申请人:Université de Bordeaux I
公开号:EP2881398A1
公开(公告)日:2015-06-10
The present invention provides a process for the preparation of aminoarylborane compounds and derivatives thereof comprising a step of arylation by reacting an aryl chloride with an aminoborane compound in the presence of a catalytic system.
Typically, the transformation comprises, converting Aryl-chloride Ar-Cl with an aminoborane such as
into an aminoarylborane compound of the following formula:
本发明提供了一种制备氨基芳基硼化合物及其衍生物的方法,包括通过在催化体系存在下,将芳基氯化物与氨基硼烷化合物反应进行芳基化的步骤。通常,该转化包括将芳基氯化物Ar-Cl与氨基硼烷化合物反应,转化为以下式的氨基芳基硼化合物: