8-chloro-N-(2-chloro-5-methylphenyl)sulfonyl-6-methylimidazo[1,2-a]pyridine-2-carboxamide

• 分子结构分类: 有机化合物 - 苯类化合物 - 苯和取代衍生物
• 英文名称: 8-chloro-N-(2-chloro-5-methylphenyl)sulfonyl-6-methylimidazo[1,2-a]pyridine-2-carboxamide
• 化学式: C₁₆H₁₃Cl₂N₃O₃S
• 分子量: 398.3
• InChiKey: JFORRFOSLLRFPA-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  4.5
• 重原子数：
  25
• 可旋转键数：
  3
• 环数：
  3.0
• sp3杂化的碳原子比例：
  0.12
• 拓扑面积：
  88.9
• 氢给体数：
  1
• 氢受体数：
  4

文献信息

• SOLID FORMS OF NEMATOCIDAL SULFONAMIDES
  申请人：E I DU PONT DE NEMOURS AND COMPANY

  公开号：US20140228393A1

  公开（公告）日：2014-08-14

  Disclosed are solid forms of 8-chloro-N-[(2-chloro-5-methoxyphenyl)sulfonyl]-6-(trifluoromethyl)-imidazo[1,2-a]pyridine-2-carboxamide (Compound 1). Methods for the preparation of solid forms of Compound 1 and for the conversion of one solid form of Compound 1 into another are disclosed. Disclosed are nematocidal compositions comprising a nematocidally effective amount of a solid form of Compound 1 and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid carriers. Compositions comprising a mixture of a solid form of Compound 1 and at least one other nematicide, insecticide and/or fungicide are also disclosed. Also disclosed are methods for protecting a plant from nematodes comprising applying to the plant, or portion, or seed thereof, or to the growing medium of the plant, a nematocidally effective amount of Compound 1 comprising the polymorph Form A.

  本发明涉及8-氯-N-[(2-氯-5-甲氧苯基)磺酰基]-6-(三氟甲基)咪唑[1,2-a]吡啶-2-羧酰胺（化合物1）的固态形式。本发明还公开了制备化合物1固态形式的方法，以及将化合物1的一种固态形式转化为另一种固态形式的方法。本发明还公开了含有化合物1固态形式的杀线虫组合物，其中该组合物包括一种线虫杀效果有效量的化合物1固态形式和至少一种选自表面活性剂、固态稀释剂和液体载体的其他成分。本发明还公开了含有化合物1固态形式和至少一种其他线虫杀剂、杀虫剂和/或杀菌剂的混合物的组合物。本发明还公开了一种保护植物免受线虫侵害的方法，包括将化合物1的多晶形式A的线虫杀效果有效量施用于植物、其部分或种子，或施用于植物的生长介质。
• METHOD FOR CONTROLLING PESTS
  申请人：Sumitomo Chemical Company, Limited

  公开号：US20170208811A1

  公开（公告）日：2017-07-27

  A method is provided which exhibits an excellent controlling effect on pests. The method includes a step of performing a soil incorporation treatment with a granule containing one or more compounds selected from the following compound group (A) and one or more compounds selected from the following compound group (B). Compound group (A) is a group consisting of clothianidin, thiamethoxam, imidacloprid, and fipronil, and Compound group (B) is a group consisting of fluopyram and a compound represented by the following formula (1)
• US9040554B2
  申请人：——

  公开号：US9040554B2

  公开（公告）日：2015-05-26