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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide —— C16H24N4O2
6-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
—— 6-methyl-2-[[4-[(2S)-oxolane-2-carbonyl]-1,4-diazepan-1-yl]methyl]-1H-quinolin-4-one —— C21H27N3O3
6-methyl-2-[[4-[(2S)-oxolane-2-carbonyl]-1,4-diazepan-1-yl]methyl]-1H-quinolin-4-one
—— (6S)-10-ethyl-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H27N5O2
(6S)-10-ethyl-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-2-cyclopropyl-8-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26FN3O2
(6S)-2-cyclopropyl-8-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R,9S)-6-(2,3-dimethoxyphenyl)-9-(4-methoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H28N2O4
(6R,9S)-6-(2,3-dimethoxyphenyl)-9-(4-methoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-9-(4-chlorophenyl)-6-(3-phenylmethoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C32H27ClN2O2
(6R,9R)-9-(4-chlorophenyl)-6-(3-phenylmethoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-9-(4-chlorophenyl)-6-(2,3-dichlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H19Cl3N2O
(6S,9R)-9-(4-chlorophenyl)-6-(2,3-dichlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-(morpholine-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H32N4O3
(6S)-10-(cyclopropylmethyl)-1-methyl-4-(morpholine-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-8-[2-(2,4-difluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26F2N2O3
(6S)-8-[2-(2,4-difluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-(2,4-difluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26F2N2O3
(6R)-8-[2-(2,4-difluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S,9R)-9-(4-chlorophenyl)-6-(3-ethoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C27H25ClN2O2
(6S,9R)-9-(4-chlorophenyl)-6-(3-ethoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-8-(2-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H28N4O2
(6S)-8-(2-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-(2-methoxyethyl)-1-methyl-9-oxo-N-propan-2-yl-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C17H32N4O3
(6S)-10-(2-methoxyethyl)-1-methyl-9-oxo-N-propan-2-yl-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— (6R)-10-(cyclopropylmethyl)-1-methyl-4-(morpholine-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H32N4O3
(6R)-10-(cyclopropylmethyl)-1-methyl-4-(morpholine-4-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-8-(2-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H28N4O2
(6R)-8-(2-methylbenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[6-methyl-4-[4-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C21H25N5O
6-[6-methyl-4-[4-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— [6-[[(3R)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-yl]-morpholin-4-ylmethanone —— C21H24N2O4
[6-[[(3R)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-yl]-morpholin-4-ylmethanone
—— (6S)-10-ethyl-1-methyl-4-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H33N5O2
(6S)-10-ethyl-1-methyl-4-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-4-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H25N5O3
(6R)-4-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-10-(2-hydroxyethyl)-1-methyl-4-(thiophene-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N3O3S
(6R)-10-(2-hydroxyethyl)-1-methyl-4-(thiophene-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S,9R)-9-(4-methoxyphenyl)-6-(4-propoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C29H30N2O3
(6S,9R)-9-(4-methoxyphenyl)-6-(4-propoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-6-[4-(diethylamino)phenyl]-9-(furan-2-yl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H39N3O3
(6S,9R)-6-[4-(diethylamino)phenyl]-9-(furan-2-yl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-10-ethyl-1-methyl-4-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H33N5O2
(6R)-10-ethyl-1-methyl-4-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R,9R)-9-(4-chlorophenyl)-6-(2-fluorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H20ClFN2O
(6R,9R)-9-(4-chlorophenyl)-6-(2-fluorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-10-(2-hydroxyethyl)-1-methyl-4-(thiophene-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H25N3O3S
(6S)-10-(2-hydroxyethyl)-1-methyl-4-(thiophene-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-1-methyl-4-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H27N5O2
