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—— 6-[(R)-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]quinoline —— C23H31N7
6-[(R)-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]quinoline
—— 6-deoxy-Tal(b1-3)[L-Tal(b1-4)]b-TalNAc —— C20H35NO15
6-deoxy-Tal(b1-3)[L-Tal(b1-4)]b-TalNAc
—— 6-methyl-3-[[[(1R)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C26H38N6O2
6-methyl-3-[[[(1R)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 6-deoxy-L-Gul(a1-3)[L-Tal(b1-4)]b-TalNAc —— C20H35NO15
6-deoxy-L-Gul(a1-3)[L-Tal(b1-4)]b-TalNAc
—— 6-deoxy-L-All(a1-3)[L-Tal(b1-4)]b-TalNAc —— C20H35NO15
6-deoxy-L-All(a1-3)[L-Tal(b1-4)]b-TalNAc
—— (6S)-N-(3-ethoxyphenyl)-2-[(Z)-1-(3-fluoro-4-methoxyphenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazinane-6-carboxamide —— C22H23FN4O4S
(6S)-N-(3-ethoxyphenyl)-2-[(Z)-1-(3-fluoro-4-methoxyphenyl)ethylidenehydrazinylidene]-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-7-cyclopropyl-1-N-(2-fluorophenyl)-6-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H26FN5O4
(6R)-7-cyclopropyl-1-N-(2-fluorophenyl)-6-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-benzyl-7-cyclopropyl-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C27H29N5O3
(6R)-1-N-benzyl-7-cyclopropyl-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-(3,4-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H35N5O4
(6S)-7-cyclopropyl-1-N-(3,4-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-(4-chlorophenyl)-7-cyclopropyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H23ClFN5O3
(6R)-1-N-(4-chlorophenyl)-7-cyclopropyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-1-N-(2-methylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C22H27N5O4
(6R)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-1-N-(2-methylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-(4-fluorophenyl)-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H23F2N5O3
(6R)-7-cyclopropyl-1-N-(4-fluorophenyl)-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-7-cyclopropyl-1-N-(4-ethoxyphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H31N5O4
(6R)-6-N-cyclopentyl-7-cyclopropyl-1-N-(4-ethoxyphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-1-N-(4-propan-2-ylphenyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C27H37N5O4
(6S)-7-cyclopropyl-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-1-N-(4-propan-2-ylphenyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-(2,5-difluorophenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H29F2N5O4
(6R)-7-cyclopropyl-1-N-(2,5-difluorophenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-(3,4-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H35N5O4
(6R)-7-cyclopropyl-1-N-(3,4-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-8-oxo-1-N-(4-propan-2-ylphenyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H31N5O4
(6S)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-8-oxo-1-N-(4-propan-2-ylphenyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-(4-ethylphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H29N5O4
(6S)-7-cyclopropyl-1-N-(4-ethylphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-1-N-(4-chlorophenyl)-7-cyclopropyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H23ClFN5O3
(6S)-1-N-(4-chlorophenyl)-7-cyclopropyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-(2-ethoxyphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H29N5O5
(6S)-7-cyclopropyl-1-N-(2-ethoxyphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-benzyl-1-N-[(3-chlorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H28ClN5O3
(6R)-6-N-benzyl-1-N-[(3-chlorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-ethyl-6-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C22H27N5O4
(6S)-7-cyclopropyl-1-N-ethyl-6-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-(2,6-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H35N5O4
(6S)-7-cyclopropyl-1-N-(2,6-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-cyclopropyl-1-N-(4-ethoxyphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H31N5O4
(6S)-6-N-cyclopentyl-7-cyclopropyl-1-N-(4-ethoxyphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-1-N-butyl-7-cyclopropyl-6-methyl-6-N-[(3-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H31N5O3
(6S)-1-N-butyl-7-cyclopropyl-6-methyl-6-N-[(3-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-butyl-7-cyclopropyl-6-methyl-6-N-[(3-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H31N5O3
(6R)-1-N-butyl-7-cyclopropyl-6-methyl-6-N-[(3-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-7-cyclopropyl-1-N-[(3-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H31N5O4
(6R)-6-N-cyclopentyl-7-cyclopropyl-1-N-[(3-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-(4-ethylphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H29N5O4
