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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[[methyl-[(1R)-1-pyridin-2-ylethyl]amino]methyl]pyridine-2-carboxylic acid —— C15H17N3O2
6-[[methyl-[(1R)-1-pyridin-2-ylethyl]amino]methyl]pyridine-2-carboxylic acid
—— 6-[5-(4-ethylpiperazin-1-yl)sulfonyl-2-propoxypyridin-3-yl]-1-propyl-3-(pyrimidin-2-ylmethyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C27H35N9O4S
6-[5-(4-ethylpiperazin-1-yl)sulfonyl-2-propoxypyridin-3-yl]-1-propyl-3-(pyrimidin-2-ylmethyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[(6R)-4-(furan-2-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]pyrazine-2-carboxamide —— C15H17N5O4
6-[(6R)-4-(furan-2-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]pyrazine-2-carboxamide
—— (6S)-1-[(4-pyrazol-1-ylphenyl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H20N4O2
(6S)-1-[(4-pyrazol-1-ylphenyl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-chloro-N-[3-oxo-2-[(1-pyridin-4-ylpiperidin-4-yl)methylamino]-3-thiomorpholin-4-ylpropyl]naphthalene-2-sulfonamide —— C28H34ClN5O3S2
6-chloro-N-[3-oxo-2-[(1-pyridin-4-ylpiperidin-4-yl)methylamino]-3-thiomorpholin-4-ylpropyl]naphthalene-2-sulfonamide
—— (6R,7R)-7-[[(2Z)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-(cyanomethoxyimino)acetyl]amino]-3-[[3-amino-2-(2-hydroxyethyl)pyrazol-1-ium-1-yl]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate —— C20H20ClN9O6S2
(6R,7R)-7-[[(2Z)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-(cyanomethoxyimino)acetyl]amino]-3-[[3-amino-2-(2-hydroxyethyl)pyrazol-1-ium-1-yl]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
—— (6R)-1-(oxan-4-yl)-4-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)-1,4-diazepan-6-ol —— C17H25N5O2
(6R)-1-(oxan-4-yl)-4-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)-1,4-diazepan-6-ol
—— (6S)-1-[3-(pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane-6-carboxylic acid —— C17H20N4O3
(6S)-1-[3-(pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane-6-carboxylic acid
—— 6-[[(1S)-1-carboxy-2-[4-[(2,6-dichloropyridine-4-carbonyl)amino]phenyl]ethyl]amino]-4-propylsulfonylpyridine-3-carboxylic acid —— C24H22Cl2N4O7S
6-[[(1S)-1-carboxy-2-[4-[(2,6-dichloropyridine-4-carbonyl)amino]phenyl]ethyl]amino]-4-propylsulfonylpyridine-3-carboxylic acid
—— 6-methoxy-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methylsulfinyl]-1H-benzimidazole;(2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid —— C31H33N3O6S
6-methoxy-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methylsulfinyl]-1H-benzimidazole;(2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid
—— (6R)-1-cyclopentyl-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane-6-carboxylic acid —— C16H23N3O3
(6R)-1-cyclopentyl-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane-6-carboxylic acid
—— 6-[2-ethoxy-5-(4-methylpiperazin-1-yl)sulfonylphenyl]-3-(phenylmethoxymethyl)-1-propyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C29H36N6O5S
6-[2-ethoxy-5-(4-methylpiperazin-1-yl)sulfonylphenyl]-3-(phenylmethoxymethyl)-1-propyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— (6R)-1-[3-(pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane-6-carboxylic acid —— C17H20N4O3
(6R)-1-[3-(pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(furan-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-6-carboxylic acid —— C17H19N3O4
(6S)-1-(furan-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-6-carboxylic acid
—— (6R)-5-[6-methyl-2-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-pyrimidin-4-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C18H17N5O3
(6R)-5-[6-methyl-2-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-pyrimidin-4-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6R,7R)-3-[(E)-3-[1,3-dihydroxypropan-2-yl(dimethyl)azaniumyl]prop-1-enyl]-7-[(2-naphthalen-2-ylsulfanylacetyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate —— C27H31N3O6S2
(6R,7R)-3-[(E)-3-[1,3-dihydroxypropan-2-yl(dimethyl)azaniumyl]prop-1-enyl]-7-[(2-naphthalen-2-ylsulfanylacetyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
—— (6R)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H16N6O2
(6R)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-ethyl-4-[(2S)-2-thiophen-2-ylazetidine-1-carbonyl]-1H-pyridin-2-one —— C15H16N2O2S
6-ethyl-4-[(2S)-2-thiophen-2-ylazetidine-1-carbonyl]-1H-pyridin-2-one
—— (6S)-5-[6-methyl-2-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-pyrimidin-4-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C18H17N5O3
(6S)-5-[6-methyl-2-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-pyrimidin-4-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic acid [(S)-2-(thiophene-2-sulfonylamino)-indan-5-yl]-amide —— C28H23F3N2O3S2
6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic acid [(S)-2-(thiophene-2-sulfonylamino)-indan-5-yl]-amide
—— (6R)-1-(furan-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-6-carboxylic acid —— C17H19N3O4
(6R)-1-(furan-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-6-carboxylic acid
—— (6R,7R)-3-chloro-7-[[2-[2,3-difluoro-4-(trifluoromethylsulfonyl)phenyl]sulfanylacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C16H10ClF5N2O6S3
(6R,7R)-3-chloro-7-[[2-[2,3-difluoro-4-(trifluoromethylsulfonyl)phenyl]sulfanylacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— [6-[4-[3-(Aminomethyl)benzoyl]piperazine-1-carbonyl]pyridin-2-yl]-[4-[3-(aminomethyl)benzoyl]piperazin-1-yl]methanone —— C31H35N7O4
[6-[4-[3-(Aminomethyl)benzoyl]piperazine-1-carbonyl]pyridin-2-yl]-[4-[3-(aminomethyl)benzoyl]piperazin-1-yl]methanone
—— (6S)-1-[(4-cyclopentyloxyphenyl)methyl]-1,4-diazepane-6-carboxylic acid —— C18H26N2O3
(6S)-1-[(4-cyclopentyloxyphenyl)methyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H16N6O2
(6S)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-1-cyclopentyl-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane-6-carboxylic acid —— C16H23N3O3
(6S)-1-cyclopentyl-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane-6-carboxylic acid
—— (6S,7S)-3-[(E)-2-[1-(2-amino-2-oxoethyl)pyridin-1-ium-4-yl]sulfanylethenyl]-7-[[(2E)-2-(2-amino-1,3-thiazol-5-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-4-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate —— C21H19N7O6S3
(6S,7S)-3-[(E)-2-[1-(2-amino-2-oxoethyl)pyridin-1-ium-4-yl]sulfanylethenyl]-7-[[(2E)-2-(2-amino-1,3-thiazol-5-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-4-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
—— (6S)-1-[2-(1H-imidazol-5-yl)acetyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H21N5O4
(6S)-1-[2-(1H-imidazol-5-yl)acetyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— (6R,7R)-7-[[2-(2,6-dichloropyridin-4-yl)sulfanylacetyl]amino]-3-[(1-methylpyridin-1-ium-4-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C21H19Cl2N4O4S3+
(6R,7R)-7-[[2-(2,6-dichloropyridin-4-yl)sulfanylacetyl]amino]-3-[(1-methylpyridin-1-ium-4-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6-Acetyl-3-cyclohexyl-4-oxo-1-phenyl-2-sulfanylidenethieno[2,3-d]pyrimidin-5-yl) 2,4-dichlorobenzoate —— C27H22Cl2N2O4S2
(6-Acetyl-3-cyclohexyl-4-oxo-1-phenyl-2-sulfanylidenethieno[2,3-d]pyrimidin-5-yl) 2,4-dichlorobenzoate
—— (6R)-1-[(4-cyclopentyloxyphenyl)methyl]-1,4-diazepane-6-carboxylic acid —— C18H26N2O3
(6R)-1-[(4-cyclopentyloxyphenyl)methyl]-1,4-diazepane-6-carboxylic acid
—— (6R)-1-[6-(2-hydroxyethylamino)pyrimidin-4-yl]-4-pent-2-ynyl-1,4-diazepane-6-carboxylic acid —— C17H25N5O3
(6R)-1-[6-(2-hydroxyethylamino)pyrimidin-4-yl]-4-pent-2-ynyl-1,4-diazepane-6-carboxylic acid
—— [6-(N-carbamoyl-2,6-difluoroanilino)-2-(2,4-difluorophenyl)pyridin-3-yl]methyl N-(2-piperazin-1-ylethyl)carbamate —— C26H26F4N6O3
[6-(N-carbamoyl-2,6-difluoroanilino)-2-(2,4-difluorophenyl)pyridin-3-yl]methyl N-(2-piperazin-1-ylethyl)carbamate
—— (6R)-1-[3-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)propanoyl]-1,4-diazepane-6-carboxylic acid —— C16H19N5O4
(6R)-1-[3-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)propanoyl]-1,4-diazepane-6-carboxylic acid
—— (6S)-6-hydroxy-N-[3-(2-methoxyphenyl)phenyl]-1,4-oxazepane-4-carboxamide —— C19H22N2O4
(6S)-6-hydroxy-N-[3-(2-methoxyphenyl)phenyl]-1,4-oxazepane-4-carboxamide
—— (6R)-6-hydroxy-N-[3-(2-methoxyphenyl)phenyl]-1,4-oxazepane-4-carboxamide —— C19H22N2O4
(6R)-6-hydroxy-N-[3-(2-methoxyphenyl)phenyl]-1,4-oxazepane-4-carboxamide
—— (6R,8R)-6-(3-fluorophenyl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]quinolin-8-amine —— C16H15FN2O2
(6R,8R)-6-(3-fluorophenyl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]quinolin-8-amine
—— (6S)-1-(1H-imidazol-2-ylmethyl)-4-[2-(5-methyl-3,4-dihydropyrazol-2-yl)acetyl]-1,4-diazepane-6-carboxylic acid —— C16H24N6O3
(6S)-1-(1H-imidazol-2-ylmethyl)-4-[2-(5-methyl-3,4-dihydropyrazol-2-yl)acetyl]-1,4-diazepane-6-carboxylic acid
—— [6-[[Tert-butyl(dimethyl)silyl]oxymethyl]-2-(4-fluorophenyl)-4-propan-2-yl-3-[[4-(trifluoromethyl)phenyl]methyl]phenyl]methanol —— C31H38F4O2Si
[6-[[Tert-butyl(dimethyl)silyl]oxymethyl]-2-(4-fluorophenyl)-4-propan-2-yl-3-[[4-(trifluoromethyl)phenyl]methyl]phenyl]methanol
—— 6-[4-[(1R)-1-(dimethylamino)ethyl]phenyl]-N-propan-2-ylpyridazin-3-amine —— C17H24N4
6-[4-[(1R)-1-(dimethylamino)ethyl]phenyl]-N-propan-2-ylpyridazin-3-amine
—— (6S)-6-(3,4-difluorophenyl)-6,7-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-8-one —— C16H11F2NO3
(6S)-6-(3,4-difluorophenyl)-6,7-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-8-one
—— (6R)-N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide —— C16H20N4O4
(6R)-N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
—— (6R)-2-amino-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one —— C8H11N3O
(6R)-2-amino-6-methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-one
—— (6S)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine —— C8H9ClN2
(6S)-4-chloro-6-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidine
—— 6-methyl-3-[(3R)-3-phenylpiperazine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one —— C20H20N4O2
6-methyl-3-[(3R)-3-phenylpiperazine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one
—— (6R,7R)-7-[[(2Z)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-3-[(E)-2-(1H-1,2,4-triazol-5-ylsulfanyl)ethenyl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C16H13ClN8O5S3
(6R,7R)-7-[[(2Z)-2-(2-amino-5-chloro-1,3-thiazol-4-yl)-2-hydroxyiminoacetyl]amino]-8-oxo-3-[(E)-2-(1H-1,2,4-triazol-5-ylsulfanyl)ethenyl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,8S)-6-(3-fluorophenyl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]quinolin-8-amine —— C16H15FN2O2
(6S,8S)-6-(3-fluorophenyl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]quinolin-8-amine
—— 6-(diaminomethylideneamino)-N-[(2S)-3-naphthalen-2-yl-1-oxo-1-[[(3S,4S)-2-oxo-4-phenoxyazetidin-3-yl]amino]propan-2-yl]hexanamide —— C29H34N6O4
6-(diaminomethylideneamino)-N-[(2S)-3-naphthalen-2-yl-1-oxo-1-[[(3S,4S)-2-oxo-4-phenoxyazetidin-3-yl]amino]propan-2-yl]hexanamide
—— (6S)-1-[3-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)propanoyl]-1,4-diazepane-6-carboxylic acid —— C16H19N5O4
(6S)-1-[3-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)propanoyl]-1,4-diazepane-6-carboxylic acid
—— (6R)-6-(3,4-difluorophenyl)-6,7-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-8-one —— C16H11F2NO3
(6R)-6-(3,4-difluorophenyl)-6,7-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-8-one