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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-8-[2-(2-amino-6-oxo-1H-pyrimidin-4-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N5O3
(6R)-8-[2-(2-amino-6-oxo-1H-pyrimidin-4-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R,7S)-3-(hydroxymethyl)-8-oxo-7-(pyridine-4-carbonylamino)-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate —— C14H12N3O5S-
(6R,7S)-3-(hydroxymethyl)-8-oxo-7-(pyridine-4-carbonylamino)-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
—— (6R)-4-[1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl]-1,4-oxazepan-6-ol —— C18H31N5O2
(6R)-4-[1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl]-1,4-oxazepan-6-ol
—— (6S)-8-[2-(2-amino-6-oxo-1H-pyrimidin-4-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N5O3
(6S)-8-[2-(2-amino-6-oxo-1H-pyrimidin-4-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C20H21NO5S
(6,7-dimethyl-2-oxochromen-4-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— 6-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-1H-benzimidazole —— C18H18N2O2
6-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-1H-benzimidazole
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C20H21NO5S
(6,7-dimethyl-2-oxochromen-4-yl)methyl (3S,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— 6-[(3R)-3-(2-fluorophenyl)-3-phenylpropanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one —— C22H20FN3O2
6-[(3R)-3-(2-fluorophenyl)-3-phenylpropanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C20H21NO5S
(6,7-dimethyl-2-oxochromen-4-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (6R)-4-[3-(1,3-benzodioxol-5-yl)propanoyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H29N3O4
(6R)-4-[3-(1,3-benzodioxol-5-yl)propanoyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3S)-3-(2-fluorophenyl)-3-phenylpropanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one —— C22H20FN3O2
6-[(3S)-3-(2-fluorophenyl)-3-phenylpropanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C17H18ClNO5S
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— [(6S)-4-(5,11-dihydro-[1]benzoxepino[3,4-d]pyrimidin-1-yl)-1,4-oxazepan-6-yl]methanol —— C18H21N3O3
[(6S)-4-(5,11-dihydro-[1]benzoxepino[3,4-d]pyrimidin-1-yl)-1,4-oxazepan-6-yl]methanol
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C17H18ClNO5S
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C17H18N2O7S
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (3R,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (6-chloro-7-methyl-2-oxochromen-4-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C19H18ClNO5S
(6-chloro-7-methyl-2-oxochromen-4-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (6S)-2-(2-hydroxyethyl)-8-(1-methylindazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O3
(6S)-2-(2-hydroxyethyl)-8-(1-methylindazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-1H-benzimidazole —— C18H18N2O2
6-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-1H-benzimidazole
—— (6-ethyl-7-hydroxy-2-oxochromen-4-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C20H21NO6S
(6-ethyl-7-hydroxy-2-oxochromen-4-yl)methyl (3R,7aS)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(1-methyl-6-oxopyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O3
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(1-methyl-6-oxopyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-7-hydroxy-2-oxochromen-4-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C20H21NO6S
(6-ethyl-7-hydroxy-2-oxochromen-4-yl)methyl (3S,7aR)-7a-methyl-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— 6-chloro-4-[(3R)-3-[1-(cyclopropylmethyl)imidazol-2-yl]piperidin-1-yl]quinoline —— C21H23ClN4
6-chloro-4-[(3R)-3-[1-(cyclopropylmethyl)imidazol-2-yl]piperidin-1-yl]quinoline
—— (6S)-1-benzyl-4-(3-pyrrol-1-ylpropyl)-1,4-diazepan-6-ol —— C19H27N3O
(6S)-1-benzyl-4-(3-pyrrol-1-ylpropyl)-1,4-diazepan-6-ol
—— (6R)-2-(2-hydroxyethyl)-8-(1-methylindazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O3
(6R)-2-(2-hydroxyethyl)-8-(1-methylindazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[3-(1,3-benzodioxol-5-yl)propanoyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H29N3O4
(6S)-4-[3-(1,3-benzodioxol-5-yl)propanoyl]-1,10-dimethyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— [6-(methoxymethyl)pyridin-2-yl]-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C22H25N5O2
[6-(methoxymethyl)pyridin-2-yl]-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (6S)-8-(5-hydroxypyridine-2-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H27N3O3
(6S)-8-(5-hydroxypyridine-2-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2S)-2-(4-chlorophenyl)morpholine-4-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H18ClN3O4
6-[(2S)-2-(4-chlorophenyl)morpholine-4-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— [(6R)-4-(5,11-dihydro-[1]benzoxepino[3,4-d]pyrimidin-1-yl)-1,4-oxazepan-6-yl]methanol —— C18H21N3O3
[(6R)-4-(5,11-dihydro-[1]benzoxepino[3,4-d]pyrimidin-1-yl)-1,4-oxazepan-6-yl]methanol
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-pyridin-2-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O2
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-pyridin-2-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H18ClN3O4
6-[(2R)-2-(4-chlorophenyl)morpholine-4-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— [(6R)-4-benzyl-6-hydroxy-1,4-diazepan-1-yl]-[5-(methylsulfanylmethyl)furan-2-yl]methanone —— C19H24N2O3S
[(6R)-4-benzyl-6-hydroxy-1,4-diazepan-1-yl]-[5-(methylsulfanylmethyl)furan-2-yl]methanone
—— (6R)-8-(5-hydroxypyridine-2-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H27N3O3
(6R)-8-(5-hydroxypyridine-2-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-4-benzyl-6-hydroxy-1,4-diazepan-1-yl]-[5-(methylsulfanylmethyl)furan-2-yl]methanone —— C19H24N2O3S
[(6S)-4-benzyl-6-hydroxy-1,4-diazepan-1-yl]-[5-(methylsulfanylmethyl)furan-2-yl]methanone
—— (6R)-1,10-dimethyl-4-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H31N5O2
(6R)-1,10-dimethyl-4-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (6R)-5-(5-methyl-4-phenylthiophene-3-carbonyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H17N3O3S
(6R)-5-(5-methyl-4-phenylthiophene-3-carbonyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(1-methyl-6-oxopyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O3
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(1-methyl-6-oxopyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-5-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H19N3O3S
(6S)-5-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— [6-(methoxymethyl)pyridin-2-yl]-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C22H25N5O2
[6-(methoxymethyl)pyridin-2-yl]-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2R)-2-(4-chlorophenyl)sulfanylpropanoate —— C18H16ClNO6S
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2R)-2-(4-chlorophenyl)sulfanylpropanoate
—— (6R)-5-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H19N3O3S
(6R)-5-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-[6-methyl-4-[4-[(5-methyl-1H-imidazol-4-yl)methylamino]piperidin-1-yl]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C21H26N6O
6-[6-methyl-4-[4-[(5-methyl-1H-imidazol-4-yl)methylamino]piperidin-1-yl]-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2S
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-1,10-dimethyl-4-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one —— C20H31N5O2
(6S)-1,10-dimethyl-4-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1,4,10-triazaspiro[5.6]dodecan-9-one
—— 6-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-7H-purin-2-amine —— C18H24N8
6-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-7H-purin-2-amine
—— (6R)-1-benzyl-4-[3-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-6-ol —— C18H20F3N3O
(6R)-1-benzyl-4-[3-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-6-ol
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H25N5O2S
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-pyridin-2-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O2
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-pyridin-2-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-5-(5-methyl-4-phenylthiophene-3-carbonyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H17N3O3S
(6S)-5-(5-methyl-4-phenylthiophene-3-carbonyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-7H-purin-2-amine —— C18H24N8
6-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-7H-purin-2-amine