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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-methyl-N-[(3S)-1-(pyrazolo[1,5-b]pyridazine-3-carbonyl)pyrrolidin-3-yl]propanamide —— C15H19N5O2
2-methyl-N-[(3S)-1-(pyrazolo[1,5-b]pyridazine-3-carbonyl)pyrrolidin-3-yl]propanamide
—— 7-oxo-2-phenyl-N-[2-(3-thiophen-3-ylphenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20N4O2S
7-oxo-2-phenyl-N-[2-(3-thiophen-3-ylphenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 2-cyclohexyl-1-[4-(pyrazolo[1,5-b]pyridazine-3-carbonyl)piperazin-1-yl]ethanone —— C19H25N5O2
2-cyclohexyl-1-[4-(pyrazolo[1,5-b]pyridazine-3-carbonyl)piperazin-1-yl]ethanone
—— 6-[4-(cyclobutanecarbonyl)piperazine-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H23N5O3
6-[4-(cyclobutanecarbonyl)piperazine-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[3-(1H-benzimidazol-2-yl)propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H20N6O2
N-[3-(1H-benzimidazol-2-yl)propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]furan-2-carboxamide —— C22H19N5O4
N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]furan-2-carboxamide
—— 6-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H21N5O4
6-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[3-(4-fluorophenoxy)propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H19FN4O3
N-[3-(4-fluorophenoxy)propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[[1-(3-methylbutanoyl)piperidin-4-yl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H29N5O3
N-[[1-(3-methylbutanoyl)piperidin-4-yl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 6-[4-(4-chlorobenzoyl)-1,4-diazepane-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H22ClN5O3
6-[4-(4-chlorobenzoyl)-1,4-diazepane-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[[3-(cyclohexylmethoxy)phenyl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H28N4O3
N-[[3-(cyclohexylmethoxy)phenyl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[1-(2-cyclohexylacetyl)piperidin-4-yl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O3
N-[1-(2-cyclohexylacetyl)piperidin-4-yl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— [(2R)-1-(2,4-difluoroanilino)-1-oxopropan-2-yl] 5-cyclopropyl-2-phenylpyrazole-3-carboxylate —— C22H19F2N3O3
[(2R)-1-(2,4-difluoroanilino)-1-oxopropan-2-yl] 5-cyclopropyl-2-phenylpyrazole-3-carboxylate
—— 7-oxo-2-phenyl-N-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H21N5O3S
7-oxo-2-phenyl-N-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 6-(4-benzoyl-1,4-diazepane-1-carbonyl)-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H23N5O3
6-(4-benzoyl-1,4-diazepane-1-carbonyl)-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 1-[4-(pyrazolo[1,5-b]pyridazine-3-carbonyl)piperazin-1-yl]propan-1-one —— C14H17N5O2
1-[4-(pyrazolo[1,5-b]pyridazine-3-carbonyl)piperazin-1-yl]propan-1-one
—— 4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-propan-2-yl-1,4-diazepane-1-carboxamide —— C22H26N6O3
4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-propan-2-yl-1,4-diazepane-1-carboxamide
—— N-[2-[4-(cyclohexylmethoxy)phenyl]ethyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H30N4O3
N-[2-[4-(cyclohexylmethoxy)phenyl]ethyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3
N-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-oxo-2-phenyl-N-[2-(4-phenylmethoxyphenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24N4O3
7-oxo-2-phenyl-N-[2-(4-phenylmethoxyphenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]-2-phenylacetamide —— C25H23N5O3
N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]-2-phenylacetamide
—— N-[[3-[2-(cyclopropylamino)-2-oxoethyl]phenyl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H23N5O3
N-[[3-[2-(cyclopropylamino)-2-oxoethyl]phenyl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-cyclohexyl-4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)piperazine-1-carboxamide —— C24H28N6O3
N-cyclohexyl-4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)piperazine-1-carboxamide
—— 7-oxo-2-phenyl-N-[(2-propan-2-yloxyphenyl)methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22N4O3
7-oxo-2-phenyl-N-[(2-propan-2-yloxyphenyl)methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 1-cyclohexyl-3-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]urea —— C24H28N6O3
1-cyclohexyl-3-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]urea
—— 7-oxo-2-phenyl-N-[[4-(pyrrolidine-1-carbonyl)phenyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H23N5O3
