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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N6O
(6S)-8-(5-ethyl-2-methylpyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-1,10-dimethyl-4-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C15H22F3N5O2
(6R)-1,10-dimethyl-4-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-(2-hydroxyethyl)-1-methyl-4-(2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C15H24N6O3
(6S)-10-(2-hydroxyethyl)-1-methyl-4-(2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-(5-ethyl-1H-pyrazole-4-carbonyl)-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H29N5O2
(6S)-4-(5-ethyl-1H-pyrazole-4-carbonyl)-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-1,10-dimethyl-4-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C15H22F3N5O2
(6S)-1,10-dimethyl-4-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-cyano-N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]pyridine-3-carboxamide —— C19H16FN5O
6-cyano-N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]pyridine-3-carboxamide
—— 6-(2,2-Dimethylpropanoylamino)-2,3-difluorobenzoate —— C12H12F2NO3-
6-(2,2-Dimethylpropanoylamino)-2,3-difluorobenzoate
—— (6R)-4-[(4-imidazol-1-ylphenyl)methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H29N5O
(6R)-4-[(4-imidazol-1-ylphenyl)methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O3
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O3
(6R)-8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-1-methyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H28N6O2
(6S)-1-methyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-8-(2-ethoxyacetyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H32N2O3
(6S)-8-(2-ethoxyacetyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O3
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-10-(2-hydroxyethyl)-1-methyl-4-(2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C15H24N6O3
(6R)-10-(2-hydroxyethyl)-1-methyl-4-(2H-triazole-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3S)-3-methyl-3-phenylpiperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C21H21N3O3
6-[(3S)-3-methyl-3-phenylpiperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione
—— (6S)-10-(2-methoxyethyl)-1-methyl-4-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H30N6O2
(6S)-10-(2-methoxyethyl)-1-methyl-4-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(7H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N8O
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(7H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-amino-N-(3-methoxypropyl)-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C21H26N5O4+
6-amino-N-(3-methoxypropyl)-2-oxo-7-[[(2S)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— (6S)-2-cyclopropyl-8-(5-fluoro-2-methylphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H25FN2O3S
(6S)-2-cyclopropyl-8-(5-fluoro-2-methylphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-10-ethyl-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H30N4O2
(6R)-10-ethyl-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-6-(pyridin-2-ylamino)-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one —— C11H9F3N4OS
(6R)-6-(pyridin-2-ylamino)-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one
—— (6S)-8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O3
(6S)-8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-amino-7-(2-methoxyethyl)-2-oxo-N-[(1R)-1-phenylethyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C23H24N5O3+
6-amino-7-(2-methoxyethyl)-2-oxo-N-[(1R)-1-phenylethyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6-amino-N-cyclohexyl-7-(3-methoxypropyl)-11-methyl-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C23H30N5O3+
6-amino-N-cyclohexyl-7-(3-methoxypropyl)-11-methyl-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— (6S)-6-(pyridin-2-ylamino)-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one —— C11H9F3N4OS
(6S)-6-(pyridin-2-ylamino)-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one
—— (6S)-8-[(4-fluoro-2-methylphenyl)methyl]-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H29FN4O
(6S)-8-[(4-fluoro-2-methylphenyl)methyl]-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-ethyl-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H30N4O2
(6S)-10-ethyl-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-Amino-7-(3-ethoxypropyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C17H20N5O3+
6-Amino-7-(3-ethoxypropyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6-amino-7-(3-methoxypropyl)-11-methyl-5-(4-methylpiperazine-1-carbonyl)-9-aza-1,7-diazoniatricyclo[8.4.0.03,8]tetradeca-1(14),3,5,7,10,12-hexaen-2-one —— C22H30N6O3+2
6-amino-7-(3-methoxypropyl)-11-methyl-5-(4-methylpiperazine-1-carbonyl)-9-aza-1,7-diazoniatricyclo[8.4.0.03,8]tetradeca-1(14),3,5,7,10,12-hexaen-2-one
—— (6R)-2-cyclopropyl-8-(5-fluoro-2-methylphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H25FN2O3S
(6R)-2-cyclopropyl-8-(5-fluoro-2-methylphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[(5-chloropyridin-2-yl)amino]-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one —— C11H8ClF3N4OS
(6R)-6-[(5-chloropyridin-2-yl)amino]-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one
—— 6-amino-7-(3-methoxypropyl)-11-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C22H28N5O4+
6-amino-7-(3-methoxypropyl)-11-methyl-2-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— [6-(4-Bromophenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylazanium —— C12H11BrN3S+
[6-(4-Bromophenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methylazanium
—— (6R)-8-(2-ethoxyacetyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H32N2O3
(6R)-8-(2-ethoxyacetyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-(cyclopropylmethyl)-4-(furan-3-ylmethyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H29N3O2
(6S)-10-(cyclopropylmethyl)-4-(furan-3-ylmethyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H30N4OS
(6S)-10-(cyclopropylmethyl)-1-methyl-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-8-[(4-fluoro-2-methylphenyl)methyl]-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H29FN4O
(6R)-8-[(4-fluoro-2-methylphenyl)methyl]-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-[4-(4-methoxyphenyl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H32N2O3
(6R)-2-cyclopropyl-8-[4-(4-methoxyphenyl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-(2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl)-10-(2-hydroxyethyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H28N6O3
(6S)-4-(2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl)-10-(2-hydroxyethyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(7H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N8O
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(7H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2-Amino-6-chloropyrimidin-4-yl)amino]hexanoate —— C10H14ClN4O2-
6-[(2-Amino-6-chloropyrimidin-4-yl)amino]hexanoate
—— (6S)-2-cyclopropyl-8-[4-(4-methoxyphenyl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H32N2O3
(6S)-2-cyclopropyl-8-[4-(4-methoxyphenyl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(4S)-4-hydroxy-4-methyl-2-oxo-1-oxa-3-azaspiro[4.5]decan-3-yl]hexanoate —— C15H24NO5-
6-[(4S)-4-hydroxy-4-methyl-2-oxo-1-oxa-3-azaspiro[4.5]decan-3-yl]hexanoate
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-(1,3-thiazol-2-ylmethyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H28N4OS
(6S)-10-(cyclopropylmethyl)-1-methyl-4-(1,3-thiazol-2-ylmethyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-Amino-7-(2-methoxyethyl)-11-methyl-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C16H18N5O3+
6-Amino-7-(2-methoxyethyl)-11-methyl-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— (6R)-3-butylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C19H19N5OS
(6R)-3-butylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (6S)-6-phenylthiazinane 1,1-dioxide —— C10H13NO2S
(6S)-6-phenylthiazinane 1,1-dioxide
—— 6-amino-7-(3-ethoxypropyl)-N-(furan-2-ylmethyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C22H24N5O4+
6-amino-7-(3-ethoxypropyl)-N-(furan-2-ylmethyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one —— C16H22N2O3S
6-[(3R,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one
—— (6S)-6-(propylamino)-3,4,5,6,7,8-hexahydro-2H-naphthalen-1-one —— C13H21NO
(6S)-6-(propylamino)-3,4,5,6,7,8-hexahydro-2H-naphthalen-1-one