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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N5O3
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-N-[(1S)-1-(4-methylsulfonylphenyl)propyl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H21N3O3S
6-methyl-N-[(1S)-1-(4-methylsulfonylphenyl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
—— (6S)-4-(1,4-dithiepan-6-yl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H29N3OS2
(6S)-4-(1,4-dithiepan-6-yl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H25N5O3
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-[2-[4-(hydroxymethyl)phenyl]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N2O3
(6R)-2-butyl-8-[2-[4-(hydroxymethyl)phenyl]acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6,8-dimethyl-2-[[2-[(2R)-1-methylpyrrolidin-2-yl]ethylamino]methyl]-1H-quinolin-4-one —— C19H27N3O
6,8-dimethyl-2-[[2-[(2R)-1-methylpyrrolidin-2-yl]ethylamino]methyl]-1H-quinolin-4-one
—— 6-fluoro-2-[[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methyl]-1H-quinolin-4-one —— C19H24FN3O2
6-fluoro-2-[[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methyl]-1H-quinolin-4-one
—— (6S)-8-[4-(difluoromethoxy)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H24F2N2O4
(6S)-8-[4-(difluoromethoxy)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N5O2
(6R)-4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-4-(1,4-dithiepan-6-yl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H29N3OS2
(6R)-4-(1,4-dithiepan-6-yl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(1S)-1-[4-(1-methylimidazol-2-yl)triazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole —— C12H12N8S
6-[(1S)-1-[4-(1-methylimidazol-2-yl)triazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole
—— 6-[(1R)-1-[4-(1-methylimidazol-2-yl)triazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole —— C12H12N8S
6-[(1R)-1-[4-(1-methylimidazol-2-yl)triazol-1-yl]ethyl]imidazo[2,1-b][1,3,4]thiadiazole
—— (6S)-N-(3-chloro-4-methylphenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C19H27ClN4O2
(6S)-N-(3-chloro-4-methylphenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— (6R)-8-[(3-methylimidazol-4-yl)methyl]-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N5O
(6R)-8-[(3-methylimidazol-4-yl)methyl]-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[4-[(4aS,7aS)-1,2,3,4,4a,5,7,7a-octahydropyrrolo[3,4-b]pyridin-6-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C18H22N4O
6-[4-[(4aS,7aS)-1,2,3,4,4a,5,7,7a-octahydropyrrolo[3,4-b]pyridin-6-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-8-[(3-methylimidazol-4-yl)methyl]-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N5O
(6S)-8-[(3-methylimidazol-4-yl)methyl]-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-(cyclopropylmethyl)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H32N4OS
(6S)-10-(cyclopropylmethyl)-4-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-fluoro-2-[[[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]amino]methyl]-1H-quinolin-4-one —— C18H21FN4O
6-fluoro-2-[[[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]amino]methyl]-1H-quinolin-4-one
—— (6S)-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H29N3O3
(6S)-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H29N3O3
(6R)-4-[1-(methoxymethyl)cyclobutanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-N-(3-chloro-4-methylphenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C19H27ClN4O2
(6R)-N-(3-chloro-4-methylphenyl)-1,10-dimethyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— 6-[(3S)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-7H-purine —— C16H21N7O
6-[(3S)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-7H-purine
—— (6S)-8-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N5O2
(6S)-8-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [6-Chloro-1-(2-hydroxyethyl)benzimidazol-2-yl]methyl 5-methyl-3-phenyl-1,2-oxazole-4-carboxylate —— C21H18ClN3O4
[6-Chloro-1-(2-hydroxyethyl)benzimidazol-2-yl]methyl 5-methyl-3-phenyl-1,2-oxazole-4-carboxylate
—— 6-fluoro-2-[[(3S)-3-(1-methylimidazole-2-carbonyl)piperidin-1-yl]methyl]-1H-quinolin-4-one —— C20H21FN4O2
6-fluoro-2-[[(3S)-3-(1-methylimidazole-2-carbonyl)piperidin-1-yl]methyl]-1H-quinolin-4-one
—— (6R)-2-[2-(dimethylamino)ethyl]-8-[4-(1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H32N6O2
(6R)-2-[2-(dimethylamino)ethyl]-8-[4-(1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O3
(6R)-2-(2-methoxyethyl)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-1-methyl-4-[(2-methyl-1-benzothiophen-3-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H27N3OS
(6S)-1-methyl-4-[(2-methyl-1-benzothiophen-3-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-8-[(2-butyl-1H-imidazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6R)-8-[(2-butyl-1H-imidazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(dimethylamino)ethyl]-8-[4-(1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H32N6O2
(6S)-2-[2-(dimethylamino)ethyl]-8-[4-(1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N5O2
(6R)-8-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-fluoro-2-[[(3R)-3-(1-methylimidazole-2-carbonyl)piperidin-1-yl]methyl]-1H-quinolin-4-one —— C20H21FN4O2
6-fluoro-2-[[(3R)-3-(1-methylimidazole-2-carbonyl)piperidin-1-yl]methyl]-1H-quinolin-4-one
—— (6S)-8-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N5O2
(6S)-8-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-1-methyl-4-[(3-methylpyridin-4-yl)methyl]-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H30N4O
(6S)-1-methyl-4-[(3-methylpyridin-4-yl)methyl]-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H21N5O2S
6-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6S)-8-[(2-butyl-1H-imidazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6S)-8-[(2-butyl-1H-imidazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O3
(6S)-2-(2-methoxyethyl)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-ethyl-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H27N5O2
(6S)-10-ethyl-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-2-(3-methylbutyl)-3-oxo-N-(thiophen-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C20H31N3O2S
(6R)-2-(3-methylbutyl)-3-oxo-N-(thiophen-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— 6-fluoro-2-[[[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]amino]methyl]-1H-quinolin-4-one —— C18H21FN4O
6-fluoro-2-[[[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]amino]methyl]-1H-quinolin-4-one
—— (6-methyl-3-nitro-2-oxo-1H-pyridin-4-yl) 3,5-dimethoxybenzoate —— C15H14N2O7
(6-methyl-3-nitro-2-oxo-1H-pyridin-4-yl) 3,5-dimethoxybenzoate
—— 6-[(3R)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-7H-purine —— C16H21N7O
6-[(3R)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-7H-purine
—— 6-[(5R)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carbonitrile —— C17H22N4O2
6-[(5R)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carbonitrile
—— 6-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H21N5O2S
6-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-[(5S)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carbonitrile —— C17H22N4O2
6-[(5S)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carbonitrile
—— (6R)-4-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H28N4O3
(6R)-4-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-8-(1-aminocyclopropanecarbonyl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N5O2
(6S)-8-(1-aminocyclopropanecarbonyl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methylbutyl)-3-oxo-N-(thiophen-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C20H31N3O2S
(6S)-2-(3-methylbutyl)-3-oxo-N-(thiophen-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— (6R)-10-ethyl-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H27N5O2
(6R)-10-ethyl-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H29N5O
(6S)-4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one