7-oxo-2-phenyl-N-[[4-(pyrrolidine-1-carbonyl)phenyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[[1-(2,2-dimethylpropanoyl)piperidin-4-yl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H29N5O3
N-[[1-(2,2-dimethylpropanoyl)piperidin-4-yl]methyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 6-(4-methylsulfonylpiperazine-1-carbonyl)-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H19N5O4S
6-(4-methylsulfonylpiperazine-1-carbonyl)-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[1-(cyclohexanecarbonyl)piperidin-4-yl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3
N-[1-(cyclohexanecarbonyl)piperidin-4-yl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 6-[4-(cyclobutanecarbonyl)-1,4-diazepane-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H25N5O3
6-[4-(cyclobutanecarbonyl)-1,4-diazepane-1-carbonyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[2-(1,3-benzodioxol-5-yloxy)ethyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H18N4O5
N-[2-(1,3-benzodioxol-5-yloxy)ethyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-oxo-2-phenyl-N-[[2-(phenylmethoxymethyl)phenyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24N4O3
7-oxo-2-phenyl-N-[[2-(phenylmethoxymethyl)phenyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-oxo-2-phenyl-N-[2-(2-thiophen-2-ylphenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20N4O2S
7-oxo-2-phenyl-N-[2-(2-thiophen-2-ylphenyl)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]benzamide —— C24H21N5O3
N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]benzamide
—— 7-oxo-2-phenyl-N-[[4-(phenylmethoxymethyl)phenyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24N4O3
7-oxo-2-phenyl-N-[[4-(phenylmethoxymethyl)phenyl]methyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 3,3-dimethyl-N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]butanamide —— C23H27N5O3
3,3-dimethyl-N-[(3S)-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidin-3-yl]butanamide
—— N-[3-(furan-2-carbonylamino)propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H19N5O4
N-[3-(furan-2-carbonylamino)propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-(3-benzamidopropyl)-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H21N5O3
N-(3-benzamidopropyl)-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[3-(3,4-dihydro-2H-quinolin-1-yl)-3-oxopropyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H23N5O3
N-[3-(3,4-dihydro-2H-quinolin-1-yl)-3-oxopropyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[3-(2,3-dihydroindol-1-yl)-3-oxopropyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H21N5O3
N-[3-(2,3-dihydroindol-1-yl)-3-oxopropyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 2-phenyl-6-[4-(2-thiophen-3-ylacetyl)piperazine-1-carbonyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H21N5O3S
2-phenyl-6-[4-(2-thiophen-3-ylacetyl)piperazine-1-carbonyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (3S)-N-cyclopentyl-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide —— C24H27N5O3
(3S)-N-cyclopentyl-1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide
—— 7-oxo-2-phenyl-N-[2-(thiophene-2-carbonylamino)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H17N5O3S
7-oxo-2-phenyl-N-[2-(thiophene-2-carbonylamino)ethyl]-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-phenylpiperazine-1-carboxamide —— C24H22N6O3
4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-phenylpiperazine-1-carboxamide
—— N-[3-[(3-chlorobenzoyl)amino]propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H20ClN5O3
N-[3-[(3-chlorobenzoyl)amino]propyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-tert-butyl-4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)piperazine-1-carboxamide —— C22H26N6O3
N-tert-butyl-4-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)piperazine-1-carboxamide
—— N-[3-(3-chloroanilino)-3-oxopropyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H18ClN5O3
N-[3-(3-chloroanilino)-3-oxopropyl]-7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-(1,3-thiazol-2-yl)piperidine-4-carboxamide —— C22H20N6O3S
1-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-(1,3-thiazol-2-yl)piperidine-4-carboxamide
—— 5-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-propan-2-yl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C24H23N5O3S
5-(7-oxo-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carbonyl)-N-propan-2-yl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— 7-oxo-N-[[4-(2-oxo-2-piperidin-1-ylethyl)phenyl]methyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H27N5O3
7-oxo-N-[[4-(2-oxo-2-piperidin-1-ylethyl)phenyl]methyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide