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—— (6S)-N-[(4R)-8-chloro-3,4-dihydro-2H-chromen-4-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C17H19ClN4O2
(6S)-N-[(4R)-8-chloro-3,4-dihydro-2H-chromen-4-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— [(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(1R)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H23N5O
[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(1R)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— 6-[4-(4-chlorophenoxy)-5-methyl-1,2-dihydropyrazol-3-ylidene]-4-ethyl-3-methoxycyclohexa-2,4-dien-1-one —— C19H19ClN2O3
6-[4-(4-chlorophenoxy)-5-methyl-1,2-dihydropyrazol-3-ylidene]-4-ethyl-3-methoxycyclohexa-2,4-dien-1-one
—— [(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(3R)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone —— C21H28N4O2
[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(3R)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone
—— (6R)-3-methyl-N-[(S)-phenyl(1,3-thiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C18H19N5OS
(6R)-3-methyl-N-[(S)-phenyl(1,3-thiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-N-(furan-2-ylmethyl)-3-methyl-N-(thiophen-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C18H20N4O2S
(6S)-N-(furan-2-ylmethyl)-3-methyl-N-(thiophen-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— 6-[(3S)-3-(azepan-1-ylmethyl)piperidin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine —— C18H28N6
6-[(3S)-3-(azepan-1-ylmethyl)piperidin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine
—— (6S)-N-[6-(benzimidazol-1-yl)pyridin-3-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H19N7O
(6S)-N-[6-(benzimidazol-1-yl)pyridin-3-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-N-[[4-(1,3-benzodioxol-5-yl)oxan-4-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C21H26N4O4
(6R)-N-[[4-(1,3-benzodioxol-5-yl)oxan-4-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— [(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(1R)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H23N5O
[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(1R)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— [(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(4S)-4-pyrazol-1-yl-3,4-dihydro-1H-isoquinolin-2-yl]methanone —— C20H22N6O
[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(4S)-4-pyrazol-1-yl-3,4-dihydro-1H-isoquinolin-2-yl]methanone
—— (6R)-N-[(4R)-8-chloro-3,4-dihydro-2H-chromen-4-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C17H19ClN4O2
(6R)-N-[(4R)-8-chloro-3,4-dihydro-2H-chromen-4-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-N-[6-(benzimidazol-1-yl)pyridin-3-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H19N7O
(6R)-N-[6-(benzimidazol-1-yl)pyridin-3-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— 6-[4-[(1R,2S,4S)-2-bicyclo[2.2.1]heptanyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine —— C17H24N6
6-[4-[(1R,2S,4S)-2-bicyclo[2.2.1]heptanyl]piperazin-1-yl]-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine
—— 6-[(5R)-5-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-1,2-oxazolidin-3-ylidene]cyclohexa-2,4-dien-1-one —— C17H20N2O5
6-[(5R)-5-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-1,2-oxazolidin-3-ylidene]cyclohexa-2,4-dien-1-one
—— [(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone —— C21H23N5O
[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(1S)-1-phenyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methanone
—— (6S)-N-[[5-(4-methoxyphenyl)-1,2,4-oxadiazol-3-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C18H20N6O3
(6S)-N-[[5-(4-methoxyphenyl)-1,2,4-oxadiazol-3-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-N-[4-chloro-2-(furan-2-carbonylamino)phenyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C19H18ClN5O3
(6R)-N-[4-chloro-2-(furan-2-carbonylamino)phenyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-N-[3-(3-methoxyphenyl)-1,2,4-thiadiazol-5-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C17H18N6O2S
(6S)-N-[3-(3-methoxyphenyl)-1,2,4-thiadiazol-5-yl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-3-methyl-N-[2-(1-phenylpyrazol-4-yl)ethyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C19H22N6O
(6S)-3-methyl-N-[2-(1-phenylpyrazol-4-yl)ethyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-N-[4-chloro-2-(furan-2-carbonylamino)phenyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C19H18ClN5O3
(6S)-N-[4-chloro-2-(furan-2-carbonylamino)phenyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C17H20N4O3
(6R)-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-N-(furan-2-ylmethyl)-3-methyl-N-(thiophen-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C18H20N4O2S
(6R)-N-(furan-2-ylmethyl)-3-methyl-N-(thiophen-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-3-methyl-N-[(R)-phenyl(1,3-thiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C18H19N5OS
(6R)-3-methyl-N-[(R)-phenyl(1,3-thiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-N,3-dimethyl-N-[3-(1-methyl-5-phenylpyrazol-3-yl)propyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C22H28N6O
(6S)-N,3-dimethyl-N-[3-(1-methyl-5-phenylpyrazol-3-yl)propyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-N-[(6-bromoimidazo[1,2-a]pyridin-2-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C16H17BrN6O
(6S)-N-[(6-bromoimidazo[1,2-a]pyridin-2-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-N-[(6-bromoimidazo[1,2-a]pyridin-2-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C16H17BrN6O
(6R)-N-[(6-bromoimidazo[1,2-a]pyridin-2-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— [(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(4R)-4-pyrazol-1-yl-3,4-dihydro-1H-isoquinolin-2-yl]methanone —— C20H22N6O
[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(4R)-4-pyrazol-1-yl-3,4-dihydro-1H-isoquinolin-2-yl]methanone
—— [(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(3R)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone —— C21H28N4O2
[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(3R)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone
—— 6-amino-4-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-2-sulfanylidene-1H-pyrimidine-5-carbonitrile —— C12H10N4O2S
6-amino-4-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-2-sulfanylidene-1H-pyrimidine-5-carbonitrile
—— [(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(3S)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone —— C21H28N4O2
[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-[(3S)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone
—— (6S)-N-[[4-(1,3-benzodioxol-5-yl)oxan-4-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C21H26N4O4
(6S)-N-[[4-(1,3-benzodioxol-5-yl)oxan-4-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6S)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C17H20N4O3
(6S)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— 6-[(3-chloroanilino)methylidene]-4-(diethylamino)cyclohexa-2,4-dien-1-one —— C17H19ClN2O
6-[(3-chloroanilino)methylidene]-4-(diethylamino)cyclohexa-2,4-dien-1-one
—— 6-bromo-1-[[(1,3,5-trimethylpyrazol-4-yl)amino]methylidene]naphthalen-2-one —— C17H16BrN3O
6-bromo-1-[[(1,3,5-trimethylpyrazol-4-yl)amino]methylidene]naphthalen-2-one
—— 6-[[[(1S,9aS)-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-yl]methylamino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C17H23N3O3
6-[[[(1S,9aS)-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-yl]methylamino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— 6-[(4-morpholin-4-ylsulfonylanilino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C17H17N3O6S
6-[(4-morpholin-4-ylsulfonylanilino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— 6-[[4-(1H-benzimidazol-2-yl)anilino]methylidene]-4-bromo-2-methoxycyclohexa-2,4-dien-1-one —— C21H16BrN3O2
6-[[4-(1H-benzimidazol-2-yl)anilino]methylidene]-4-bromo-2-methoxycyclohexa-2,4-dien-1-one
—— 6-[[4-(5-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C21H15N3O4
6-[[4-(5-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— 6-[[[2-(3-fluorophenyl)-1,3-benzoxazol-6-yl]amino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C20H12FN3O4
6-[[[2-(3-fluorophenyl)-1,3-benzoxazol-6-yl]amino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— 6-[(4-acetylanilino)methylidene]-3-ethoxycyclohexa-2,4-dien-1-one —— C17H17NO3
6-[(4-acetylanilino)methylidene]-3-ethoxycyclohexa-2,4-dien-1-one
—— 6-[4-(1-benzofuran-2-yl)-3-(trifluoromethyl)-2H-1,2-oxazol-5-ylidene]-3-methoxycyclohexa-2,4-dien-1-one —— C19H12F3NO4
6-[4-(1-benzofuran-2-yl)-3-(trifluoromethyl)-2H-1,2-oxazol-5-ylidene]-3-methoxycyclohexa-2,4-dien-1-one
—— 6-[[4-(6-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C21H15N3O4
6-[[4-(6-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— 6-tert-butyl-2-[(3S)-3-pyridin-3-yloxypyrrolidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole —— C17H21N5OS
6-tert-butyl-2-[(3S)-3-pyridin-3-yloxypyrrolidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole
—— 6-[(2,3-dihydro-1,4-benzodioxin-6-ylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C15H12N2O5
6-[(2,3-dihydro-1,4-benzodioxin-6-ylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6R)-N-(2-hydroxy-2-methylpropyl)-2-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C15H20F3N3O2
(6R)-N-(2-hydroxy-2-methylpropyl)-2-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide
—— [(6R)-2-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-6-yl]-piperidin-1-ylmethanone —— C16H20F3N3O
[(6R)-2-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-6-yl]-piperidin-1-ylmethanone
—— 6-(11-azatetracyclo[8.7.0.02,7.013,17]heptadeca-1(10),2,4,6,8,13(17)-hexaen-12-ylidene)cyclohexa-2,4-dien-1-one —— C22H17NO
6-(11-azatetracyclo[8.7.0.02,7.013,17]heptadeca-1(10),2,4,6,8,13(17)-hexaen-12-ylidene)cyclohexa-2,4-dien-1-one
—— 6-[[2-(3-fluorophenoxy)-5-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C20H13F4NO2
6-[[2-(3-fluorophenoxy)-5-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6S)-N-(2,2-dimethylpropyl)-N,2-dimethyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide —— C17H24F3N3O
(6S)-N-(2,2-dimethylpropyl)-N,2-dimethyl-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline-6-carboxamide