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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[methyl-[(2R)-1-[(R)-methylsulfinyl]propan-2-yl]amino]pyridine-3-carbonitrile —— C11H15N3OS
6-[methyl-[(2R)-1-[(R)-methylsulfinyl]propan-2-yl]amino]pyridine-3-carbonitrile
—— 6-[methyl-[(2S)-1-[(R)-methylsulfinyl]propan-2-yl]amino]pyridine-3-carbonitrile —— C11H15N3OS
6-[methyl-[(2S)-1-[(R)-methylsulfinyl]propan-2-yl]amino]pyridine-3-carbonitrile
—— (6-fluoro-1H-benzimidazol-4-yl)-[(3R)-3-(2-methyl-1,3-dioxolan-2-yl)piperidin-1-yl]methanone —— C17H20FN3O3
(6-fluoro-1H-benzimidazol-4-yl)-[(3R)-3-(2-methyl-1,3-dioxolan-2-yl)piperidin-1-yl]methanone
—— (6-fluoro-1H-benzimidazol-4-yl)-[(3S)-3-(2-methyl-1,3-dioxolan-2-yl)piperidin-1-yl]methanone —— C17H20FN3O3
(6-fluoro-1H-benzimidazol-4-yl)-[(3S)-3-(2-methyl-1,3-dioxolan-2-yl)piperidin-1-yl]methanone
—— 6,8-dibromo-3-[(Z)-3-(2-chlorophenyl)prop-2-enoyl]chromen-2-one —— C18H9Br2ClO3
6,8-dibromo-3-[(Z)-3-(2-chlorophenyl)prop-2-enoyl]chromen-2-one
—— 6-[4-[[(3S)-thian-3-yl]amino]cyclohexyl]oxypyridine-3-carbonitrile —— C17H23N3OS
6-[4-[[(3S)-thian-3-yl]amino]cyclohexyl]oxypyridine-3-carbonitrile
—— 6-[4-[[(3R)-thian-3-yl]amino]cyclohexyl]oxypyridine-3-carbonitrile —— C17H23N3OS
6-[4-[[(3R)-thian-3-yl]amino]cyclohexyl]oxypyridine-3-carbonitrile
—— 6-[4-[[(3R)-thian-3-yl]amino]piperidin-1-yl]pyridine-3-carbonitrile —— C16H22N4S
6-[4-[[(3R)-thian-3-yl]amino]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[4-[[(3S)-thian-3-yl]amino]piperidin-1-yl]pyridine-3-carbonitrile —— C16H22N4S
6-[4-[[(3S)-thian-3-yl]amino]piperidin-1-yl]pyridine-3-carbonitrile
—— (6R)-1-[(2-aminopyridin-3-yl)methyl]-4-(7H-purin-6-yl)-1,4-diazepan-6-ol —— C16H20N8O
(6R)-1-[(2-aminopyridin-3-yl)methyl]-4-(7H-purin-6-yl)-1,4-diazepan-6-ol
—— (6R)-5-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H22N6O2
(6R)-5-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6R)-1-(1H-imidazol-5-ylmethyl)-4-(2-methoxyacetyl)-1,4-diazepane-6-carboxylic acid —— C13H20N4O4
(6R)-1-(1H-imidazol-5-ylmethyl)-4-(2-methoxyacetyl)-1,4-diazepane-6-carboxylic acid
—— (6S)-1-(1H-imidazol-5-ylmethyl)-4-(2-methoxyacetyl)-1,4-diazepane-6-carboxylic acid —— C13H20N4O4
(6S)-1-(1H-imidazol-5-ylmethyl)-4-(2-methoxyacetyl)-1,4-diazepane-6-carboxylic acid
—— 6-[(5S)-9-acetyl-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyrazine-2-carboxylic acid —— C17H24N4O4
6-[(5S)-9-acetyl-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyrazine-2-carboxylic acid
—— (6S)-5-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C17H22N6O2
(6S)-5-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— 6-[(5R)-9-acetyl-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyrazine-2-carboxylic acid —— C17H24N4O4
6-[(5R)-9-acetyl-5-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyrazine-2-carboxylic acid
—— (6R)-1-cyclopentyl-4-[(5-methyl-1H-imidazol-4-yl)methyl]-1,4-diazepane-6-carboxylic acid —— C16H26N4O2
(6R)-1-cyclopentyl-4-[(5-methyl-1H-imidazol-4-yl)methyl]-1,4-diazepane-6-carboxylic acid
—— 6-(dimethylamino)-N-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]pyridine-3-carboxamide —— C16H23N5O
6-(dimethylamino)-N-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]pyridine-3-carboxamide
—— [6-[4-[(1R)-1-ethoxyethyl]phenyl]pyridin-3-yl]-morpholin-4-ylmethanone —— C20H24N2O3
[6-[4-[(1R)-1-ethoxyethyl]phenyl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-propyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H31N3O4S
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-propyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— [6-[4-[(1S)-1-ethoxyethyl]phenyl]pyridin-3-yl]-morpholin-4-ylmethanone —— C20H24N2O3
[6-[4-[(1S)-1-ethoxyethyl]phenyl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-propyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H31N3O4S
6-cyclopropyl-3-(2,2-dimethylpropyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-propyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-cyclopropyl-N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C22H32N4O4S
6-cyclopropyl-N-[3-(dimethylamino)propyl]-N-[(3R)-1,1-dioxothiolan-3-yl]-3-propan-2-yl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6S)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one —— C28H38N4O3
(6S)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
—— (6R)-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-1-[(1-methylpyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one —— C26H31N5O4
(6R)-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-1-[(1-methylpyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
