N-(2-carbamoyl-4-cyano-6-methylphenyl)-2-(3-chloropyridin-2-yl)-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide | 1229654-71-0

• 分子结构分类: 有机化合物 - 苯类化合物 - 苯和取代衍生物
• 英文名称: N-(2-carbamoyl-4-cyano-6-methylphenyl)-2-(3-chloropyridin-2-yl)-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide
• CAS: 1229654-71-0
• 化学式: C₂₁H₁₄ClF₃N₁₀O₂
• 分子量: 530.856
• InChiKey: SLEBRVSWNGIMJO-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  3.2
• 重原子数：
  37
• 可旋转键数：
  6
• 环数：
  4.0
• sp3杂化的碳原子比例：
  0.14
• 拓扑面积：
  170
• 氢给体数：
  2
• 氢受体数：
  11

文献信息

• METHOD FOR PRODUCING SUBSTITUTED ANTHRANILIC ACID DERIVATIVES
  申请人：BAYER INTELLECTUAL PROPERTY GMBH

  公开号：US20150011772A1

  公开（公告）日：2015-01-08

  The present invention relates to a process for preparing substituted anthranilic acid derivatives of the formula (I) in which R 1 , R 2 , R 3 and R 4 are each as defined in the description, by conversion of compounds of the general formula (IV) in the presence of a palladium catalyst and carbon monoxide. The present invention likewise relates to compounds of the general formula (IV).

  本发明涉及一种制备式（I）的取代蒽酸衍生物的方法，其中R1、R2、R3和R4的定义如描述中所述，通过在钯催化剂和一氧化碳存在下转化通式（IV）化合物。本发明还涉及通式（IV）的化合物。
• Tetrazole-substituted anthranilamides as pesticides
  申请人：Fischer Rüdiger

  公开号：US20100256195A1

  公开（公告）日：2010-10-07

  The present invention relates to tetrazole-substituted anthranilamides of the formula (I) in which R 1 , R 2 , R 3 R 4 , R 5 , n, X and Q have the meanings given in the description—and to their use as insecticides and/or acaricides, also in combination with other agents such as penetrants and/or ammonium salts or phosphonium salts.

  本发明涉及公式（I）中的四唑取代的蒽酰胺，其中R1，R2，R3R4，R5，n，X和Q具有说明书中给出的含义，并且它们的用途是作为杀虫剂和/或杀螨剂，也可以与其他剂如渗透剂和/或铵盐或膦盐组合使用。
• Tetrazolsubstituierte Anthranilsäureamide als Pestizide
  申请人：Bayer CropScience AG

  公开号：EP2484676A2

  公开（公告）日：2012-08-08

  Die vorliegende Erfindung betrifft tetrazolsubstituierte Anthranilsäureamide der Formel (I) - in welcher R1, R2, R3 R4, R5 n, X und Q die in der Beschreibung angegebenen Bedeutungen haben - und ihre Verwendung als Insektizide und / oder Akarizide auch in Kombination mit weiteren Mitteln wie Penetrationsförderern und/oder Ammonium-oder Phoshoniumsalzen.

  本发明涉及式（I）的四唑取代的蒽酸酰胺 - 其中 R1、R2、R3、R4、R5 n、X 和 Q 的含义见说明 - 以及它们作为杀虫剂和/或杀螨剂的用途，也可与其他药剂如渗透促进剂和/或铵盐或磷鎓盐结合使用。
• Active ingredient combinations having insecticidal and acaricidal properties
  申请人：FUNKE Christian

  公开号：US20110311503A1

  公开（公告）日：2011-12-22

  The novel active ingredient combinations which consist of the compounds of the formula (I) in combination with further active insecticidal ingredients (II) are very suitable for control of animal pests such as insects and/or unwanted acarids.
• Anthranilamides in combination with fungicides
  申请人：FUNKE Christian

  公开号：US20120010073A1

  公开（公告）日：2012-01-12

  The present invention relates to novel active compound combinations which include of the insecticidally active compounds of the formula (I) in combination with fungicidally active compounds (II) and are highly suitable for controlling unwanted animal pests, such as insects, and unwanted phytopathogenic fungi.