(6R)-7-cyclopropyl-1-N-(4-ethylphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-8-oxo-1-N-[4-(trifluoromethoxy)phenyl]-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C22H24F3N5O5
(6S)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-8-oxo-1-N-[4-(trifluoromethoxy)phenyl]-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-cyclopropyl-1-N-[(3-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H31N5O4
(6S)-6-N-cyclopentyl-7-cyclopropyl-1-N-[(3-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-7-cyclopropyl-1-N-(2-methoxy-5-methylphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H31N5O4
(6S)-6-N-cyclopentyl-7-cyclopropyl-1-N-(2-methoxy-5-methylphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N,6-dimethyl-6-N-[(4-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C21H25N5O3
(6R)-7-cyclopropyl-1-N,6-dimethyl-6-N-[(4-methylphenyl)methyl]-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-7-cyclopropyl-1-N-(2-methoxy-5-methylphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H31N5O4
(6R)-6-N-cyclopentyl-7-cyclopropyl-1-N-(2-methoxy-5-methylphenyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-(2-fluorophenyl)-6-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H26FN5O4
(6S)-7-cyclopropyl-1-N-(2-fluorophenyl)-6-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-(2-ethoxyphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H29N5O5
(6R)-7-cyclopropyl-1-N-(2-ethoxyphenyl)-6-N-(2-methoxyethyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— 6-fluoro-3-[3-[4-(trifluoromethyl)phenyl]-2H-1,2,4-oxadiazol-5-ylidene]quinolin-4-one —— C18H9F4N3O2
6-fluoro-3-[3-[4-(trifluoromethyl)phenyl]-2H-1,2,4-oxadiazol-5-ylidene]quinolin-4-one
—— (6S)-7-cyclopropyl-1-N-(4-fluorophenyl)-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H23F2N5O3
(6S)-7-cyclopropyl-1-N-(4-fluorophenyl)-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-8-oxo-1-N-[4-(trifluoromethoxy)phenyl]-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C22H24F3N5O5
(6R)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-8-oxo-1-N-[4-(trifluoromethoxy)phenyl]-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-1-N-(2-methylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C22H27N5O4
(6S)-7-cyclopropyl-6-N-(2-methoxyethyl)-6-methyl-1-N-(2-methylphenyl)-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-(2,6-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H35N5O4
(6R)-7-cyclopropyl-1-N-(2,6-dimethylphenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-7-cyclopropyl-1-N-ethyl-6-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C22H27N5O4
(6R)-7-cyclopropyl-1-N-ethyl-6-N-[(2-methoxyphenyl)methyl]-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-7-propyl-1-N-(2-thiophen-2-ylethyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H31N5O3S
(6R)-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-7-propyl-1-N-(2-thiophen-2-ylethyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-N-[(4-fluorophenyl)methyl]-6-methyl-1-(4-methylpiperazine-1-carbonyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-6-carboxamide —— C24H31FN6O3
(6R)-N-[(4-fluorophenyl)methyl]-6-methyl-1-(4-methylpiperazine-1-carbonyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-6-carboxamide
—— (6S)-1-N,1-N-diethyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H30FN5O3
(6S)-1-N,1-N-diethyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N,1-N-diethyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H30FN5O3
(6R)-1-N,1-N-diethyl-6-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-6-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-1-N-propan-2-yl-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H31N5O4
(6R)-6-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-1-N-propan-2-yl-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-7-cyclopropyl-1-N-(2,5-difluorophenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H29F2N5O4
(6S)-7-cyclopropyl-1-N-(2,5-difluorophenyl)-6-methyl-8-oxo-6-N-(3-propan-2-yloxypropyl)-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-benzyl-6-methyl-8-oxo-1-N-(2-phenylethyl)-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C27H31N5O3
(6S)-6-N-benzyl-6-methyl-8-oxo-1-N-(2-phenylethyl)-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-(azepane-1-carbonyl)-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-6-carboxamide —— C26H35N5O4
(6R)-1-(azepane-1-carbonyl)-N-[(4-methoxyphenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-6-carboxamide
—— (6R)-6-N-cyclopentyl-7-ethyl-1-N-(3-methoxypropyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C20H31N5O4
(6R)-6-N-cyclopentyl-7-ethyl-1-N-(3-methoxypropyl)-6-methyl-8-oxo-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide