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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-fluoro-2-[[[(1S)-1-(4-methoxyphenyl)ethyl]-methylamino]methyl]-1H-quinolin-4-one —— C20H21FN2O2
6-fluoro-2-[[[(1S)-1-(4-methoxyphenyl)ethyl]-methylamino]methyl]-1H-quinolin-4-one
—— (6R)-6-(3,3-diphenylpiperidine-1-carbonyl)piperazin-2-one —— C22H25N3O2
(6R)-6-(3,3-diphenylpiperidine-1-carbonyl)piperazin-2-one
—— 6-fluoro-2-[[[(1R)-1-(4-methoxyphenyl)ethyl]-methylamino]methyl]-1H-quinolin-4-one —— C20H21FN2O2
6-fluoro-2-[[[(1R)-1-(4-methoxyphenyl)ethyl]-methylamino]methyl]-1H-quinolin-4-one
—— (6S)-4-[6-(methoxymethyl)pyrimidin-4-yl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H27N5O2
(6S)-4-[6-(methoxymethyl)pyrimidin-4-yl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-2-cyclopropyl-8-(3-methoxyphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4S
(6S)-2-cyclopropyl-8-(3-methoxyphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N5O2
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-fluoro-2-[[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-1H-quinolin-4-one —— C18H18FN3O2
6-fluoro-2-[[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-1H-quinolin-4-one
—— (6R)-4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C15H25N3O3
(6R)-4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-cyclopropyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrimidin-4-amine —— C18H24N4O2
6-cyclopropyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrimidin-4-amine
—— (6R)-4-[6-(methoxymethyl)pyrimidin-4-yl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H27N5O2
(6R)-4-[6-(methoxymethyl)pyrimidin-4-yl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-cyclopropyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrimidin-4-amine —— C18H24N4O2
6-cyclopropyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrimidin-4-amine
—— (6S)-6-(3,3-diphenylpiperidine-1-carbonyl)piperazin-2-one —— C22H25N3O2
(6S)-6-(3,3-diphenylpiperidine-1-carbonyl)piperazin-2-one
—— (6R)-8-(1-tert-butylpyrrole-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H33N3O2
(6R)-8-(1-tert-butylpyrrole-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-pyridin-2-ylethyl)-8-[2-(tetrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N7O2
(6S)-2-(2-pyridin-2-ylethyl)-8-[2-(tetrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C15H25N3O3
(6S)-4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-8-(1-tert-butylpyrrole-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H33N3O2
(6S)-8-(1-tert-butylpyrrole-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(2,5-dichlorothiophene-3-carbonyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C15H14Cl2N2O2S2
(6R)-2-[(2,5-dichlorothiophene-3-carbonyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-(3-methylbutyl)-8-(2-morpholin-4-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H35N3O3
(6S)-2-(3-methylbutyl)-8-(2-morpholin-4-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methylbutyl)-8-(2-morpholin-4-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H35N3O3
(6R)-2-(3-methylbutyl)-8-(2-morpholin-4-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[[5-(2-fluorophenyl)furan-2-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H26FN3O2
(6S)-4-[[5-(2-fluorophenyl)furan-2-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-tert-butyl-4-[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-1H-pyrimidin-2-one —— C18H27N3O4
6-tert-butyl-4-[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-1H-pyrimidin-2-one
—— (6S)-2-cyclopropyl-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H29N3O2
(6S)-2-cyclopropyl-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(1H-imidazol-5-ylmethyl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O
(6S)-8-(1H-imidazol-5-ylmethyl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H29N3O2
(6R)-2-cyclopropyl-8-(2-pyrrolidin-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-10-(2-hydroxyethyl)-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C17H27N5O3
(6S)-10-(2-hydroxyethyl)-4-(6-methoxypyrimidin-4-yl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-1-methyl-4-[2-(4-propoxyphenoxy)ethyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H33N3O3
