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—— 6-[(5R,10bS)-9-bromo-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid —— C26H23BrN2O6
6-[(5R,10bS)-9-bromo-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid
—— (6R,9R)-6-(4-tert-butylphenyl)-9-(4-methoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C32H31F3N2O3
(6R,9R)-6-(4-tert-butylphenyl)-9-(4-methoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(5S,10bS)-2-(4-phenylsulfanylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid —— C31H26N2O5S
6-[(5S,10bS)-2-(4-phenylsulfanylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid
—— 6-[(5R,10bR)-9-bromo-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid —— C26H23BrN2O6
6-[(5R,10bR)-9-bromo-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid
—— (6S)-5-benzoyl-9,9-dimethyl-6-[5-(2-methyl-4-nitrophenyl)furan-2-yl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C33H29N3O5
(6S)-5-benzoyl-9,9-dimethyl-6-[5-(2-methyl-4-nitrophenyl)furan-2-yl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H19F7N2O2
(6R,9R)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H19F7N2O2
(6S,9R)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(5R,10bS)-9-bromo-2-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid —— C26H23BrN2O6
6-[(5R,10bS)-9-bromo-2-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid
—— (6R,9S)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H19F7N2O2
(6R,9S)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(5R,10bS)-9-bromo-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid —— C26H23BrN2O5
6-[(5R,10bS)-9-bromo-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-2,3-dimethoxybenzoic acid
—— 6-(aminomethyl)-4-(4-but-2-ynoxyphenyl)sulfonyl-N-hydroxy-2,2-dimethylthiomorpholine-3-carboxamide —— C18H25N3O5S2
6-(aminomethyl)-4-(4-but-2-ynoxyphenyl)sulfonyl-N-hydroxy-2,2-dimethylthiomorpholine-3-carboxamide
—— 6-(p-Anisyl)-2,3-dimethoxy-5,6-dihydro-5,11-diketo-8,9-methylenedioxy-11H-indeno[1,2-c]isoquinoline —— C26H19NO7
6-(p-Anisyl)-2,3-dimethoxy-5,6-dihydro-5,11-diketo-8,9-methylenedioxy-11H-indeno[1,2-c]isoquinoline
—— (6S,9S)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H19F7N2O2
(6S,9S)-9-(4-fluorophenyl)-5-(2,2,2-trifluoroacetyl)-6-[4-(trifluoromethyl)phenyl]-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— [6-(Chloromethyl)-2-(4-fluorophenyl)-4-propan-2-yl-3-[[4-(trifluoromethyl)phenyl]methyl]phenyl]methanol —— C25H23ClF4O
[6-(Chloromethyl)-2-(4-fluorophenyl)-4-propan-2-yl-3-[[4-(trifluoromethyl)phenyl]methyl]phenyl]methanol
—— 6-Methoxy-1-methyl-7-[[(2-phenylpiperidin-3-yl)amino]methyl]-1-(trifluoromethyl)-3,4-dihydroisochromen-4-ol —— C24H29F3N2O3
6-Methoxy-1-methyl-7-[[(2-phenylpiperidin-3-yl)amino]methyl]-1-(trifluoromethyl)-3,4-dihydroisochromen-4-ol
—— 6-(3,5-diphenylpyrazol-4-ylidene)-2-[(3-methoxyphenyl)methyl]-1H-pyridazin-3-one —— C27H22N4O2
6-(3,5-diphenylpyrazol-4-ylidene)-2-[(3-methoxyphenyl)methyl]-1H-pyridazin-3-one
—— 6-methoxy-4-(4-methylquinolin-7-yloxy)-7-(3-(pyrrolidin-1-yl)propoxy)quinazoline —— C26H28N4O3
6-methoxy-4-(4-methylquinolin-7-yloxy)-7-(3-(pyrrolidin-1-yl)propoxy)quinazoline
—— 6-tert-butyl-2-[4-chloro-3-[(4-fluorophenyl)methoxy]phenyl]-1H-benzimidazole —— C24H22ClFN2O
6-tert-butyl-2-[4-chloro-3-[(4-fluorophenyl)methoxy]phenyl]-1H-benzimidazole
—— 6-[6-[6-[Acetyl(hydroxy)amino]hexanoyl-hydroxyamino]hexanoyl-hydroxyamino]hexanoic acid —— C20H37N3O8
6-[6-[6-[Acetyl(hydroxy)amino]hexanoyl-hydroxyamino]hexanoyl-hydroxyamino]hexanoic acid
—— 6-[2-[4-(4-Tert-butylphenoxy)-3-(trifluoromethyl)phenyl]ethynyl]pyridine-3-carboxylic acid —— C25H20F3NO3
6-[2-[4-(4-Tert-butylphenoxy)-3-(trifluoromethyl)phenyl]ethynyl]pyridine-3-carboxylic acid
—— [6-Hydroxy-2-(4-hydroxyphenyl)-1-benzofuran-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]methanone —— C27H25NO5
[6-Hydroxy-2-(4-hydroxyphenyl)-1-benzofuran-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]methanone
—— 6-tert-butyl-2-[4-chloro-3-[(4-fluorophenyl)methoxy]phenyl]-1H-benzimidazole;hydrochloride —— C24H23Cl2FN2O
6-tert-butyl-2-[4-chloro-3-[(4-fluorophenyl)methoxy]phenyl]-1H-benzimidazole;hydrochloride
—— 6-(4-Chlorophenyl)-1-methyl-4-(pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-a][1,3,4]benzotriazepine;hydrochloride —— C22H18Cl2N6
6-(4-Chlorophenyl)-1-methyl-4-(pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-a][1,3,4]benzotriazepine;hydrochloride
—— (6S,9S)-9-[4-(diethylamino)phenyl]-6-phenyl-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C31H30F3N3O2
(6S,9S)-9-[4-(diethylamino)phenyl]-6-phenyl-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(4-Chlorophenyl)-(3-methylimidazol-4-yl)methyl]-1-methyl-4-(3-methylbut-1-ynyl)quinolin-2-one —— C26H24ClN3O
6-[(4-Chlorophenyl)-(3-methylimidazol-4-yl)methyl]-1-methyl-4-(3-methylbut-1-ynyl)quinolin-2-one
—— [6-(N-carbamoyl-2,6-difluoroanilino)-2-(2,4-difluorophenyl)pyridin-3-yl]methyl carbamate —— C20H14F4N4O3
[6-(N-carbamoyl-2,6-difluoroanilino)-2-(2,4-difluorophenyl)pyridin-3-yl]methyl carbamate
—— 6-bromo-3-[(5S)-1-(furan-2-carbonyl)-5-phenylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one —— C29H20BrN3O3
6-bromo-3-[(5S)-1-(furan-2-carbonyl)-5-phenylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one
—— 6-chloro-2-{1-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-piperidin-4-yl}-3H-quinazolin-4-one —— C23H22ClFN4O
6-chloro-2-{1-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-piperidin-4-yl}-3H-quinazolin-4-one
—— (6R)-9,9-dimethyl-6-[5-(4-nitrophenyl)furan-2-yl]-5-(2-phenylacetyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C33H29N3O5
(6R)-9,9-dimethyl-6-[5-(4-nitrophenyl)furan-2-yl]-5-(2-phenylacetyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-(3-methylphenoxy)-2-phenyl-4H-indeno[1,2-d][1,3]thiazole;hydrobromide —— C23H18BrNOS
6-(3-methylphenoxy)-2-phenyl-4H-indeno[1,2-d][1,3]thiazole;hydrobromide
—— 6-bromo-3-[(5R)-1-(furan-2-carbonyl)-5-phenylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one —— C29H20BrN3O3
6-bromo-3-[(5R)-1-(furan-2-carbonyl)-5-phenylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one
—— (6S,9S)-9-(2-ethoxyphenyl)-5-hexanoyl-6-(4-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H38N2O4
(6S,9S)-9-(2-ethoxyphenyl)-5-hexanoyl-6-(4-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6Z)-3-benzyl-6-[[2-bromo-5-(2-methylbut-3-en-2-yl)-1H-imidazol-4-yl]methylidene]piperazine-2,5-dione —— C20H21BrN4O2
(6Z)-3-benzyl-6-[[2-bromo-5-(2-methylbut-3-en-2-yl)-1H-imidazol-4-yl]methylidene]piperazine-2,5-dione
—— 6-[(E)-2-[2,2-diethyl-4-(4-fluorophenyl)-3,4-dihydrochromen-3-yl]ethenyl]-4-hydroxyoxan-2-one —— C26H29FO4
6-[(E)-2-[2,2-diethyl-4-(4-fluorophenyl)-3,4-dihydrochromen-3-yl]ethenyl]-4-hydroxyoxan-2-one
—— (6R,9S)-9-(2-ethoxyphenyl)-5-hexanoyl-6-(4-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H38N2O4
(6R,9S)-9-(2-ethoxyphenyl)-5-hexanoyl-6-(4-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(1E)-4,4-bis(4-fluorophenyl)-3-(furan-2-yl)buta-1,3-dienyl]-4-hydroxyoxan-2-one —— C25H20F2O4
6-[(1E)-4,4-bis(4-fluorophenyl)-3-(furan-2-yl)buta-1,3-dienyl]-4-hydroxyoxan-2-one
—— (6R,9R)-9-(2-ethoxyphenyl)-5-hexanoyl-6-(4-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C34H38N2O4
(6R,9R)-9-(2-ethoxyphenyl)-5-hexanoyl-6-(4-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[[[4-(aminomethyl)phenyl]methylamino]methyl]-2-methyl-2H-1,4-benzoxazin-3-amine —— C18H22N4O
6-[[[4-(aminomethyl)phenyl]methylamino]methyl]-2-methyl-2H-1,4-benzoxazin-3-amine
—— (6R)-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-N-(3,4-dichlorophenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C37H34Cl3N3O4
(6R)-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-N-(3,4-dichlorophenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S,7R)-7-[3-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C21H20BrF3N6O4S3
(6S,7R)-7-[3-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,9S)-5-[2-(1,3-benzothiazol-2-ylsulfanyl)acetyl]-9-(4-methoxyphenyl)-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H27N3O3S3
(6R,9S)-5-[2-(1,3-benzothiazol-2-ylsulfanyl)acetyl]-9-(4-methoxyphenyl)-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,7S)-7-[[(2R)-2-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C21H20BrF3N6O4S3
(6R,7S)-7-[[(2R)-2-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,9R)-5-benzoyl-6,9-bis(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C38H38N2O8
(6S,9R)-5-benzoyl-6,9-bis(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-5-benzoyl-6,9-bis(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C38H38N2O8
(6S,9S)-5-benzoyl-6,9-bis(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,7S)-7-[[(2R)-2-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C21H20BrF3N6O4S3
(6S,7S)-7-[[(2R)-2-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoyl]amino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,9S)-9-phenyl-5-(3,4,5-trimethoxybenzoyl)-6-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C38H38N2O8
(6R,9S)-9-phenyl-5-(3,4,5-trimethoxybenzoyl)-6-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,7S)-7-[3-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C21H20BrF3N6O4S3
(6S,7S)-7-[3-[4-bromo-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]propanoylamino]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6R,9R)-9-phenyl-5-(3,4,5-trimethoxybenzoyl)-6-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C38H38N2O8
(6R,9R)-9-phenyl-5-(3,4,5-trimethoxybenzoyl)-6-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-9-(4-tert-butylphenyl)-6-(3,5-ditert-butyl-4-hydroxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C39H45F3N2O3
(6R,9S)-9-(4-tert-butylphenyl)-6-(3,5-ditert-butyl-4-hydroxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-9-(4-fluorophenyl)-5-(4-methoxybenzoyl)-6-(4-pentoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C38H37FN2O4
(6R,9R)-9-(4-fluorophenyl)-5-(4-methoxybenzoyl)-6-(4-pentoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one