(6S)-1-methyl-4-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S,9R)-9-(4-chlorophenyl)-6-(4-methylsulfanylphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H23ClN2OS
(6S,9R)-9-(4-chlorophenyl)-6-(4-methylsulfanylphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— [6-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-yl]-morpholin-4-ylmethanone —— C21H24N2O4
[6-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-yl]-morpholin-4-ylmethanone
—— (6R)-4-(2-cyclopentylacetyl)-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H33N3O2
(6R)-4-(2-cyclopentylacetyl)-1-methyl-10-prop-2-enyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S,9S)-6-(2-butoxyphenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C29H29ClN2O2
(6S,9S)-6-(2-butoxyphenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-6-(2-chlorophenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H20Cl2N2O
(6S,9S)-6-(2-chlorophenyl)-9-(4-chlorophenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-4-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H25N5O3
(6S)-4-(2-cyclopropyl-6-oxo-1H-pyrimidine-5-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-8-(4-ethylthiadiazole-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H26N4O3S
(6S)-8-(4-ethylthiadiazole-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-ethyl-1-methyl-4-pyridazin-3-yl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H25N5O
(6S)-10-ethyl-1-methyl-4-pyridazin-3-yl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[6-methyl-4-[methyl-[[(3R)-oxolan-3-yl]methyl]amino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H21N3O2
6-[6-methyl-4-[methyl-[[(3R)-oxolan-3-yl]methyl]amino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R,9S)-9-(4-chlorophenyl)-6-(2-propan-2-yloxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H27ClN2O2
(6R,9S)-9-(4-chlorophenyl)-6-(2-propan-2-yloxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-1-methyl-4-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H27N5O2
(6R)-1-methyl-4-[1-(pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[6-methyl-4-[methyl-[[(3S)-oxolan-3-yl]methyl]amino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H21N3O2
6-[6-methyl-4-[methyl-[[(3S)-oxolan-3-yl]methyl]amino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R,9S)-6-[4-(diethylamino)phenyl]-9-(furan-2-yl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H39N3O3
(6R,9S)-6-[4-(diethylamino)phenyl]-9-(furan-2-yl)-5-hexanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-1,10-dimethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H26N4O3
(6R)-1,10-dimethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[[(3S)-1,1-dioxothiolan-3-yl]amino]hexanoic acid —— C10H19NO4S
6-[[(3S)-1,1-dioxothiolan-3-yl]amino]hexanoic acid
—— (6R)-10-ethyl-1-methyl-4-pyridazin-3-yl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H25N5O
(6R)-10-ethyl-1-methyl-4-pyridazin-3-yl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R,9S)-9-(4-methoxyphenyl)-6-(3-methoxy-4-propoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C30H32N2O4
(6R,9S)-9-(4-methoxyphenyl)-6-(3-methoxy-4-propoxyphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-methyl-N-(4-methylphenyl)-2-(phenylcarbamothioylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C24H25N3OS2
(6S)-6-methyl-N-(4-methylphenyl)-2-(phenylcarbamothioylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-1-methyl-9-oxo-10-prop-2-enyl-N-(thiophen-2-ylmethyl)-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C19H28N4O2S
(6S)-1-methyl-9-oxo-10-prop-2-enyl-N-(thiophen-2-ylmethyl)-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— (6R)-1-methyl-9-oxo-10-prop-2-enyl-N-(thiophen-2-ylmethyl)-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide —— C19H28N4O2S
(6R)-1-methyl-9-oxo-10-prop-2-enyl-N-(thiophen-2-ylmethyl)-1,4,10-triazaspiro[5.6]dodecane-4-carboxamide
—— (6R)-8-(4-ethylthiadiazole-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H26N4O3S
(6R)-8-(4-ethylthiadiazole-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O3
(6R)-8-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-1-ethyl-6-oxopiperidine-3-carbonyl]-N,N,1-trimethyl-5,7-dihydro-4H-pyrrolo[2,3-c]pyridine-2-carboxamide —— C19H28N4O3
6-[(3S)-1-ethyl-6-oxopiperidine-3-carbonyl]-N,N,1-trimethyl-5,7-dihydro-4H-pyrrolo[2,3-c]pyridine-2-carboxamide
—— (6S)-8-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O3
(6S)-8-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one