—— (6S)-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-1-[(1-methylpyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one —— C26H31N5O4
(6S)-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-1-[(1-methylpyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
—— (6R)-1-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-1,4-diazepane-6-carboxylic acid —— C16H21N3O3
(6R)-1-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-1,4-diazepane-6-carboxylic acid
—— 6-[[(2R)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid —— C17H19N5O3
6-[[(2R)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
—— (6S)-1-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-1,4-diazepane-6-carboxylic acid —— C16H21N3O3
(6S)-1-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-1,4-diazepane-6-carboxylic acid
—— 6-[[(2S)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid —— C17H19N5O3
6-[[(2S)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
—— 6-[4-[(1S)-1-(dimethylamino)ethyl]phenyl]-N,N-dimethylpyrazine-2-carboxamide —— C17H22N4O
6-[4-[(1S)-1-(dimethylamino)ethyl]phenyl]-N,N-dimethylpyrazine-2-carboxamide
—— (6S)-1-cyclohexyl-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one —— C27H35N3O4
(6S)-1-cyclohexyl-4-[(Z)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
—— [(6S)-6-hydroxy-4-(7H-purin-6-yl)-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone —— C15H17N7O2
[(6S)-6-hydroxy-4-(7H-purin-6-yl)-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone
—— (6S)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one —— C27H33N5O2S
(6S)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
—— 6-(oxan-4-yl)-3-[(Z)-2-phenylethenyl]-1-(pyridin-2-ylmethyl)-7,8-dihydro-5H-1,6-naphthyridin-2-one —— C27H29N3O2
6-(oxan-4-yl)-3-[(Z)-2-phenylethenyl]-1-(pyridin-2-ylmethyl)-7,8-dihydro-5H-1,6-naphthyridin-2-one
—— 6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(Z)-3-phenylprop-2-enyl]-3-pyridin-4-yl-7,8-dihydro-5H-1,6-naphthyridin-2-one —— C31H29N3O2
6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(Z)-3-phenylprop-2-enyl]-3-pyridin-4-yl-7,8-dihydro-5H-1,6-naphthyridin-2-one
—— (6R)-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-[(Z)-3-phenylprop-2-enyl]-1,4-diazepan-2-one —— C22H31N3O3
(6R)-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-[(Z)-3-phenylprop-2-enyl]-1,4-diazepan-2-one
—— 6-[4-[(1R)-1-(dimethylamino)ethyl]phenyl]-N,N-dimethylpyrazine-2-carboxamide —— C17H22N4O
6-[4-[(1R)-1-(dimethylamino)ethyl]phenyl]-N,N-dimethylpyrazine-2-carboxamide
—— (6S)-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-[(Z)-3-phenylprop-2-enyl]-1,4-diazepan-2-one —— C22H31N3O3
(6S)-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-[(Z)-3-phenylprop-2-enyl]-1,4-diazepan-2-one
—— (6S)-1-benzyl-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-6-methoxy-1,4-diazepan-2-one —— C24H31N3O2
(6S)-1-benzyl-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-6-methoxy-1,4-diazepan-2-one
—— (6R)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one —— C27H33N5O2S
(6R)-4-[(Z)-3-[4-(dimethylamino)phenyl]prop-2-enyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
—— 6-chloro-N-[3-[(3S)-3-(hydroxymethyl)piperidin-1-yl]propyl]-2-methylquinoline-4-carboxamide —— C20H26ClN3O2
6-chloro-N-[3-[(3S)-3-(hydroxymethyl)piperidin-1-yl]propyl]-2-methylquinoline-4-carboxamide
—— 6-methyl-3-[(2E)-2-[1-(4-methyl-3-nitrophenyl)ethylidene]hydrazinyl]-4H-1,2,4-triazin-5-one —— C13H14N6O3
6-methyl-3-[(2E)-2-[1-(4-methyl-3-nitrophenyl)ethylidene]hydrazinyl]-4H-1,2,4-triazin-5-one
—— (6R)-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C15H18N4O2S
(6R)-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— [(6R)-4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone —— C19H23N3O2
[(6R)-4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone
—— (6S)-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C15H18N4O2S
(6S)-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (6S)-1-[2-(methylamino)acetyl]-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid —— C14H25N3O4
(6S)-1-[2-(methylamino)acetyl]-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
—— [(6S)-4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone —— C19H23N3O2
[(6S)-4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-(1H-pyrrol-3-yl)methanone
—— 6-chloro-N-[3-[(3R)-3-(hydroxymethyl)piperidin-1-yl]propyl]-2-methylquinoline-4-carboxamide —— C20H26ClN3O2
6-chloro-N-[3-[(3R)-3-(hydroxymethyl)piperidin-1-yl]propyl]-2-methylquinoline-4-carboxamide
—— 6-(2-hydroxyethyl)-N-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H22N4O2
6-(2-hydroxyethyl)-N-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide