Fluoro 4-azido-2,3,5-trifluoro-6-phenylbenzoate

• 分子结构分类: 有机化合物 - 苯类化合物 - 苯和取代衍生物
• 英文名称: Fluoro 4-azido-2,3,5-trifluoro-6-phenylbenzoate
• 英文别名: fluoro 4-azido-2,3,5-trifluoro-6-phenylbenzoate
• 化学式: C13H5F4N3O2
• 分子量: 311.19
• InChiKey: CXZIPQLKDSCGRZ-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  5.2
• 重原子数：
  22
• 可旋转键数：
  3
• 环数：
  2.0
• sp3杂化的碳原子比例：
  0.0
• 拓扑面积：
  40.7
• 氢给体数：
  0
• 氢受体数：
  8

文献信息

• [EN] COMPOUNDS AND BIOLOGICAL MATERIALS AND USES THEREOF<br/>[FR] MATÉRIAUX BIOLOGIQUES ET COMPOSÉS, ET UTILISATIONS CORRESPONDANTES
  申请人：PHOTOBIOTICS LTD

  公开号：WO2010106341A1

  公开（公告）日：2010-09-23

  The invention provides compounds of Formula (I): wherein b, D, R1, R2, G, Ra and Rb have meanings given in the description, or pharmaceutically-acceptable salts or solvates, or pharmaceutically functional derivatives thereof. The invention further provides process for conjugating the compounds to carrier molecules and uses of such compounds and conjugates in the treatment of disease.

  该发明提供了Formula (I)的化合物：其中b，D，R1，R2，G，Ra和Rb的含义如描述中所述，或其在药学上可接受的盐或溶剂，或其药学功能衍生物。该发明还提供了将这些化合物与载体分子结合的方法以及在治疗疾病中使用这些化合物和结合物的方法。
• COMPOUNDS AND BIOLOGICAL MATERIALS AND USES THEREOF
  申请人：Yahioglu Gokhan

  公开号：US20120070377A1

  公开（公告）日：2012-03-22

  The invention provides compounds of Formula (I): wherein b, D, R 1 , R 2 , G, R a and R b have meanings given in the description, or pharmaceutically-acceptable salts or solvates, or pharmaceutically functional derivatives thereof. The invention further provides process for conjugating the compounds to carrier molecules and uses of such compounds and conjugates in the treatment of disease.

  本发明提供公式（I）的化合物：其中b，D，R1，R2，G，Ra和Rb具有描述中给出的含义，或其药学上可接受的盐或溶剂或药学上的功能衍生物。本发明还提供将该化合物与载体分子结合的过程以及在治疗疾病中使用这些化合物和结合物的用途。
• CONJUGATES OF PHOTOSENSITISERS AND ANTIBODy-FRAGMENTS
  申请人：Photobiotics Limited

  公开号：EP1933875B1

  公开（公告）日：2014-02-19
• CONJUGATES OF PHOTOSENSITISERS AND ANTIBODIES
  申请人：Photobiotics Limited

  公开号：EP1933875A2

  公开（公告）日：2008-06-25
• BIOLOGICAL MATERIALS AND USES THEREOF
  申请人：Deonarain Mahendra

  公开号：US20090053247A1

  公开（公告）日：2009-02-26

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