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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-8-(5-methyl-1,3,4-oxadiazol-2-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C15H24N4O2
(6S)-8-(5-methyl-1,3,4-oxadiazol-2-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-fluoro-4-[[(3R)-1-methylpiperidin-3-yl]methyl]-1,4-benzoxazin-3-one —— C15H19FN2O2
6-fluoro-4-[[(3R)-1-methylpiperidin-3-yl]methyl]-1,4-benzoxazin-3-one
—— (6R)-4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H25N5O2
(6R)-4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-2-methylpyridazin-3-one —— C16H23N3O4
6-[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-2-methylpyridazin-3-one
—— 6-[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-2-methylpyridazin-3-one —— C16H23N3O4
6-[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-2-methylpyridazin-3-one
—— (6S)-4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H25N5O2
(6S)-4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-7H-purin-2-amine —— C15H22N6O2
6-[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-7H-purin-2-amine
—— 6-[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-7H-purin-2-amine —— C15H22N6O2
6-[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-7H-purin-2-amine
—— 6-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylchromen-2-one —— C16H19NO4S
6-[(3S,5S)-3,5-dimethylpiperidin-1-yl]sulfonylchromen-2-one
—— 6-[5-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C19H18ClN5O2
6-[5-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H29N5O2
(6S)-10-(cyclopropylmethyl)-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-tert-butyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6S)-10-(2-methoxyethyl)-1-methyl-4-methylsulfonyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C14H27N3O4S
(6S)-10-(2-methoxyethyl)-1-methyl-4-methylsulfonyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-tert-butyl-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6R)-4-isoquinolin-1-yl-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H26N4O
(6R)-4-isoquinolin-1-yl-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-chloro-4-N-(2-morpholin-4-ium-4-ylethyl)-2-N-propan-2-yl-1,3,5-triazine-2,4-diamine —— C12H22ClN6O+
6-chloro-4-N-(2-morpholin-4-ium-4-ylethyl)-2-N-propan-2-yl-1,3,5-triazine-2,4-diamine
—— (6R)-10-ethyl-1-methyl-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H29N5O2
(6R)-10-ethyl-1-methyl-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-tert-butyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H28N4O3
(6S)-10-(cyclopropylmethyl)-1-methyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-tert-butyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6R)-10-(cyclopropylmethyl)-1-methyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H28N4O3
(6R)-10-(cyclopropylmethyl)-1-methyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-ethyl-1-methyl-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H29N5O2
(6S)-10-ethyl-1-methyl-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(R)-[1-(2-phenylethyl)tetrazol-5-yl]-pyrrolidin-1-ium-1-ylmethyl]quinoline —— C23H25N6+
6-[(R)-[1-(2-phenylethyl)tetrazol-5-yl]-pyrrolidin-1-ium-1-ylmethyl]quinoline
—— (6S)-4-isoquinolin-1-yl-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H26N4O
(6S)-4-isoquinolin-1-yl-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-4-[3-(2-chlorophenyl)propanoyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H26ClN3O2
(6R)-4-[3-(2-chlorophenyl)propanoyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-(cyclopropylmethyl)-4-(6-methoxyhexanoyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H37N3O3
(6S)-10-(cyclopropylmethyl)-4-(6-methoxyhexanoyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-8-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3S
(6R)-8-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-10-ethyl-1-methyl-4-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H29N5O2S
(6R)-10-ethyl-1-methyl-4-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-ethyl-1-methyl-4-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H29N5O2S
(6S)-10-ethyl-1-methyl-4-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-8-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3S
(6S)-8-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-10-(cyclopropylmethyl)-4-(6-methoxyhexanoyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H37N3O3
(6R)-10-(cyclopropylmethyl)-4-(6-methoxyhexanoyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-fluoro-2-[[[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]methyl]-1H-quinolin-4-one —— C15H16FN5O
6-fluoro-2-[[[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]methyl]-1H-quinolin-4-one
—— 6-[(S)-azepan-1-ium-1-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]quinoline —— C25H29N6+
6-[(S)-azepan-1-ium-1-yl-[1-(2-phenylethyl)tetrazol-5-yl]methyl]quinoline
—— 6-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyrimidin-4-amine —— C15H17N3O2
6-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyrimidin-4-amine
—— 6-[3-oxo-2-[[(2R)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid —— C20H27N3O4
6-[3-oxo-2-[[(2R)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid
—— (6R)-1-methyl-4-(1-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H25N5O2S
(6R)-1-methyl-4-(1-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-fluoro-2-[[[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]methyl]-1H-quinolin-4-one —— C15H16FN5O
6-fluoro-2-[[[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]methyl]-1H-quinolin-4-one
—— (6S)-1-methyl-4-(1-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H25N5O2S
(6S)-1-methyl-4-(1-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(3-hydroxypropyl)-[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]azanium —— C22H31N6O3+
(6,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(3-hydroxypropyl)-[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]azanium
—— (6,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(3-hydroxypropyl)-[(1R)-1-[1-(2-methoxyethyl)tetrazol-5-yl]ethyl]azanium —— C21H31N6O3+
(6,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(3-hydroxypropyl)-[(1R)-1-[1-(2-methoxyethyl)tetrazol-5-yl]ethyl]azanium
—— 6-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyrimidin-4-amine —— C15H17N3O2
6-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyrimidin-4-amine
—— (6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl-(3-hydroxypropyl)-[[1-(2-methoxyethyl)tetrazol-5-yl]methyl]azanium —— C20H29N6O4+
(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl-(3-hydroxypropyl)-[[1-(2-methoxyethyl)tetrazol-5-yl]methyl]azanium
—— 6-[3-oxo-2-[[(2S)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid —— C20H27N3O4
6-[3-oxo-2-[[(2S)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid
—— 6-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-N,N-dimethylpyrazin-2-amine —— C17H21N3O2
6-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-N,N-dimethylpyrazin-2-amine
—— [6-[(2R)-butan-2-yl]sulfonyl-2-(methylamino)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]-pyrrolidin-1-ylmethanone —— C17H27N5O3S
[6-[(2R)-butan-2-yl]sulfonyl-2-(methylamino)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]-pyrrolidin-1-ylmethanone
—— (6S)-4-[(2-aminopyridin-3-yl)methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C16H25N5O
(6S)-4-[(2-aminopyridin-3-yl)methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-ethoxy-3-[(R)-(4-methylpiperidin-1-ium-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one —— C22H31N6O2+
6-ethoxy-3-[(R)-(4-methylpiperidin-1-ium-1-yl)-(1-propan-2-yltetrazol-5-yl)methyl]-1H-quinolin-2-one
—— (6S)-2-methyl-6-[2-(2-phenylethyl)-1,2,4-triazol-3-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H20N6O
(6S)-2-methyl-6-[2-(2-phenylethyl)-1,2,4-triazol-3-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— (6R)-2-methyl-6-[2-(2-phenylethyl)-1,2,4-triazol-3-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H20N6O
(6R)-2-methyl-6-[2-(2-phenylethyl)-1,2,4-triazol-3-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— (6R)-10-(cyclopropylmethyl)-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H28N4O2
(6R)-10-(cyclopropylmethyl)-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one