1,2-二甲基-3,3a,4,5,6,6a-六氢-2H-环戊并[b]吡咯 | 74195-76-9

• 分子结构分类: 有机化合物 - 有机杂环化合物 - 吡咯烷类
• 中文名称: 1,2-二甲基-3,3a,4,5,6,6a-六氢-2H-环戊并[b]吡咯
• 英文名称: 1,2-Dimethyl-2,3,3a,6a-tetrahydrocyclopenta(b)pyrrole
• 英文别名: 1,2-dimethyl-3,3a,4,5,6,6a-hexahydro-2H-cyclopenta[b]pyrrole
• CAS: 74195-76-9
• 化学式: C₉H₁₇N
• 分子量: 139.24
• InChiKey: RDFOURSPNBBXIY-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  2
• 重原子数：
  10
• 可旋转键数：
  0
• 环数：
  2.0
• sp3杂化的碳原子比例：
  1.0
• 拓扑面积：
  3.2
• 氢给体数：
  0
• 氢受体数：
  1

文献信息

• ANTIVIRAL COMPOUNDS
  申请人：Gilead Sciences, Inc.

  公开号：US20140178336A1

  公开（公告）日：2014-06-26

  The disclosure is related to anti-viral compounds, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.

  该披露涉及抗病毒化合物，含有这种化合物的组合物，包括给予这种化合物的治疗方法，以及用于制备这种化合物的有用过程和中间体。
• Biphenyl-Substituted Cyclic Ketoenols
  申请人：FISCHER Reiner

  公开号：US20110230346A1

  公开（公告）日：2011-09-22

  The invention relates to novel compounds of the formula (I) in which W, X, Y, Z, and CKE have the meanings given above, to a plurality of processes and intermediates for their preparation and to their use as pesticides and/or herbicides and/or fungicides. Moreover, the invention relates to selectively herbicidal compositions comprising, firstly, the biphenyl-substituted cyclic ketoenols and, secondly, a crop plant compatibility-improving compound. The present invention furthermore relates to the boosting of the action of crop protection compositions comprising in particular biphenyl-substituted cyclic ketoenols through the addition of ammonium or phosphium salts and optionally penetrants, to the corresponding compositions, to processes for their preparation and to their use in crop protection as insecticides and/or nematicides and/or acaricides and/or fungicides and/or for preventing unwanted plant growth.

  该发明涉及以下式(I)的新化合物，其中W、X、Y、Z和CKE具有上述给定的含义，涉及它们的制备的多种过程和中间体，以及它们作为杀虫剂和/或除草剂和/或杀菌剂的用途。此外，该发明涉及包括第一，二苯基取代的环状酮烯醇和第二，一种改善作物植物相容性的化合物的选择性除草剂组合物。本发明还涉及通过添加铵盐或磷盐和可选的渗透剂，提高尤其是二苯基取代的环状酮烯醇的作物保护组合物的作用，以及相应的组合物、其制备的过程以及它们在作物保护中作为杀虫剂和/或线虫剂和/或螨虫剂和/或杀菌剂以及用于防止不受欢迎的植物生长的用途。
• Haloalkylmethyleneoxyphenyl-substituted ketoenols
  申请人：Fischer Reiner

  公开号：US20100311593A1

  公开（公告）日：2010-12-09

  The invention relates to novel compounds of the formula (I), in which W, X, Y, Z and CKE are each as defined above, to several methods and intermediates for preparation thereof and to the use thereof as pesticides and/or herbicides. The invention also relates to selective herbicidal compositions which comprise firstly haloalkylmethyleneoxyphenyl-substituted ketoenols and secondly a compound which improves crop plant compatibility. The present invention further relates to the enhancement of the action of crop protection compositions comprising especially haloalkylmethyleneoxyphenyl-substituted ketoenols, by the addition of ammonium or phosphonium salts and optionally penetration enhancers, to the corresponding compositions, to methods for production thereof and to the use thereof in crop protection as insecticides and/or acaricides and/or for preventing undesired plant growth.

  该发明涉及公式（I）中的新化合物，其中W、X、Y、Z和CKE各自如上所定义，以及其制备的几种方法和中间体，以及将其用作杀虫剂和/或除草剂的用途。该发明还涉及选择性除草剂组合物，其首先包括卤代烷基亚甲氧基苯基取代酮烯醇，其次包括改善作物植物相容性的化合物。本发明还涉及通过添加铵盐或磷盐以及必要时的渗透增效剂，增强特别是卤代烷基亚甲氧基苯基取代酮烯醇的作物保护组合物的作用，以及相应组合物的制备方法和将其用于作物保护作为杀虫剂和/或螨虫剂和/或预防不受欢迎的植物生长。
• CYCLOALKYLPHENYL SUBSTITUTED CYCLIC KETOENOLS
  申请人：Fischer Reiner

  公开号：US20090305891A1

  公开（公告）日：2009-12-10

  The disclosure relates to novel cycloalkylphenyl-substituted cyclic ketoenols of the formula (I) in which J, X, Y, m and CKE are as defined above, to processes and intermediates for their preparation and to their use as pesticides and/or herbicides. Moreover, the disclosure relates to selective herbicidal compositions comprising, firstly, the cycloalkylphenyl-substituted cyclic ketoenols and, secondly, a crop plant compatibility-improving compound. The disclosure furthermore relates to increasing the activity of crop protection compositions comprising compounds of the formula (I) by adding ammonium or phosphonium salts and, if appropriate, penetrants.

  该披露涉及到具有以下结构的新型环烷基苯基取代的环状酮烯醇（I）的公式，其中J、X、Y、m和CKE的定义如上所述，以及它们的制备过程和中间体，以及它们作为杀虫剂和/或除草剂的用途。此外，该披露涉及包括第一部分为环烷基苯基取代的环状酮烯醇和第二部分为作物植物相容性改进化合物的选择性除草剂组合物。该披露还涉及通过添加铵盐或膦盐以及必要时渗透剂来增加公式（I）化合物的作物保护组合物的活性。
• Trifluromethoxyphenyl-Substituted Tetramic Acid Derivatives Pesticides and/or Herbicides
  申请人：Fischer Reiner

  公开号：US20120015807A1

  公开（公告）日：2012-01-19

  The present invention relates to novel trifluoromethoxyphenyl-substituted tetramic acid derivatives of the formula (I), in which J, X, Y, A, B, D and G have the meanings given above, to a number of processes for their preparation, and to their use as pesticides and/or herbicides. The invention further provides selective herbicidal compositions which comprise, firstly, trifluoromethoxyphenyl-substituted tetramic acid derivatives and, secondly, a crop plant compatibility-improving compound. The invention further relates to the boosting of the action of crop protection compositions comprising compounds of the formula (I) through the additions of ammonium salts or phosphonium salts and optionally penetrants.

  本发明涉及一种新型的三氟甲氧基苯基取代的四酰胺酸衍生物，其化学式为(I)，其中J、X、Y、A、B、D和G具有上述给定的含义，以及它们的制备方法，以及它们作为杀虫剂和/或除草剂的用途。该发明进一步提供了选择性除草剂组合物，其包括首先为三氟甲氧基苯基取代的四酰胺酸衍生物，其次为一种改善作物植物兼容性的化合物。该发明还涉及通过添加铵盐或磷盐以及可选的渗透剂来增强化合物(I)的作物保护组合物的作用。