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中文名称 英文名称 CAS号 化学式 结构式图片
—— [2-Bromo-4-methoxy-3-[(1-oxothian-1-ylidene)amino]phenyl]-[1-methyl-5-(naphthalen-2-ylmethoxy)pyrazol-4-yl]methanone 1207343-49-4 C28H28BrN3O4S
[2-Bromo-4-methoxy-3-[(1-oxothian-1-ylidene)amino]phenyl]-[1-methyl-5-(naphthalen-2-ylmethoxy)pyrazol-4-yl]methanone
—— 2,4-dimethyl-1-oxazol-2-ylmethyl-6-oxo-1,6-dihydro-pyridine-3-carboxylic acid 1310923-79-5 C12H12N2O4
2,4-dimethyl-1-oxazol-2-ylmethyl-6-oxo-1,6-dihydro-pyridine-3-carboxylic acid
—— phenylmethyl 4-{4-[6-amino-2-(butylamino)-8-(methyloxy)-9H-purin-9-yl]butyl}-1-piperidinecarboxylate 1208369-09-8 C27H39N7O3
phenylmethyl 4-{4-[6-amino-2-(butylamino)-8-(methyloxy)-9H-purin-9-yl]butyl}-1-piperidinecarboxylate
—— 2-(5-fluoro-4-hydroxy-1H-indol-3-yl)acetic acid 1227605-03-9 C10H8FNO3
2-(5-fluoro-4-hydroxy-1H-indol-3-yl)acetic acid
—— (2R)-2-[5-[[5-[4-(methylamino)piperidin-1-yl]pyridin-2-yl]amino]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-8-yl]propan-1-ol 1169697-41-9 C23H28N8O
(2R)-2-[5-[[5-[4-(methylamino)piperidin-1-yl]pyridin-2-yl]amino]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-8-yl]propan-1-ol
—— (2S)-2-[5-[[6-[(3S)-3-methylpiperazin-1-yl]pyridazin-3-yl]amino]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-8-yl]propan-1-ol 1169697-37-3 C21H25N9O
(2S)-2-[5-[[6-[(3S)-3-methylpiperazin-1-yl]pyridazin-3-yl]amino]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-8-yl]propan-1-ol
—— [(3S,4R)-4-(4-chloro-phenyl)-1-(1-cyclopropanecarbonyl-pyrrolidine-3-carbonyl)-pyrrolidin-3-yl]-methyl-carbamic acid 4-fluoro-phenyl ester 1310820-33-7 C27H29ClFN3O4
[(3S,4R)-4-(4-chloro-phenyl)-1-(1-cyclopropanecarbonyl-pyrrolidine-3-carbonyl)-pyrrolidin-3-yl]-methyl-carbamic acid 4-fluoro-phenyl ester
—— 2-(6-(5-(2-aminoacetamido)-1,3,4-thiadiazol-2-yloxy)-1-hydroxy-4-methyl-1,3-dhydrobenzo[c][1,2]oxaborol-3-yl)acetic acid 1265358-81-3 C14H15BN4O6S
2-(6-(5-(2-aminoacetamido)-1,3,4-thiadiazol-2-yloxy)-1-hydroxy-4-methyl-1,3-dhydrobenzo[c][1,2]oxaborol-3-yl)acetic acid
—— 6-[(3S,4R)-3-{[4-acetyl-5-(4-methoxyphenyl)-1,4-diazocan-1-yl]carbonyl}-4-(2,4-difluorophenyl)pyrrolidin-1-yl]pyridazine-3-carbonitrile 1207511-07-6 C31H32F2N6O3
6-[(3S,4R)-3-{[4-acetyl-5-(4-methoxyphenyl)-1,4-diazocan-1-yl]carbonyl}-4-(2,4-difluorophenyl)pyrrolidin-1-yl]pyridazine-3-carbonitrile
—— (2R)-N-[2-[(3S)-3-(3,4-dichlorophenyl)piperidin-3-yl]ethyl]-1,1,1-trifluoropropan-2-amine 1231957-41-7 C16H21Cl2F3N2
(2R)-N-[2-[(3S)-3-(3,4-dichlorophenyl)piperidin-3-yl]ethyl]-1,1,1-trifluoropropan-2-amine
—— methyl N-[[(5S)-3-[3-fluoro-4-[4-[2-[(2-methylimidazo[1,2-a]pyrazine-3-carbonyl)amino]acetyl]piperazin-1-yl]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]carbamate 1227685-94-0 C26H29FN8O6
methyl N-[[(5S)-3-[3-fluoro-4-[4-[2-[(2-methylimidazo[1,2-a]pyrazine-3-carbonyl)amino]acetyl]piperazin-1-yl]phenyl]-2-oxo-1,3-oxazolidin-5-yl]methyl]carbamate
—— (S)-7-(tert-butyldimethylsilyloxy)-3-methoxyheptanal 1185341-90-5 C14H30O3Si
(S)-7-(tert-butyldimethylsilyloxy)-3-methoxyheptanal
—— 3,4-Di-O-methyl-(-)-inosit 19647-43-9 C8H16O6
3,4-Di-O-methyl-(-)-inosit
—— methyl (5S,7R)-5,7-dihydroxyoct-2-ynoate 1141411-82-6 C9H14O4
methyl (5S,7R)-5,7-dihydroxyoct-2-ynoate
—— (R)-benzyl(5-phenylpent-1-en-3-yl)sulfane 1402974-72-4 C18H20S
(R)-benzyl(5-phenylpent-1-en-3-yl)sulfane
—— 3-(4-tert-butylphenyl)-5-(6-methoxynaphthalen-2-yl)-1H-pyrazole 1204427-40-6 C24H24N2O
3-(4-tert-butylphenyl)-5-(6-methoxynaphthalen-2-yl)-1H-pyrazole
—— (2R,5S)-1-(tert-butyloxycarbonyl)-5-(hydroxymethyl)-2-[2-(ethyloxycarbonyl)ethyl]pyrrolidine 1203491-23-9 C15H27NO5
(2R,5S)-1-(tert-butyloxycarbonyl)-5-(hydroxymethyl)-2-[2-(ethyloxycarbonyl)ethyl]pyrrolidine
—— N-[4-(2-methylimidazo[1,2-a]pyrimidin-3-yl)-1,3-thiazol-2-yl]-N-[4-(trifluoromethyl)phenyl]amine 1116555-62-4 C17H12F3N5S
N-[4-(2-methylimidazo[1,2-a]pyrimidin-3-yl)-1,3-thiazol-2-yl]-N-[4-(trifluoromethyl)phenyl]amine
—— 1-ethyl-6,7-difluoro-3-(4-fluorophenyl)quinoxalin-2(1H)-one 1186527-63-8 C16H11F3N2O
1-ethyl-6,7-difluoro-3-(4-fluorophenyl)quinoxalin-2(1H)-one
—— 17-(2,6-dimethoxy-pyrimidin-4-yloxy)-13-methyl-2,14-dioxo-3,13-diaza-tricyclo[13.3.0.0*4,6*]octadec-7-ene-4-carboxylic acid ethyl ester 1044560-84-0 C26H36N4O7
17-(2,6-dimethoxy-pyrimidin-4-yloxy)-13-methyl-2,14-dioxo-3,13-diaza-tricyclo[13.3.0.0*4,6*]octadec-7-ene-4-carboxylic acid ethyl ester
—— tert-butyl N-[[2-(2-chloro-4-methoxybenzoyl)-3-oxocyclohexen-1-yl]amino]-N-methylcarbamate 1356597-11-9 C20H25ClN2O5
tert-butyl N-[[2-(2-chloro-4-methoxybenzoyl)-3-oxocyclohexen-1-yl]amino]-N-methylcarbamate
—— 1-(Cyclopropanesulfonyl)-1,4-diazepane hydrochloride 1403952-62-4 C8H17ClN2O2S
1-(Cyclopropanesulfonyl)-1,4-diazepane hydrochloride
—— (4-{6-[(2-morpholin-4-ylethylcarbamoyl)methyl]-7-oxo-3-phenyl-2,6,7,8-tetrahydro-4H-pyrazolo[3,4-e][1,4]thiazepin-4-yl}phenoxy)acetic acid methyl ester 1221172-85-5 C29H33N5O6S
(4-{6-[(2-morpholin-4-ylethylcarbamoyl)methyl]-7-oxo-3-phenyl-2,6,7,8-tetrahydro-4H-pyrazolo[3,4-e][1,4]thiazepin-4-yl}phenoxy)acetic acid methyl ester
—— 7-tert-butyl-3-(3-cyanophenyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-b]quinoline-2-carboxamide 1036650-75-5 C23H24N4O
7-tert-butyl-3-(3-cyanophenyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-b]quinoline-2-carboxamide
—— 3-(2-Methoxyphenyl)-5,5-dimethyl-1-[(2-phenoxyphenyl)methyl]imidazolidine-2,4-dione 1181079-38-8 C25H24N2O4
3-(2-Methoxyphenyl)-5,5-dimethyl-1-[(2-phenoxyphenyl)methyl]imidazolidine-2,4-dione
—— (2S)-N-[(3,5-difluorophenyl)methyl]-3,3,3-trifluoro-2-methyl-N-[2-[[(2S)-1'-methyl-2',4'-dioxospiro[1,3-dihydroindene-2,5'-imidazolidine]-5-yl]amino]-2-oxoethyl]-2-phenylmethoxypropanamide 1072446-24-2 C32H29F5N4O5
(2S)-N-[(3,5-difluorophenyl)methyl]-3,3,3-trifluoro-2-methyl-N-[2-[[(2S)-1'-methyl-2',4'-dioxospiro[1,3-dihydroindene-2,5'-imidazolidine]-5-yl]amino]-2-oxoethyl]-2-phenylmethoxypropanamide
—— 3-[4-(6-oxo-1H-pyridazin-3-yl)-2-(trifluoromethyl)phenyl]-1,3-thiazolidine-2,4-dione 1187874-27-6 C14H8F3N3O3S
3-[4-(6-oxo-1H-pyridazin-3-yl)-2-(trifluoromethyl)phenyl]-1,3-thiazolidine-2,4-dione
—— N-(2-(4-(dimethylamino)-4-phenylcyclohexyl)ethyl)-2-((1-(4-methoxy-2,6-dimethylphenylsulfonyl)piperidin-2-yl)methoxy)-N-methylacetamide 1187962-11-3 C34H51N3O5S
N-(2-(4-(dimethylamino)-4-phenylcyclohexyl)ethyl)-2-((1-(4-methoxy-2,6-dimethylphenylsulfonyl)piperidin-2-yl)methoxy)-N-methylacetamide
—— propane-1-sulfonic acid {2-fluoro-3-[hydroxy-(4-isopropylamino-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-methyl]-phenyl}-amide 1309432-12-9 C19H24FN5O3S
propane-1-sulfonic acid {2-fluoro-3-[hydroxy-(4-isopropylamino-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-methyl]-phenyl}-amide
—— 3-azido-1-cyclopentene-1,2-dicarboxylic acid dimethylester 149140-92-1 C9H11N3O4
3-azido-1-cyclopentene-1,2-dicarboxylic acid dimethylester
—— {3-[4-Benzo[1,3]dioxol-5-yl-2-hydroxy-2-(4-methoxyphenyl)-5-oxo-2,5-dihydro-furan-3-ylmethyl]phenyl}-acetic acid methyl ester 169805-08-7 C28H24O8
{3-[4-Benzo[1,3]dioxol-5-yl-2-hydroxy-2-(4-methoxyphenyl)-5-oxo-2,5-dihydro-furan-3-ylmethyl]phenyl}-acetic acid methyl ester
—— 5-[4-(3,3,3-Triphenylpropoxy)phenyl]-1H-tetrazole 193282-85-8 C28H24N4O
5-[4-(3,3,3-Triphenylpropoxy)phenyl]-1H-tetrazole
—— US8653087, III-148 1213244-33-7 C31H30F3N9O2
US8653087, III-148
—— 4-fluoro-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide 1150462-69-3 C34H31F4N5O5S
4-fluoro-N-[6-(1-methyl-2-{4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl}-1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide
—— ethyl (2S)-2-[[methyl(propan-2-yl)carbamoyl]amino]-4-morpholin-4-ylbutanoate 1383570-32-8 C15H29N3O4
ethyl (2S)-2-[[methyl(propan-2-yl)carbamoyl]amino]-4-morpholin-4-ylbutanoate
—— 3-fluoro-4-[[5-fluoro-7-[1-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]piperidin-4-yl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-N,N-dimethylbenzamide 1236284-35-7 C24H26F2N8O3
3-fluoro-4-[[5-fluoro-7-[1-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]piperidin-4-yl]pyrrolo[2,3-d]pyrimidin-4-yl]amino]-N,N-dimethylbenzamide
—— 2-[4-(3-{1-[4-(5-amino-3-methyl-pyrazin-2-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]-N,N-dimethyl-acetamide 1360551-33-2 C25H28N8O2
2-[4-(3-{1-[4-(5-amino-3-methyl-pyrazin-2-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]-N,N-dimethyl-acetamide
—— 2-(5,6-dimethoxypyridin-3-yl)-6-[1-[2-(5-methylpyrazol-1-yl)ethyl]pyrazol-4-yl]-7H-pyrrolo[3,4-b]pyridin-5-one 1315536-27-6 C23H23N7O3
2-(5,6-dimethoxypyridin-3-yl)-6-[1-[2-(5-methylpyrazol-1-yl)ethyl]pyrazol-4-yl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— 5-Amino-4-(N-((methoxycarbonyl)methyl)carbamoyl)-1-(2,3,5-tri-O-benzoyl-β-D-ribofuranosyl)imidazole 129966-73-0 C33H30N4O10
5-Amino-4-(N-((methoxycarbonyl)methyl)carbamoyl)-1-(2,3,5-tri-O-benzoyl-β-D-ribofuranosyl)imidazole
—— (Z)-1,3-diphenyl-4-octen-6-yne-1-one 151259-79-9 C20H18O
(Z)-1,3-diphenyl-4-octen-6-yne-1-one
—— dihydroligujapone 130848-40-7 C14H18O2
dihydroligujapone
—— L-Phenylalanin-methylamid-acetat 15368-71-5 C2H4O2*C10H14N2O
L-Phenylalanin-methylamid-acetat
—— 9-cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-6-ol 1169692-41-4 C23H26N8O
9-cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-9H-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-6-ol
—— 4-(1-Pyridin-3-ylpyrazol-4-yl)pyrimidine 1292295-70-5 C12H9N5
4-(1-Pyridin-3-ylpyrazol-4-yl)pyrimidine
—— 3-hydroxy-4-methyl-3-pyrimidin-5-yl-1-(2-trifluoromethoxyphenyl)-pent-1-yne 131910-57-1 C17H15F3N2O2
3-hydroxy-4-methyl-3-pyrimidin-5-yl-1-(2-trifluoromethoxyphenyl)-pent-1-yne
—— propyl [3-({4-oxo-1-[1-(tetrahydro-2H-puran-4-ylmethyl)-1H-pyrazol-4-yl]-1,4-dihydropyridazin-3-yl}methyl)phenyl]carbamate 1314381-58-2 C24H29N5O4
propyl [3-({4-oxo-1-[1-(tetrahydro-2H-puran-4-ylmethyl)-1H-pyrazol-4-yl]-1,4-dihydropyridazin-3-yl}methyl)phenyl]carbamate
—— 5-({[9-(3-fluorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]carbonyl}amino)-2,2-dimethylpentanoic acid 1354803-82-9 C25H29FN4O3
5-({[9-(3-fluorobenzyl)-5,6,8,9-tetrahydro-7H-pyrido[4',3':4,5]pyrrolo[2,3-b]pyridin-7-yl]carbonyl}amino)-2,2-dimethylpentanoic acid
—— N-(2-aminoethyl)-4-chloro-3-methylbenzamide 1252974-34-7 C10H13ClN2O
N-(2-aminoethyl)-4-chloro-3-methylbenzamide
—— 2-chloro-5-((dimethylamino)methyl)-N-(6-(methylsulfonyl)benzo[d]thiazol-2-ylcarbamoyl)benzamide 1143024-40-1 C19H19ClN4O4S2
2-chloro-5-((dimethylamino)methyl)-N-(6-(methylsulfonyl)benzo[d]thiazol-2-ylcarbamoyl)benzamide
—— 2-(4-acetylpiperazin-1-yl)-4-[2-ethyl-2-(4-methylphenyl)hydrazino]-6-isopropyl-5,6-dihydro-7H-pyrrolo[3,4-d]pyrimidin-7-one 1079653-87-4 C24H33N7O2
2-(4-acetylpiperazin-1-yl)-4-[2-ethyl-2-(4-methylphenyl)hydrazino]-6-isopropyl-5,6-dihydro-7H-pyrrolo[3,4-d]pyrimidin-7-one