-oxopyridine-3-carbonitrile
—— 6-(4-benzylpiperazin-1-yl)-5-[(Z)-[3-(3-ethoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1-ethyl-4-methyl-2-oxopyridine-3-carbonitrile —— C29H35N5O3S2
6-(4-benzylpiperazin-1-yl)-5-[(Z)-[3-(3-ethoxypropyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1-ethyl-4-methyl-2-oxopyridine-3-carbonitrile
—— (6,8-dichloro-3,4-dihydro-1H-isoquinolin-2-yl)-[(2S)-4-methylmorpholin-2-yl]methanone —— C15H18Cl2N2O2
(6,8-dichloro-3,4-dihydro-1H-isoquinolin-2-yl)-[(2S)-4-methylmorpholin-2-yl]methanone
—— 6-(4-benzylpiperazin-1-yl)-1-ethyl-4-methyl-5-[(Z)-(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-2-oxopyridine-3-carbonitrile —— C25H27N5O2S2
6-(4-benzylpiperazin-1-yl)-1-ethyl-4-methyl-5-[(Z)-(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-2-oxopyridine-3-carbonitrile
—— 6-(4-benzylpiperazin-1-yl)-5-[(Z)-[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile —— C33H35N5O4S2
6-(4-benzylpiperazin-1-yl)-5-[(Z)-[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile
—— 6-(2,6-dimethylmorpholin-4-yl)-5-[(Z)-[3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile —— C29H30N6O4S2
6-(2,6-dimethylmorpholin-4-yl)-5-[(Z)-[3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile
—— 6-[(5Z)-5-[[5-cyano-2-(4-ethoxycarbonylpiperidin-1-yl)-1-ethyl-4-methyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C27H34N4O6S2
6-[(5Z)-5-[[5-cyano-2-(4-ethoxycarbonylpiperidin-1-yl)-1-ethyl-4-methyl-6-oxopyridin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-chloro-8-[[(R)-[3-(trifluoromethyl)phenyl]methylsulfinyl]methyl]-3,4-dihydro-2H-1,5-benzodioxepine —— C18H16ClF3O3S
6-chloro-8-[[(R)-[3-(trifluoromethyl)phenyl]methylsulfinyl]methyl]-3,4-dihydro-2H-1,5-benzodioxepine
—— 6-(4-benzylpiperidin-1-yl)-5-[(Z)-[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile —— C34H36N4O4S2
6-(4-benzylpiperidin-1-yl)-5-[(Z)-[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-1,4-dimethyl-2-oxopyridine-3-carbonitrile
—— 6-(4-ethylpiperazin-1-yl)-1,4-dimethyl-5-[(Z)-(3-octyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-2-oxopyridine-3-carbonitrile —— C26H37N5O2S2
6-(4-ethylpiperazin-1-yl)-1,4-dimethyl-5-[(Z)-(3-octyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-2-oxopyridine-3-carbonitrile
—— (6Z)-6-(4-{2-[4-(butan-2-yl)phenoxy]ethoxy}-3-ethoxybenzylidene)-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H34N4O4S
(6Z)-6-(4-{2-[4-(butan-2-yl)phenoxy]ethoxy}-3-ethoxybenzylidene)-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[(2-phenylsulfanylethylamino)methylidene]cyclohexa-2,4-dien-1-one —— C15H15NOS
(6E)-6-[(2-phenylsulfanylethylamino)methylidene]cyclohexa-2,4-dien-1-one
—— (6,9-dihydroxy-5,8a-dimethyl-1-methylidene-2-oxo-4,5,5a,6,7,8,9,9a-octahydro-3aH-azuleno[6,7-b]furan-8-yl) (E)-2-methylbut-2-enoate —— C20H28O6
(6,9-dihydroxy-5,8a-dimethyl-1-methylidene-2-oxo-4,5,5a,6,7,8,9,9a-octahydro-3aH-azuleno[6,7-b]furan-8-yl) (E)-2-methylbut-2-enoate
—— (6Z)-6-[4-(benzyloxy)-3-bromo-5-methoxybenzylidene]-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H21BrN4O3S
(6Z)-6-[4-(benzyloxy)-3-bromo-5-methoxybenzylidene]-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-6-{[1-(naphthalen-1-ylmethyl)-1H-pyrrol-2-yl]methylidene}-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H14F3N5OS
(6Z)-5-imino-6-{[1-(naphthalen-1-ylmethyl)-1H-pyrrol-2-yl]methylidene}-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-6-{4-[(2-methylbenzyl)oxy]benzylidene}-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H27N5O3S
(6Z)-5-imino-6-{4-[(2-methylbenzyl)oxy]benzylidene}-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-(butylaminomethylidene)-3-methoxycyclohexa-2,4-dien-1-one —— C12H17NO2
(6E)-6-(butylaminomethylidene)-3-methoxycyclohexa-2,4-dien-1-one
—— 6,8-dichloro-3-[2-[(S)-(2,5-dichlorophenyl)sulfinyl]ethylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine —— C14H9Cl4N3OS2
6,8-dichloro-3-[2-[(S)-(2,5-dichlorophenyl)sulfinyl]ethylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine
—— 6,8-dichloro-3-[2-[(R)-(2,5-dichlorophenyl)sulfinyl]ethylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine —— C14H9Cl4N3OS2
6,8-dichloro-3-[2-[(R)-(2,5-dichlorophenyl)sulfinyl]ethylsulfanyl]-[1,2,4]triazolo[4,3-a]pyridine
—— (6E)-6-(3H-1,3-benzoxazol-2-ylidene)-4-[[5-(3-methylphenyl)furan-2-yl]methylideneamino]cyclohexa-2,4-dien-1-one —— C25H18N2O3
(6E)-6-(3H-1,3-benzoxazol-2-ylidene)-4-[[5-(3-methylphenyl)furan-2-yl]methylideneamino]cyclohexa-2,4-dien-1-one
—— [(6Z,10E)-9-acetyloxy-5-hydroxy-6,10-dimethyl-3-methylidene-2-oxo-3a,4,5,8,9,11a-hexahydrocyclodeca[b]furan-4-yl] 2-methylbutanoate —— C22H30O7
[(6Z,10E)-9-acetyloxy-5-hydroxy-6,10-dimethyl-3-methylidene-2-oxo-3a,4,5,8,9,11a-hexahydrocyclodeca[b]furan-4-yl] 2-methylbutanoate
—— (6Z)-4-methyl-6-[1-(2-phenylhydrazinyl)ethylidene]cyclohexa-2,4-dien-1-one —— C15H16N2O
(6Z)-4-methyl-6-[1-(2-phenylhydrazinyl)ethylidene]cyclohexa-2,4-dien-1-one
—— 6-tert-butyl-8-[(Z)-[4-[(4-chlorophenyl)methoxy]phenyl]methylideneamino]-[1,2,4]triazolo[4,3-b][1,2,4]triazin-7-one —— C22H21ClN6O2
6-tert-butyl-8-[(Z)-[4-[(4-chlorophenyl)methoxy]phenyl]methylideneamino]-[1,2,4]triazolo[4,3-b][1,2,4]triazin-7-one
—— (6Z)-5-imino-6-[[2-methyl-1-[2-(4-methylphenoxy)ethyl]indol-3-yl]methylidene]-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H27N5O2S
(6Z)-5-imino-6-[[2-methyl-1-[2-(4-methylphenoxy)ethyl]indol-3-yl]methylidene]-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{[1-(4-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-methyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H21N5O2S
(6Z)-6-{[1-(4-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-methyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(5-bromofuran-2-yl)prop-2-enoate —— C16H12BrNO7
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(5-bromofuran-2-yl)prop-2-enoate
—— (6E)-3-(3,4-dimethoxyphenyl)-6-[(2-methoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C20H17N3O4S
(6E)-3-(3,4-dimethoxyphenyl)-6-[(2-methoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-nitro-2-[(E)-2-[3-[(E)-2-(6-nitro-1,3-benzothiazol-2-yl)ethenyl]phenyl]ethenyl]-1,3-benzothiazole —— C24H14N4O4S2
6-nitro-2-[(E)-2-[3-[(E)-2-(6-nitro-1,3-benzothiazol-2-yl)ethenyl]phenyl]ethenyl]-1,3-benzothiazole
—— 6-{[1-(3-chloro-4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylene}-5-imino-2-pentyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H26ClN5O2S
6-{[1-(3-chloro-4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylene}-5-imino-2-pentyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[(2,6-dichlorophenyl)methylidene]-3-(3,4,5-trimethoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C20H15Cl2N3O4S
(6Z)-6-[(2,6-dichlorophenyl)methylidene]-3-(3,4,5-trimethoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— (6E)-4-chloro-6-[[4-chloro-3-(6-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C21H14Cl2N2O2
(6E)-4-chloro-6-[[4-chloro-3-(6-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one