(6S)-1-methyl-4-[2-(4-propoxyphenoxy)ethyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[6-methyl-4-[[(2S)-oxan-2-yl]methylamino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H21N3O2
6-[6-methyl-4-[[(2S)-oxan-2-yl]methylamino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6-methylimidazo[1,2-a]pyridin-2-yl)-[(2S)-2-thiophen-2-ylazetidin-1-yl]methanone —— C16H15N3OS
(6-methylimidazo[1,2-a]pyridin-2-yl)-[(2S)-2-thiophen-2-ylazetidin-1-yl]methanone
—— (6S)-4-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H26FN5O
(6S)-4-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6-methylimidazo[1,2-a]pyridin-2-yl)-[(2R)-2-thiophen-2-ylazetidin-1-yl]methanone —— C16H15N3OS
(6-methylimidazo[1,2-a]pyridin-2-yl)-[(2R)-2-thiophen-2-ylazetidin-1-yl]methanone
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(6-methylpyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O2
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(6-methylpyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C21H22N6
6-methyl-2-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-methyl-2-[[(2-oxo-2-pyrrolidin-1-ylethyl)amino]methyl]-1H-quinolin-4-one —— C17H21N3O2
6-methyl-2-[[(2-oxo-2-pyrrolidin-1-ylethyl)amino]methyl]-1H-quinolin-4-one
—— (6S)-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N6O2
(6S)-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6-methylimidazo[1,2-a]pyridin-2-yl)-[(1R)-1-pyridin-3-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H19N5O
(6-methylimidazo[1,2-a]pyridin-2-yl)-[(1R)-1-pyridin-3-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— 6-[6-methyl-4-[[(2R)-oxan-2-yl]methylamino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H21N3O2
6-[6-methyl-4-[[(2R)-oxan-2-yl]methylamino]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H26FN5O
(6S)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-methyl-2-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C21H22N6
6-methyl-2-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[(3S)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]pyridine-2-carboxylic acid —— C15H22N2O3
6-[(3S)-3-(hydroxymethyl)-3-propylpiperidin-1-yl]pyridine-2-carboxylic acid
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-(4,4,4-trifluorobutyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C18H30F3N3O
(6S)-10-(cyclopropylmethyl)-1-methyl-4-(4,4,4-trifluorobutyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3S)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carbonitrile —— C16H23N3O2
6-[(3S)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carbonitrile
—— 6-[(3R)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carbonitrile —— C16H23N3O2
6-[(3R)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyridine-2-carbonitrile
—— (6-aminopyridin-3-yl)-[(4R)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl]methanone —— C22H28N4O
(6-aminopyridin-3-yl)-[(4R)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl]methanone
—— (6S)-N-cyclopentyl-2-[2-(1H-imidazol-5-yl)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C20H31N5O2
(6S)-N-cyclopentyl-2-[2-(1H-imidazol-5-yl)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— (6R)-4-(2,3-dihydro-1H-indene-5-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H27N3O2
(6R)-4-(2,3-dihydro-1H-indene-5-carbonyl)-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6S)-10-(cyclopropylmethyl)-1-methyl-4-[(1-methylimidazol-2-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C19H31N5O
(6S)-10-(cyclopropylmethyl)-1-methyl-4-[(1-methylimidazol-2-yl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-methyl-2-[[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1H-quinolin-4-one —— C19H22N4O2
6-methyl-2-[[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1H-quinolin-4-one
—— (6-aminopyridin-3-yl)-[(4S)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl]methanone —— C22H28N4O
(6-aminopyridin-3-yl)-[(4S)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl]methanone
—— 6-tert-butyl-4-[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-1H-pyrimidin-2-one —— C18H27N3O4
6-tert-butyl-4-[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl]-1H-pyrimidin-2-one
—— (6-methylimidazo[1,2-a]pyridin-2-yl)-[(1S)-1-pyridin-3-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H19N5O
(6-methylimidazo[1,2-a]pyridin-2-yl)-[(1S)-1-pyridin-3-yl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone