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—— (6-aminopyridin-3-yl)-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C18H20N6OS
(6-aminopyridin-3-yl)-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (6S)-4-(2-indazol-1-ylacetyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H27N5O2
(6S)-4-(2-indazol-1-ylacetyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[4-[(2R)-2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazin-1-yl]pyridine-3-carbonitrile —— C21H25N5O
6-[4-[(2R)-2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazin-1-yl]pyridine-3-carbonitrile
—— (6R)-4-(1,7-dimethylindole-2-carbonyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C22H30N4O2
(6R)-4-(1,7-dimethylindole-2-carbonyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— [6-oxo-6-[4-[(1R)-1-(4-oxo-3-propylquinazolin-2-yl)propyl]piperazin-4-ium-1-yl]hexyl]azanium —— C24H39N5O2+2
[6-oxo-6-[4-[(1R)-1-(4-oxo-3-propylquinazolin-2-yl)propyl]piperazin-4-ium-1-yl]hexyl]azanium
—— (6S)-4-[3-(3,4-dihydro-2H-quinolin-1-yl)-3-oxopropyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C22H32N4O2
(6S)-4-[3-(3,4-dihydro-2H-quinolin-1-yl)-3-oxopropyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-(3-chlorophenyl)sulfonyl-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H22ClN3O3S
(6S)-4-(3-chlorophenyl)sulfonyl-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(6R)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylic acid —— C22H27N3O2
6-[(6R)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylic acid
—— 6-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C18H20N8
6-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— (6S)-4-[(4-fluoro-3-methylphenyl)methyl]-10-(2-methoxyethyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H32FN3O2
(6S)-4-[(4-fluoro-3-methylphenyl)methyl]-10-(2-methoxyethyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile —— C18H20N8
6-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-2-carbonitrile
—— (6R)-4-(2-indazol-1-ylacetyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H27N5O2
(6R)-4-(2-indazol-1-ylacetyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-ethyl-N-[[(3R)-1-(3-methylphenyl)pyrrolidin-3-yl]methyl]pyrimidin-4-amine —— C18H24N4
6-ethyl-N-[[(3R)-1-(3-methylphenyl)pyrrolidin-3-yl]methyl]pyrimidin-4-amine
—— (6R)-10-ethyl-4-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H33N3O3
(6R)-10-ethyl-4-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-methyl-2-[2-[(3S)-1-methylpyrrolidin-3-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid —— C21H30N4O3
6-methyl-2-[2-[(3S)-1-methylpyrrolidin-3-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid
—— (6R)-10-ethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H30N4O2S
(6R)-10-ethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3S)-1-(2-methoxyacetyl)piperidine-3-carbonyl]-2,3-dimethyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-one —— C17H24N4O4
6-[(3S)-1-(2-methoxyacetyl)piperidine-3-carbonyl]-2,3-dimethyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-one
—— (6R)-4-[2-(4-chloropyrazol-1-yl)ethyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H26ClN5O
(6R)-4-[2-(4-chloropyrazol-1-yl)ethyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-methyl-2-[2-[(3R)-1-methylpyrrolidin-3-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid —— C21H30N4O3
6-methyl-2-[2-[(3R)-1-methylpyrrolidin-3-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid
—— 6-Amino-5-[2-[[5-(3,4-dimethylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione —— C19H21N5O4S
6-Amino-5-[2-[[5-(3,4-dimethylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione
—— (6R)-2-[[(E)-2-cyano-3-(2-fluorophenyl)prop-2-enoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C20H18FN3O2S
(6R)-2-[[(E)-2-cyano-3-(2-fluorophenyl)prop-2-enoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-10-ethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H30N4O2S
(6S)-10-ethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(6S)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylic acid —— C22H27N3O2
6-[(6S)-8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylic acid
—— (6S)-10-ethyl-4-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H33N3O3
(6S)-10-ethyl-4-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-[2-(4-chloropyrazol-1-yl)ethyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H26ClN5O
(6S)-4-[2-(4-chloropyrazol-1-yl)ethyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H27N5O2
(6S)-4-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-ethyl-N-[(1S)-1-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)ethyl]pyrimidin-4-amine —— C13H19N5O
6-ethyl-N-[(1S)-1-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)ethyl]pyrimidin-4-amine
—— (6S)-4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H26ClN3O3
(6S)-4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-(cyclopropylmethyl)-4-(3-methoxypyrazin-2-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H29N5O2
(6S)-10-(cyclopropylmethyl)-4-(3-methoxypyrazin-2-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-10-ethyl-4-[2-(2-methoxyphenyl)acetyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H31N3O3
(6R)-10-ethyl-4-[2-(2-methoxyphenyl)acetyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3R)-1-(2-methoxyacetyl)piperidine-3-carbonyl]-2,3-dimethyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-one —— C17H24N4O4
6-[(3R)-1-(2-methoxyacetyl)piperidine-3-carbonyl]-2,3-dimethyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-4-one
—— (6R)-4-[3-(difluoromethoxy)benzoyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H23F2N3O3
(6R)-4-[3-(difluoromethoxy)benzoyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-cyclopropyl-N-[2-[(2R)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-4-amine —— C15H24N4O2S
6-cyclopropyl-N-[2-[(2R)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-4-amine
—— 6-ethyl-N-[(1R)-1-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)ethyl]pyrimidin-4-amine —— C13H19N5O
6-ethyl-N-[(1R)-1-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)ethyl]pyrimidin-4-amine
—— 6-ethyl-N-[[(3S)-1-(3-methylphenyl)pyrrolidin-3-yl]methyl]pyrimidin-4-amine —— C18H24N4
6-ethyl-N-[[(3S)-1-(3-methylphenyl)pyrrolidin-3-yl]methyl]pyrimidin-4-amine
—— (6S)-4-[3-(difluoromethoxy)benzoyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H23F2N3O3
(6S)-4-[3-(difluoromethoxy)benzoyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-cyclopropyl-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-4-amine —— C15H24N4O2S
6-cyclopropyl-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-4-amine
—— (6R)-4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H26ClN3O3
(6R)-4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-ethyl-4-[2-(2-methoxyphenyl)acetyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H31N3O3
(6S)-10-ethyl-4-[2-(2-methoxyphenyl)acetyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-4-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H27N5O2
(6R)-4-[[2-(furan-2-yl)pyrimidin-5-yl]methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-fluoro-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]-1H-benzimidazole-4-carboxamide —— C15H14FN3OS
6-fluoro-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]-1H-benzimidazole-4-carboxamide
—— 6-fluoro-N-methyl-N-[(1R)-1-thiophen-2-ylethyl]-1H-benzimidazole-4-carboxamide —— C15H14FN3OS
6-fluoro-N-methyl-N-[(1R)-1-thiophen-2-ylethyl]-1H-benzimidazole-4-carboxamide
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-N-[[2-(4-ethoxyphenoxy)pyridin-4-yl]methyl]pyridine-3-carboxamide —— C26H30N4O4
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-N-[[2-(4-ethoxyphenoxy)pyridin-4-yl]methyl]pyridine-3-carboxamide
—— (6R)-10-(cyclopropylmethyl)-4-[2-[2-methoxyethyl(methyl)amino]acetyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H36N4O3
(6R)-10-(cyclopropylmethyl)-4-[2-[2-methoxyethyl(methyl)amino]acetyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(5S)-4-[hydroxy-(4-methoxyphenyl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]hexanoate —— C24H24NO6-
6-[(5S)-4-[hydroxy-(4-methoxyphenyl)methylidene]-2,3-dioxo-5-phenylpyrrolidin-1-yl]hexanoate
—— 6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-N-[[2-(4-ethoxyphenoxy)pyridin-4-yl]methyl]pyridine-3-carboxamide —— C26H30N4O4
6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-N-[[2-(4-ethoxyphenoxy)pyridin-4-yl]methyl]pyridine-3-carboxamide
—— 6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[[2-(4-ethoxyphenoxy)pyridin-4-yl]methyl]pyridine-3-carboxamide —— C26H30N4O4
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[[2-(4-ethoxyphenoxy)pyridin-4-yl]methyl]pyridine-3-carboxamide
—— (6S)-4-[(3-hydroxy-4-methoxyphenyl)methyl]-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H31N3O3
(6S)-4-[(3-hydroxy-4-methoxyphenyl)methyl]-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[[[(3S)-3-[(4R)-2,2-dimethyloxan-4-yl]-3-phenylpropyl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C23H29NO2
6-[[[(3S)-3-[(4R)-2,2-dimethyloxan-4-yl]-3-phenylpropyl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6S)-10-(cyclopropylmethyl)-4-(3-hydroxybenzoyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H29N3O3
(6S)-10-(cyclopropylmethyl)-4-(3-hydroxybenzoyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one