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—— (6S)-2-methyl-N-[(1S,3S)-3-methylsulfanylcyclohexyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C18H24F3N3OS
(6S)-2-methyl-N-[(1S,3S)-3-methylsulfanylcyclohexyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— (6S)-2-methyl-N-[4-(5-propan-2-yl-1,3-oxazol-2-yl)phenyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C23H23F3N4O2
(6S)-2-methyl-N-[4-(5-propan-2-yl-1,3-oxazol-2-yl)phenyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— (6R)-2-methyl-N-[(1S)-1-(1-propan-2-ylbenzimidazol-2-yl)ethyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C23H26F3N5O
(6R)-2-methyl-N-[(1S)-1-(1-propan-2-ylbenzimidazol-2-yl)ethyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— 6-(4-bromophenoxy)-N-[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]pyridine-3-carboxamide —— C17H15BrN4O3
6-(4-bromophenoxy)-N-[(1S)-1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]pyridine-3-carboxamide
—— (6R)-N-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-2-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C20H20F5N3O3
(6R)-N-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-2-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— (6E)-6-[4-(2-fluorophenoxy)-1H-quinazolin-2-ylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C21H15FN2O3
(6E)-6-[4-(2-fluorophenoxy)-1H-quinazolin-2-ylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-tert-butyl-N-[[(2S)-1,4-dioxan-2-yl]methyl]-1H-indole-2-carboxamide —— C18H24N2O3
6-tert-butyl-N-[[(2S)-1,4-dioxan-2-yl]methyl]-1H-indole-2-carboxamide
—— (6R)-2-methyl-N-[4-(5-propan-2-yl-1,3-oxazol-2-yl)phenyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C23H23F3N4O2
(6R)-2-methyl-N-[4-(5-propan-2-yl-1,3-oxazol-2-yl)phenyl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— (6E)-5-imino-6-{[1-(naphthalen-1-ylmethyl)-1H-indol-3-yl]methylidene}-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H23N5OS
(6E)-5-imino-6-{[1-(naphthalen-1-ylmethyl)-1H-indol-3-yl]methylidene}-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[5-(3-chlorophenyl)furan-2-yl]methylidene}-5-imino-2-methyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C18H12ClN3O2S
(6E)-6-{[5-(3-chlorophenyl)furan-2-yl]methylidene}-5-imino-2-methyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-6-[[1-(2-methoxy-5-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-methylpropyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H27N5O2S
(6Z)-5-imino-6-[[1-(2-methoxy-5-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-methylpropyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[2-(6-morpholin-4-ylpyridazin-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C15H17N5O2
(6Z)-6-[[2-(6-morpholin-4-ylpyridazin-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-[(2-hydroxy-4-methylanilino)methylidene]-4-methyl-2-nitrocyclohexa-2,4-dien-1-one —— C15H14N2O4
(6E)-6-[(2-hydroxy-4-methylanilino)methylidene]-4-methyl-2-nitrocyclohexa-2,4-dien-1-one
—— (6Z)-6-[[4-[2-(4-butan-2-ylphenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-imino-2-(phenoxymethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C32H32N4O5S
(6Z)-6-[[4-[2-(4-butan-2-ylphenoxy)ethoxy]-3-methoxyphenyl]methylidene]-5-imino-2-(phenoxymethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-4-chloro-6-[5-(4-methoxyphenyl)pyrazolidin-3-ylidene]cyclohexa-2,4-dien-1-one —— C16H15ClN2O2
(6Z)-4-chloro-6-[5-(4-methoxyphenyl)pyrazolidin-3-ylidene]cyclohexa-2,4-dien-1-one
—— (6E)-4-chloro-2-methoxy-6-[(2-methylanilino)methylidene]cyclohexa-2,4-dien-1-one —— C15H14ClNO2
(6E)-4-chloro-2-methoxy-6-[(2-methylanilino)methylidene]cyclohexa-2,4-dien-1-one
—— (6R)-N-[(5-methylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H16N6
(6R)-N-[(5-methylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6E)-2-heptyl-5-imino-6-[[1-[(2-methylphenyl)methyl]indol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H31N5OS
(6E)-2-heptyl-5-imino-6-[[1-[(2-methylphenyl)methyl]indol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[4-(4-methylpiperidin-1-yl)sulfonylanilino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C19H21N3O5S
(6E)-6-[[4-(4-methylpiperidin-1-yl)sulfonylanilino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6S)-N-[(5-methylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H16N6
(6S)-N-[(5-methylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6Z)-2-butyl-6-[3-ethoxy-4-(2-phenoxyethoxy)benzylidene]-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N4O4S
(6Z)-2-butyl-6-[3-ethoxy-4-(2-phenoxyethoxy)benzylidene]-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-methylpyrazol-1-yl)-N-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridazin-3-amine —— C15H19F3N6
6-(3-methylpyrazol-1-yl)-N-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridazin-3-amine
—— (6R)-3-methyl-N-[4-(8-methylimidazo[1,2-a]pyridin-2-yl)phenyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C22H22N6O
(6R)-3-methyl-N-[4-(8-methylimidazo[1,2-a]pyridin-2-yl)phenyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-2-methylsulfanyl-5,6,7,8-tetrahydroquinazoline-6-carboxylic acid —— C10H12N2O2S
(6R)-2-methylsulfanyl-5,6,7,8-tetrahydroquinazoline-6-carboxylic acid
—— 6-tert-butyl-2-[(2R)-1,4-dithian-2-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C14H18N2OS3
6-tert-butyl-2-[(2R)-1,4-dithian-2-yl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (6S)-2-methylsulfanyl-5,6,7,8-tetrahydroquinazoline-6-carboxylic acid —— C10H12N2O2S
(6S)-2-methylsulfanyl-5,6,7,8-tetrahydroquinazoline-6-carboxylic acid
—— 6-(3-methylpyrazol-1-yl)-N-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridazin-3-amine —— C15H19F3N6
6-(3-methylpyrazol-1-yl)-N-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridazin-3-amine
—— (6S)-3-methyl-N-[4-(8-methylimidazo[1,2-a]pyridin-2-yl)phenyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C22H22N6O
(6S)-3-methyl-N-[4-(8-methylimidazo[1,2-a]pyridin-2-yl)phenyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6Z)-6-[(3-hydroxyanilino)methylidene]cyclohexa-2,4-dien-1-one —— C13H11NO2
(6Z)-6-[(3-hydroxyanilino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-(3-methylpyrazol-1-yl)-N-[(9R)-6-oxaspiro[4.5]decan-9-yl]pyridazin-3-amine —— C17H23N5O
6-(3-methylpyrazol-1-yl)-N-[(9R)-6-oxaspiro[4.5]decan-9-yl]pyridazin-3-amine
—— 6-tert-butyl-4-[(Z)-[(1R)-cyclohex-3-en-1-yl]methylideneamino]-3-methylsulfanyl-1,2,4-triazin-5-one —— C15H22N4OS
6-tert-butyl-4-[(Z)-[(1R)-cyclohex-3-en-1-yl]methylideneamino]-3-methylsulfanyl-1,2,4-triazin-5-one
—— 6-(3-methylpyrazol-1-yl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyridazin-3-amine —— C18H18N8
6-(3-methylpyrazol-1-yl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyridazin-3-amine
—— 6-(3-methylpyrazol-1-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyridazin-3-amine —— C18H18N8
6-(3-methylpyrazol-1-yl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyridazin-3-amine
—— (6Z)-3-[(4-bromophenyl)methylideneamino]-6-(6-methyl-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,4-dien-1-one —— C21H15BrN2O2
(6Z)-3-[(4-bromophenyl)methylideneamino]-6-(6-methyl-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,4-dien-1-one
—— 6-tert-butyl-4-[(Z)-[(1S)-cyclohex-3-en-1-yl]methylideneamino]-3-methylsulfanyl-1,2,4-triazin-5-one —— C15H22N4OS
6-tert-butyl-4-[(Z)-[(1S)-cyclohex-3-en-1-yl]methylideneamino]-3-methylsulfanyl-1,2,4-triazin-5-one
—— (6Z)-6-[4-(benzyloxy)-3-methoxybenzylidene]-5-imino-2-[2-(morpholin-4-yl)-2-oxoethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H25N5O5S
(6Z)-6-[4-(benzyloxy)-3-methoxybenzylidene]-5-imino-2-[2-(morpholin-4-yl)-2-oxoethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-tert-butyl-2-[(2S)-1,4-dithian-2-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C14H18N2OS3
6-tert-butyl-2-[(2S)-1,4-dithian-2-yl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (1S,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C18H16N2O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (1S,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— (6E)-2-ethoxy-6-[[2-[6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C24H30N4O2S
(6E)-2-ethoxy-6-[[2-[6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (1S,2S)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C18H16N2O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (1S,2S)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— (6Z)-6-(1H-pyrrol-2-ylhydrazinylidene)cyclohexa-2,4-dien-1-one —— C10H9N3O
(6Z)-6-(1H-pyrrol-2-ylhydrazinylidene)cyclohexa-2,4-dien-1-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (1R,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate —— C18H16N2O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (1R,2R)-2-(furan-2-yl)cyclopropane-1-carboxylate
—— (6S)-N-[2-(2,6-dimethylphenoxy)ethyl]-2,2,6-trimethylmorpholine-4-carboxamide —— C18H28N2O3
(6S)-N-[2-(2,6-dimethylphenoxy)ethyl]-2,2,6-trimethylmorpholine-4-carboxamide
—— 6-methyl-2-oxo-N-[(5R)-2,3,4,5-tetrahydrobenzo[i][1]benzoxepin-5-yl]-1H-pyridine-3-carboxamide —— C21H20N2O3
6-methyl-2-oxo-N-[(5R)-2,3,4,5-tetrahydrobenzo[i][1]benzoxepin-5-yl]-1H-pyridine-3-carboxamide
—— (6E)-4-hydroxy-6-[[2-[(E)-(3-hydroxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C14H12N2O4
(6E)-4-hydroxy-6-[[2-[(E)-(3-hydroxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-4-chloro-6-[(oxolan-2-ylmethylamino)methylidene]cyclohexa-2,4-dien-1-one —— C12H14ClNO2
(6E)-4-chloro-6-[(oxolan-2-ylmethylamino)methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-[(4-bromo-2-methylanilino)methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C15H14BrNO2
(6Z)-6-[(4-bromo-2-methylanilino)methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— (6E)-6-[[(1,1-dioxothiolan-3-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C11H13NO3S
(6E)-6-[[(1,1-dioxothiolan-3-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[2-[(Z)-(2-methylindol-3-ylidene)methyl]hydrazinyl]-2-N,4-N-diphenyl-1,3,5-triazine-2,4-diamine —— C25H22N8
6-[2-[(Z)-(2-methylindol-3-ylidene)methyl]hydrazinyl]-2-N,4-N-diphenyl-1,3,5-triazine-2,4-diamine
—— (6E)-2,4-dibromo-6-[[(1-octylbenzimidazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C22H25Br2N3O
(6E)-2,4-dibromo-6-[[(1-octylbenzimidazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one