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—— 6-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C36H44N2O7
6-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine —— C16H25N7
6-[4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine
—— 6-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C30H33NO6S
6-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C33H36N4O6S
6-[[3-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C29H38N2O7
6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-methoxy-5-[[[(2R,3S)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]methyl]pyrimidin-4-amine —— C17H25N5OS
6-methoxy-5-[[[(2R,3S)-1-methyl-2-thiophen-2-ylpiperidin-3-yl]methylamino]methyl]pyrimidin-4-amine
—— 6-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C40H51N3O6
6-[[2-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C35H48N2O6
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl)methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[3-[4-[(2R,4R,6S)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C39H44N2O6
6-[[3-[4-[(2R,4R,6S)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C32H42N2O8
6-[[4-[(2R,4R,6S)-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(pyrimidin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C35H37N3O6S
6-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(pyrimidin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C31H35NO6S
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C36H44N2O7
6-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-chloro-N-[(2S,3R)-2-(4-chlorophenyl)-1-methylpyrrolidin-3-yl]pyridine-3-carboxamide —— C17H17Cl2N3O
6-chloro-N-[(2S,3R)-2-(4-chlorophenyl)-1-methylpyrrolidin-3-yl]pyridine-3-carboxamide
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C33H41N3O6
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(2-pyridin-2-ylethyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C26H30N4O6S
6-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-chloro-N-[(2S,3S)-2-(4-chlorophenyl)-1-methylpyrrolidin-3-yl]pyridine-3-carboxamide —— C17H17Cl2N3O
6-chloro-N-[(2S,3S)-2-(4-chlorophenyl)-1-methylpyrrolidin-3-yl]pyridine-3-carboxamide
—— 6-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C35H42N2O7
6-[[3-[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(morpholin-4-ylmethyl)-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C29H38N2O7
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-(morpholin-4-ylmethyl)-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[methyl-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]amino]-N-prop-2-enylpyridine-3-carboxamide —— C15H20N4O2
6-[methyl-[(3R)-1-methyl-2-oxopyrrolidin-3-yl]amino]-N-prop-2-enylpyridine-3-carboxamide
—— 6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C28H36N2O7
6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-[methyl-[(3S)-1-methyl-2-oxopyrrolidin-3-yl]amino]-N-prop-2-enylpyridine-3-carboxamide —— C15H20N4O2
6-[methyl-[(3S)-1-methyl-2-oxopyrrolidin-3-yl]amino]-N-prop-2-enylpyridine-3-carboxamide
—— 6-[4-[(2R,4R,6S)-4-(2-hydroxyethylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C26H33NO7S
6-[4-[(2R,4R,6S)-4-(2-hydroxyethylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid —— C29H38N2O7
6-[[4-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methylamino]-6-oxohexanoic acid
—— 6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid —— C28H36N2O6
6-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]anilino]-6-oxohexanoic acid
—— 6-[(4aR,7aR)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H21N3O2
6-[(4aR,7aR)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-[(4aR,7aS)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H21N3O2
6-[(4aR,7aS)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-[(4aS,7aR)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H21N3O2
6-[(4aS,7aR)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-[(4aS,7aS)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H21N3O2
6-[(4aS,7aS)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyridine-1-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-[(3aS,7aR)-1,3,3a,4,5,6,7,7a-octahydroisoindole-2-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H21N3O2
6-[(3aS,7aR)-1,3,3a,4,5,6,7,7a-octahydroisoindole-2-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-[(3aS,7aS)-1,3,3a,4,5,6,7,7a-octahydroisoindole-2-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H21N3O2
6-[(3aS,7aS)-1,3,3a,4,5,6,7,7a-octahydroisoindole-2-carbonyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-methyl-N-[(1S,2R)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide —— C18H28N2O3
6-methyl-N-[(1S,2R)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide
—— 6-methyl-N-[(1S,2S)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide —— C18H28N2O3
6-methyl-N-[(1S,2S)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide
—— 6-methyl-N-[(1R,2S)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide —— C18H28N2O3
6-methyl-N-[(1R,2S)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide
—— 6-methyl-N-[(1R,2R)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide —— C18H28N2O3
6-methyl-N-[(1R,2R)-2-(3-methylbutoxy)cyclohexyl]-4-oxo-1H-pyridine-3-carboxamide
—— 6-[(3aS,6R,11aS,11bR)-6-(2-hydroxynaphthalen-1-yl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C33H31NO7
6-[(3aS,6R,11aS,11bR)-6-(2-hydroxynaphthalen-1-yl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(6-hydroxy-4H-chromen-3-yl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C32H31NO8
6-[(3aS,6R,11aS,11bR)-6-(6-hydroxy-4H-chromen-3-yl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(4-hydroxy-3,5-dimethoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C31H33NO9
6-[(3aS,6R,11aS,11bR)-6-(4-hydroxy-3,5-dimethoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,6aS,10aR,11aS,11bR)-6-(2-hydroxy-3-prop-2-enylphenyl)-6a,8-dimethyl-1,3,7,10-tetraoxo-4,6,10a,11,11a,11b-hexahydro-3aH-naphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C33H37NO7
6-[(3aS,6R,6aS,10aR,11aS,11bR)-6-(2-hydroxy-3-prop-2-enylphenyl)-6a,8-dimethyl-1,3,7,10-tetraoxo-4,6,10a,11,11a,11b-hexahydro-3aH-naphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(2-hydroxy-3-prop-2-enylphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C32H33NO7
6-[(3aS,6R,11aS,11bR)-6-(2-hydroxy-3-prop-2-enylphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(4-hydroxy-3-methylphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C30H31NO7
6-[(3aS,6R,11aS,11bR)-6-(4-hydroxy-3-methylphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6S,11aS,11bR)-6-[2-(4-hydroxy-3,5-dimethoxyphenyl)ethenyl]-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C33H35NO9
6-[(3aS,6S,11aS,11bR)-6-[2-(4-hydroxy-3,5-dimethoxyphenyl)ethenyl]-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6S,11aS,11bR)-6-(2-chloro-4-hydroxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C29H28ClNO7
6-[(3aS,6S,11aS,11bR)-6-(2-chloro-4-hydroxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(4-hydroxynaphthalen-1-yl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C33H31NO7
6-[(3aS,6R,11aS,11bR)-6-(4-hydroxynaphthalen-1-yl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(2-hydroxy-3-methoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C30H31NO8
6-[(3aS,6R,11aS,11bR)-6-(2-hydroxy-3-methoxyphenyl)-8-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(5-chloro-2-hydroxyphenyl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C29H28ClNO7
6-[(3aS,6R,11aS,11bR)-6-(5-chloro-2-hydroxyphenyl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3aS,6R,11aS,11bR)-6-(3-fluoro-2-hydroxyphenyl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C29H28FNO7
6-[(3aS,6R,11aS,11bR)-6-(3-fluoro-2-hydroxyphenyl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid
—— 6-[(3R,4S)-3-(dimethylamino)-4-methylsulfanylpyrrolidin-1-yl]-N-(oxan-4-yl)pyridazine-3-carboxamide —— C17H27N5O2S
6-[(3R,4S)-3-(dimethylamino)-4-methylsulfanylpyrrolidin-1-yl]-N-(oxan-4-yl)pyridazine-3-carboxamide
—— 6-[(3S,4S)-3-(dimethylamino)-4-methylsulfanylpyrrolidin-1-yl]-N-(oxan-4-yl)pyridazine-3-carboxamide —— C17H27N5O2S
6-[(3S,4S)-3-(dimethylamino)-4-methylsulfanylpyrrolidin-1-yl]-N-(oxan-4-yl)pyridazine-3-carboxamide
—— 6-[(3aS,6S,11aS,11bR)-6-(4-hydroxyphenyl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid —— C29H29NO7
6-[(3aS,6S,11aS,11bR)-6-(4-hydroxyphenyl)-9-methyl-1,3,7,10-tetraoxo-3a,4,6,11,11a,11b-hexahydronaphtho[2,3-e]isoindol-2-yl]hexanoic acid